piperidines and efaproxiral

piperidines has been researched along with efaproxiral* in 2 studies

Other Studies

2 other study(ies) available for piperidines and efaproxiral

ArticleYear
Trimethylaluminium mediated amide bond formation in a continuous flow microreactor as key to the synthesis of rimonabant and efaproxiral.
    Chemical communications (Cambridge, England), 2008, Mar-07, Issue:9

    A safe, functional-group-tolerant and high-throughput version of the trimethylaluminium mediated amide bond formation reaction has been developed in a microreactor system; rimonabant and efaproxiral were prepared to illustrate the utility of the method.

    Topics: Alkanes; Aluminum; Amides; Aniline Compounds; Equipment Design; Microwaves; Miniaturization; Molecular Structure; Piperidines; Propionates; Pyrazoles; Rimonabant; Stereoisomerism

2008
Hit to Lead Success Stories--IBC Conference: Effective chemistry strategies for reducing attrition rates and speeding lead compounds into the pipeline. 31 January-1 February 2005, San Diego, CA, USA.
    IDrugs : the investigational drugs journal, 2005, Volume: 8, Issue:3

    Topics: Aniline Compounds; Bradykinin; Drug Approval; Drug Design; Drug Evaluation; Humans; Molecular Structure; Piperidines; Propionates; Pyridines; Time Factors

2005