Page last updated: 2024-08-16

pindolol and idazoxan

pindolol has been researched along with idazoxan in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (60.00)18.2507
2000's3 (20.00)29.6817
2010's3 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Hjorth, S; Tao, R1
Gustafson, I; Westerberg, EJ; Wieloch, T1
Atgie, C; Carpene, C; Lafontan, M; Quideau, N; Saulnier-Blache, JS1
Carpéné, C; Dauzats, M; Lafontan, M; Larrouy, D; Quideau, N; Saulnier-Blache, JS1
Paré, WP; Tejani-Butt, SM; Yang, J1
Tejani-Butt, SM; Yang, J1
Herman, CA; Luczy, G; Uhlén, S; Wikberg, JE1
Leander, JD; Wolff, MC1
Butterworth, RF; Buu, PN; Michalak, A; Rose, C1
Bylund, DB; Happe, HK; Murrin, LC; Sanders, JD; Szot, P; Weinshenker, D1
Chen, HX; Jiang, XZ; Li, J; Li, YF; Wang, NP; Zhang, YZ1

Other Studies

15 other study(ies) available for pindolol and idazoxan

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Alpha 2-adrenoceptor modulation of rat ventral hippocampal 5-hydroxytryptamine release in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Hippocampus; Idazoxan; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Thiazoles; Tyrosine 3-Monooxygenase

1992
Effects of ischemia on regional ligand binding to adrenoceptors in the rat brain.
    Journal of the neurological sciences, 1992, Volume: 113, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Brain; Dioxanes; Idazoxan; Ischemic Attack, Transient; Male; Pindolol; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic; Time Factors

1992
Hamster adipocyte alpha 2-adrenoceptor changes during fat mass modifications are not directly dependent on adipose tissue norepinephrine content.
    Endocrinology, 1990, Volume: 126, Issue:5

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cricetinae; Dioxanes; Energy Intake; Food Deprivation; Hydroxydopamines; Idazoxan; Lipolysis; Male; Mesocricetus; Norepinephrine; Oxidopamine; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha; Sympathectomy, Chemical

1990
Photoperiodic control of adipocyte alpha 2-adrenoceptors in Syrian hamsters: role of testosterone.
    Endocrinology, 1990, Volume: 127, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Brimonidine Tartrate; Cricetinae; Dioxanes; Idazoxan; Isoproterenol; Kidney; Light; Lipolysis; Male; Mesocricetus; Periodicity; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha; Testosterone

1990
Effect of repeated novel stressors on depressive behavior and brain norepinephrine receptor system in Sprague-Dawley and Wistar Kyoto (WKY) rats.
    Brain research, 1994, Jun-27, Volume: 649, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Body Weight; Brain; Carrier Proteins; Depression; Dioxanes; Fluoxetine; Idazoxan; Male; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Pindolol; Rats; Rats, Inbred WKY; Rats, Sprague-Dawley; Receptors, Adrenergic; Species Specificity; Stress, Psychological; Swimming; Symporters

1994
A time course of altered thyroid states on the noradrenergic system in rat brain by quantitative autoradiography.
    Neuroendocrinology, 1994, Volume: 59, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Autoradiography; Body Weight; Brain Chemistry; Dioxanes; Fluoxetine; Idazoxan; Male; Norepinephrine; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Presynaptic; Thyroid Gland; Thyroidectomy; Time Factors

1994
Characterization of adrenoceptor types and subtypes in American bullfrogs acclimated to warm or cold temperature.
    General and comparative endocrinology, 1996, Volume: 104, Issue:2

    Topics: Acclimatization; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Humans; Idazoxan; Kidney; Membrane Proteins; Myocardium; Pindolol; Prazosin; Radioligand Assay; Rana catesbeiana; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Spinal Cord; Temperature

1996
Differentiation of 5-HT1A receptor ligands by drug discrimination.
    European journal of pharmacology, 1997, Aug-27, Volume: 333, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aminopyridines; Animals; Behavior, Animal; Buspirone; Columbidae; Cyclohexylamines; Discrimination Learning; Dose-Response Relationship, Drug; Idazoxan; Ligands; Male; Pindolol; Piperazines; Pyridines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists

1997
Evidence for altered central noradrenergic function in experimental acute liver failure in the rat.
    Hepatology (Baltimore, Md.), 1998, Volume: 27, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Cerebral Cortex; Chromatography, High Pressure Liquid; Coma; Dopamine; Frontal Lobe; Hippocampus; Hypothalamus; Idazoxan; Liver Failure, Acute; Microdialysis; Norepinephrine; Pindolol; Prazosin; Propanolamines; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Serotonin; Thalamus

1998
Analysis of brain adrenergic receptors in dopamine-beta-hydroxylase knockout mice.
    Brain research, 2006, Sep-13, Volume: 1109, Issue:1

    Topics: Analysis of Variance; Animals; Animals, Newborn; Autoradiography; Brain; Dopamine beta-Hydroxylase; Gene Expression Regulation, Developmental; Guanosine 5'-O-(3-Thiotriphosphate); Idazoxan; Isotopes; Mice; Mice, Inbred C57BL; Mice, Knockout; Pindolol; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2

2006
[5-HT1A/1B receptors, alpha2-adrenoceptors and the post-receptor adenylate cyclase activation in the mice brain are involved in the antidepressant-like action of agmatine].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2008, Volume: 43, Issue:5

    Topics: Adenylyl Cyclases; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Agmatine; Animals; Antidepressive Agents; Behavior, Animal; Depression; Dose-Response Relationship, Drug; Fenclonine; Idazoxan; Male; Mice; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Biogenic Amine; Serotonin 5-HT1 Receptor Antagonists; Swimming; Synapses; Yohimbine

2008