pindolol has been researched along with colforsin in 61 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 19 (31.15) | 18.7374 |
1990's | 39 (63.93) | 18.2507 |
2000's | 3 (4.92) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Mader, SL | 1 |
Bylund, DB; Pleus, RC | 1 |
Molinoff, PB; Unsworth, CD | 1 |
Armata, MG; Crescimanno, M; D'Alessandro, N; D'Amico, C; Leonardi, V; Palazzoadriano, M | 1 |
Bohmaker, K; Chalfin, M; Meller, E | 1 |
Atkinson, BN; Minneman, KP | 1 |
Asano, M; Asano, T; Masuzawa, K; Matsuda, T | 1 |
Emmerich, B; Göhly, U; Haen, E; Hallek, M; Kamp, T; Remien, J | 1 |
Pracyk, JB; Slotkin, TA | 1 |
Insel, PA; Jasper, JR; Michel, MC | 2 |
Beusenberg, FD; Bonta, IL; Leurs, R; van Amsterdam, JG; van Schaik, A | 1 |
Ciaranello, RD; Dean, R; Tan, GL | 1 |
Buckenmeyer, PJ; Dax, EM; Goldfarb, AH; Partilla, JS; Piñeyro, MA | 1 |
Hui, KK; Yu, JL | 1 |
McCook, EC; Navarro, HA; Seidler, FJ; Slotkin, TA | 1 |
De Vivo, M; Maayani, S | 1 |
Hoffman, BB; Lee, CH; Tsujimoto, G | 1 |
Linden, J | 1 |
Callens-el Amrani, F; Chevalier, B; Mansier, P; Swynghedauw, B | 1 |
Baughman, KL; Cates, AE; Feldman, AM; Levine, MA; Van Dop, C | 1 |
Hintze, TH; Homcy, CJ; Nejima, J; Susanni, EE; Uemura, N; Vatner, DE; Vatner, SF | 1 |
Cornfield, LJ; Martin, AR; Nelson, DL; Taylor, EW | 1 |
Insel, PA; Maisel, AS; Motulsky, HJ; Ziegler, MG | 1 |
Crooke, ST; Stadel, JM | 1 |
Kelvie, SL; Sundaresan, PR | 1 |
Boland, SR; Katz, MS; Schmidt, SJ | 1 |
Oksenberg, D; Peroutka, SJ | 1 |
Ebstein, RP; Lipshitz, I; Mintzer, J; Steinitz, M; Stessman, J | 1 |
Goldie, RG; Papadimitriou, JM; Paterson, JW; Rigby, PJ; Self, HM; Spina, D | 1 |
Ballard, PL; Dattel, BJ; Davis, DJ; Roberts, JM | 1 |
Dax, EM; Gregerman, RI; Partilla, JS; Piñeyro, MA | 1 |
Crooke, ST; Nakada, MT; Poksay, KS; Stadel, JM | 1 |
Keshles, O; Levitzki, A | 1 |
Ichihara, A; Kato, S; Nakamura, T; Noda, C; Shinjyo, F; Tomomura, A | 1 |
Björntorp, P; Edén, S; Xu, X; Yang, S | 1 |
Blankesteijn, WM; de Pont, JJ; Graafsma, SJ; Thien, T; Willems, PH | 1 |
Merryman, J; Orloff, M; Park, PG; Schuller, HM | 1 |
Davis, DJ; Lefebvre, CA; Lyon, ME | 1 |
Benovic, JL; Higgins, NC; Kelsen, SG; Mardini, IA; Zhou, S | 1 |
Blin, N; Drumare, MF; Nahmias, C; Strosberg, AD | 1 |
Adham, N; Branchek, T; Ellerbrock, B; Hartig, P; Weinshank, RL | 1 |
Clark, CJ; Connell, JM; Milligan, G | 1 |
Fay, FS; Moore, ED | 1 |
Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
Christoffersen, T; Jacobsen, FW; Refsnes, M; Sandnes, D | 1 |
Martyn, JA; Wang, C | 1 |
Pantuck, CB; Smiley, RM | 1 |
Droms, KA | 1 |
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H | 1 |
Asano, M; Azuma, H; Hashimoto, S; Ito, Y; Kato, H; Morikawa, K; Ohashi, T | 1 |
Díaz-Laviada, I; Guillén, A; Haro, A; Nieto, JL | 1 |
Bolofo, ML; Giles, H; Lansdell, SJ; Martin, GR; Wilson, HL | 1 |
Bertin, B; Jockers, R; Marullo, S; Strosberg, AD | 1 |
Bungay, PJ; George, SE; Naylor, LH | 1 |
Cohen-Tannoudji, J; Coudouel, N; Lécrivain, JL; Legrand, C; Maltier, JP; Robin, MT | 1 |
Branchek, TA; Zgombick, JM | 1 |
Dhalla, NS; Elimban, V; Persad, S; Siddiqui, F | 1 |
Ishii, K; Karikomi, Y; Kubota, Y; Nakahara, T; Sakamoto, K | 1 |
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B | 1 |
61 other study(ies) available for pindolol and colforsin
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Influence of animal age on the beta-adrenergic system in cultured rat aortic and mesenteric artery smooth muscle cells.
Topics: Aging; Alprostadil; Animals; Aorta, Thoracic; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Iodocyanopindolol; Isoproterenol; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Pindolol; Propranolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta | 1992 |
Desensitization and down-regulation of the 5-hydroxytryptamine1B receptor in the opossum kidney cell line.
Topics: Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Down-Regulation; Iodocyanopindolol; Kidney; Opossums; Pindolol; Radioligand Assay; Receptors, Serotonin; Serotonin | 1992 |
Regulation of the 5-hydroxytryptamine1B receptor in opossum kidney cells after exposure to agonists.
Topics: Animals; Cells, Cultured; Colforsin; Cyclic AMP; Down-Regulation; Iodine Radioisotopes; Iodocyanopindolol; Kidney; Kinetics; Opossums; Pindolol; Piperazines; Radioligand Assay; Receptors, Serotonin; Serotonin; Stimulation, Chemical; Up-Regulation | 1992 |
Number and functionality of beta-adrenergic receptors in the mouse lymphocytic P388 leukemia as a doxorubicin-sensitive and -resistant variant.
Topics: Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Doxorubicin; Drug Resistance; Leukemia P388; Mice; Pindolol | 1992 |
Serotonin 5-HT1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Body Temperature; Colforsin; Drug Tolerance; Fenclonine; Hypothermia; Male; Mice; Pindolol; Piperazines; Quinolines; Receptors, Serotonin; Serotonin | 1992 |
Occupancy-response relationships for beta- and alpha 2-adrenergic receptors exerting opposing effects on cAMP production.
Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Isoproterenol; Kinetics; Neuroglia; Norepinephrine; Pindolol; Quinolines; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1992 |
Decreased responsiveness to beta-adrenoceptor agonists in arterial strips from spontaneously hypertensive rats is not associated with alterations in beta-adrenoceptors.
Topics: Animals; Arteries; Colforsin; Femoral Artery; In Vitro Techniques; Iodocyanopindolol; Male; Mesenteric Arteries; Norepinephrine; Pindolol; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Vasoconstriction | 1991 |
Reduced responsiveness of adenylate cyclase to forskolin in human lymphoma cells.
Topics: Adenylyl Cyclase Inhibitors; Aged; B-Lymphocytes; Binding Sites; Cholera Toxin; Colforsin; Cyclic AMP; Female; Humans; Isoproterenol; Lymphoma, Non-Hodgkin; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured | 1991 |
Thyroid hormone differentially regulates development of beta-adrenergic receptors, adenylate cyclase and ornithine decarboxylase in rat heart and kidney.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Animals, Newborn; Body Weight; Bucladesine; Colforsin; Heart; Isoproterenol; Kidney; Myocardium; Organ Size; Ornithine Decarboxylase; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Triiodothyronine | 1991 |
Partial agonistic activity of two irreversible beta-adrenergic receptor ligands, bromoacetylated derivatives of alprenolol and pindolol.
Topics: Adrenergic beta-Agonists; Alprenolol; Cell Line; Colforsin; Cyclic AMP; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Humans; Pindolol | 1991 |
Sensitization enhances the adenylyl cyclase responsiveness in alveolar macrophages. Changes induced at post-receptor level.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cholera Toxin; Colforsin; Dinoprostone; Enzyme Activation; GTP-Binding Proteins; Guinea Pigs; Iodocyanopindolol; Isoproterenol; Macrophage Activation; Macrophages; Male; Ovalbumin; Pindolol; Pulmonary Alveoli; Signal Transduction; Timolol | 1991 |
G-protein-linked serotonin receptors in mouse kidney exhibit identical properties to 5-HT1b receptors in brain.
Topics: Alkylation; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Colforsin; Ethylmaleimide; GTP-Binding Proteins; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Kidney; Male; Mice; Mice, Inbred BALB C; Pindolol; Receptors, Serotonin | 1990 |
Endurance training, not acute exercise, differentially alters beta-receptors and cyclase in skeletal fiber types.
Topics: Adenylyl Cyclases; Animals; Colforsin; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Muscles; Organ Specificity; Physical Conditioning, Animal; Physical Exertion; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reference Values; Sodium Fluoride; Succinate Cytochrome c Oxidoreductase | 1990 |
Protein kinase A and/or C inhibitors potentiate isoproterenol-induced cyclic AMP accumulation in intact human lymphocytes.
Topics: Alprostadil; Colforsin; Cyclic AMP; Drug Synergism; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lymphocytes; Phorbol Esters; Pindolol; Protein Kinase C; Protein Kinase Inhibitors | 1990 |
Fetal nicotine exposure produces postnatal up-regulation of adenylate cyclase activity in peripheral tissues.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Colforsin; Female; Fetal Resorption; Isoproterenol; Kidney; Myocardium; Nicotine; Pindolol; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Up-Regulation | 1990 |
Stimulation and inhibition of adenylyl cyclase by distinct 5-hydroxytryptamine receptors.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Membrane; Cerebral Cortex; Colforsin; Drug Interactions; Enzyme Activation; Fluphenazine; Guinea Pigs; Hippocampus; Mathematics; Mianserin; Pindolol; Piperazines; Rats; Receptors, Serotonin; Spiperone | 1990 |
Age-related decrease in beta adrenergic receptor-mediated vascular smooth muscle relaxation.
Topics: 1-Methyl-3-isobutylxanthine; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Acetylcholine; Aging; Bucladesine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Iodocyanopindolol; Isoproterenol; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroglycerin; Pindolol; Receptors, Adrenergic, beta; Serotonin | 1986 |
Enhanced cAMP accumulation after termination of cholinergic action in the heart.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Heart; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Myocardial Contraction; Myocardium; Parasympathomimetics; Pindolol; Receptors, Muscarinic | 1987 |
Beta-adrenergic system is modified in compensatory pressure cardiac overload in rats: physiological and biochemical evidence.
Topics: Animals; Binding Sites; Cardiac Pacing, Artificial; Cardiomegaly; Colforsin; Coronary Circulation; Isoproterenol; Male; Myocardial Contraction; Perfusion; Pindolol; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1989 |
Multiple effects of ethanol on cardiac adenylate cyclase.
Topics: Adenosine Diphosphate; Adenylyl Cyclases; Animals; Cholera Toxin; Colforsin; Ethanol; Female; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Manganese; Myocardium; NAD; Pindolol; Rabbits; Receptors, Adrenergic, beta | 1989 |
Chronic norepinephrine elicits desensitization by uncoupling the beta-receptor.
Topics: Adenylyl Cyclases; Animals; Colforsin; Dogs; Drug Tolerance; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart Ventricles; Hemodynamics; Isoproterenol; Norepinephrine; Organ Size; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Sodium-Potassium-Exchanging ATPase; Ventricular Function | 1989 |
MDL 73005EF: partial agonist at the 5-HT1A receptor negatively linked to adenylate cyclase.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenosine Triphosphate; Adenylyl Cyclase Inhibitors; Animals; Buspirone; Colforsin; Cyclic AMP; Dioxins; Hippocampus; In Vitro Techniques; Male; Membranes; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiro Compounds; Tetrahydronaphthalenes; Tryptamines | 1989 |
Ischemia- and agonist-induced changes in alpha- and beta-adrenergic receptor traffic in guinea pig hearts.
Topics: Animals; Colforsin; Epinephrine; Guanylyl Imidodiphosphate; Guinea Pigs; Iodocyanopindolol; Male; Microscopy, Electron; Myocardium; Pindolol; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1987 |
Differential effects of fluoride on adenylate cyclase activity and guanine nucleotide regulation of agonist high-affinity receptor binding.
Topics: Adenylyl Cyclases; Alprostadil; Animals; Anura; Cell Membrane; Cells, Cultured; Colforsin; Dihydroalprenolol; Epinephrine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Iodocyanopindolol; Isoproterenol; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Yohimbine | 1988 |
Beta-adrenergic receptor coupled adenylate cyclase in rat kidney. Differential coupling in glomeruli and tubules.
Topics: Adenylyl Cyclases; Animals; Betaxolol; Colforsin; Cyclic AMP; Guanylyl Imidodiphosphate; Iodocyanopindolol; Kidney Glomerulus; Kidney Tubules; Male; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stereoisomerism | 1988 |
Developmental changes of beta-adrenergic receptor-linked adenylate cyclase of rat liver.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding Sites; Colforsin; Diterpenes; Female; Fluorides; Growth Inhibitors; Guanosine Triphosphate; Iodine Radioisotopes; Liver; Male; Pindolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Stimulation, Chemical | 1985 |
Molecular mechanism of beta-adrenergic receptor blockers with intrinsic sympathomimetic activity.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Celiprolol; Colforsin; Cyclic AMP; Drug Synergism; Isoproterenol; Lymphoma; Pindolol; Propanolamines; Propranolol; Sympathomimetics; Tumor Cells, Cultured | 1988 |
Antagonism of 5-hydroxytryptamine1A (5-HT1A) receptor-mediated modulation of adenylate cyclase activity by pindolol and propranolol isomers.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Colforsin; GTP-Binding Proteins; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Pindolol; Propranolol; Rats; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism; Tetrahydronaphthalenes | 1988 |
Beta-adrenergic-stimulated adenylate cyclase activity in normal and EBV-transformed lymphocytes.
Topics: Adenylyl Cyclases; Cell Line; Cell Transformation, Viral; Colforsin; Cyclic AMP; Herpesvirus 4, Human; Iodocyanopindolol; Isoproterenol; Lymphocytes; Pindolol; Receptors, Adrenergic, beta | 1985 |
Influence of the epithelium on responsiveness of guinea-pig isolated trachea to contractile and relaxant agonists.
Topics: Acetylcholine; Animals; Asthma; Autoradiography; Carbachol; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Epithelium; Female; Guinea Pigs; Histamine; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Muscle Contraction; Nitroglycerin; Pindolol; Potassium; Receptors, Adrenergic, beta; Theophylline; Trachea | 1986 |
Beta-adrenergic receptors and cyclic adenosine monophosphate generation in human fetal lung.
Topics: Alprostadil; Colforsin; Cyclic AMP; Gestational Age; Humans; Iodocyanopindolol; Isoproterenol; Lung; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1987 |
Beta-adrenergic receptors, glucagon receptors, and their relationship to adenylate cyclase in rat liver during aging.
Topics: Adenylyl Cyclases; Aging; Animals; Colforsin; Enzyme Activation; Glucagon; Guanine Nucleotides; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Gastrointestinal Hormone; Receptors, Glucagon; Sodium Fluoride | 1987 |
Glucocorticoid regulation of beta-adrenergic receptors in 3T3-L1 preadipocytes.
Topics: Adipose Tissue; Alprenolol; Animals; Binding, Competitive; Cell Line; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Dexamethasone; Epinephrine; Glucocorticoids; Iodocyanopindolol; Kinetics; Membranes; Mice; Norepinephrine; Pindolol; Receptors, Adrenergic, beta; Tunicamycin | 1987 |
The ontogenesis of beta-adrenergic receptors and of adenylate cyclase in the developing rat brain.
Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Brain; Colforsin; Diterpenes; Guanylyl Imidodiphosphate; Iodocyanopindolol; Manganese; Pindolol; Rats; Receptors, Adrenergic, beta | 1984 |
Mechanism of heterologous desensitization of the adenylate cyclase system by glucagon in primary cultures of adult rat hepatocytes.
Topics: Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Diterpenes; Glucagon; Guanylyl Imidodiphosphate; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sodium Fluoride | 1984 |
Additive effects of growth hormone and testosterone on lipolysis in adipocytes of hypophysectomized rats.
Topics: Adipocytes; Adrenergic beta-Antagonists; Animals; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Drug Synergism; Growth Hormone; Hypophysectomy; Lipolysis; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Testosterone; Weight Gain | 1995 |
Forskolin-stimulated adenylyl cyclase activity is decreased but beta 2-adrenoceptor function is unchanged in primary hypertension.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Colforsin; Female; Hemodynamics; Humans; Hypertension; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Sex Factors | 1993 |
Beta-adrenergic mitogenic signal transduction in peripheral lung adenocarcinoma: implications for individuals with preexisting chronic lung disease.
Topics: Adenocarcinoma; Cell Division; Colforsin; Cyclic AMP; Epinephrine; Humans; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Lung Diseases; Lung Neoplasms; Mitogens; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured | 1995 |
Characterisation of the beta adrenergic response cascade in fetal guinea pig lung.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Membrane; Choline; Colforsin; Cyclic AMP; Gestational Age; Guinea Pigs; Isoproterenol; Lung; Models, Biological; Phosphatidylcholines; Pindolol; Radioimmunoassay; Receptors, Adrenergic, beta | 1994 |
Functional behavior of the beta-adrenergic receptor-adenylyl cyclase system in rabbit airway epithelium.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Betaxolol; Binding, Competitive; Bradykinin; Colforsin; Cyclic AMP; Dinoprostone; Epithelial Cells; Epithelium; Glycerol; Isoproterenol; Kinetics; Pindolol; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Tetradecanoylphorbol Acetate; Trachea | 1994 |
Mediation of most atypical effects by species homologues of the beta 3-adrenoceptor.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Colforsin; Cricetinae; Epinephrine; Humans; Iodocyanopindolol; Isoproterenol; Ligands; Mice; Norepinephrine; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Species Specificity | 1994 |
Receptor reserve masks partial agonist activity of drugs in a cloned rat 5-hydroxytryptamine1B receptor expression system.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; Iodocyanopindolol; Pindolol; Quinolines; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Transfection; Virulence Factors, Bordetella | 1993 |
Guanine nucleotide regulatory protein alterations in young Milan hypertensive strain rats.
Topics: Adenylyl Cyclases; Alprostadil; Amino Acid Sequence; Animals; Cell Membrane; Cells, Cultured; Colforsin; GTP-Binding Proteins; Hypertension; Immune Sera; Isoproterenol; Molecular Sequence Data; Muscle, Smooth, Vascular; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Signal Transduction | 1994 |
Isoproterenol stimulates rapid extrusion of sodium from isolated smooth muscle cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzofurans; Bufo marinus; Carbachol; Colforsin; Ethers, Cyclic; Fluorescent Dyes; Gastric Mucosa; In Vitro Techniques; Isoproterenol; Kinetics; Microscopy, Fluorescence; Muscle, Smooth; Ouabain; Pindolol; Potassium; Sodium; Stomach; Time Factors | 1993 |
Activity of serotonin (5-HT) receptor agonists, partial agonists and antagonists at cloned human 5-HT1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HeLa cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Colforsin; Cyclic AMP; HeLa Cells; Humans; Indoles; Lysergic Acid Diethylamide; Models, Biological; Pindolol; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Transfection | 1993 |
Long-term inhibitory effect of cAMP on beta-adrenoceptor acquisition and nonselective attenuation of adenylyl cyclase in hepatocytes.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Down-Regulation; Glucagon; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Thionucleotides | 1993 |
Burn injury alters beta-adrenergic receptor and second messenger function in rat ventricular muscle.
Topics: Adrenergic beta-Agonists; Animals; Burns; Cell Membrane; Colforsin; Cyclic AMP; Heart Ventricles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Myocardium; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Second Messenger Systems; Signal Transduction | 1996 |
Effect of cesarean delivery on perioperative regulation of the beta-adrenergic receptor system of human lymphocytes.
Topics: Abdomen; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Alprostadil; Anesthesia, Obstetrical; Anesthesia, Spinal; Cesarean Section; Colforsin; Cyclic AMP; Down-Regulation; Female; Humans; Iodine Radioisotopes; Isoproterenol; Lymphocytes; Pindolol; Pregnancy; Receptors, Adrenergic, beta; Stress, Physiological; Thoracic Surgery; Vasodilator Agents | 1996 |
Beta-adrenergic signalling in neoplastic lung type 2 cells: glucocorticoid-dependent and -independent defects.
Topics: Adenylyl Cyclases; Animals; Cell Line; Colforsin; Dexamethasone; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Iodocyanopindolol; Isoproterenol; Lung Neoplasms; Mice; Pindolol; Receptors, Adrenergic, beta | 1996 |
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured | 1996 |
Potent inhibition of spontaneous rhythmic contraction by a novel beta 2-adrenoceptor agonist, HSR-81, in pregnant rat uterus.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Benzyl Alcohols; Binding, Competitive; Colforsin; Diestrus; Female; Gestational Age; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Isotope Labeling; Kinetics; Pindolol; Pregnancy; Propanolamines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Ritodrine; Uterine Contraction | 1996 |
Effect of endurance physical training on rat liver adenylyl cyclase system.
Topics: Adaptation, Physiological; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Colforsin; Enzyme Activation; Fluorides; Glucagon; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Manganese; Physical Conditioning, Animal; Physical Endurance; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1996 |
Characterization of a 5-HT1B receptor on CHO cells: functional responses in the absence of radioligand binding.
Topics: Animals; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Pindolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1996 |
Activation of a beta 2-adrenergic receptor/Gs alpha fusion protein elicits a desensitization-resistant cAMP signal capable of inhibiting proliferation of two cancer cell lines.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Albuterol; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Colforsin; Cyclic AMP; Down-Regulation; Gene Expression Regulation, Neoplastic; GTP-Binding Protein alpha Subunits, Gs; Iodocyanopindolol; Isoproterenol; Mice; Pindolol; ras Proteins; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Salmeterol Xinafoate; Signal Transduction; Transfection; Tumor Cells, Cultured | 1997 |
Functional coupling of endogenous serotonin (5-HT1B) and calcitonin (C1a) receptors in CHO cells to a cyclic AMP-responsive luciferase reporter gene.
Topics: Animals; Calcitonin; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine; Gene Expression; Genes, Reporter; Kinetics; Luciferases; Pindolol; Receptor, Serotonin, 5-HT1B; Receptors, Calcitonin; Receptors, Serotonin; Recombinant Fusion Proteins; Serotonin; Serotonin Receptor Agonists; Somatostatin; Transfection | 1997 |
Molecular mechanisms of adenylyl cyclase desensitization in pregnant rat myometrium following in vivo administration of the beta-adrenergic agonist, isoproterenol.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Drug Tolerance; Female; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Myometrium; Pindolol; Pregnancy; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger | 1998 |
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella | 1998 |
Alterations in cardiac membrane beta-adrenoceptors and adenylyl cyclase due to hypochlorous acid.
Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hypochlorous Acid; Immunoblotting; Isoproterenol; Lipid Peroxidation; Methionine; Myocardium; Pertussis Toxin; Pindolol; Propane; Rats; Receptors, Adrenergic; Sodium Fluoride; Virulence Factors, Bordetella | 1999 |
Characterization of mexiletine as an antagonist of beta-adrenoceptor in Chinese hamster ovary cells expressing cloned human beta-adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Female; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lidocaine; Mexiletine; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection | 2004 |
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 2008 |