pipequaline has been researched along with pk 9084 in 13 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 12 (92.31) | 18.7374 |
1990's | 1 (7.69) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
File, SE; Wilks, L | 1 |
File, SE; Pellow, S | 1 |
Gee, KW | 1 |
Le Fur, G | 1 |
File, SE; Lister, RG | 1 |
Gee, KW; Yamamura, HI | 1 |
Keane, PE; Morre, M; Simiand, J | 1 |
File, SE | 2 |
Burgevin, MC; Ferris, O; Gauthier, A; Guérémy, C; Heaulme, M; Le Fur, G; Mizoule, J; Uzan, A | 1 |
Brinton, RE; Gee, KW; Yamamura, HI | 1 |
File, SE; Simmonds, MA | 1 |
Chen, JS; Gee, KW; Johnson, D; Lan, NC | 1 |
13 other study(ies) available for pipequaline and pk 9084
Article | Year |
---|---|
Effects of acute and chronic treatment on the pro- and anti-convulsant actions of CL 218, 872, PK 8165 and PK 9084, putative ligands for the benzodiazepine receptor.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Male; Mice; Pentylenetetrazole; Picrotoxin; Pyridazines; Quinolines; Receptors, GABA-A; Time Factors | 1985 |
The effects of putative anxiolytic compounds (PK 8165, PK 9084 and tracazolate) on the rat corticosterone response.
Topics: Animals; Anti-Anxiety Agents; Corticosterone; Male; Pyrazoles; Quinolines; Rats; Receptors, GABA-A; Stress, Psychological | 1985 |
Phenylquinolines PK 8165 and PK 9084 allosterically modulate [35S]t-butylbicyclophosphorothionate binding to a chloride ionophore in rat brain via a novel Ro5 4864 binding site.
Topics: Animals; Anticonvulsants; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Convulsants; gamma-Aminobutyric Acid; Kinetics; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
[Anxiety receptors: new pharmacological approach (author's transl)].
Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Binding, Competitive; Brain; Chlordiazepoxide; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Quinolines; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Seizures | 1982 |
Quinolines and anxiety: anxiogenic effects of CGS 8216 and partial anxiolytic profile of PK 9084.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Humans; Male; Motor Activity; Pyrazoles; Quinolines; Rats; Social Behavior | 1983 |
Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes?
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Cerebral Cortex; Drug Interactions; Flunitrazepam; Male; Postural Balance; Pyrazoles; Pyridazines; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Temperature | 1983 |
The quinolines PK 8165 and PK 9084 possess benzodiazepine-like activity in vitro but not in vivo.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Modification of seizures elicited by the benzodiazepine Ro 5-3663--a comparison with picrotoxin.
Topics: Animals; Benzodiazepinones; Chemical Phenomena; Chemistry; Convulsants; Diazepam; Drug Synergism; Flumazenil; Male; Mice; Picrotoxin; Pyrazoles; Quinolines; Seizures | 1984 |
Multiple benzodiazepine receptors: evidence of dissociation between anticonflict and anticonvulsant properties by PK 8165 and PK 9084 (two quinoline derivatives).
Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Cerebellar Cortex; Chlordiazepoxide; Conflict, Psychological; Cyclic AMP; Cyclic GMP; Diazepam; Hypnotics and Sedatives; Kinetics; Male; Motor Activity; Piperazines; Quinolines; Rats; Receptors, Drug; Receptors, GABA-A | 1981 |
PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam.
Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Diazepam; Drug Antagonism; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Quinolines; Receptors, Cell Surface; Receptors, GABA-A; Seizures | 1983 |
Interactions of two phenylquinolines with picrotoxin and benzodiazepines in vivo and in vitro.
Topics: Animals; Anticonvulsants; Benzodiazepines; Drug Interactions; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Myoclonus; Pentylenetetrazole; Picrotoxin; Quinolines; Rats; Rats, Inbred Strains; Seizures | 1984 |
Sedative effects of PK 9084 and PK 8165, alone and in combination with chlordiazepoxide.
Topics: Animals; Behavior, Animal; Body Temperature; Chlordiazepoxide; Drug Interactions; Exploratory Behavior; Hypnotics and Sedatives; Male; Motor Activity; Quinolines; Rats | 1983 |
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection | 1995 |