piperidines and chloroethylnorapomorphine

piperidines has been researched along with chloroethylnorapomorphine* in 1 studies

Other Studies

1 other study(ies) available for piperidines and chloroethylnorapomorphine

Article	Year
Assessment of the chloroethyl analog of 3-PPP (N-n-propyl-3-(3-hydroxyphenyl)-piperidine), 3-PPP-C1 as an irreversible ligand for central dopaminergic recognition sites. European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3 NCA, the chloro analog of the potent dopamine agonist NPA is an irreversible ligand at dopamine receptors in mammalian brain. The chloroethyl analog of the recently described putative dopamine autoreceptor agonist 3-PPP, 3-PPP-C1, was evaluated for its potential use as an irreversible autoreceptor ligand. N-Chloroethylation of 3-PPP reduced the intrinsic affinity of the agonist seven-fold and, consequently, in contrast to NCA, it was found that 3-PPP-C1 was not a good irreversible ligand at dopamine receptors. Topics: Animals; Aporphines; Brain; In Vitro Techniques; Ligands; Piperidines; Rats; Receptors, Dopamine	1983

Article

Year

Assessment of the chloroethyl analog of 3-PPP (N-n-propyl-3-(3-hydroxyphenyl)-piperidine), 3-PPP-C1 as an irreversible ligand for central dopaminergic recognition sites.

European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

NCA, the chloro analog of the potent dopamine agonist NPA is an irreversible ligand at dopamine receptors in mammalian brain. The chloroethyl analog of the recently described putative dopamine autoreceptor agonist 3-PPP, 3-PPP-C1, was evaluated for its potential use as an irreversible autoreceptor ligand. N-Chloroethylation of 3-PPP reduced the intrinsic affinity of the agonist seven-fold and, consequently, in contrast to NCA, it was found that 3-PPP-C1 was not a good irreversible ligand at dopamine receptors.

Topics: Animals; Aporphines; Brain; In Vitro Techniques; Ligands; Piperidines; Rats; Receptors, Dopamine

1983