Page last updated: 2024-08-18

piperidine and sr 142801

piperidine has been researched along with sr 142801 in 1 studies

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bissantz, C; Kratzeisen, C; Malherbe, P; Marcuz, A; Nettekoven, MH; Ratni, H; Wettstein, JG; Zenner, MT1

Other Studies

1 other study(ies) available for piperidine and sr 142801

ArticleYear
Identification of a critical residue in the transmembrane domain 2 of tachykinin neurokinin 3 receptor affecting the dissociation kinetics and antagonism mode of osanetant (SR 142801) and piperidine-based structures.
    Journal of medicinal chemistry, 2009, Nov-26, Volume: 52, Issue:22

    Topics: Amino Acid Sequence; Animals; Cattle; Cell Line; Cell Membrane; Dogs; Guinea Pigs; Humans; Inositol Phosphates; Isotope Labeling; Kinetics; Models, Molecular; Molecular Conformation; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Piperidines; Protein Structure, Tertiary; Rats; Receptors, Neurokinin-3; Reproducibility of Results; Tritium

2009