Page last updated: 2024-08-16

pindolol and colforsin

pindolol has been researched along with colforsin in 61 studies

Research

Studies (61)

TimeframeStudies, this research(%)All Research%
pre-199019 (31.15)18.7374
1990's39 (63.93)18.2507
2000's3 (4.92)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Mader, SL1
Bylund, DB; Pleus, RC1
Molinoff, PB; Unsworth, CD1
Armata, MG; Crescimanno, M; D'Alessandro, N; D'Amico, C; Leonardi, V; Palazzoadriano, M1
Bohmaker, K; Chalfin, M; Meller, E1
Atkinson, BN; Minneman, KP1
Asano, M; Asano, T; Masuzawa, K; Matsuda, T1
Emmerich, B; Göhly, U; Haen, E; Hallek, M; Kamp, T; Remien, J1
Pracyk, JB; Slotkin, TA1
Insel, PA; Jasper, JR; Michel, MC2
Beusenberg, FD; Bonta, IL; Leurs, R; van Amsterdam, JG; van Schaik, A1
Ciaranello, RD; Dean, R; Tan, GL1
Buckenmeyer, PJ; Dax, EM; Goldfarb, AH; Partilla, JS; Piñeyro, MA1
Hui, KK; Yu, JL1
McCook, EC; Navarro, HA; Seidler, FJ; Slotkin, TA1
De Vivo, M; Maayani, S1
Hoffman, BB; Lee, CH; Tsujimoto, G1
Linden, J1
Callens-el Amrani, F; Chevalier, B; Mansier, P; Swynghedauw, B1
Baughman, KL; Cates, AE; Feldman, AM; Levine, MA; Van Dop, C1
Hintze, TH; Homcy, CJ; Nejima, J; Susanni, EE; Uemura, N; Vatner, DE; Vatner, SF1
Cornfield, LJ; Martin, AR; Nelson, DL; Taylor, EW1
Insel, PA; Maisel, AS; Motulsky, HJ; Ziegler, MG1
Crooke, ST; Stadel, JM1
Kelvie, SL; Sundaresan, PR1
Boland, SR; Katz, MS; Schmidt, SJ1
Oksenberg, D; Peroutka, SJ1
Ebstein, RP; Lipshitz, I; Mintzer, J; Steinitz, M; Stessman, J1
Goldie, RG; Papadimitriou, JM; Paterson, JW; Rigby, PJ; Self, HM; Spina, D1
Ballard, PL; Dattel, BJ; Davis, DJ; Roberts, JM1
Dax, EM; Gregerman, RI; Partilla, JS; Piñeyro, MA1
Crooke, ST; Nakada, MT; Poksay, KS; Stadel, JM1
Keshles, O; Levitzki, A1
Ichihara, A; Kato, S; Nakamura, T; Noda, C; Shinjyo, F; Tomomura, A1
Björntorp, P; Edén, S; Xu, X; Yang, S1
Blankesteijn, WM; de Pont, JJ; Graafsma, SJ; Thien, T; Willems, PH1
Merryman, J; Orloff, M; Park, PG; Schuller, HM1
Davis, DJ; Lefebvre, CA; Lyon, ME1
Benovic, JL; Higgins, NC; Kelsen, SG; Mardini, IA; Zhou, S1
Blin, N; Drumare, MF; Nahmias, C; Strosberg, AD1
Adham, N; Branchek, T; Ellerbrock, B; Hartig, P; Weinshank, RL1
Clark, CJ; Connell, JM; Milligan, G1
Fay, FS; Moore, ED1
Leysen, JE; Pauwels, PJ; Van Gompel, P1
Christoffersen, T; Jacobsen, FW; Refsnes, M; Sandnes, D1
Martyn, JA; Wang, C1
Pantuck, CB; Smiley, RM1
Droms, KA1
Esbenshade, TA; Guerrero, SW; Minneman, KP; Zhong, H1
Asano, M; Azuma, H; Hashimoto, S; Ito, Y; Kato, H; Morikawa, K; Ohashi, T1
Díaz-Laviada, I; Guillén, A; Haro, A; Nieto, JL1
Bolofo, ML; Giles, H; Lansdell, SJ; Martin, GR; Wilson, HL1
Bertin, B; Jockers, R; Marullo, S; Strosberg, AD1
Bungay, PJ; George, SE; Naylor, LH1
Cohen-Tannoudji, J; Coudouel, N; Lécrivain, JL; Legrand, C; Maltier, JP; Robin, MT1
Branchek, TA; Zgombick, JM1
Dhalla, NS; Elimban, V; Persad, S; Siddiqui, F1
Ishii, K; Karikomi, Y; Kubota, Y; Nakahara, T; Sakamoto, K1
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B1

Other Studies

61 other study(ies) available for pindolol and colforsin

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Influence of animal age on the beta-adrenergic system in cultured rat aortic and mesenteric artery smooth muscle cells.
    Journal of gerontology, 1992, Volume: 47, Issue:2

    Topics: Aging; Alprostadil; Animals; Aorta, Thoracic; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Iodocyanopindolol; Isoproterenol; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Pindolol; Propranolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta

1992
Desensitization and down-regulation of the 5-hydroxytryptamine1B receptor in the opossum kidney cell line.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:1

    Topics: Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Down-Regulation; Iodocyanopindolol; Kidney; Opossums; Pindolol; Radioligand Assay; Receptors, Serotonin; Serotonin

1992
Regulation of the 5-hydroxytryptamine1B receptor in opossum kidney cells after exposure to agonists.
    Molecular pharmacology, 1992, Volume: 42, Issue:3

    Topics: Animals; Cells, Cultured; Colforsin; Cyclic AMP; Down-Regulation; Iodine Radioisotopes; Iodocyanopindolol; Kidney; Kinetics; Opossums; Pindolol; Piperazines; Radioligand Assay; Receptors, Serotonin; Serotonin; Stimulation, Chemical; Up-Regulation

1992
Number and functionality of beta-adrenergic receptors in the mouse lymphocytic P388 leukemia as a doxorubicin-sensitive and -resistant variant.
    Pharmacological research, 1992, Volume: 26 Suppl 2

    Topics: Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Doxorubicin; Drug Resistance; Leukemia P388; Mice; Pindolol

1992
Serotonin 5-HT1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Body Temperature; Colforsin; Drug Tolerance; Fenclonine; Hypothermia; Male; Mice; Pindolol; Piperazines; Quinolines; Receptors, Serotonin; Serotonin

1992
Occupancy-response relationships for beta- and alpha 2-adrenergic receptors exerting opposing effects on cAMP production.
    Receptor, 1992,Fall, Volume: 2, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Isoproterenol; Kinetics; Neuroglia; Norepinephrine; Pindolol; Quinolines; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1992
Decreased responsiveness to beta-adrenoceptor agonists in arterial strips from spontaneously hypertensive rats is not associated with alterations in beta-adrenoceptors.
    Journal of hypertension, 1991, Volume: 9, Issue:7

    Topics: Animals; Arteries; Colforsin; Femoral Artery; In Vitro Techniques; Iodocyanopindolol; Male; Mesenteric Arteries; Norepinephrine; Pindolol; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Vasoconstriction

1991
Reduced responsiveness of adenylate cyclase to forskolin in human lymphoma cells.
    Biochemical pharmacology, 1991, Sep-12, Volume: 42, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Aged; B-Lymphocytes; Binding Sites; Cholera Toxin; Colforsin; Cyclic AMP; Female; Humans; Isoproterenol; Lymphoma, Non-Hodgkin; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured

1991
Thyroid hormone differentially regulates development of beta-adrenergic receptors, adenylate cyclase and ornithine decarboxylase in rat heart and kidney.
    Journal of developmental physiology, 1991, Volume: 16, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Animals, Newborn; Body Weight; Bucladesine; Colforsin; Heart; Isoproterenol; Kidney; Myocardium; Organ Size; Ornithine Decarboxylase; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Triiodothyronine

1991
Partial agonistic activity of two irreversible beta-adrenergic receptor ligands, bromoacetylated derivatives of alprenolol and pindolol.
    Biochemical pharmacology, 1991, Dec-11, Volume: 42 Suppl

    Topics: Adrenergic beta-Agonists; Alprenolol; Cell Line; Colforsin; Cyclic AMP; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Humans; Pindolol

1991
Sensitization enhances the adenylyl cyclase responsiveness in alveolar macrophages. Changes induced at post-receptor level.
    Biochemical pharmacology, 1991, Jul-15, Volume: 42, Issue:3

    Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cholera Toxin; Colforsin; Dinoprostone; Enzyme Activation; GTP-Binding Proteins; Guinea Pigs; Iodocyanopindolol; Isoproterenol; Macrophage Activation; Macrophages; Male; Ovalbumin; Pindolol; Pulmonary Alveoli; Signal Transduction; Timolol

1991
G-protein-linked serotonin receptors in mouse kidney exhibit identical properties to 5-HT1b receptors in brain.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:3

    Topics: Alkylation; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Colforsin; Ethylmaleimide; GTP-Binding Proteins; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Kidney; Male; Mice; Mice, Inbred BALB C; Pindolol; Receptors, Serotonin

1990
Endurance training, not acute exercise, differentially alters beta-receptors and cyclase in skeletal fiber types.
    The American journal of physiology, 1990, Volume: 258, Issue:1 Pt 1

    Topics: Adenylyl Cyclases; Animals; Colforsin; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Muscles; Organ Specificity; Physical Conditioning, Animal; Physical Exertion; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reference Values; Sodium Fluoride; Succinate Cytochrome c Oxidoreductase

1990
Protein kinase A and/or C inhibitors potentiate isoproterenol-induced cyclic AMP accumulation in intact human lymphocytes.
    Life sciences, 1990, Volume: 47, Issue:4

    Topics: Alprostadil; Colforsin; Cyclic AMP; Drug Synergism; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lymphocytes; Phorbol Esters; Pindolol; Protein Kinase C; Protein Kinase Inhibitors

1990
Fetal nicotine exposure produces postnatal up-regulation of adenylate cyclase activity in peripheral tissues.
    Life sciences, 1990, Volume: 47, Issue:17

    Topics: Adenylyl Cyclases; Animals; Cell Membrane; Colforsin; Female; Fetal Resorption; Isoproterenol; Kidney; Myocardium; Nicotine; Pindolol; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Up-Regulation

1990
Stimulation and inhibition of adenylyl cyclase by distinct 5-hydroxytryptamine receptors.
    Biochemical pharmacology, 1990, Oct-01, Volume: 40, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Membrane; Cerebral Cortex; Colforsin; Drug Interactions; Enzyme Activation; Fluphenazine; Guinea Pigs; Hippocampus; Mathematics; Mianserin; Pindolol; Piperazines; Rats; Receptors, Serotonin; Spiperone

1990
Age-related decrease in beta adrenergic receptor-mediated vascular smooth muscle relaxation.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Acetylcholine; Aging; Bucladesine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Iodocyanopindolol; Isoproterenol; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroglycerin; Pindolol; Receptors, Adrenergic, beta; Serotonin

1986
Enhanced cAMP accumulation after termination of cholinergic action in the heart.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1987, Volume: 1, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Heart; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Myocardial Contraction; Myocardium; Parasympathomimetics; Pindolol; Receptors, Muscarinic

1987
Beta-adrenergic system is modified in compensatory pressure cardiac overload in rats: physiological and biochemical evidence.
    Journal of cardiovascular pharmacology, 1989, Volume: 13, Issue:3

    Topics: Animals; Binding Sites; Cardiac Pacing, Artificial; Cardiomegaly; Colforsin; Coronary Circulation; Isoproterenol; Male; Myocardial Contraction; Perfusion; Pindolol; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1989
Multiple effects of ethanol on cardiac adenylate cyclase.
    Journal of cardiovascular pharmacology, 1989, Volume: 13, Issue:5

    Topics: Adenosine Diphosphate; Adenylyl Cyclases; Animals; Cholera Toxin; Colforsin; Ethanol; Female; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Manganese; Myocardium; NAD; Pindolol; Rabbits; Receptors, Adrenergic, beta

1989
Chronic norepinephrine elicits desensitization by uncoupling the beta-receptor.
    The Journal of clinical investigation, 1989, Volume: 84, Issue:6

    Topics: Adenylyl Cyclases; Animals; Colforsin; Dogs; Drug Tolerance; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart Ventricles; Hemodynamics; Isoproterenol; Norepinephrine; Organ Size; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Sodium-Potassium-Exchanging ATPase; Ventricular Function

1989
MDL 73005EF: partial agonist at the 5-HT1A receptor negatively linked to adenylate cyclase.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenosine Triphosphate; Adenylyl Cyclase Inhibitors; Animals; Buspirone; Colforsin; Cyclic AMP; Dioxins; Hippocampus; In Vitro Techniques; Male; Membranes; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiro Compounds; Tetrahydronaphthalenes; Tryptamines

1989
Ischemia- and agonist-induced changes in alpha- and beta-adrenergic receptor traffic in guinea pig hearts.
    The American journal of physiology, 1987, Volume: 253, Issue:5 Pt 2

    Topics: Animals; Colforsin; Epinephrine; Guanylyl Imidodiphosphate; Guinea Pigs; Iodocyanopindolol; Male; Microscopy, Electron; Myocardium; Pindolol; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1987
Differential effects of fluoride on adenylate cyclase activity and guanine nucleotide regulation of agonist high-affinity receptor binding.
    The Biochemical journal, 1988, Aug-15, Volume: 254, Issue:1

    Topics: Adenylyl Cyclases; Alprostadil; Animals; Anura; Cell Membrane; Cells, Cultured; Colforsin; Dihydroalprenolol; Epinephrine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Iodocyanopindolol; Isoproterenol; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Yohimbine

1988
Beta-adrenergic receptor coupled adenylate cyclase in rat kidney. Differential coupling in glomeruli and tubules.
    Biochemical pharmacology, 1988, Dec-01, Volume: 37, Issue:23

    Topics: Adenylyl Cyclases; Animals; Betaxolol; Colforsin; Cyclic AMP; Guanylyl Imidodiphosphate; Iodocyanopindolol; Kidney Glomerulus; Kidney Tubules; Male; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stereoisomerism

1988
Developmental changes of beta-adrenergic receptor-linked adenylate cyclase of rat liver.
    The American journal of physiology, 1985, Volume: 248, Issue:6 Pt 1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding Sites; Colforsin; Diterpenes; Female; Fluorides; Growth Inhibitors; Guanosine Triphosphate; Iodine Radioisotopes; Liver; Male; Pindolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Stimulation, Chemical

1985
Molecular mechanism of beta-adrenergic receptor blockers with intrinsic sympathomimetic activity.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1988, Volume: 2, Issue:13

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Celiprolol; Colforsin; Cyclic AMP; Drug Synergism; Isoproterenol; Lymphoma; Pindolol; Propanolamines; Propranolol; Sympathomimetics; Tumor Cells, Cultured

1988
Antagonism of 5-hydroxytryptamine1A (5-HT1A) receptor-mediated modulation of adenylate cyclase activity by pindolol and propranolol isomers.
    Biochemical pharmacology, 1988, Sep-15, Volume: 37, Issue:18

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Colforsin; GTP-Binding Proteins; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Pindolol; Propranolol; Rats; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism; Tetrahydronaphthalenes

1988
Beta-adrenergic-stimulated adenylate cyclase activity in normal and EBV-transformed lymphocytes.
    Experientia, 1985, Dec-15, Volume: 41, Issue:12

    Topics: Adenylyl Cyclases; Cell Line; Cell Transformation, Viral; Colforsin; Cyclic AMP; Herpesvirus 4, Human; Iodocyanopindolol; Isoproterenol; Lymphocytes; Pindolol; Receptors, Adrenergic, beta

1985
Influence of the epithelium on responsiveness of guinea-pig isolated trachea to contractile and relaxant agonists.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Acetylcholine; Animals; Asthma; Autoradiography; Carbachol; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Epithelium; Female; Guinea Pigs; Histamine; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Muscle Contraction; Nitroglycerin; Pindolol; Potassium; Receptors, Adrenergic, beta; Theophylline; Trachea

1986
Beta-adrenergic receptors and cyclic adenosine monophosphate generation in human fetal lung.
    Pediatric research, 1987, Volume: 21, Issue:2

    Topics: Alprostadil; Colforsin; Cyclic AMP; Gestational Age; Humans; Iodocyanopindolol; Isoproterenol; Lung; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1987
Beta-adrenergic receptors, glucagon receptors, and their relationship to adenylate cyclase in rat liver during aging.
    Endocrinology, 1987, Volume: 120, Issue:4

    Topics: Adenylyl Cyclases; Aging; Animals; Colforsin; Enzyme Activation; Glucagon; Guanine Nucleotides; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Gastrointestinal Hormone; Receptors, Glucagon; Sodium Fluoride

1987
Glucocorticoid regulation of beta-adrenergic receptors in 3T3-L1 preadipocytes.
    Molecular pharmacology, 1987, Volume: 31, Issue:4

    Topics: Adipose Tissue; Alprenolol; Animals; Binding, Competitive; Cell Line; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Dexamethasone; Epinephrine; Glucocorticoids; Iodocyanopindolol; Kinetics; Membranes; Mice; Norepinephrine; Pindolol; Receptors, Adrenergic, beta; Tunicamycin

1987
The ontogenesis of beta-adrenergic receptors and of adenylate cyclase in the developing rat brain.
    Biochemical pharmacology, 1984, Oct-15, Volume: 33, Issue:20

    Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Brain; Colforsin; Diterpenes; Guanylyl Imidodiphosphate; Iodocyanopindolol; Manganese; Pindolol; Rats; Receptors, Adrenergic, beta

1984
Mechanism of heterologous desensitization of the adenylate cyclase system by glucagon in primary cultures of adult rat hepatocytes.
    The Journal of biological chemistry, 1984, Jun-25, Volume: 259, Issue:12

    Topics: Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Diterpenes; Glucagon; Guanylyl Imidodiphosphate; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sodium Fluoride

1984
Additive effects of growth hormone and testosterone on lipolysis in adipocytes of hypophysectomized rats.
    The Journal of endocrinology, 1995, Volume: 147, Issue:1

    Topics: Adipocytes; Adrenergic beta-Antagonists; Animals; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Drug Synergism; Growth Hormone; Hypophysectomy; Lipolysis; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Testosterone; Weight Gain

1995
Forskolin-stimulated adenylyl cyclase activity is decreased but beta 2-adrenoceptor function is unchanged in primary hypertension.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:5

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Colforsin; Female; Hemodynamics; Humans; Hypertension; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Pindolol; Receptors, Adrenergic, beta; Sex Factors

1993
Beta-adrenergic mitogenic signal transduction in peripheral lung adenocarcinoma: implications for individuals with preexisting chronic lung disease.
    Cancer research, 1995, Aug-15, Volume: 55, Issue:16

    Topics: Adenocarcinoma; Cell Division; Colforsin; Cyclic AMP; Epinephrine; Humans; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Lung Diseases; Lung Neoplasms; Mitogens; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Signal Transduction; Tumor Cells, Cultured

1995
Characterisation of the beta adrenergic response cascade in fetal guinea pig lung.
    Thorax, 1994, Volume: 49, Issue:7

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Membrane; Choline; Colforsin; Cyclic AMP; Gestational Age; Guinea Pigs; Isoproterenol; Lung; Models, Biological; Phosphatidylcholines; Pindolol; Radioimmunoassay; Receptors, Adrenergic, beta

1994
Functional behavior of the beta-adrenergic receptor-adenylyl cyclase system in rabbit airway epithelium.
    American journal of respiratory cell and molecular biology, 1994, Volume: 11, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Betaxolol; Binding, Competitive; Bradykinin; Colforsin; Cyclic AMP; Dinoprostone; Epithelial Cells; Epithelium; Glycerol; Isoproterenol; Kinetics; Pindolol; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Tetradecanoylphorbol Acetate; Trachea

1994
Mediation of most atypical effects by species homologues of the beta 3-adrenoceptor.
    British journal of pharmacology, 1994, Volume: 112, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Colforsin; Cricetinae; Epinephrine; Humans; Iodocyanopindolol; Isoproterenol; Ligands; Mice; Norepinephrine; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Species Specificity

1994
Receptor reserve masks partial agonist activity of drugs in a cloned rat 5-hydroxytryptamine1B receptor expression system.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; Iodocyanopindolol; Pindolol; Quinolines; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Transfection; Virulence Factors, Bordetella

1993
Guanine nucleotide regulatory protein alterations in young Milan hypertensive strain rats.
    Biochimica et biophysica acta, 1994, Jan-11, Volume: 1225, Issue:2

    Topics: Adenylyl Cyclases; Alprostadil; Amino Acid Sequence; Animals; Cell Membrane; Cells, Cultured; Colforsin; GTP-Binding Proteins; Hypertension; Immune Sera; Isoproterenol; Molecular Sequence Data; Muscle, Smooth, Vascular; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Signal Transduction

1994
Isoproterenol stimulates rapid extrusion of sodium from isolated smooth muscle cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Sep-01, Volume: 90, Issue:17

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzofurans; Bufo marinus; Carbachol; Colforsin; Ethers, Cyclic; Fluorescent Dyes; Gastric Mucosa; In Vitro Techniques; Isoproterenol; Kinetics; Microscopy, Fluorescence; Muscle, Smooth; Ouabain; Pindolol; Potassium; Sodium; Stomach; Time Factors

1993
Activity of serotonin (5-HT) receptor agonists, partial agonists and antagonists at cloned human 5-HT1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HeLa cells.
    Biochemical pharmacology, 1993, Jan-26, Volume: 45, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Colforsin; Cyclic AMP; HeLa Cells; Humans; Indoles; Lysergic Acid Diethylamide; Models, Biological; Pindolol; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Transfection

1993
Long-term inhibitory effect of cAMP on beta-adrenoceptor acquisition and nonselective attenuation of adenylyl cyclase in hepatocytes.
    European journal of pharmacology, 1993, Jul-15, Volume: 246, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Down-Regulation; Glucagon; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Thionucleotides

1993
Burn injury alters beta-adrenergic receptor and second messenger function in rat ventricular muscle.
    Critical care medicine, 1996, Volume: 24, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Burns; Cell Membrane; Colforsin; Cyclic AMP; Heart Ventricles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Myocardium; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Second Messenger Systems; Signal Transduction

1996
Effect of cesarean delivery on perioperative regulation of the beta-adrenergic receptor system of human lymphocytes.
    Anesthesia and analgesia, 1996, Volume: 82, Issue:5

    Topics: Abdomen; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Alprostadil; Anesthesia, Obstetrical; Anesthesia, Spinal; Cesarean Section; Colforsin; Cyclic AMP; Down-Regulation; Female; Humans; Iodine Radioisotopes; Isoproterenol; Lymphocytes; Pindolol; Pregnancy; Receptors, Adrenergic, beta; Stress, Physiological; Thoracic Surgery; Vasodilator Agents

1996
Beta-adrenergic signalling in neoplastic lung type 2 cells: glucocorticoid-dependent and -independent defects.
    British journal of cancer, 1996, Volume: 74, Issue:3

    Topics: Adenylyl Cyclases; Animals; Cell Line; Colforsin; Dexamethasone; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Iodocyanopindolol; Isoproterenol; Lung Neoplasms; Mice; Pindolol; Receptors, Adrenergic, beta

1996
Inducible expression of beta 1- and beta 2-adrenergic receptors in rat C6 glioma cells: functional interactions between closely related subtypes.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Gene Expression Regulation, Neoplastic; Genomic Library; Glioma; Imidazoles; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Norepinephrine; Pindolol; Radioligand Assay; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Tumor Cells, Cultured

1996
Potent inhibition of spontaneous rhythmic contraction by a novel beta 2-adrenoceptor agonist, HSR-81, in pregnant rat uterus.
    European journal of pharmacology, 1996, Jul-04, Volume: 307, Issue:3

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Benzyl Alcohols; Binding, Competitive; Colforsin; Diestrus; Female; Gestational Age; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Isotope Labeling; Kinetics; Pindolol; Pregnancy; Propanolamines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Ritodrine; Uterine Contraction

1996
Effect of endurance physical training on rat liver adenylyl cyclase system.
    Cellular signalling, 1996, Volume: 8, Issue:4

    Topics: Adaptation, Physiological; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Colforsin; Enzyme Activation; Fluorides; Glucagon; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Liver; Male; Manganese; Physical Conditioning, Animal; Physical Endurance; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1996
Characterization of a 5-HT1B receptor on CHO cells: functional responses in the absence of radioligand binding.
    British journal of pharmacology, 1996, Volume: 117, Issue:6

    Topics: Animals; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Pindolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1996
Activation of a beta 2-adrenergic receptor/Gs alpha fusion protein elicits a desensitization-resistant cAMP signal capable of inhibiting proliferation of two cancer cell lines.
    Receptors & channels, 1997, Volume: 5, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Albuterol; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Colforsin; Cyclic AMP; Down-Regulation; Gene Expression Regulation, Neoplastic; GTP-Binding Protein alpha Subunits, Gs; Iodocyanopindolol; Isoproterenol; Mice; Pindolol; ras Proteins; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Salmeterol Xinafoate; Signal Transduction; Transfection; Tumor Cells, Cultured

1997
Functional coupling of endogenous serotonin (5-HT1B) and calcitonin (C1a) receptors in CHO cells to a cyclic AMP-responsive luciferase reporter gene.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Animals; Calcitonin; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine; Gene Expression; Genes, Reporter; Kinetics; Luciferases; Pindolol; Receptor, Serotonin, 5-HT1B; Receptors, Calcitonin; Receptors, Serotonin; Recombinant Fusion Proteins; Serotonin; Serotonin Receptor Agonists; Somatostatin; Transfection

1997
Molecular mechanisms of adenylyl cyclase desensitization in pregnant rat myometrium following in vivo administration of the beta-adrenergic agonist, isoproterenol.
    Biology of reproduction, 1998, Volume: 59, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colforsin; Drug Tolerance; Female; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Myometrium; Pindolol; Pregnancy; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger

1998
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:5

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella

1998
Alterations in cardiac membrane beta-adrenoceptors and adenylyl cyclase due to hypochlorous acid.
    Journal of molecular and cellular cardiology, 1999, Volume: 31, Issue:1

    Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hypochlorous Acid; Immunoblotting; Isoproterenol; Lipid Peroxidation; Methionine; Myocardium; Pertussis Toxin; Pindolol; Propane; Rats; Receptors, Adrenergic; Sodium Fluoride; Virulence Factors, Bordetella

1999
Characterization of mexiletine as an antagonist of beta-adrenoceptor in Chinese hamster ovary cells expressing cloned human beta-adrenoceptors.
    Biochemical pharmacology, 2004, Mar-01, Volume: 67, Issue:5

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Female; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lidocaine; Mexiletine; Pindolol; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

2004
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
    Anesthesia and analgesia, 2008, Volume: 107, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

2008