Page last updated: 2024-09-03

piperaquine and nitd 609

piperaquine has been researched along with nitd 609 in 5 studies

Compound Research Comparison

Studies
(piperaquine)
Trials
(piperaquine)
Recent Studies (post-2010)
(piperaquine)
Studies
(nitd 609)
Trials
(nitd 609)
Recent Studies (post-2010) (nitd 609)
63822749746742

Protein Interaction Comparison

ProteinTaxonomypiperaquine (IC50)nitd 609 (IC50)
Adenosine receptor A3Homo sapiens (human)8.3

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (80.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Biamonte, MA; Le Roch, KG; Wanner, J1
Fidock, DA; Flannery, EL; Winzeler, EA1
Ashton, TD; Burrows, JN; Charman, SA; Creek, DJ; Devine, SM; Laleu, B; Möhrle, JJ; Sleebs, BE1
Griffin, P; Jain, JP; Kangas, M; Lefèvre, G; Lickliter, J; Machineni, S; Stein, DS1
Akakpo, S; Chalon, S; Chughlay, MF; Csermak-Renner, K; Djeriou, E; Gaur, AH; Leboulleux, D; McCarthy, J; Odedra, A; Shanks, GD; Winnips, C1

Reviews

3 review(s) available for piperaquine and nitd 609

ArticleYear
Recent advances in malaria drug discovery.
    Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure

2013
Using genetic methods to define the targets of compounds with antimalarial activity.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum

2013
The Development Process for Discovery and Clinical Advancement of Modern Antimalarials.
    Journal of medicinal chemistry, 2019, 12-12, Volume: 62, Issue:23

    Topics: Antimalarials; Drug Discovery; Humans; Malaria; Molecular Structure; Plasmodium

2019

Trials

1 trial(s) available for piperaquine and nitd 609

ArticleYear
Open-label, single-dose, parallel-group study in healthy volunteers to determine the drug-drug interaction potential between KAE609 (cipargamin) and piperaquine.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:6

    Topics: Adolescent; Adult; Dose-Response Relationship, Drug; Drug Interactions; Female; Healthy Volunteers; Humans; Indoles; Male; Middle Aged; Quinolines; Spiro Compounds; Young Adult

2015

Other Studies

1 other study(ies) available for piperaquine and nitd 609

ArticleYear
Liver Enzyme Elevations in
    The American journal of tropical medicine and hygiene, 2020, Volume: 103, Issue:1

    Topics: Acrylamides; Adamantane; Adult; Alanine Transaminase; Aminopyridines; Aminoquinolines; Antimalarials; Aspartate Aminotransferases; Chemical and Drug Induced Liver Injury; Erythrocyte Transfusion; Erythrocytes; Female; Ferrous Compounds; Healthy Volunteers; Heterocyclic Compounds, 4 or More Rings; Humans; Indoles; Isoquinolines; Malaria, Falciparum; Male; Metallocenes; Parasitemia; Peroxides; Piperazines; Plasmodium falciparum; Primaquine; Pyrimidines; Quinolines; Spiro Compounds; Sulfones; Triazoles; Young Adult

2020