Page last updated: 2024-08-16

piperazine and pyrazole

piperazine has been researched along with pyrazole in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Fotsch, C; St Jean, DJ1
Batista, DC; Cardoso, CS; Costa, EA; Florentino, IF; Gonçalves, MP; Lião, LM; Menegatti, R; Sanz, G; Silva, DPB; Valadares, MC; Vaz, BG1
Mekky, AEM; Sanad, SMH1

Reviews

1 review(s) available for piperazine and pyrazole

ArticleYear
Mitigating heterocycle metabolism in drug discovery.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats

2012

Other Studies

2 other study(ies) available for piperazine and pyrazole

ArticleYear
Anti-inflammatory effect of a new piperazine derivative: (4-methylpiperazin-1-yl)(1-phenyl-1H-pyrazol-4-yl)methanone.
    Inflammopharmacology, 2018, Volume: 26, Issue:1

    Topics: Analgesics; Animals; Anti-Inflammatory Agents; BALB 3T3 Cells; Carrageenan; Cell Line; Cell Movement; Edema; Female; Interleukin-1beta; Mice; Pain; Pain Measurement; Piperazine; Piperazines; Pleurisy; Pyrazoles; Tumor Necrosis Factor-alpha

2018
Novel bis(pyrazole-benzofuran) hybrids possessing piperazine linker: Synthesis of potent bacterial biofilm and MurB inhibitors.
    Bioorganic chemistry, 2020, Volume: 102

    Topics: Anti-Bacterial Agents; Antineoplastic Agents; Benzofurans; Biofilms; Carbohydrate Dehydrogenases; Cell Line; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Bacterial; Drug Screening Assays, Antitumor; Enterococcus faecalis; Escherichia coli; Humans; Microbial Sensitivity Tests; Molecular Structure; Piperazine; Pyrazoles; Staphylococcus aureus; Structure-Activity Relationship

2020