Page last updated: 2024-08-16

pindolol and cyanopindolol

pindolol has been researched along with cyanopindolol in 233 studies

Research

Studies (233)

TimeframeStudies, this research(%)All Research%
pre-199055 (23.61)18.7374
1990's125 (53.65)18.2507
2000's41 (17.60)29.6817
2010's12 (5.15)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Crino, PB; Jensen, EL; Vogt, BA1
Kompa, AR; Molenaar, P; Pak, HS; Roberts, SJ; Summers, RJ1
Tran, VT1
Liggett, SB1
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P1
Danilo, P; Malfatto, G; Rosen, MR; Rosen, TS; Steinberg, SF1
McNeel, RL; Mersmann, HJ1
Houslay, MD; Milligan, G; Strassheim, D1
Chiyotani, A; Kondo, M; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F1
Molenaar, P; Russell, FD; Summers, RJ1
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL1
Gustafson, I; Westerberg, EJ; Wieloch, T1
Hamblin, MW; McGuffin, RW; Metcalf, MA1
Grignaschi, G; Samanin, R1
Cornett, LE; Rossby, SP1
Anlar, B; Arnason, BG; Karaszewski, JW; Kim, WC; Reder, AT1
Emmerich, B; Göhly, U; Haen, E; Hallek, M; Kamp, T; Remien, J1
Amenta, F; Coppola, L; Ferrante, F; Forlani, A; Gallo, P; Monopoli, A; Napoleone, P1
Crino, PB; Vogt, BA; Volicer, L1
Doran, AR; Fregeau, DR; Gietzen, DW; Goodman, TA; Graf, K; Maddock, RJ; Magliozzi, JR; Weiler, PG1
Anderson, DR; Ferrari-Dileo, G; Feuer, WJ; Grajewski, AL1
MacDonald, A; McLaughlin, DP1
Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS1
Kim, YS; Molenaar, P; Sainz, RD; Summers, RJ1
Otto, J; Pohl, A; Urbanek, R1
Molenaar, P; Russell, FD; Shimada, T; Summers, RJ1
Kostowski, W; Pałejko, W; Płaźnik, A; Stefański, R1
Ulrichsen, J1
Aihara, K; Homma, I; Inazu, M; Inoue, K; Sakai, Y1
De Felipe, MC; Del Río, J; Montero, D1
Druse, MJ; Kuo, A; Tajuddin, N1
Atgie, C; Carpene, C; Lafontan, M; Quideau, N; Saulnier-Blache, JS1
Jeffery, PK; Sharma, RK1
Fraeyman, N; Van de Velde, E; Vanscheeuwijck, P1
Fortin, TL; Sundaresan, PR1
Moudry, R; Porzig, H1
Carpéné, C; Dauzats, M; Lafontan, M; Larrouy, D; Quideau, N; Saulnier-Blache, JS1
Lerea, LS; McCarthy, KD1
Borst, SE; Conolly, ME; Hui, KK1
Kahle, G; Kaulen, P; Wollensak, J1
Folléa, N; Fortier, MA; Labrie, F; Marchetti, B; Pelletier, G; Poyet, P1
Labrie, F; Marchetti, B1
Caron, MG; Hausdorff, WP; Hnatowich, M; Lefkowitz, RJ; O'Dowd, BF1
Arnason, BG; Brown, M; Karaszewski, JW; Maselli, R; Reder, AT1
el-Yassir, N; Fleetwood-Walker, SM1
Borton, M; Docherty, JR1
Goldie, RG; Passarelli, MC; Rigby, PJ; Self, GJ1
Cooper, SJ; Neill, JC1
Ariani, K; Ciaranello, RD; Hamblin, MW; Stratford, CA; Tan, GL1
Dalpé, M; de Montigny, C; Lal, S; Martial, J; Olivier, A; Quirion, R1
De Boer, SF; Nijkamp, FP; Thijssen, JH; Van Heuven-Nolsen, D; Van Oosterhout, AJ1
Grogan, DM; Hatjis, CG; Koritnik, DR2
Davis, JN; Nishino, K1
Hintze, TH; Homcy, CJ; Nejima, J; Susanni, EE; Uemura, N; Vatner, DE; Vatner, SF1
Henricks, PA; Nijkamp, FP; van Esch, B; van Oosterhout, AJ1
Murphree, SS; Saffitz, JE1
Booze, RM; Crisostomo, EA; Davis, JN2
Korichneva, IL; Krasnikova, TL; Radiukhin, VA1
Cardone, F; Cignarelli, M; Corso, M; De Pergola, G; Di Paolo, S; Garruti, G; Giorgino, R; Nardelli, G1
Folléa, N; Labrie, F; Marchetti, B; Pelletier, G; Plante, M; Poyet, P; Spinola, PG1
Daniel, EE; Kostka, P; Kwan, CY; Niles, LP; Sipos, SN1
Grogan, DM; Hatjis, CG1
Hamon, M; Ruiz, G; Vergé, D1
Chung, MK; Gulick, T; Lange, LG; Pieper, SJ; Schreiner, GF1
Davis, JM; Janicak, PG; Pandey, GN1
Caron, MG; Daniel, K; Kobilka, BK; Kobilka, TS; Lefkowitz, RJ; Regan, JW1
Crews, A; Hatjis, CG1
Caron, MG; Collins, S; French, FS; Lefkowitz, RJ; Quarmby, VE1
Levitzki, A; Marbach, I1
Klaassen, AB; Rodrigues de Miranda, JF; van den Broek, P; van Ginneken, CA; van Megen, YJ; van Ratingen, CJ1
Pelletier, G; Tolszczuk, M1
Cooke, R; Ellis, PM; McIntosh, CJ; Stowell, LI1
Butina, D; Coates, LH; Connor, HE; Feniuk, W; Humphrey, PP; Oxford, AW; Perren, MJ1
Davis, EA; Hall, S; Handberg, GM; Molenaar, P; Pennefather, JN; Summers, RJ1
Göthert, M; Hillenbrand, K; Schlicker, E1
Malta, E; Molenaar, P1
Crooke, ST; Gotlib, L; Minnich, MD; Shorr, RG; Strohsacker, MW; Varrichio, A1
Gagne, B; Labrie, F; Lavoie, M; Poyet, P1
Edwards, E; Whitaker-Azmitia, PM1
Kusiak, JW; Pitha, J1
Lew, R; Summers, RJ2
Lange, F; Lange, J; Morin, D; Tillement, JP; Zini, R1
Levitzki, A; Marbach, I; Shiloach, J1
Earley, KJ; Gunasegaram, S; Tenner, TE1
Bittera, I; Eck, E; Falkay, G; Gyurkovits, K; Koltai, M1
Deighton, N; Elfellah, MS; Reid, JL1
Curzon, G; Kennett, GA1
Engel, G; Göthert, M; Hillenbrand, K; Hoyer, D; Schlicker, E1
Feuerstein, TJ; Hertting, G; Lupp, A1
Houston, DS; Vanhoutte, PM1
el-Yassir, N; Fleetwood-Walker, SM; Mitchell, R1
Caron, MG; Dickinson, KE; Leeb-Lundberg, LM; Lefkowitz, RJ; Strasser, RH1
Crooke, ST; Heckman, GD; Nambi, P; Schmidt, DB; Stassen, FL; Whitman, MH1
Lipe, S; Summers, RJ1
Molenaar, P; Summers, RJ1
Canale, E; Molenaar, P; Summers, RJ1
Beld, AJ; Hermanussen, MW; Lammers, JW; Rodrigues de Miranda, JF; van Ginneken, CA; van Koppen, CJ; Verrijp, KN1
Candelore, MR; Dixon, RA; Rands, E; Strader, CD1
Maura, G; Raiteri, M; Ulivi, M1
Classen, K; Fink, K; Göthert, M; Schlicker, E1
Björntorp, P; Edén, S; Xu, X; Yang, S1
Blankesteijn, WM; de Pont, JJ; Graafsma, SJ; Thien, T; Willems, PH1
Bejarano, P; Green, SA; Hall, IP; Liggett, SB; Turki, J1
Kim, KR; Maia, AL; Raasmaja, A; Rubio, A; Silva, JE1
Bax, WA; Bos, E; Renzenbrink, GJ; Saxena, PR; Thijssen, EJ; Van Heuven-Nolsen, D1
Aryana, A; Emala, CW; Hirshman, CA; Levine, MA; Margolick, JB1
Grignaschi, G; Samanin, R; Sironi, F1
Aller, MI; Candelas, MA; Fernández-López, A; Pazos, A; Revilla, V; Soria, C1
Chaudhry, A; Cohen, ML; Cushing, DJ; Granneman, JG; Palkowitz, AD; Schenck, KW1
Breslow, MJ; Clarkson, K; Tobin, JR1
Anciones, B; Berciano, J; Grijalba, B; Pascual, J; Pazos, A1
Haugen, AH; Opstad, PK; Skrede, KK; Wiik, P1
Cazaux, C; Cremaschi, GA; Miguel, S; Sterin-Borda, L1
Minneman, KP; Zhong, H1
Hirsch, DJ; Morgunov, NS; You, YD1
Kahle, G; Kaulen, P; Scherer, V; Wollensak, J1
Elnatan, J; Molenaar, P; Rosenfeldt, FL; Summers, RJ1
Chojnacka-Wójcik, E; Filip, M; Przegaliński, E; Tatarczyńska, E1
Kompa, AR; Molenaar, P; Russell, FD; Summers, RJ1
Esposito, E; Pagannone, S; Prisco, S1
Amara, DA; Buhot, MC; Dierich, A; Hen, R; LeMeur, M; Ramboz, S; Saudou, F; Segu, L1
Chiyotani, A; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F; Yamawaki, I1
Dombrowski, MP; Gauvin, JM; Hayashi, RH; Hurd, WW1
Birnbaumer, L; Kaumann, AJ; Levy, FO; Zhu, X1
Clark, CJ; Connell, JM; Milligan, G1
Futuro-Neto, HA; Pires, JG; Ramage, AG; Silva, SR1
Craig, DA; Martin, GR1
Ikegaya, T; Kaneko, M; Kobayashi, A; Nishiyama, T; Yamazaki, N1
Grignaschi, G; Mantelli, B; Samanin, R1
Chojnacka-Wójcik, E; Przegalinski, E; Tatarczyńska, E1
Molenaar, P; Sarsero, D1
Molenaar, P; Roberts, SJ; Russell, FD; Summers, RJ1
Crick, H; Manuel, NA; Wallis, DI1
Oriowo, MA1
Hoey, A; Jackson, C; Pegg, G; Sillence, M1
Browning, RA; Dailey, JW; Jobe, PC; Statnick, MA1
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H1
Calvo, JR; Caraballo, MI; Garcia-Macias, JF; Guerrero, JM; Harmouch, A; Molinero, P; Osuna, C; Pozo, D; Rafii-el-Idrissi, M1
Brown, AM; Kaumann, AJ; Lynham, JA1
Cui, Y; Iwase, M; Kalthof, B; Sato, N; Shen, YT; Uechi, M; Vatner, DE; Vatner, SF1
Fillion, G; Fillion, MP; Massot, O; Prudhomme, N; Rousselle, JC; Zifa, E1
Abraini, JH; Kriem, B; Rostain, JC1
Bouanani, NE; Crozatier, B; Su, JB; Xiong, L1
Gabilondo, AM; Krasel, C; Lohse, MJ1
Díaz-Laviada, I; Guillén, A; Haro, A; Nieto, JL1
El Hadri, K; Fève, B; Pairault, J1
Malinowska, B; Schlicker, E2
Kaumann, AJ; Molenaar, P1
Bolofo, ML; Giles, H; Lansdell, SJ; Martin, GR; Wilson, HL1
Björntorp, P; Edén, S; Liu, X; Yang, S1
Hoey, AJ; Jackson, CM; Pegg, GG; Sillence, MN1
Herman, CA; Luczy, G; Uhlén, S; Wikberg, JE1
Feuerstein, TJ; Gleichauf, O; Landwehrmeyer, GB1
Houston, G; Kelly, J1
Dutta, PK; Eraundorfer, P; Patil, PN1
Lohse, MJ; Oesterhelt, D; Söhlemann, P; Soppa, J1
Bado, A; Laigneau, JP; Levasseur, S; Lewin, MJ; Moizo, L; Reyl-Desmars, F1
Ouyang, A; Yu, O1
Bernstein, D; Chruscinski, A; Desai, KH; Kobilka, BK; Rohrer, DK; Schauble, E1
Gjerstad, J; Hole, K; Tjølsen, A1
Audigier, Y; Caput, D; Devic, E; Paquereau, L; Steinberg, R1
Conti, P; Dallanoce, C; De Amici, M; De Micheli, C; Klotz, KN1
Cohen-Tannoudji, J; Coudouel, N; Lécrivain, JL; Legrand, C; Maltier, JP; Robin, MT1
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F1
Isono, K; Nagai, A; Tagaya, E; Tamaoki, J1
Branchek, TA; Zgombick, JM1
Centurión, D; Rabelo, G; Sánchez-López, A; Villalón, CM1
Dhalla, NS; Elimban, V; Persad, S; Siddiqui, F1
Baranski, TJ; Bourne, HR; Iiri, T; Lichtarge, O; Meng, EC; Nissenson, RA; Sheikh, SP; Vilardarga, JP1
Arnold, PB; Cardenas, CG; Cardenas, LM; Mar, LP; Scroggs, RS; Surmeier, DJ; Vysokanov, AV1
Bouzeghrane, F; Fagette, S; Gallo-Bona, N; Gauquelin-Koch, G; Gharib, C; Somody, L1
Guerrero, SW; Minneman, KP1
Daws, LC; Frazer, A; Gerhardt, GA1
MacDonald, A; Watt, K1
Cherian, A; Mustafa, SM; Oriowo, MA; Yousif, M1
Dorn, GW; Liggett, SB; Tepe, NM; Wu, G; Yatani, A1
Boege, F; Haase, W; Hampe, W; Michel, H; Reiländer, H; Voss, RH1
Brawley, L; MacDonald, A; Shaw, AM2
Brink, CB; Neubig, RR; Wade, SM1
Töneke, K1
Ando, M; Ando, Y; Nakamura, M; Obayashi, K; Suga, M; Terazaki, H; Uchino, M; Yamashita, T1
Daws, LC; Frazer, A; Gerhardt, GA; Gould, GG; Teicher, SD1
Ammer, H; Schulz, R1
Evans, BA; Hutchinson, DS; Summers, RJ1
Engelhardt, S; Hein, L; Kaumann, AJ; Lohse, M; Molenaar, P1
Yan, QS; Yan, SE2
Ase, AR; Descarries, L; Hen, R; Reader, TA; Riad, M1
Aubert, N; Burlet, C; Devaux, Y; Mertes, PM; Seguin, C; Siaghy, EM; Ungureanu-Longrois, D; Zannad, F1
Green, SA; Liggett, SB; Rathz, DA; Schuster, AJ1
Hussein, SM; Khan, I; Oriowo, M1
Chi, J; Stephens, RL; Varanasi, S1
Cremaschi, GA; Edgar, VA; Genaro, AM; Sterin-Borda, L1
Möck, M; Schwarz, C; Thier, P1
Hrupka, BJ; Langhans, W; von Meyenburg, C1
Banks, ML; Cook, VJ; Mills, EM; Sprague, JE1
Andrade, R; Béïque, JC; Chapin-Penick, EM; Mladenovic, L1
Barakat, H; Christian, B; Davis, J; Hickner, R; McConnaughey, MM; Privette, J; Sheets, KA1
Ishii, K; Karikomi, Y; Kubota, Y; Nakahara, T; Sakamoto, K1
Brahmadevara, N; MacDonald, A; Shaw, AM1
Jackman, GP; Louis, SN; Louis, WJ; Machida, CA; Nero, TL; Rezmann-Vitti, LA1
Brown, MJ; O'Shaughnessy, KM; Sandilands, A; Yeo, G1
Cremaschi, G; Fernández, MM; Fossati, CA; Goin, JC; Gorelik, G; Malchiodi, EL; Zwirner, NW1
Desfontis, JC; Gauthier, C; Gautier, F; Gogny, M; Mallem, MY; Serpillon, S; Toumaniantz, G1
Christopoulos, A; Evans, BA; Hutchinson, DS; Sato, M; Summers, RJ1
Chandrasekhar, B; Fatinikun, T; Kadavil, EA; Khan, I; Omu, AE; Oriowo, MA1
Desfontis, JC; Gogny, M; Holopherne, D; Le Coz, O; Mallem, Y; Reculeau, O1
Desfontis, JC; Gogny, M; Le Coz, O; Mallem, MY; Reculeau, O1
Kozłowska, H; Kwolek, G; Malinowska, B; Schlicker, E; Zakrzeska, A1
Clark, RB; Dai, W; Friedman, J; Godines, V; Knoll, BJ; Millman, EE; Moore, RH; Tran, TM; Vaughan, DJ1
Odagaki, Y; Toyoshima, R1
Baranowska, M; Kozłowska, H; Kozłowski, M; Malinowska, B; Schlicker, E1
Chan, YS; Chen, L; Yung, KK; Yung, WH1
Baker, JG; Edwards, PC; Henderson, R; Leslie, AG; Moukhametzianov, R; Schertler, GF; Serrano-Vega, MJ; Tate, CG; Warne, T1
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B1
Sabio, M; Topiol, S1
Chess-Williams, R; Kay, LJ; Peachell, PT; Rostami-Hodjegan, A; Scola, AM; Suvarna, SK1
Balaraman, GS; Bhattacharya, S; Vaidehi, N1
Miller, JL; Tate, CG1
Ribeiro, CA; Silva, SA1
Bai, F; Cherezov, V; Gao, X; Han, GW; Huang, XP; Jiang, H; Jiang, Y; Katritch, V; Liu, W; Ma, J; McCorvy, JD; Melcher, K; Roth, BL; Stevens, RC; Vardy, E; Wacker, D; Wang, C; Wu, H; Xu, HE; Yang, H; Yang, L; Zhang, C; Zhou, XE1
Daws, LC; Horton, RE; Montañez, S; Munn, JL; Owens, WA1
Edwards, PC; Leslie, AG; Miller-Gallacher, JL; Nehmé, R; Schertler, GF; Tate, CG; Warne, T1
Ahmari, SE; Barr, MM; Blanco, C; David, DJ; Gardier, AM; Hen, R; Le Dantec, Y; Nautiyal, KM; Tanaka, KF; Tritschler, L1
Baker, J; Brown, GA; Congreve, M; Leslie, AG; Sato, T; Tate, CG; Warne, T1
Dong, X; Wang, Y1
Ahmari, SE; David, DJ; Gardier, AM; Hen, R; Nautiyal, KM; Tritschler, L1
Bregman, T; Diwan, M; Fletcher, PJ; Hamani, C; Nobrega, JN; Raymond, R; Scott, B; Volle, J1

Reviews

3 review(s) available for pindolol and cyanopindolol

ArticleYear
Experimental QT interval prolongation.
    Annals of the New York Academy of Sciences, 1992, Jan-27, Volume: 644

    Topics: Adrenergic beta-Antagonists; Animals; Animals, Newborn; Electrocardiography; Heart Conduction System; Long QT Syndrome; Nerve Growth Factors; Phenethylamines; Pindolol; Tetralones

1992
Chimeric alpha 2-,beta 2-adrenergic receptors: delineation of domains involved in effector coupling and ligand binding specificity.
    Science (New York, N.Y.), 1988, Jun-03, Volume: 240, Issue:4857

    Topics: Amino Acid Sequence; Animals; Chimera; Cloning, Molecular; GTP-Binding Proteins; Humans; Molecular Sequence Data; Pindolol; Protein Conformation; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

1988
X-ray structure breakthroughs in the GPCR transmembrane region.
    Biochemical pharmacology, 2009, Jul-01, Volume: 78, Issue:1

    Topics: Animals; Cell Membrane; Humans; Models, Molecular; Molecular Conformation; Pindolol; Propanolamines; Protein Conformation; Receptor, Adenosine A2A; Receptors, Adrenergic, beta-2; Receptors, G-Protein-Coupled; Retinaldehyde; Rhodopsin; X-Ray Diffraction

2009

Trials

1 trial(s) available for pindolol and cyanopindolol

ArticleYear
Differences in beta-adrenergic receptor densities in omental and subcutaneous adipose tissue from obese African American and Caucasian women.
    Metabolism: clinical and experimental, 2004, Volume: 53, Issue:2

    Topics: Adipose Tissue; Adrenergic beta-Agonists; Adult; Black or African American; Cell Membrane; Female; Humans; Immunoblotting; Isoproterenol; Kinetics; Lipolysis; Obesity, Morbid; Omentum; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; White People

2004

Other Studies

229 other study(ies) available for pindolol and cyanopindolol

ArticleYear
Multiple heteroreceptors on limbic thalamic axons: M2 acetylcholine, serotonin1B, beta 2-adrenoceptors, mu-opioid, and neurotensin.
    Synapse (New York, N.Y.), 1992, Volume: 10, Issue:1

    Topics: Atenolol; Autoradiography; Axons; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethanolamines; Limbic System; Neurotensin; Oxotremorine; Pindolol; Pirenzepine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Receptors, Neurotensin; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, mu; Receptors, Serotonin; Thalamus; Tritium

1992
Localization of (-)-[125I]cyanopindolol binding in guinea-pig heart: characteristics of non-beta-adrenoceptor related binding in cardiac pacemaker and conducting regions.
    Neuroscience letters, 1992, Feb-17, Volume: 136, Issue:1

    Topics: Alprenolol; Animals; Ascorbic Acid; Binding Sites; Ethanolamines; Female; Guinea Pigs; Haloperidol; Heart Conduction System; Isoproterenol; Male; Myocardium; Peroxidase; Phentolamine; Pindolol; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta; Serotonin; Thiophenes; Trachea

1992
Human retinal pigment epithelial cells possess beta 2-adrenergic receptors.
    Experimental eye research, 1992, Volume: 55, Issue:3

    Topics: Adenylyl Cyclases; Betaxolol; Cells, Cultured; Cyclic AMP; Epinephrine; Humans; Isoproterenol; Norepinephrine; Pigment Epithelium of Eye; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1992
Functional properties of the rat and human beta 3-adrenergic receptors: differential agonist activation of recombinant receptors in Chinese hamster ovary cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Enzyme Activation; Humans; Isoproterenol; Pindolol; Rats; Receptors, Adrenergic, beta; Recombinant Proteins

1992
Influence of age on the beta 1- and beta 2-adrenergic receptors in rat liver.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Cell Membrane; Imidazoles; Liver; Liver Glycogen; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1992
Ligand binding to the porcine adipose tissue beta-adrenergic receptor.
    Journal of animal science, 1992, Volume: 70, Issue:3

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Kinetics; Ligands; Molecular Conformation; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Swine; Temperature; Time Factors

1992
Regulation of cardiac adenylate cyclase activity in rodent models of obesity.
    The Biochemical journal, 1992, Apr-01, Volume: 283 ( Pt 1)

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding, Competitive; Disease Models, Animal; GTP-Binding Proteins; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Membranes; Mice; Mice, Obese; Myocardium; Obesity; Pindolol; Rats; Rats, Zucker; Receptors, Adrenergic, beta; Stimulation, Chemical

1992
[Airway epithelial beta 3-adrenergic receptor--effect on bioelectric properties and its mechanism of action].
    Nihon Kyobu Shikkan Gakkai zasshi, 1992, Volume: 30, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Bumetanide; Calcium; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Epithelium; Ethanolamines; Membrane Potentials; Pindolol; Receptors, Adrenergic, beta; Trachea

1992
Absence of mitochondrial beta-adrenoceptors in guinea pig myocardium: evidence for tissue disparity.
    General pharmacology, 1992, Volume: 23, Issue:5

    Topics: 5'-Nucleotidase; Adrenergic beta-Antagonists; Animals; Autoradiography; Azides; Ca(2+) Mg(2+)-ATPase; Cell Membrane; Female; Guinea Pigs; Male; Mitochondria, Heart; Myocardium; Ouabain; Pindolol; Receptors, Adrenergic, beta; Sarcolemma; Sodium Azide; Sodium-Potassium-Exchanging ATPase

1992
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured

1992
Effects of ischemia on regional ligand binding to adrenoceptors in the rat brain.
    Journal of the neurological sciences, 1992, Volume: 113, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Brain; Dioxanes; Idazoxan; Ischemic Attack, Transient; Male; Pindolol; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic; Time Factors

1992
Conversion of the human 5-HT1D beta serotonin receptor to the rat 5-HT1B ligand-binding phenotype by Thr355Asn site directed mutagenesis.
    Biochemical pharmacology, 1992, Nov-17, Volume: 44, Issue:10

    Topics: Amino Acid Sequence; Animals; Asparagine; Binding Sites; Cell Line; Humans; Molecular Sequence Data; Mutagenesis, Site-Directed; Phenotype; Pindolol; Rats; Receptors, Serotonin; Recombinant Proteins; Threonine

1992
Role of 5-HT receptors in the effect of d-fenfluramine on feeding patterns in the rat.
    European journal of pharmacology, 1992, Mar-03, Volume: 212, Issue:2-3

    Topics: Animals; Feeding Behavior; Fenfluramine; Male; Metergoline; Pindolol; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereoisomerism

1992
Steady state levels of hepatic alpha 1- and beta 2-adrenergic receptors and gene transcripts during development of the male rat.
    Journal of cellular physiology, 1991, Volume: 147, Issue:1

    Topics: Age Factors; Animals; Blotting, Northern; Gene Expression; Liver; Male; Pindolol; Prazosin; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; RNA, Messenger

1991
Increased lymphocyte beta-adrenergic receptor density in progressive multiple sclerosis is specific for the CD8+, CD28- suppressor cell.
    Annals of neurology, 1991, Volume: 30, Issue:1

    Topics: Adult; Antigens, CD; Antigens, Differentiation, T-Lymphocyte; Autoimmune Diseases; CD28 Antigens; CD8 Antigens; Cells, Cultured; Humans; Interleukin-2; Lymphocyte Activation; Middle Aged; Models, Biological; Multiple Sclerosis; Neurons, Afferent; Pindolol; Receptors, Adrenergic, beta; Recombinant Proteins; T-Lymphocyte Subsets; Up-Regulation

1991
Reduced responsiveness of adenylate cyclase to forskolin in human lymphoma cells.
    Biochemical pharmacology, 1991, Sep-12, Volume: 42, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Aged; B-Lymphocytes; Binding Sites; Cholera Toxin; Colforsin; Cyclic AMP; Female; Humans; Isoproterenol; Lymphoma, Non-Hodgkin; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured

1991
Autoradiographic localization of beta-adrenergic receptors in human large coronary arteries.
    Circulation research, 1991, Volume: 68, Issue:6

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Autoradiography; Binding, Competitive; Coronary Vessels; Female; Humans; Imidazoles; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Silver; Tissue Distribution

1991
Laminar alterations in gamma-aminobutyric acidA, muscarinic, and beta adrenoceptors and neuron degeneration in cingulate cortex in Alzheimer's disease.
    Journal of neurochemistry, 1991, Volume: 57, Issue:1

    Topics: Adrenergic beta-Antagonists; Aged; Alzheimer Disease; Gyrus Cinguli; Humans; Muscimol; Nerve Degeneration; Neurons; Pindolol; Pirenzepine; Receptors, Adrenergic, beta; Receptors, GABA-A; Receptors, Muscarinic

1991
Beta receptor density in human lymphocyte membranes: changing with aging?
    Journal of gerontology, 1991, Volume: 46, Issue:4

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Aging; Binding Sites; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Female; Humans; Lymphocytes; Male; Middle Aged; Norepinephrine; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta

1991
Beta-adrenergic responsiveness of choroidal vasculature.
    Ophthalmology, 1991, Volume: 98, Issue:6

    Topics: Administration, Topical; Adrenergic beta-Antagonists; Adult; Animals; Autoradiography; Choroid; Female; Hemodynamics; Humans; Intraocular Pressure; Male; Middle Aged; Pigment Epithelium of Eye; Pindolol; Rabbits; Receptors, Adrenergic, beta; Retinal Vessels; Timolol

1991
Characterization of catecholamine-mediated relaxations in rat isolated gastric fundus: evidence for an atypical beta-adrenoceptor.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Catecholamines; Ethanolamines; Gastric Fundus; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Norepinephrine; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
    European journal of pharmacology, 1991, Jul-09, Volume: 199, Issue:3

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Characterization of beta 1- and beta 2-adrenoceptors in rat skeletal muscles.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Imidazoles; Male; Membranes; Muscles; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Beta-2-adrenoceptors of polymorphonuclear leukocytes in children with atopic dermatitis. Their number and affinity to the radioligand [125I]-cyanopindolol.
    International archives of allergy and applied immunology, 1991, Volume: 95, Issue:2-3

    Topics: Adolescent; Adrenergic beta-Antagonists; Binding Sites; Child; Child, Preschool; Dermatitis, Atopic; Female; Humans; Infant; Male; Neutrophils; Pindolol; Receptors, Adrenergic, beta

1991
Densitometric analysis of beta 1- and beta 2-adrenoceptors in guinea-pig atrioventricular conducting system.
    Journal of molecular and cellular cardiology, 1990, Volume: 22, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Atrioventricular Node; Autoradiography; Densitometry; Female; Guinea Pigs; Heart Conduction System; Male; Pindolol; Propranolol; Proteins; Purkinje Cells; Receptors, Adrenergic, beta; Rosaniline Dyes; Staining and Labeling

1990
Serotonergic mechanisms in the nucleus accumbens affected by chronic desipramine treatment.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Buspirone; Chromans; Desipramine; Dose-Response Relationship, Drug; Methysergide; Microinjections; Nucleus Accumbens; Pindolol; Quipazine; Rats; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Alterations in serotonin receptor subtypes in ethanol-dependent rats.
    Alcohol and alcoholism (Oxford, Oxfordshire), 1991, Volume: 26, Issue:5-6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alcohol Withdrawal Delirium; Alcoholic Intoxication; Alcoholism; Animals; Brain; Ethanol; Ketanserin; Pindolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Relations between contractile responses and beta-adrenoceptors in gastric fundus of diabetic rats.
    Life sciences, 1991, Volume: 48, Issue:11

    Topics: Animals; Diabetes Mellitus, Experimental; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stomach

1991
Acute or chronic antidepressants do not modify [125I]cyanopindolol binding to 5-HT1B receptors in rat brain.
    European journal of pharmacology, 1991, Apr-24, Volume: 196, Issue:3

    Topics: Animals; Antidepressive Agents, Tricyclic; Biogenic Monoamines; Brain; Clomipramine; Female; Iodine Radioisotopes; Iprindole; Male; Pindolol; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Thiazepines; Time Factors

1991
Effects of in utero ethanol exposure on the developing serotonergic system.
    Alcoholism, clinical and experimental research, 1991, Volume: 15, Issue:4

    Topics: Animals; Animals, Newborn; Brain Stem; Cerebral Cortex; Chromatography, High Pressure Liquid; Ethanol; Female; Iodine Radioisotopes; Male; Pindolol; Pregnancy; Prenatal Exposure Delayed Effects; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1991
Hamster adipocyte alpha 2-adrenoceptor changes during fat mass modifications are not directly dependent on adipose tissue norepinephrine content.
    Endocrinology, 1990, Volume: 126, Issue:5

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cricetinae; Dioxanes; Energy Intake; Food Deprivation; Hydroxydopamines; Idazoxan; Lipolysis; Male; Mesocricetus; Norepinephrine; Oxidopamine; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha; Sympathectomy, Chemical

1990
Airway beta-adrenoceptor number in cystic fibrosis and asthma.
    Clinical science (London, England : 1979), 1990, Volume: 78, Issue:4

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Aged; Asthma; Bronchi; Bronchial Neoplasms; Bronchiectasis; Cell Membrane; Child; Child, Preschool; Cystic Fibrosis; Female; Humans; Lung; Male; Middle Aged; Muscle, Smooth; Pindolol; Receptors, Adrenergic, beta

1990
Characterization of the beta-adrenergic transduction system in spleen mononuclear leukocyte membranes of young and senescent rats.
    Biochemical pharmacology, 1990, Jun-15, Volume: 39, Issue:12

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Aging; Animals; Binding, Competitive; Cell Membrane; Cyclic AMP; Leukocytes, Mononuclear; Ligands; Male; Pindolol; Rats; Receptors, Adrenergic, beta; Signal Transduction; Spleen

1990
Reserpine up-regulation of rat renal cortical beta adrenergic receptors is independent of its effect on the sympathetic nervous system.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Catecholamines; Guanethidine; Kidney Cortex; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reserpine; Sympathetic Nervous System; Up-Regulation

1990
Regulation of beta-adrenergic responsiveness during erythroid differentiation of Friend erythroleukemia cells.
    Biomedica biochimica acta, 1990, Volume: 49, Issue:2-3

    Topics: Adrenergic beta-Antagonists; Animals; Cell Differentiation; Cell Membrane; Dimethyl Sulfoxide; Friend murine leukemia virus; GTP-Binding Proteins; Leukemia, Erythroblastic, Acute; Mice; Pindolol; Poly(ADP-ribose) Polymerases; Receptors, Adrenergic, beta; Tumor Cells, Cultured

1990
Photoperiodic control of adipocyte alpha 2-adrenoceptors in Syrian hamsters: role of testosterone.
    Endocrinology, 1990, Volume: 127, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Brimonidine Tartrate; Cricetinae; Dioxanes; Idazoxan; Isoproterenol; Kidney; Light; Lipolysis; Male; Mesocricetus; Periodicity; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha; Testosterone

1990
Neuron-associated astroglial cells express beta- and alpha 1-adrenergic receptors in vitro.
    Brain research, 1990, Jun-25, Volume: 521, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Cells, Cultured; Hippocampus; Pindolol; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1990
Beta-adrenergic receptors on human lymphocytes: comparison of down-regulation in vivo and in vitro.
    Pharmacology, 1990, Volume: 40, Issue:6

    Topics: Adrenergic beta-Antagonists; Down-Regulation; Humans; Isoproterenol; Lymphocytes; Pindolol; Receptors, Adrenergic, beta; Terbutaline; Time Factors

1990
Quantitative autoradiography of beta-adrenergic receptors in rabbit eyes.
    Experimental eye research, 1990, Volume: 51, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Ciliary Body; Cornea; Endothelium, Corneal; Epithelium; Eye; Female; Frozen Sections; Iris; Male; Pindolol; Rabbits; Receptors, Adrenergic, beta

1990
Beta-adrenergic receptors in the rat mammary gland during pregnancy and lactation: characterization, distribution, and coupling to adenylate cyclase.
    Endocrinology, 1990, Volume: 126, Issue:1

    Topics: Adenylyl Cyclases; Animals; Autoradiography; Cytosol; Female; Gonadal Steroid Hormones; Kinetics; Lactation; Mammary Glands, Animal; Pindolol; Pregnancy; Pregnancy, Animal; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Progesterone; Tissue Distribution

1990
Hormonal regulation of beta-adrenergic receptors in the rat mammary gland during the estrous cycle and lactation: role of sex steroids and prolactin.
    Endocrinology, 1990, Volume: 126, Issue:1

    Topics: Animals; Estrus; Female; Gonadal Steroid Hormones; Hormones; Lactation; Mammary Glands, Animal; Membranes; Ovariectomy; Pindolol; Pregnancy; Prolactin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1990
A mutation of the beta 2-adrenergic receptor impairs agonist activation of adenylyl cyclase without affecting high affinity agonist binding. Distinct molecular determinants of the receptor are involved in physical coupling to and functional activation of
    The Journal of biological chemistry, 1990, Jan-25, Volume: 265, Issue:3

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Cell Compartmentation; DNA Mutational Analysis; Endocytosis; Enzyme Activation; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Isoproterenol; Macromolecular Substances; Molecular Sequence Data; Mutation; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Structure-Activity Relationship

1990
Sympathetic skin responses are decreased and lymphocyte beta-adrenergic receptors are increased in progressive multiple sclerosis.
    Annals of neurology, 1990, Volume: 27, Issue:4

    Topics: Adult; Binding, Competitive; Cyclic AMP; Electric Stimulation; Female; Humans; Male; Membrane Potentials; Middle Aged; Multiple Sclerosis; Pindolol; Receptors, Adrenergic, beta; Skin; Sympathetic Nervous System; T-Lymphocytes

1990
A 5-HT1-type receptor mediates the antinociceptive effect of nucleus raphe magnus stimulation in the rat.
    Brain research, 1990, Jul-16, Volume: 523, Issue:1

    Topics: Animals; Electric Stimulation; Evoked Potentials; Iontophoresis; Ketanserin; Nociceptors; Pindolol; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord

1990
The effects of ageing on prejunctional 5-hydroxytryptamine receptors in the rat vas deferens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:2

    Topics: Aging; Animals; Electric Stimulation; In Vitro Techniques; Male; Muscle, Smooth; Myocardial Contraction; Pertussis Toxin; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vas Deferens; Virulence Factors, Bordetella; Yohimbine

1990
Characteristics and localisation of 125I ion binding in mammalian airways.
    European journal of pharmacology, 1990, Feb-06, Volume: 176, Issue:2

    Topics: Animals; Ascorbic Acid; Dithiothreitol; Guinea Pigs; Humans; In Vitro Techniques; Iodides; Iodine Radioisotopes; Lung; Macaca fascicularis; Mice; Mice, Inbred CBA; Muscle, Smooth; Pindolol; Protein Binding; Rats; Rats, Inbred Strains; Sodium Iodide; Species Specificity; Swine; Trachea

1990
Evidence that d-fenfluramine anorexia is mediated by 5-HT1 receptors.
    Psychopharmacology, 1989, Volume: 97, Issue:2

    Topics: Amidines; Animals; Appetite Depressants; Fenfluramine; Male; Metergoline; Pindolol; Piperidines; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1989
G protein dependent alterations in [125I]iodocyanopindolol and +/- cyanopindolol binding at 5-HT1B binding sites in rat brain membranes.
    Neurochemical research, 1989, Volume: 14, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Dihydroergotamine; Ethylmaleimide; GTP-Binding Proteins; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Iodocyanopindolol; Magnesium Sulfate; Pindolol; Rats; Receptors, Serotonin

1989
Apparent absence of serotonin1B receptors in biopsied and post-mortem human brain.
    Synapse (New York, N.Y.), 1989, Volume: 4, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Biopsy; Brain; Female; Humans; Male; Pindolol; Postmortem Changes; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Tissue Preservation

1989
Endotoxin-induced reduction of beta-adrenergic binding sites on splenic lymphocytes in vivo and in vitro: its modulation by anterior hypothalamic lesions.
    Life sciences, 1989, Volume: 44, Issue:1

    Topics: Animals; Catecholamines; Cell Membrane; Endotoxins; Escherichia coli; Glucocorticoids; Guinea Pigs; Hypothalamic Hormones; Hypothalamus, Anterior; In Vitro Techniques; Lipopolysaccharides; Lymphocyte Activation; Lymphocytes; Male; Pindolol; Receptors, Adrenergic, beta; Spleen; Thyroid Hormones

1989
Up-regulation of guinea pig myometrial beta-adrenergic receptors by intrauterine estradiol and progesterone pellets.
    American journal of obstetrics and gynecology, 1989, Volume: 160, Issue:3

    Topics: Animals; Drug Implants; Estradiol; Female; Guinea Pigs; Myometrium; Osmolar Concentration; Pindolol; Progesterone; Receptors, Adrenergic, beta; Uterus

1989
Rapid reduction in [3H]prazosin binding to gerbil forebrain membranes during bilateral common carotid artery occlusion.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1989, Volume: 9, Issue:3

    Topics: Animals; Carotid Arteries; Cell Membrane; Cell Survival; Diencephalon; Gerbillinae; Ischemic Attack, Transient; Kinetics; Male; Neurons; Phospholipases A; Phospholipases A2; Pindolol; Prazosin; Quinuclidinyl Benzilate; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Muscarinic; Telencephalon

1989
Chronic norepinephrine elicits desensitization by uncoupling the beta-receptor.
    The Journal of clinical investigation, 1989, Volume: 84, Issue:6

    Topics: Adenylyl Cyclases; Animals; Colforsin; Dogs; Drug Tolerance; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart Ventricles; Hemodynamics; Isoproterenol; Norepinephrine; Organ Size; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Sodium-Potassium-Exchanging ATPase; Ventricular Function

1989
Guinea pig alveolar macrophages possess beta-adrenergic receptors.
    Agents and actions, 1989, Volume: 26, Issue:1-2

    Topics: Adrenergic beta-Antagonists; Animals; Guinea Pigs; Macrophages; Pindolol; Pulmonary Alveoli; Receptors, Adrenergic, beta; Timolol

1989
Distribution of beta-adrenergic receptors in failing human myocardium. Implications for mechanisms of down-regulation.
    Circulation, 1989, Volume: 79, Issue:6

    Topics: Adrenergic beta-Antagonists; Adult; Autoradiography; Female; Heart Failure; Heart Transplantation; Humans; Iodine Radioisotopes; Male; Myocardium; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta

1989
Species differences in the localization and number of CNS beta adrenergic receptors: rat versus guinea pig.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Brain; Guinea Pigs; Iodine Radioisotopes; Male; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Species Specificity

1989
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used].
    Biokhimiia (Moscow, Russia), 1989, Volume: 54, Issue:2

    Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature

1989
Influence of lactate on isoproterenol-induced lipolysis and beta-adrenoceptors distribution in human fat cells.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1989, Volume: 21, Issue:4

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Cell Membrane; Cells, Cultured; Humans; Isoproterenol; Lactates; Lipolysis; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Serotonin Antagonists

1989
Beta-adrenergic receptors in DMBA-induced rat mammary tumors: correlation with progesterone receptor and tumor growth.
    Breast cancer research and treatment, 1989, Volume: 13, Issue:3

    Topics: 9,10-Dimethyl-1,2-benzanthracene; Adrenergic beta-Antagonists; Aging; Animals; Catecholamines; Female; Hormones; Iodine Radioisotopes; Kinetics; Mammary Neoplasms, Experimental; Neoplasm Regression, Spontaneous; Neoplasms, Hormone-Dependent; Ovariectomy; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Progesterone; Substrate Specificity

1989
Identification and characterization of presynaptic and postsynaptic beta adrenoreceptors in the longitudinal smooth muscle/myenteric plexus of dog ileum.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dogs; Ileum; In Vitro Techniques; Muscle, Smooth; Myenteric Plexus; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Subcellular Fractions

1989
Treatment of oophorectomized guinea pigs with intrauterine 17 beta-estradiol pellets may modulate myometrial beta-adrenergic receptor binding properties.
    American journal of obstetrics and gynecology, 1989, Volume: 161, Issue:6 Pt 1

    Topics: Adrenergic beta-Antagonists; Animals; Estradiol; Female; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Myometrium; Ovariectomy; Pindolol; Progesterone; Receptors, Adrenergic, beta

1989
Pregnancy-induced changes in the interaction of guinea pig myometrial beta-adrenergic receptors with l-isoproterenol.
    American journal of obstetrics and gynecology, 1989, Volume: 161, Issue:6 Pt 1

    Topics: Adrenergic beta-Antagonists; Animals; Female; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Myometrium; Pindolol; Pregnancy; Pregnancy, Animal; Receptors, Adrenergic, beta

1989
Chronic phenytoin treatment decreases GABAA but not beta-adrenoceptors in the cerebellum of young rats.
    European journal of pharmacology, 1989, Sep-13, Volume: 168, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Cerebellum; Female; Flunitrazepam; Kinetics; Muscimol; Phenytoin; Pindolol; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, GABA-A; Tritium

1989
Immune cytokine inhibition of beta-adrenergic agonist stimulated cyclic AMP generation in cardiac myocytes.
    Biochemical and biophysical research communications, 1988, Jan-15, Volume: 150, Issue:1

    Topics: Animals; Animals, Newborn; Biological Products; Cells, Cultured; Culture Media; Cyclic AMP; Cytokines; Isoproterenol; Lymphocyte Activation; Lymphocytes; Macrophages; Myocardium; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Spleen

1988
Decreased beta-adrenergic receptors in the leukocytes of depressed patients.
    Psychiatry research, 1987, Volume: 22, Issue:4

    Topics: Adult; Depressive Disorder; Dexamethasone; Humans; Hydrocortisone; Iodine Radioisotopes; Leukocytes; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Schizophrenia

1987
Regulation of guinea pig myometrial beta-adrenoreceptors by guanosine triphosphate and magnesium ion.
    Biology of reproduction, 1988, Volume: 38, Issue:3

    Topics: Animals; Female; Guanosine Triphosphate; Guinea Pigs; Iodine Radioisotopes; Isoproterenol; Magnesium; Myometrium; Pindolol; Pregnancy; Propranolol; Radioimmunoassay; Receptors, Adrenergic, beta

1988
Regulation of the beta 2-adrenergic receptor and its mRNA in the rat ventral prostate by testosterone.
    FEBS letters, 1988, Jun-06, Volume: 233, Issue:1

    Topics: Animals; Binding, Competitive; Cell Membrane; Gene Expression Regulation; Male; Nucleic Acid Hybridization; Orchiectomy; Pindolol; Prostate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; RNA, Messenger; Testosterone; Transcription, Genetic

1988
Use of electrofocusing for the analysis and purification of turkey erythrocytes beta 1-adrenoceptors.
    FEBS letters, 1988, Jun-06, Volume: 233, Issue:1

    Topics: Acrylic Resins; Animals; Binding, Competitive; Chromatography, Affinity; Digitonin; Electrophoresis, Polyacrylamide Gel; Erythrocytes; Hydrogen-Ion Concentration; Iodine Radioisotopes; Isoelectric Focusing; Pindolol; Receptors, Adrenergic, beta; Turkeys

1988
Demonstration of beta-adrenergic receptors in rat nasal glands by an in vitro autoradiographic technique.
    Neuroscience letters, 1988, Jul-19, Volume: 90, Issue:1-2

    Topics: Adrenergic Fibers; Animals; Autoradiography; In Vitro Techniques; Nasal Mucosa; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1988
Autoradiographic localization of beta-adrenoreceptors in rat uterus.
    The journal of histochemistry and cytochemistry : official journal of the Histochemistry Society, 1988, Volume: 36, Issue:12

    Topics: Animals; Autoradiography; Binding, Competitive; Epithelium; Ethanolamines; Female; Iodine Radioisotopes; Myometrium; Pindolol; Practolol; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Tissue Distribution; Uterus

1988
Adrenoceptor and imipramine receptor binding during the menstrual cycle.
    Acta psychiatrica Scandinavica, 1988, Volume: 78, Issue:3

    Topics: Adult; Blood Platelets; Carrier Proteins; Dihydroergotoxine; Female; Humans; Imipramine; Lymphocytes; Menstrual Cycle; Pindolol; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Drug; Receptors, Neurotransmitter

1988
GR43175, a selective agonist for the 5-HT1-like receptor in dog isolated saphenous vein.
    British journal of pharmacology, 1988, Volume: 94, Issue:4

    Topics: Animals; Cats; Dogs; Female; In Vitro Techniques; Indoles; Male; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Rabbits; Rats; Receptors, Serotonin; Saphenous Vein; Serotonin Antagonists; Sulfonamides; Sumatriptan; Swine; Tropanes; Vagus Nerve

1988
Beta-adrenoceptors in circular and longitudinal myometrial membranes and in lung membranes from dioestrous and post-partum guinea-pigs.
    Clinical and experimental pharmacology & physiology, 1988, Volume: 15, Issue:9

    Topics: Animals; Autoradiography; Diestrus; Extraembryonic Membranes; Female; Guinea Pigs; Lung; Myometrium; Pindolol; Pregnancy; Receptors, Adrenergic, beta

1988
Cyanopindolol is a highly potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Isoproterenol; Male; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Stereoisomerism

1985
Analysis of agonist dissociation constants as assessed by functional antagonism in guinea pig left atria.
    Journal of pharmacological methods, 1986, Volume: 15, Issue:2

    Topics: Adenosine; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Benzofurans; Carbachol; Catechols; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Myocardial Contraction; Nifedipine; Pindolol; Propanolamines

1986
Evidence for tyrosine at the ligand binding center of beta-adrenergic receptors.
    Biochemical pharmacology, 1986, Nov-01, Volume: 35, Issue:21

    Topics: Adrenergic beta-Antagonists; Animals; Anura; Binding Sites; Cattle; Cell Membrane; Guinea Pigs; Ligands; Pindolol; Rabbits; Rats; Receptors, Adrenergic, beta; Species Specificity; Turkeys; Tyrosine

1986
Characteristics of the beta-adrenergic receptor in the rat ventral prostate using [125I]cyanopindolol.
    Molecular and cellular endocrinology, 1986, Volume: 48, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Chemical Precipitation; Epinephrine; Isoproterenol; Male; Norepinephrine; Pindolol; Polyethylene Glycols; Prostate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1986
Selective beta-antagonists are equally and highly potent at 5-HT sites in the rat hippocampus.
    Neuropharmacology, 1987, Volume: 26, Issue:1

    Topics: 5-Methoxytryptamine; 5,7-Dihydroxytryptamine; Adrenergic beta-Antagonists; Animals; Atenolol; Binding, Competitive; Ethanolamines; Hippocampus; In Vitro Techniques; Male; Membranes; Pindolol; Propranolol; Rats; Receptors, Serotonin; Serotonin

1987
A bromoacetylated analogue of cyanopindolol: an irreversible antagonist at rat beta-adrenoceptors.
    Life sciences, 1987, Jul-06, Volume: 41, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Brain; Dihydroalprenolol; Erythrocytes; Lung; Metabolic Clearance Rate; Myocardium; Pindolol; Rats; Receptors, Adrenergic, beta; Time Factors

1987
The distribution of beta-adrenoceptors in dog kidney: an autoradiographic analysis.
    European journal of pharmacology, 1987, Aug-04, Volume: 140, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Dogs; Female; In Vitro Techniques; Iodine Radioisotopes; Kidney; Male; Pindolol; Receptors, Adrenergic, beta

1987
Alterations of beta-adrenergic, muscarinic cholinergic receptors and imipramine binding sites in human lung tumors.
    International journal of clinical pharmacology, therapy, and toxicology, 1987, Volume: 25, Issue:11

    Topics: Adenocarcinoma; Adrenergic beta-Antagonists; Carcinoma, Squamous Cell; Humans; Imipramine; In Vitro Techniques; Lung Neoplasms; Pindolol; Quinuclidinyl Benzilate; Receptors, Adrenergic, beta; Receptors, Cholinergic; Receptors, Muscarinic

1987
Gi affects the agonist-binding properties of beta-adrenoceptors in the presence of Gs.
    European journal of biochemistry, 1988, Feb-15, Volume: 172, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Catalysis; Cholera Toxin; Erythrocyte Membrane; GTP-Binding Proteins; Isoproterenol; Lymphoma; Pertussis Toxin; Pindolol; Receptors, Adrenergic, beta; Turkeys; Virulence Factors, Bordetella

1988
Characterization and localization of (-)[125I]-cyanopindolol binding to non-beta-adrenoceptor sites in dog kidney.
    Clinical and experimental pharmacology & physiology, 1987, Volume: 14, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding, Competitive; Dogs; Female; In Vitro Techniques; Iodine Radioisotopes; Kidney; Kinetics; Male; Membranes; Pindolol; Radioligand Assay

1987
Determination of beta adrenoceptor density on rabbit mononuclear leukocytes.
    Journal of pharmacological methods, 1988, Volume: 19, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Atropine; Cell Membrane; Cell Separation; Cimetidine; Leukocytes, Mononuclear; Male; Pindolol; Propranolol; Rabbits; Receptors, Adrenergic, beta

1988
Beta-adrenergic receptors of lymphocytes in children with allergic respiratory diseases.
    Pediatric pulmonology, 1988, Volume: 5, Issue:2

    Topics: Adrenergic beta-Antagonists; Asthma; Bronchial Provocation Tests; Child; Female; Humans; Immunoglobulin E; Iodine Radioisotopes; Lymphocytes; Male; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Rhinitis, Allergic, Seasonal

1988
Regulation of beta-adrenoceptors by catecholamines in the rabbit skeletal muscle.
    European journal of pharmacology, 1988, Nov-22, Volume: 157, Issue:2-3

    Topics: Adrenergic beta-Antagonists; Animals; Epinephrine; Male; Metoprolol; Muscles; Norepinephrine; Pindolol; Propanolamines; Rabbits; Receptors, Adrenergic, beta

1988
Evidence that hypophagia induced by mCPP and TFMPP requires 5-HT1C and 5-HT1B receptors; hypophagia induced by RU 24969 only requires 5-HT1B receptors.
    Psychopharmacology, 1988, Volume: 96, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Ergolines; Feeding Behavior; Food Deprivation; Indoles; Male; Mianserin; Motor Activity; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tropisetron

1988
Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1

    Topics: Animals; Cerebral Cortex; In Vitro Techniques; Isoproterenol; Ketanserin; Kinetics; Male; Pindolol; Piperidines; Rats; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Swine

1986
The serotonin (5-HT) autoreceptor in the hippocampus of the rabbit: role of 5-HT biophase concentration.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Hippocampus; Mathematics; Metergoline; Methiothepin; Methoxydimethyltryptamines; Methysergide; Phentolamine; Pindolol; Quipazine; Rabbits; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1987
Comparison of serotonergic receptor subtypes on the smooth muscle and endothelium of the canine coronary artery.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Ketanserin; Male; Metergoline; Methiothepin; Muscle, Smooth, Vascular; Pindolol; Receptors, Serotonin; Tetrahydronaphthalenes; Vasodilation

1988
Heterogeneous effects of serotonin in the dorsal horn of rat: the involvement of 5-HT1 receptor subtypes.
    Brain research, 1988, Jul-19, Volume: 456, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Indoles; Ketanserin; Male; Neurons, Afferent; Pain; Physical Stimulation; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spinal Cord; Tetrahydronaphthalenes

1988
Identification of the subunit structure of rat pineal adrenergic receptors by photoaffinity labeling.
    Journal of neurochemistry, 1986, Volume: 46, Issue:4

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Cell Membrane; Liver; Molecular Weight; Phenethylamines; Photochemistry; Pindolol; Pineal Gland; Propanolamines; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Spleen; Tetralones

1986
Induction of functional beta-adrenergic receptors in rat aortic smooth muscle cells by sodium butyrate.
    Biochemical pharmacology, 1986, Nov-01, Volume: 35, Issue:21

    Topics: Adenylyl Cyclases; Animals; Butyrates; Butyric Acid; Cell Membrane; Cells, Cultured; Isoproterenol; Kinetics; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta

1986
Autoradiographic analysis of the distribution of beta-adrenoceptors in the dog splenic vasculature.
    British journal of pharmacology, 1986, Volume: 87, Issue:3

    Topics: Animals; Autoradiography; Dogs; In Vitro Techniques; Iodine Radioisotopes; Muscle, Smooth, Vascular; Pindolol; Receptors, Adrenergic, beta; Spleen; Splenic Artery

1986
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus

1987
Autoradiographic localization of beta-1 and beta-2 adrenoceptors in guinea pig atrium and regions of the conducting system.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Autoradiography; Binding, Competitive; Guinea Pigs; Heart Atria; Heart Conduction System; Imidazoles; Isomerism; Kinetics; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1987
Beta-adrenoceptors in human tracheal smooth muscle: characteristics of binding and relaxation.
    Life sciences, 1987, Jun-29, Volume: 40, Issue:26

    Topics: Atenolol; Binding, Competitive; Humans; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pindolol; Propranolol; Receptors, Adrenergic, beta; Sarcolemma; Stereoisomerism; Trachea

1987
Beta-adrenergic receptor subtype is an intrinsic property of the receptor gene product.
    Molecular pharmacology, 1987, Volume: 32, Issue:1

    Topics: Animals; Cricetinae; Gene Expression Regulation; Mice; Pindolol; Protein Processing, Post-Translational; Receptors, Adrenergic, beta; Transfection

1987
(-)-Propranolol and (+/-)-cyanopindolol are mixed agonists-antagonists at serotonin autoreceptors in the hippocampus of the rat brain.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Hippocampus; Male; Pindolol; Potassium; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stereoisomerism; Synaptosomes

1987
Effects of RU 24969 on serotonin release in rat brain cortex: further support for the identity of serotonin autoreceptors with 5-HT1B sites.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 288, Issue:1

    Topics: Animals; Cerebral Cortex; Electric Stimulation; In Vitro Techniques; Indoles; Male; Monoamine Oxidase; Pindolol; Potassium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Synaptosomes

1987
Additive effects of growth hormone and testosterone on lipolysis in adipocytes of hypophysectomized rats.
    The Journal of endocrinology, 1995, Volume: 147, Issue:1

    Topics: Adipocytes; Adrenergic beta-Antagonists; Animals; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Drug Synergism; Growth Hormone; Hypophysectomy; Lipolysis; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Testosterone; Weight Gain

1995
Forskolin-stimulated adenylyl cyclase activity is decreased but beta 2-adrenoceptor function is unchanged in primary hypertension.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:5

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Colforsin; Female; Hemodynamics; Humans; Hypertension; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Sex Factors

1993
Influence of beta 2-adrenergic receptor genotypes on signal transduction in human airway smooth muscle cells.
    American journal of respiratory cell and molecular biology, 1995, Volume: 13, Issue:1

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Genotype; Humans; Isoproterenol; Muscle, Smooth; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta-2; Second Messenger Systems; Signal Transduction; Trachea

1995
Effects of thyroid hormone on norepinephrine signaling in brown adipose tissue. I. Beta 1- and beta 2-adrenergic receptors and cyclic adenosine 3',5'-monophosphate generation.
    Endocrinology, 1995, Volume: 136, Issue:8

    Topics: Adipose Tissue, Brown; Adrenergic Agents; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Hypothyroidism; Norepinephrine; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Reference Values; Signal Transduction; Temperature; Thyroid Hormones

1995
5-HT receptors mediating contractions of the isolated human coronary artery.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Adolescent; Adult; Arteries; Blood Platelets; Child; Child, Preschool; Coronary Vessels; Dose-Response Relationship, Drug; Ergotamine; Female; Humans; In Vitro Techniques; Infant; Ketanserin; Male; Metergoline; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Pindolol; Potassium; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Substance P; Sumatriptan; Yohimbine

1993
Reduced adenylyl cyclase activation with no decrease in beta-adrenergic receptors in basenji greyhound leukocytes: relevance to beta-adrenergic responses in airway smooth muscle.
    The Journal of allergy and clinical immunology, 1995, Volume: 95, Issue:4

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Dogs; Enzyme Activation; Flow Cytometry; GTP-Binding Proteins; Immunoblotting; Leukocytes; Lymphocyte Subsets; Muscle, Smooth; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Trachea

1995
The 5-HT1B receptor mediates the effect of d-fenfluramine on eating caused by intra-hypothalamic injection of neuropeptide Y.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Analysis of Variance; Animals; Antiparkinson Agents; Drug Interactions; Eating; Ergolines; Fenfluramine; Hyperphagia; Hypothalamus; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Male; Metergoline; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Pindolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists

1995
Identification of beta-adrenoceptors in rat lymph nodes and spleen: an autoradiographic study.
    European journal of pharmacology, 1994, Sep-12, Volume: 262, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Image Processing, Computer-Assisted; Ligands; Lymph Nodes; Male; Pindolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Serotonin; Spleen

1994
Is the "atypical" beta-receptor in the rat stomach fundus the rat beta 3 receptor?
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:1

    Topics: Adenylyl Cyclases; Animals; CHO Cells; Cricetinae; Dioxoles; Enzyme Activation; Gene Expression; In Vitro Techniques; Male; Muscle Relaxation; Pindolol; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger; Stomach

1995
Atypical beta-adrenoceptor in bovine adrenal medulla.
    European journal of pharmacology, 1994, Oct-03, Volume: 263, Issue:3

    Topics: Adrenal Medulla; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cattle; Cell Degranulation; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta

1994
Adrenergic receptors in the cerebellum of olivopontocerebellar atrophy.
    Journal of neural transmission. General section, 1994, Volume: 96, Issue:2

    Topics: Aged; Brimonidine Tartrate; Cerebellar Cortex; Cerebellum; Humans; Nerve Tissue Proteins; Norepinephrine; Olivopontocerebellar Atrophies; Pindolol; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta

1994
Adrenaline stimulated cyclic adenosine monophosphate response in leucocytes is reduced after prolonged physical activity combined with sleep and energy deprivation.
    European journal of applied physiology and occupational physiology, 1994, Volume: 69, Issue:5

    Topics: Adrenergic beta-Antagonists; Adult; Binding Sites; Binding, Competitive; Cells, Cultured; Cyclic AMP; Epinephrine; Fasting; Granulocytes; Humans; Leukocytes; Male; Monocytes; Physical Exertion; Pindolol; Sleep Deprivation; Time Factors; Timolol

1994
Increased proliferative activity, loss of beta-adrenergic receptor function and class I major histocompatibility complex antigen surface expression in a modified lymphoma cell line.
    Cellular signalling, 1994, Volume: 6, Issue:7

    Topics: Adrenergic beta-Antagonists; Animals; Biomarkers; Cell Division; Histocompatibility Antigens Class I; Lymphoma; Mice; Pindolol; Receptors, Adrenergic, beta; Tumor Cells, Cultured

1994
Coexisting beta-1 and beta-2-adrenergic receptors with differential receptor reserves in rat C6 glioma cells.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:3

    Topics: Animals; Cyclohexane Monoterpenes; Dexamethasone; Glioma; Guanosine Triphosphate; In Vitro Techniques; Pindolol; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tumor Cells, Cultured

1995
Response of mouse proximal straight tubule and medullary thick ascending limb to beta-agonist.
    Journal of the American Society of Nephrology : JASN, 1993, Volume: 4, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Electrophysiology; Furosemide; In Vitro Techniques; Isoproterenol; Kidney Medulla; Kidney Tubules; Kidney Tubules, Proximal; Kinetics; Membrane Potentials; Mice; Perfusion; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta

1993
[Increase in beta-adrenergic receptors in rabbits in long-term local administration of beta-blockers].
    Der Ophthalmologe : Zeitschrift der Deutschen Ophthalmologischen Gesellschaft, 1993, Volume: 90, Issue:6

    Topics: Administration, Topical; Adrenergic beta-Antagonists; Animals; Autoradiography; Ciliary Body; Cornea; Long-Term Care; Male; Pindolol; Rabbits; Receptors, Adrenergic, beta-2; Timolol

1993
Autoradiographic localization and quantitation of beta 1- and beta 2-adrenoceptors in the human atrioventricular conducting system: a comparison of patients with idiopathic dilated cardiomyopathy and ischemic heart disease.
    Journal of molecular and cellular cardiology, 1994, Volume: 26, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Atrioventricular Node; Binding, Competitive; Bundle of His; Cardiomyopathy, Dilated; Down-Regulation; Female; Heart Septum; Humans; Imidazoles; Male; Middle Aged; Muscle Proteins; Myocardial Ischemia; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1994
The role of 5-hydroxytryptamine1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Anxiety; Betaxolol; Conflict, Psychological; Disease Models, Animal; Drug Interactions; Male; p-Chloroamphetamine; Pindolol; Piperazines; Prazosin; Propanolamines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists

1994
Regulation of beta-adrenoceptors in the guinea-pig sinoatrial node.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Catechols; Chromatography, High Pressure Liquid; Densitometry; Down-Regulation; Drug Interactions; Female; Guinea Pigs; Heart Atria; Isoproterenol; Male; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Sinoatrial Node

1994
Serotonin-dopamine interaction in the rat ventral tegmental area: an electrophysiological study in vivo.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Ergolines; Male; Motor Activity; Pindolol; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Ventral Tegmental Area

1994
Enhanced aggressive behavior in mice lacking 5-HT1B receptor.
    Science (New York, N.Y.), 1994, Sep-23, Volume: 265, Issue:5180

    Topics: Aggression; Animals; Brain Chemistry; Chimera; Female; Indoles; Male; Mice; Motor Activity; Mutation; Pindolol; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombination, Genetic; Serotonin Receptor Agonists

1994
Atypical beta-adrenoceptor- (beta 3-adrenoceptor) mediated relaxation of canine isolated bronchial smooth muscle.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 74, Issue:1

    Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bronchi; Cyclic AMP; Dogs; Ethanolamines; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1993
Beta-adrenergic receptors in the hippocampal and retrohippocampal regions of rats and guinea pigs: autoradiographic and immunohistochemical studies.
    Synapse (New York, N.Y.), 1993, Volume: 13, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Guinea Pigs; Hippocampus; Immunohistochemistry; Limbic System; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Tissue Distribution; Tyrosine 3-Monooxygenase

1993
Cocaine selectively inhibits beta-adrenergic receptor binding in pregnant human myometrium.
    American journal of obstetrics and gynecology, 1993, Volume: 169, Issue:3

    Topics: Adrenergic beta-Antagonists; Binding, Competitive; Cocaine; Dihydroergotoxine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Isoproterenol; Least-Squares Analysis; Molecular Structure; Myometrium; Pindolol; Pregnancy; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1993
Studies on the intrinsic activity (efficacy) of human adrenergic receptors. Co-expression of beta 1 and beta 2 reveals a lower efficacy for the beta 1 receptor.
    Texas Heart Institute journal, 1994, Volume: 21, Issue:1

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Cell Line; Humans; L Cells; Mice; Molecular Sequence Data; Myocardium; Pindolol; Receptors, Adrenergic, beta

1994
Guanine nucleotide regulatory protein alterations in young Milan hypertensive strain rats.
    Biochimica et biophysica acta, 1994, Jan-11, Volume: 1225, Issue:2

    Topics: Adenylyl Cyclases; Alprostadil; Amino Acid Sequence; Animals; Cell Membrane; Cells, Cultured; Colforsin; GTP-Binding Proteins; Hypertension; Immune Sera; Isoproterenol; Molecular Sequence Data; Muscle, Smooth, Vascular; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Signal Transduction

1994
Effects of the 5-HT receptor antagonists cyanopindolol, ICI 169,369, cisapride and granisetron on neuroleptic-induced catalepsy in mice.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1993, Volume: 26, Issue:8

    Topics: Animals; Buspirone; Catalepsy; Cisapride; Female; Granisetron; Haloperidol; Male; Mice; Pindolol; Piperidines; Quinolines; Serotonin Antagonists; Time Factors

1993
5-HT1B receptors mediate potent contractile responses to 5-HT in rat caudal artery.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arteries; Ergolines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Pindolol; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Vasoconstrictor Agents

1993
Verapamil induced reduction of the myocardial beta-adrenoceptor density in BIO 14.6 cardiomyopathic Syrian hamsters.
    Molecular and cellular biochemistry, 1993, Apr-07, Volume: 121, Issue:1

    Topics: Animals; Binding, Competitive; Calcium Channels; Cardiomyopathies; Cricetinae; Disease Models, Animal; Heart; Mesocricetus; Myocardium; Pindolol; Receptors, Adrenergic, beta; Verapamil

1993
The hypophagic effect of restraint stress in rats can be mediated by 5-HT2 receptors in the paraventricular nucleus of the hypothalamus.
    Neuroscience letters, 1993, Apr-02, Volume: 152, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amidines; Animals; Anorexia; Anorexia Nervosa; Disease Models, Animal; Feeding Behavior; Ketanserin; Male; Paraventricular Hypothalamic Nucleus; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Restraint, Physical; Ritanserin; Stress, Physiological

1993
The role of hippocampal 5-hydroxytryptamine 1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists.
    Neuropharmacology, 1995, Volume: 34, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Hippocampus; Male; Pindolol; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1995
Effects of chronic infusion of (-)-isoprenaline on rat cardiac muscarinic (M2)-cholinoceptors and beta 1- and beta 2-adrenoceptors.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Binding, Competitive; Down-Regulation; Heart Ventricles; Imidazoles; Infusion Pumps, Implantable; Isoproterenol; Male; Myocardium; N-Methylscopolamine; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Scopolamine Derivatives

1995
Characterization and localization of atypical beta-adrenoceptors in rat ileum.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Female; Ileum; Iodine Radioisotopes; Isoproterenol; Kinetics; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

1995
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan

1995
Different atypical beta-adrenoceptors mediate isoprenaline-induced relaxation in vascular and non-vascular smooth muscles.
    Life sciences, 1995, Mar-03, Volume: 56, Issue:15

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta

1995
Atypical responses of rat ileum to pindolol, cyanopindolol and iodocyanopindolol.
    British journal of pharmacology, 1996, Volume: 117, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Female; Ileum; In Vitro Techniques; Iodocyanopindolol; Male; Muscle Relaxation; Pindolol; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1996
Abnormalities in 5-HT1A and 5-HT1B receptor binding in severe-seizure genetically epilepsy-prone rats (GEPR-9s).
    Neuropharmacology, 1996, Volume: 35, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Epilepsy; Male; Pindolol; Rats; Receptors, Serotonin; Serotonin Antagonists

1996
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured

1996
Characterization of binding sites for beta-adrenergic agonists and vasoactive intestinal peptide in the rat harderian gland.
    Microscopy research and technique, 1996, Jun-01, Volume: 34, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Harderian Gland; Male; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Vasoactive Intestinal Peptide; Vasoactive Intestinal Peptide

1996
Comparison of the densities of 5-HT4 receptors, beta 1- and beta 2-adrenoceptors in human atrium: functional implications.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Binding, Competitive; Catecholamines; Dioxanes; Heart Atria; Humans; Iodine Radioisotopes; Isotope Labeling; Male; Middle Aged; Myocardial Contraction; Pindolol; Piperidines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Regression Analysis; Serotonin Antagonists

1996
Identification and functional role of beta-adrenergic receptor subtypes in primate and rodent: in vivo versus isolated myocytes.
    Journal of molecular and cellular cardiology, 1996, Volume: 28, Issue:6

    Topics: Adrenergic beta-Antagonists; Animals; Betaxolol; Blood Pressure; Cells, Cultured; Coronary Vessels; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardium; Papio; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Vascular Resistance; Ventricular Function, Left; Ventricular Function, Right

1996
A new peptide, 5-HT-moduline, isolated and purified from mammalian brain specifically interacts with 5-HT1B/1D receptors.
    Behavioural brain research, 1996, Volume: 73, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Binding Sites; Brain Chemistry; Cell Line; Cerebral Cortex; Chromatography, High Pressure Liquid; In Vitro Techniques; Membranes; Mice; Molecular Sequence Data; Neuropeptides; Oligopeptides; Pindolol; Rats; Receptors, Serotonin

1996
Role of 5-HT1b receptor in the pressure-induced behavioral and neurochemical disorders in rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Atmospheric Pressure; Behavior, Animal; Brain Chemistry; Calibration; Dopamine; Electrochemistry; Electrodes; High Pressure Neurological Syndrome; Isoproterenol; Male; Motor Activity; Neostriatum; Pindolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Propranolol therapy in experimental heart failure in rabbits improves cardiac response to catecholamines without beta-adrenoceptor up-regulation.
    Fundamental & clinical pharmacology, 1995, Volume: 9, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Cardiac Output, Low; Catecholamines; Female; Heart; Heart Function Tests; Heart Rate; Hemodynamics; Isoproterenol; Male; Myocardium; Norepinephrine; Pindolol; Propranolol; Rabbits; Receptors, Adrenergic, beta; Up-Regulation; Ventricular Function

1995
Mutations of Tyr326 in the beta 2-adrenoceptor disrupt multiple receptor functions.
    European journal of pharmacology, 1996, Jun-27, Volume: 307, Issue:2

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alanine; Animals; Cell Membrane; CHO Cells; Cloning, Molecular; Cricetinae; Gene Expression; Humans; Iodine Radioisotopes; Isoproterenol; Mutagenesis, Site-Directed; Mutation; Phenylalanine; Pindolol; Protein Binding; Radioligand Assay; Receptors, Adrenergic, beta-2; Transfection; Tyrosine

1996
Effect of endurance physical training on rat liver adenylyl cyclase system.
    Cellular signalling, 1996, Volume: 8, Issue:4

    Topics: Adaptation, Physiological; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Colforsin; Enzyme Activation; Fluorides; Glucagon; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Manganese; Physical Conditioning, Animal; Physical Endurance; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1996
Developmental expression and functional activity of beta 1- and beta 3-adrenoceptors in murine 3T3-F442A differentiating adipocytes.
    European journal of pharmacology, 1996, Feb-15, Volume: 297, Issue:1-2

    Topics: Adenylyl Cyclases; Adipocytes; Animals; Base Sequence; Cell Differentiation; Cell Line; Lipolysis; Membranes; Molecular Sequence Data; Pindolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; RNA, Messenger; Signal Transduction

1996
Mediation of the positive chronotropic effect of CGP 12177 and cyanopindolol in the pithed rat by atypical beta-adrenoceptors, different from beta 3-adrenoceptors.
    British journal of pharmacology, 1996, Volume: 117, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stimulation, Chemical

1996
Differences between the third cardiac beta-adrenoceptor and the colonic beta 3-adrenoceptor in the rat.
    British journal of pharmacology, 1996, Volume: 118, Issue:8

    Topics: Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Female; Heart; Male; Norepinephrine; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

1996
Characterization of a 5-HT1B receptor on CHO cells: functional responses in the absence of radioligand binding.
    British journal of pharmacology, 1996, Volume: 117, Issue:6

    Topics: Animals; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Pindolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1996
Growth hormone treatment of hypophysectomized rats increases catecholamine-induced lipolysis and the number of beta-adrenergic receptors in adipocytes: no differences in the effects of growth hormone on different fat depots.
    Obesity research, 1996, Volume: 4, Issue:5

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Female; Growth Hormone; Hypophysectomy; Iodine Radioisotopes; Isoproterenol; Lipolysis; Male; Norepinephrine; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

1996
Characteristics of cyanopindolol analogues active at the beta 3-adrenoceptor in rat ileum.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Ethanolamines; Female; Ileum; Iodocyanopindolol; Linear Models; Male; Muscle Relaxation; Pindolol; Rats

1996
Characterization of adrenoceptor types and subtypes in American bullfrogs acclimated to warm or cold temperature.
    General and comparative endocrinology, 1996, Volume: 104, Issue:2

    Topics: Acclimatization; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Humans; Idazoxan; Kidney; Membrane Proteins; Myocardium; Pindolol; Prazosin; Radioligand Assay; Rana catesbeiana; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Spinal Cord; Temperature

1996
Modulation of cortical acetylcholine release by serotonin: the role of substance P interneurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:5

    Topics: Acetylcholine; Animals; Capsaicin; Hippocampus; Humans; Indoles; Isoindoles; Neurokinin-1 Receptor Antagonists; Pindolol; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Substance P; Tetrodotoxin

1996
Beta 3-adrenoceptors mediating relaxation of the oesophageal tunica muscularis mucosae and distal colon in the rat: comparative pharmacology and their desensitization by BRL 37344.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Esophagus; Ethanolamines; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1996
Stereoselective modification of circular dichroism spectra of rat lung beta-adrenoceptor protein preparation by enantiomers of epinephrine.
    Chirality, 1996, Volume: 8, Issue:7

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cattle; Circular Dichroism; Epinephrine; In Vitro Techniques; Lung; Membranes; Pindolol; Rats; Receptors, Adrenergic, beta; Serum Albumin, Bovine; Stereoisomerism

1996
Expression of beta 2-adrenoceptors in halobacteria.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:2

    Topics: Adrenergic Antagonists; Animals; Bacteriorhodopsins; Blotting, Northern; Blotting, Western; Genetic Vectors; Halobacterium; Humans; Pindolol; Polymerase Chain Reaction; Receptors, Adrenergic, beta-2; Recombinant Proteins

1997
Characterization of a beta 3-adrenoceptor stimulating gastrin and somatostatin secretions in rat antrum.
    The American journal of physiology, 1997, Volume: 272, Issue:5 Pt 1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; DNA, Complementary; Female; Gastrins; Pindolol; Pyloric Antrum; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Somatostatin; Tetrahydronaphthalenes

1997
Distribution of beta-adrenoceptor subtypes in gastrointestinal tract of nondiabetic and diabetic BB rats. A longitudinal study.
    Digestive diseases and sciences, 1997, Volume: 42, Issue:6

    Topics: Adrenergic beta-Antagonists; Aging; Animals; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Digestive System; Male; Pindolol; Rats; Rats, Inbred BB; Receptors, Adrenergic, beta; Time Factors

1997
The developmental and physiological consequences of disrupting genes encoding beta 1 and beta 2 adrenoceptors.
    Advances in pharmacology (San Diego, Calif.), 1998, Volume: 42

    Topics: Adrenergic beta-Antagonists; Animals; Crosses, Genetic; Homozygote; Imidazoles; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stem Cells

1998
A dual effect of 5-HT1B receptor stimulation on nociceptive dorsal horn neurones in rats.
    European journal of pharmacology, 1997, Sep-24, Volume: 335, Issue:2-3

    Topics: Action Potentials; Animals; Drug Interactions; Electric Stimulation; Female; Neurons; Pain; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission

1997
Early expression of a beta1-adrenergic receptor and catecholamines in Xenopus oocytes and embryos.
    FEBS letters, 1997, Nov-10, Volume: 417, Issue:2

    Topics: Animals; Base Sequence; Catecholamines; DNA, Complementary; Gene Expression; Gene Expression Regulation, Developmental; Molecular Sequence Data; Oocytes; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta-1; Sequence Alignment; Sequence Homology, Amino Acid; Xenopus laevis

1997
Further evidence for differences between cardiac atypical beta-adrenoceptors and brown adipose tissue beta3-adrenoceptors in the pithed rat.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Temperature

1997
Synthesis of new delta 2-isoxazoline derivatives and their pharmacological characterization as beta-adrenergic receptor antagonists.
    Bioorganic & medicinal chemistry, 1998, Volume: 6, Issue:4

    Topics: Adenylyl Cyclases; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; CHO Cells; Chromatography, Thin Layer; Cricetinae; Glioma; Humans; Isoxazoles; Magnetic Resonance Spectroscopy; Pindolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tumor Cells, Cultured

1998
Molecular mechanisms of adenylyl cyclase desensitization in pregnant rat myometrium following in vivo administration of the beta-adrenergic agonist, isoproterenol.
    Biology of reproduction, 1998, Volume: 59, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Drug Tolerance; Female; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Myometrium; Pindolol; Pregnancy; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger

1998
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
    Respiration physiology, 1998, Volume: 112, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

1998
Atypical adrenoceptor-mediated relaxation of canine pulmonary artery through a cAMP-dependent pathway.
    Biochemical and biophysical research communications, 1998, Jul-30, Volume: 248, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dioxoles; Dogs; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Pulmonary Artery; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1998
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:5

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella

1998
Pharmacological profile of the prejunctional 5-HT1 receptors mediating inhibition of sympathetic vasopressor outflow in the pithed rat.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Central Nervous System; Oxadiazoles; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathetic Nervous System

1998
Alterations in cardiac membrane beta-adrenoceptors and adenylyl cyclase due to hypochlorous acid.
    Journal of molecular and cellular cardiology, 1999, Volume: 31, Issue:1

    Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hypochlorous Acid; Immunoblotting; Isoproterenol; Lipid Peroxidation; Methionine; Myocardium; Pertussis Toxin; Pindolol; Propane; Rats; Receptors, Adrenergic; Sodium Fluoride; Virulence Factors, Bordetella

1999
Similar structures and shared switch mechanisms of the beta2-adrenoceptor and the parathyroid hormone receptor. Zn(II) bridges between helices III and VI block activation.
    The Journal of biological chemistry, 1999, Jun-11, Volume: 274, Issue:24

    Topics: Animals; Binding, Competitive; Evolution, Molecular; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Histidine; Humans; Isoproterenol; Models, Molecular; Mutation; Pindolol; Protein Engineering; Protein Structure, Secondary; Receptors, Adrenergic, beta-2; Receptors, Parathyroid Hormone; Rod Opsins; Secretin; Sequence Alignment; Signal Transduction; Zinc

1999
Serotonergic modulation of hyperpolarization-activated current in acutely isolated rat dorsal root ganglion neurons.
    The Journal of physiology, 1999, Jul-15, Volume: 518 ( Pt 2)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Cell Size; Cyclic Nucleotide-Gated Cation Channels; Dopamine Antagonists; Ganglia, Spinal; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Neurons, Afferent; Patch-Clamp Techniques; Pindolol; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Effect of a 14-day hindlimb suspension on beta-adrenoreceptors in rats.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1999, Volume: 123, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Heart Atria; Heart Ventricles; Hindlimb Suspension; Kidney; Male; Pindolol; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1999
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

1999
5-HT1B antagonists modulate clearance of extracellular serotonin in rat hippocampus.
    Neuroscience letters, 1999, May-14, Volume: 266, Issue:3

    Topics: Analysis of Variance; Animals; Corpus Callosum; Hippocampus; Male; Metabolic Clearance Rate; Methiothepin; Neuropeptides; Oligopeptides; Pindolol; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists

1999
Characterisation of the atypical beta-adrenoceptor in rabbit isolated jejunum using BRL 37344, cyanopindolol and SR 59230A.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Jejunum; Male; Pindolol; Propanolamines; Propranolol; Rabbits; Receptors, Adrenergic, beta

1999
Beta1- and beta3-adrenoceptors mediate relaxation in ovine trachealis smooth muscle.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Ethanolamines; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; Sheep; Trachea

1999
Mechanisms of impaired beta-adrenergic receptor signaling in G(alphaq)-mediated cardiac hypertrophy and ventricular dysfunction.
    Molecular pharmacology, 2000, Volume: 57, Issue:2

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Cardiomegaly; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Humans; Iodine Radioisotopes; Mice; Mice, Transgenic; Patch-Clamp Techniques; Pindolol; Receptors, Adrenergic, beta; Signal Transduction; Ventricular Dysfunction

2000
Engineering of a proteolytically stable human beta 2-adrenergic receptor/maltose-binding protein fusion and production of the chimeric protein in Escherichia coli and baculovirus-infected insect cells.
    Journal of biotechnology, 2000, Feb-17, Volume: 77, Issue:2-3

    Topics: Adrenergic beta-Antagonists; Animals; ATP-Binding Cassette Transporters; Baculoviridae; Carrier Proteins; Chromatography, Affinity; Diazomethane; Escherichia coli; Escherichia coli Proteins; Genetic Engineering; GTP-Binding Proteins; Humans; Maltose-Binding Proteins; Monosaccharide Transport Proteins; Periplasmic Binding Proteins; Photoaffinity Labels; Pindolol; Receptors, Adrenergic, beta; Recombinant Fusion Proteins; Spodoptera; Transfection

2000
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents

2000
Role of endothelium/nitric oxide in atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    European journal of pharmacology, 2000, Jun-16, Volume: 398, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Norepinephrine; Oxadiazoles; Phenoxyacetates; Phenoxypropanolamines; Phenylacetates; Pindolol; Propanolamines; Propranolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasodilation

2000
Agonist-directed trafficking of porcine alpha(2A)-adrenergic receptor signaling in Chinese hamster ovary cells: l-isoproterenol selectively activates G(s).
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Binding Sites; Brimonidine Tartrate; CHO Cells; Cricetinae; Drug Interactions; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Isoproterenol; Kinetics; Oxymetazoline; Pindolol; Protein Binding; Quinoxalines; Receptors, Adrenergic, alpha-2; Serotonin Antagonists; Signal Transduction; Swine; Yohimbine

2000
Beta-adrenoceptors in equine trachea and heart.
    Veterinary research communications, 1999, Volume: 23, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Heart Atria; Heart Ventricles; Horses; Imidazoles; Iodine Radioisotopes; Ligands; Male; Muscle, Smooth; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Regression Analysis; Spectrometry, Gamma; Trachea

1999
Mechanism of anemia associated with autonomic dysfunction in rats.
    Autonomic neuroscience : basic & clinical, 2000, Aug-14, Volume: 82, Issue:3

    Topics: Adrenergic beta-Antagonists; Anemia; Animals; Autonomic Nervous System Diseases; Blood Cell Count; Blood Pressure; Epinephrine; Erythrocytes; Erythropoietin; Female; Hematocrit; Hemoglobins; Norepinephrine; Oxidopamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Sympatholytics

2000
5-HT(1B) receptor-mediated regulation of serotonin clearance in rat hippocampus in vivo.
    Journal of neurochemistry, 2000, Volume: 75, Issue:5

    Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Drug Synergism; Electrochemistry; Extracellular Space; Fenclonine; Fluvoxamine; Hippocampus; Male; Metabolic Clearance Rate; Microinjections; Pindolol; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

2000
Opioid tolerance/dependence in neuroblastoma x glioma (NG108-15) hybrid cells is associated with a reduction in spontaneous stimulatory receptor activity.
    FEBS letters, 2000, Nov-24, Volume: 485, Issue:2-3

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; COS Cells; Drug Tolerance; Enzyme Inhibitors; Glioma; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hybrid Cells; Iodine Radioisotopes; Morphine; Narcotics; Neuroblastoma; Pindolol; Propanolamines; Receptors, Adrenergic, beta-2; Signal Transduction; Transfection

2000
beta(1)-Adrenoceptors compensate for beta(3)-adrenoceptors in ileum from beta(3)-adrenoceptor knock-out mice.
    British journal of pharmacology, 2001, Volume: 132, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Genotype; Ileum; In Vitro Techniques; Isoproterenol; Mice; Mice, Knockout; Muscle Relaxation; Muscle, Smooth; Pindolol; Propranolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2001
Abolition of (-)-CGP 12177-evoked cardiostimulation in double beta1/beta2-adrenoceptor knockout mice. Obligatory role of beta1-adrenoceptors for putative beta4-adrenoceptor pharmacology.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Binding, Competitive; Bucladesine; Dose-Response Relationship, Drug; Female; Genotype; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Membranes; Mice; Mice, Knockout; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sinoatrial Node; Tritium

2001
Activation of 5-HT(1B/1D) receptors in the mesolimbic dopamine system increases dopamine release from the nucleus accumbens: a microdialysis study.
    European journal of pharmacology, 2001, Apr-20, Volume: 418, Issue:1-2

    Topics: Animals; Dopamine; Male; Microdialysis; Nucleus Accumbens; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Time Factors; Ventral Tegmental Area

2001
Regional changes in density of serotonin transporter in the brain of 5-HT1A and 5-HT1B knockout mice, and of serotonin innervation in the 5-HT1B knockout.
    Journal of neurochemistry, 2001, Volume: 78, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Behavior, Animal; Brain; Carrier Proteins; Citalopram; Female; Immunohistochemistry; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons; Pindolol; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists

2001
Consequences of labetalol administration on myocardial beta adrenergic receptors in the brain dead pig.
    Annals of transplantation, 2000, Volume: 5, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Brain Death; Heart; Hemodynamics; In Vitro Techniques; Kinetics; Labetalol; Myocardium; Pindolol; Receptors, Adrenergic, beta; Swine

2000
The Ile164 beta(2)-adrenoceptor polymorphism alters salmeterol exosite binding and conventional agonist coupling to G(s).
    European journal of pharmacology, 2001, Jun-15, Volume: 421, Issue:3

    Topics: Adrenergic beta-Agonists; Albuterol; Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Genotype; Humans; Iodine Radioisotopes; Isoproterenol; Metaproterenol; Pindolol; Polymorphism, Genetic; Radioligand Assay; Receptors, Adrenergic, beta-2; Salmeterol Xinafoate; Terbutaline

2001
Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices.
    Journal of neurochemistry, 2001, Volume: 79, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Oxadiazoles; Pindolol; Piperazines; Potassium; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Ventral Tegmental Area

2001
Studies on the expression and function of beta-3-adrenoceptors in the colon of rats with acetic acid-induced colitis.
    Pharmacology, 2002, Volume: 64, Issue:2

    Topics: Acetic Acid; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colitis, Ulcerative; Colon; Dose-Response Relationship, Drug; Ethanolamines; Female; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Peroxidase; Pindolol; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-3; RNA, Messenger

2002
Methiothepin attenuates gastric secretion and motility effects of vagal stimulants at the dorsal vagal complex.
    European journal of pharmacology, 2002, Feb-01, Volume: 436, Issue:1-2

    Topics: Animals; Dose-Response Relationship, Drug; Gastric Acid; Gastrointestinal Motility; Glutamic Acid; Kainic Acid; Male; Methiothepin; Methysergide; Pindolol; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Ritanserin; Serotonin Antagonists; Solitary Nucleus; Time Factors; Vagus Nerve

2002
Altered expression of autonomic neurotransmitter receptors and proliferative responses in lymphocytes from a chronic mild stress model of depression: effects of fluoxetine.
    Brain, behavior, and immunity, 2002, Volume: 16, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Antidepressive Agents, Second-Generation; Autonomic Nervous System; B-Lymphocytes; CD4-CD8 Ratio; Cell Division; Chronic Disease; Cyclic AMP; Cyclic GMP; Disease Models, Animal; Female; Fluoxetine; Iodine Radioisotopes; Mice; Mice, Inbred BALB C; Mitogens; Muscarinic Antagonists; Pindolol; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Muscarinic; Stress, Psychological; T-Lymphocytes; Tritium

2002
Serotonergic control of cerebellar mossy fiber activity by modulation of signal transfer by rat pontine nuclei neurons.
    Journal of neurophysiology, 2002, Volume: 88, Issue:2

    Topics: Animals; Cinanserin; Electrophysiology; Nerve Fibers; Pindolol; Pons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Synaptic Transmission

2002
Evidence that the anorexia induced by lipopolysaccharide is mediated by the 5-HT2C receptor.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 74, Issue:2

    Topics: Adrenergic beta-Antagonists; Aminopyridines; Animals; Anorexia; Dopamine Antagonists; Dose-Response Relationship, Drug; Indoles; Lipopolysaccharides; Male; Metoclopramide; Pindolol; Piperidones; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiro Compounds; Sulfonamides

2003
Hypothalamic-pituitary-thyroid axis and sympathetic nervous system involvement in hyperthermia induced by 3,4-methylenedioxymethamphetamine (Ecstasy).
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:1

    Topics: 3,4-Methylenedioxyamphetamine; Adrenergic alpha-Antagonists; Animals; Drug Interactions; Fever; Hypophysectomy; Hypothalamo-Hypophyseal System; Male; Muscle, Skeletal; N-Methyl-3,4-methylenedioxyamphetamine; Neurotoxicity Syndromes; Pindolol; Prazosin; Rats; Rats, Sprague-Dawley; Rectum; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Thyroid Gland; Thyroxine

2003
Serotonergic facilitation of synaptic activity in the developing rat prefrontal cortex.
    The Journal of physiology, 2004, May-01, Volume: 556, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amphetamines; Animals; Bicuculline; Fluorobenzenes; GABA-A Receptor Antagonists; Glutamic Acid; Indoles; Lidocaine; Male; Patch-Clamp Techniques; Phenols; Pindolol; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sodium Channel Blockers; Sulfonamides; Synapses; Tetrodotoxin; Time Factors

2004
Characterization of mexiletine as an antagonist of beta-adrenoceptor in Chinese hamster ovary cells expressing cloned human beta-adrenoceptors.
    Biochemical pharmacology, 2004, Mar-01, Volume: 67, Issue:5

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Female; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lidocaine; Mexiletine; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

2004
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Site-directed mutagenesis of the rat beta1-adrenoceptor. Involvement of Tyr356 (7.43) in (+/-)cyanopindolol but not (+/-)[125Iodo]cyanopindolol binding.
    European journal of medicinal chemistry, 2004, Volume: 39, Issue:7

    Topics: Adrenergic beta-Antagonists; Animals; Iodine Radioisotopes; Models, Molecular; Mutagenesis, Site-Directed; Pindolol; Protein Binding; Protein Conformation; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Tyrosine

2004
Functional responses of human beta1 adrenoceptors with defined haplotypes for the common 389R>G and 49S>G polymorphisms.
    Pharmacogenetics, 2004, Volume: 14, Issue:6

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cells, Cultured; Cyclic AMP; DNA, Complementary; Down-Regulation; Genotype; Haplotypes; Humans; Iodine Radioisotopes; Isoproterenol; Kidney; Ligands; Pindolol; Polymorphism, Genetic; Receptors, Adrenergic, beta-1

2004
Modulatory effects on myocardial physiology induced by an anti-Trypanosoma cruzi monoclonal antibody involve recognition of major antigenic epitopes from beta1-adrenergic and M2-muscarinic cholinergic receptors without requiring receptor cross-linking.
    Journal of neuroimmunology, 2004, Volume: 153, Issue:1-2

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Animals; Antibodies, Monoclonal; Antibodies, Protozoan; Binding, Competitive; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Epitopes; Immunoglobulin Fab Fragments; In Vitro Techniques; Iodine Isotopes; Mice; Mice, Inbred BALB C; Muscarinic Antagonists; Myocardial Contraction; Pindolol; Quinuclidinyl Benzilate; Radioimmunoassay; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Adrenergic, beta-1; Titrimetry; Trypanosoma cruzi

2004
Impairment of the low-affinity state beta1-adrenoceptor-induced relaxation in spontaneously hypertensive rats.
    British journal of pharmacology, 2004, Volume: 143, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hypertension; Immunohistochemistry; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; omega-N-Methylarginine; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta-1

2004
Evidence for pleiotropic signaling at the mouse beta3-adrenoceptor revealed by SR59230A [3-(2-Ethylphenoxy)-1-[(1,S)-1,2,3,4-tetrahydronapth-1-ylamino]-2S-2-propanol oxalate].
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 312, Issue:3

    Topics: 3T3 Cells; Adipocytes; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclic AMP; Dioxoles; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Ileum; Mice; Pindolol; Propanolamines

2005
Evidence for the presence of beta-3-adrenoceptors mediating relaxation in the human oviduct.
    Pharmacology, 2005, Volume: 74, Issue:3

    Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adult; Dose-Response Relationship, Drug; Ethanolamines; Fallopian Tubes; Female; Humans; In Vitro Techniques; Isoproterenol; Middle Aged; Muscle Relaxation; Pindolol; Propranolol; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2005
Beta-adrenoceptor-mediated vascular relaxation in spontaneously hypertensive rats.
    Autonomic neuroscience : basic & clinical, 2005, Mar-31, Volume: 118, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Tetrahydronaphthalenes

2005
Low-affinity state beta1-adrenoceptor-induced vasodilation in SHR.
    Peptides, 2005, Volume: 26, Issue:8

    Topics: Adrenergic beta-1 Receptor Agonists; Alprenolol; Animals; Aorta; Blood Pressure; Dose-Response Relationship, Drug; Enalapril; Losartan; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta-1; Vasodilation

2005
Positive inotropic and lusitropic effects mediated via the low-affinity state of beta1-adrenoceptors in pithed rats.
    British journal of pharmacology, 2005, Volume: 146, Issue:5

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Animals; Decerebrate State; Humans; Male; Myocardial Contraction; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1

2005
Role of the G protein-coupled receptor kinase site serine cluster in beta2-adrenergic receptor internalization, desensitization, and beta-arrestin translocation.
    The Journal of biological chemistry, 2006, Mar-17, Volume: 281, Issue:11

    Topics: Adenylyl Cyclases; Alanine; Arrestins; Aspartic Acid; beta-Arrestin 1; beta-Arrestin 2; beta-Arrestins; Binding Sites; Blotting, Western; Cell Line; Cell Membrane; Cyclic AMP-Dependent Protein Kinases; DNA, Complementary; Epinephrine; G-Protein-Coupled Receptor Kinase 1; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Mutation; Phosphorylation; Pindolol; Protein Structure, Tertiary; Protein Transport; Receptors, Adrenergic, beta-2; Serine; Time Factors; Transfection

2006
5-HT-stimulated [35S]guanosine-5'-O-(3-thio)triphosphate binding as an assay for functional activation of G proteins coupled with 5-HT1B receptors in rat striatal membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:5

    Topics: Animals; Binding, Competitive; Corpus Striatum; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Oxadiazoles; Pindolol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Agents; Sulfur Radioisotopes; Tryptamines

2006
Potential involvement of a propranolol-insensitive atypical beta-adrenoceptor the vasodilator effect of cyanopindolol in the human pulmonary artery.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2006, Volume: 57, Issue:3

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Bupranolol; Dose-Response Relationship, Drug; Female; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Pindolol; Pulmonary Artery; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction; Vasodilation; Vasodilator Agents

2006
5-HT excites globus pallidus neurons by multiple receptor mechanisms.
    Neuroscience, 2008, Jan-24, Volume: 151, Issue:2

    Topics: Animals; Cations; Electrophysiology; Excitatory Postsynaptic Potentials; Globus Pallidus; In Vitro Techniques; Ion Channels; Male; Neurons; Patch-Clamp Techniques; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Presynaptic; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Synapses; Synaptic Transmission

2008
Structure of a beta1-adrenergic G-protein-coupled receptor.
    Nature, 2008, Jul-24, Volume: 454, Issue:7203

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Amino Acid Motifs; Animals; Binding Sites; Crystallization; Crystallography, X-Ray; Ligands; Models, Molecular; Mutant Proteins; Mutation; Pindolol; Propanolamines; Protein Conformation; Receptors, Adrenergic, beta-1; Thermodynamics; Turkeys

2008
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
    Anesthesia and analgesia, 2008, Volume: 107, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

2008
Influence of beta2-adrenoceptor gene polymorphisms on beta2-adrenoceptor expression in human lung.
    Pulmonary pharmacology & therapeutics, 2010, Volume: 23, Issue:2

    Topics: Female; Gene Expression; Genotype; Humans; Lung; Male; Pindolol; Polymorphism, Single Nucleotide; Promoter Regions, Genetic; Protein Binding; Radioligand Assay; Receptors, Adrenergic, beta-2

2010
Structural insights into conformational stability of wild-type and mutant beta1-adrenergic receptor.
    Biophysical journal, 2010, Jul-21, Volume: 99, Issue:2

    Topics: Adrenergic beta-1 Receptor Agonists; Amino Acid Substitution; Animals; Models, Molecular; Mutant Proteins; Mutation; Norepinephrine; Pindolol; Protein Stability; Protein Structure, Secondary; Receptors, Adrenergic, beta-1; Salts; Transition Temperature; Turkeys

2010
Engineering an ultra-thermostable β(1)-adrenoceptor.
    Journal of molecular biology, 2011, Oct-28, Volume: 413, Issue:3

    Topics: Animals; Cells, Cultured; Crystallography, X-Ray; Disulfides; Humans; Models, Molecular; Mutagenesis, Site-Directed; Mutation; Pindolol; Protein Binding; Protein Conformation; Protein Engineering; Protein Stability; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, G-Protein-Coupled; Temperature; Turkey; Zinc

2011
Tachyphylaxis to the sumatriptan-induced contractile effect in the human uterine artery but not in human cerebral blood vessels: pharmacological demonstration of the 5-HT(1B) receptor functionality loss.
    Pharmacology, 2012, Volume: 89, Issue:1-2

    Topics: Adult; Basilar Artery; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Interactions; Female; Humans; In Vitro Techniques; Male; Middle Aged; Middle Cerebral Artery; Muscle, Smooth, Vascular; Pindolol; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Tachyphylaxis; Time Factors; Uterine Artery

2012
Structural basis for molecular recognition at serotonin receptors.
    Science (New York, N.Y.), 2013, May-03, Volume: 340, Issue:6132

    Topics: Amino Acid Sequence; Binding Sites; Crystallography, X-Ray; Dihydroergotamine; Ergotamine; Humans; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Ligands; Lysergic Acid Diethylamide; Models, Molecular; Molecular Docking Simulation; Molecular Sequence Data; Mutagenesis; Norfenfluramine; Pindolol; Propranolol; Protein Conformation; Protein Folding; Protein Structure, Secondary; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Tryptamines

2013
5-HT1B receptor modulation of the serotonin transporter in vivo: studies using KO mice.
    Neurochemistry international, 2014, Volume: 73

    Topics: Animals; Fluvoxamine; Hippocampus; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Pindolol; Receptor, Serotonin, 5-HT1B; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

2014
The 2.1 Å resolution structure of cyanopindolol-bound β1-adrenoceptor identifies an intramembrane Na+ ion that stabilises the ligand-free receptor.
    PloS one, 2014, Volume: 9, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Binding Sites; Cell Membrane; Crystallography, X-Ray; Models, Molecular; Mutation; Pindolol; Protein Binding; Protein Conformation; Protein Stability; Receptor, Adenosine A2A; Receptors, Adrenergic, beta-1; Sodium; Temperature; Turkeys

2014
Distinct Circuits Underlie the Effects of 5-HT1B Receptors on Aggression and Impulsivity.
    Neuron, 2015, May-06, Volume: 86, Issue:3

    Topics: Actins; Aggression; Animals; Animals, Newborn; Brain; Choice Behavior; Conditioning, Operant; Dopamine; Dopamine Uptake Inhibitors; Doxycycline; Gene Expression Regulation, Developmental; Impulsive Behavior; Iodine Isotopes; Mice; Mice, Transgenic; Pindolol; Piperazines; Protein Binding; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists

2015
Pharmacological Analysis and Structure Determination of 7-Methylcyanopindolol-Bound β1-Adrenergic Receptor.
    Molecular pharmacology, 2015, Volume: 88, Issue:6

    Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Humans; Pindolol; Protein Binding; Protein Structure, Secondary; Receptors, Adrenergic, beta-1; Structure-Activity Relationship; Turkey

2015
Nebivolol ameliorates asymmetric dimethylarginine-induced vascular response in rat aorta via β3 adrenoceptor-mediated mechanism.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2016, Volume: 38, Issue:2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Antagonists; Animals; Aorta; Arginine; Butoxamine; Enzyme Inhibitors; In Vitro Techniques; Nebivolol; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Pindolol; Rats; Receptors, Adrenergic, beta-3

2016
A Lack of Serotonin 1B Autoreceptors Results in Decreased Anxiety and Depression-Related Behaviors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2016, Volume: 41, Issue:12

    Topics: Animals; Animals, Newborn; Anxiety; Autoreceptors; Depression; Disease Models, Animal; Exploratory Behavior; Food Preferences; Hippocampus; Iodine Isotopes; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Transgenic; Pindolol; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

2016
Deep brain stimulation and fluoxetine exert different long-term changes in the serotonergic system.
    Neuropharmacology, 2018, Volume: 135

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Deep Brain Stimulation; Fluoxetine; Hippocampus; Iodine Radioisotopes; Pindolol; Prefrontal Cortex; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Plasma Membrane Transport Proteins; Time Factors; Tritium

2018