Page last updated: 2024-09-03

piperaquine and halofantrine

piperaquine has been researched along with halofantrine in 5 studies

Compound Research Comparison

Studies
(piperaquine)
Trials
(piperaquine)
Recent Studies (post-2010)
(piperaquine)
Studies
(halofantrine)
Trials
(halofantrine)
Recent Studies (post-2010) (halofantrine)
6382274974866849

Protein Interaction Comparison

ProteinTaxonomypiperaquine (IC50)halofantrine (IC50)
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)1.9
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)1.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.1622
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)1.9
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)1.9

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19902 (40.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's1 (20.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Masseno, V; Muriithi, S; Nzila, A1
Coulanges, P; Deloron, P; Le Bras, J; Ramanamirija, JA1
Biaud, JM; Coulanges, P; Deloron, P; Le Bras, J; Ramanamirija, JA1
Raju, KS; Singh, SP; Taneja, I; Wahajuddin, M1
Amalvict, R; Benoit, N; Chevalier, A; Delaunay, P; Fonta, I; Jeandel, PY; Madamet, M; Marty, P; Massamba, L; Mondain, V; Mosnier, J; Pomares, C; Pradines, B1

Other Studies

5 other study(ies) available for piperaquine and halofantrine

ArticleYear
In vitro chemosensitization of Plasmodium falciparum to antimalarials by verapamil and probenecid.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:7

    Topics: Adjuvants, Pharmaceutic; Animals; Antimalarials; Parasitic Sensitivity Tests; Plasmodium falciparum; Probenecid; Verapamil

2009
Plasmodium falciparum in Madagascar: in vivo and in vitro sensitivity to seven drugs.
    Annals of tropical medicine and parasitology, 1985, Volume: 79, Issue:4

    Topics: Adolescent; Adult; Aged; Amodiaquine; Antimalarials; Child; Child, Preschool; Chloroquine; Humans; Infant; Madagascar; Malaria; Mefloquine; Microbial Sensitivity Tests; Middle Aged; Phenanthrenes; Piperazines; Plasmodium falciparum; Quinine; Quinolines

1985
[In vivo and in vitro sensitivity to 4-aminoquinolines of Plasmodium falciparum in Madagascar: results of 2 years' study].
    Bulletin de la Societe de pathologie exotique et de ses filiales, 1985, Volume: 78, Issue:5

    Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; In Vitro Techniques; Madagascar; Malaria; Phenanthrenes; Piperazines; Plasmodium falciparum; Quinine; Quinolines

1985
Assessment of pharmacokinetic compatibility of short acting CDRI candidate trioxane derivative, 99-411, with long acting prescription antimalarials, lumefantrine and piperaquine.
    Scientific reports, 2015, Nov-25, Volume: 5

    Topics: Animals; Antimalarials; Chromatography, High Pressure Liquid; Ethanolamines; Fluorenes; Half-Life; Heterocyclic Compounds; Humans; Lumefantrine; Microsomes, Liver; Phenanthrenes; Quinolines; Rats; Spiro Compounds; Tandem Mass Spectrometry

2015
Late clinical failure associated with cytochrome b codon 268 mutation during treatment of falciparum malaria with atovaquone-proguanil in traveller returning from Congo.
    Malaria journal, 2020, Jan-21, Volume: 19, Issue:1

    Topics: Antimalarials; Artemisinins; Atovaquone; Codon; Congo; Cytochromes b; Drug Combinations; Drug Resistance; Female; France; Humans; Malaria, Falciparum; Middle Aged; Mutation; Phenanthrenes; Plasmodium falciparum; Proguanil; Quinolines; Tetrahydrofolate Dehydrogenase; Travel

2020