Page last updated: 2024-08-16

piperazine and amg 511

piperazine has been researched along with amg 511 in 1 studies

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, KL; Cee, VJ; Hong, FT; Hughes, PE; Jiang, J; Lanman, BA; McCarter, JD; Mullady, EL; Norman, MH; Pettus, LH; Reed, AB; San Miguel, T; Subramanian, R; Tasker, AS; Wang, L; Whittington, DA; Wu, T; Wurz, RP; Zalameda, L; Zhang, N1

Other Studies

1 other study(ies) available for piperazine and amg 511

ArticleYear
Phosphoinositide-3-kinase inhibitors: evaluation of substituted alcohols as replacements for the piperazine sulfonamide portion of AMG 511.
    Bioorganic & medicinal chemistry letters, 2014, Dec-15, Volume: 24, Issue:24

    Topics: Alcohols; Animals; Female; Half-Life; Liver; Male; Mice; Mice, Nude; Molecular Conformation; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Piperazine; Piperazines; Protein Binding; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Pyridines; Rats; Rats, Sprague-Dawley; Signal Transduction; Structure-Activity Relationship; Sulfonamides; TOR Serine-Threonine Kinases; Triazines

2014