Page last updated: 2024-08-25

pipequaline and pk 9084

pipequaline has been researched along with pk 9084 in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-199012 (92.31)18.7374
1990's1 (7.69)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
File, SE; Wilks, L1
File, SE; Pellow, S1
Gee, KW1
Le Fur, G1
File, SE; Lister, RG1
Gee, KW; Yamamura, HI1
Keane, PE; Morre, M; Simiand, J1
File, SE2
Burgevin, MC; Ferris, O; Gauthier, A; Guérémy, C; Heaulme, M; Le Fur, G; Mizoule, J; Uzan, A1
Brinton, RE; Gee, KW; Yamamura, HI1
File, SE; Simmonds, MA1
Chen, JS; Gee, KW; Johnson, D; Lan, NC1

Other Studies

13 other study(ies) available for pipequaline and pk 9084

ArticleYear
Effects of acute and chronic treatment on the pro- and anti-convulsant actions of CL 218, 872, PK 8165 and PK 9084, putative ligands for the benzodiazepine receptor.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Male; Mice; Pentylenetetrazole; Picrotoxin; Pyridazines; Quinolines; Receptors, GABA-A; Time Factors

1985
The effects of putative anxiolytic compounds (PK 8165, PK 9084 and tracazolate) on the rat corticosterone response.
    Physiology & behavior, 1985, Volume: 35, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Corticosterone; Male; Pyrazoles; Quinolines; Rats; Receptors, GABA-A; Stress, Psychological

1985
Phenylquinolines PK 8165 and PK 9084 allosterically modulate [35S]t-butylbicyclophosphorothionate binding to a chloride ionophore in rat brain via a novel Ro5 4864 binding site.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:3

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Convulsants; gamma-Aminobutyric Acid; Kinetics; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
[Anxiety receptors: new pharmacological approach (author's transl)].
    L'Encephale, 1982, Volume: 8, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Binding, Competitive; Brain; Chlordiazepoxide; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Quinolines; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Seizures

1982
Quinolines and anxiety: anxiogenic effects of CGS 8216 and partial anxiolytic profile of PK 9084.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Humans; Male; Motor Activity; Pyrazoles; Quinolines; Rats; Social Behavior

1983
Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes?
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Cerebral Cortex; Drug Interactions; Flunitrazepam; Male; Postural Balance; Pyrazoles; Pyridazines; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Temperature

1983
The quinolines PK 8165 and PK 9084 possess benzodiazepine-like activity in vitro but not in vivo.
    Neuroscience letters, 1984, Mar-09, Volume: 45, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A

1984
Modification of seizures elicited by the benzodiazepine Ro 5-3663--a comparison with picrotoxin.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:12

    Topics: Animals; Benzodiazepinones; Chemical Phenomena; Chemistry; Convulsants; Diazepam; Drug Synergism; Flumazenil; Male; Mice; Picrotoxin; Pyrazoles; Quinolines; Seizures

1984
Multiple benzodiazepine receptors: evidence of dissociation between anticonflict and anticonvulsant properties by PK 8165 and PK 9084 (two quinoline derivatives).
    Life sciences, 1981, Mar-30, Volume: 28, Issue:13

    Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Cerebellar Cortex; Chlordiazepoxide; Conflict, Psychological; Cyclic AMP; Cyclic GMP; Diazepam; Hypnotics and Sedatives; Kinetics; Male; Motor Activity; Piperazines; Quinolines; Rats; Receptors, Drug; Receptors, GABA-A

1981
PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam.
    Brain research, 1983, Mar-28, Volume: 264, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Diazepam; Drug Antagonism; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Quinolines; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
Interactions of two phenylquinolines with picrotoxin and benzodiazepines in vivo and in vitro.
    European journal of pharmacology, 1984, Jan-27, Volume: 97, Issue:3-4

    Topics: Animals; Anticonvulsants; Benzodiazepines; Drug Interactions; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Myoclonus; Pentylenetetrazole; Picrotoxin; Quinolines; Rats; Rats, Inbred Strains; Seizures

1984
Sedative effects of PK 9084 and PK 8165, alone and in combination with chlordiazepoxide.
    British journal of pharmacology, 1983, Volume: 79, Issue:1

    Topics: Animals; Behavior, Animal; Body Temperature; Chlordiazepoxide; Drug Interactions; Exploratory Behavior; Hypnotics and Sedatives; Male; Motor Activity; Quinolines; Rats

1983
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection

1995