piperaquine has been researched along with nitd 609 in 5 studies
Studies (piperaquine) | Trials (piperaquine) | Recent Studies (post-2010) (piperaquine) | Studies (nitd 609) | Trials (nitd 609) | Recent Studies (post-2010) (nitd 609) |
---|---|---|---|---|---|
638 | 227 | 497 | 46 | 7 | 42 |
Protein | Taxonomy | piperaquine (IC50) | nitd 609 (IC50) |
---|---|---|---|
Adenosine receptor A3 | Homo sapiens (human) | 8.3 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 4 (80.00) | 24.3611 |
2020's | 1 (20.00) | 2.80 |
Authors | Studies |
---|---|
Biamonte, MA; Le Roch, KG; Wanner, J | 1 |
Fidock, DA; Flannery, EL; Winzeler, EA | 1 |
Ashton, TD; Burrows, JN; Charman, SA; Creek, DJ; Devine, SM; Laleu, B; Möhrle, JJ; Sleebs, BE | 1 |
Griffin, P; Jain, JP; Kangas, M; Lefèvre, G; Lickliter, J; Machineni, S; Stein, DS | 1 |
Akakpo, S; Chalon, S; Chughlay, MF; Csermak-Renner, K; Djeriou, E; Gaur, AH; Leboulleux, D; McCarthy, J; Odedra, A; Shanks, GD; Winnips, C | 1 |
3 review(s) available for piperaquine and nitd 609
Article | Year |
---|---|
Recent advances in malaria drug discovery.
Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure | 2013 |
Using genetic methods to define the targets of compounds with antimalarial activity.
Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum | 2013 |
The Development Process for Discovery and Clinical Advancement of Modern Antimalarials.
Topics: Antimalarials; Drug Discovery; Humans; Malaria; Molecular Structure; Plasmodium | 2019 |
1 trial(s) available for piperaquine and nitd 609
Article | Year |
---|---|
Open-label, single-dose, parallel-group study in healthy volunteers to determine the drug-drug interaction potential between KAE609 (cipargamin) and piperaquine.
Topics: Adolescent; Adult; Dose-Response Relationship, Drug; Drug Interactions; Female; Healthy Volunteers; Humans; Indoles; Male; Middle Aged; Quinolines; Spiro Compounds; Young Adult | 2015 |
1 other study(ies) available for piperaquine and nitd 609
Article | Year |
---|---|
Liver Enzyme Elevations in
Topics: Acrylamides; Adamantane; Adult; Alanine Transaminase; Aminopyridines; Aminoquinolines; Antimalarials; Aspartate Aminotransferases; Chemical and Drug Induced Liver Injury; Erythrocyte Transfusion; Erythrocytes; Female; Ferrous Compounds; Healthy Volunteers; Heterocyclic Compounds, 4 or More Rings; Humans; Indoles; Isoquinolines; Malaria, Falciparum; Male; Metallocenes; Parasitemia; Peroxides; Piperazines; Plasmodium falciparum; Primaquine; Pyrimidines; Quinolines; Spiro Compounds; Sulfones; Triazoles; Young Adult | 2020 |