Page last updated: 2024-08-16

pindolol and brl 37344

pindolol has been researched along with brl 37344 in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19901 (4.17)18.7374
1990's18 (75.00)18.2507
2000's5 (20.83)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kompa, AR; Molenaar, P; Pak, HS; Roberts, SJ; Summers, RJ1
Chiyotani, A; Kondo, M; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F1
Esbenshade, TA; Granneman, JG; Han, C; Minneman, KP; Theroux, TL1
MacDonald, A; McLaughlin, DP1
Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS1
Baude, B; Blin, N; Emorine, LJ; Fève, B; Lasnier, F; Nahmias, C; Pairault, J; Strosberg, AD1
Bast, A; Rademaker, B; van der Vliet, A1
Fraser, C; Giacobino, JP; Muzzin, P; Seydoux, J; Venter, JC1
Amend, A; Guan, XM; Strader, CD1
Chiyotani, A; Konno, K; Takeuchi, S; Tamaoki, J; Yamauchi, F; Yamawaki, I1
Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD; Zilberfarb, V1
Oriowo, MA1
el Borai, N; Ito, K; Nakano, S; Nakazawa, H; Tanaka, E; Yamakawa, A; Yamamura, M1
Feller, DR; Konkar, AA; Lezama, EJ; Miller, DD; Salazar-Bookaman, MM1
Hoey, AJ; Jackson, CM; Pegg, GG; Sillence, MN1
Houston, G; Kelly, J1
Isono, K; Nagai, A; Tagaya, E; Tamaoki, J1
MacDonald, A; Watt, K1
Cherian, A; Mustafa, SM; Oriowo, MA; Yousif, M1
Horinouchi, T; Koike, K2
Hussein, SM; Khan, I; Oriowo, M1
Brahmadevara, N; MacDonald, A; Shaw, AM1
Chandrasekhar, B; Fatinikun, T; Kadavil, EA; Khan, I; Omu, AE; Oriowo, MA1

Other Studies

24 other study(ies) available for pindolol and brl 37344

ArticleYear
Localization of (-)-[125I]cyanopindolol binding in guinea-pig heart: characteristics of non-beta-adrenoceptor related binding in cardiac pacemaker and conducting regions.
    Neuroscience letters, 1992, Feb-17, Volume: 136, Issue:1

    Topics: Alprenolol; Animals; Ascorbic Acid; Binding Sites; Ethanolamines; Female; Guinea Pigs; Haloperidol; Heart Conduction System; Isoproterenol; Male; Myocardium; Peroxidase; Phentolamine; Pindolol; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta; Serotonin; Thiophenes; Trachea

1992
[Airway epithelial beta 3-adrenergic receptor--effect on bioelectric properties and its mechanism of action].
    Nihon Kyobu Shikkan Gakkai zasshi, 1992, Volume: 30, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Bumetanide; Calcium; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Epithelium; Ethanolamines; Membrane Potentials; Pindolol; Receptors, Adrenergic, beta; Trachea

1992
Coexisting beta 1- and atypical beta-adrenergic receptors cause redundant increases in cyclic AMP in human neuroblastoma cells.
    Molecular pharmacology, 1992, Volume: 42, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Neuroblastoma; Pindolol; Radioligand Assay; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured

1992
Characterization of catecholamine-mediated relaxations in rat isolated gastric fundus: evidence for an atypical beta-adrenoceptor.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Catecholamines; Ethanolamines; Gastric Fundus; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Norepinephrine; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
    European journal of pharmacology, 1991, Jul-09, Volume: 199, Issue:3

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Atypical beta-adrenergic receptor in 3T3-F442A adipocytes. Pharmacological and molecular relationship with the human beta 3-adrenergic receptor.
    The Journal of biological chemistry, 1991, Oct-25, Volume: 266, Issue:30

    Topics: 3T3 Cells; Adipose Tissue; Adrenergic beta-Antagonists; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; DNA; Ethanolamines; Humans; Imidazoles; Mice; Molecular Sequence Data; Oxprenolol; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; RNA, Messenger

1991
A beta adrenoceptor with atypical characteristics is involved in the relaxation of the rat small intestine.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:1

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Ethanolamines; In Vitro Techniques; Intestine, Small; Iodocyanopindolol; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Pindolol; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1990
Discrepancies between the affinities of binding and action of the novel beta-adrenergic agonist BRL 37344 in rat brown adipose tissue.
    Biochemical and biophysical research communications, 1988, Oct-14, Volume: 156, Issue:1

    Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Animals; Binding, Competitive; Cell Membrane; Ethanolamines; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Oxygen Consumption; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reference Values

1988
Determination of structural domains for G protein coupling and ligand binding in beta 3-adrenergic receptor.
    Molecular pharmacology, 1995, Volume: 48, Issue:3

    Topics: Adrenergic beta-Agonists; Amino Acid Sequence; Base Sequence; Binding, Competitive; Cell Membrane; Ethanolamines; GTP-Binding Proteins; Humans; Iodine Radioisotopes; Iodocyanopindolol; Ligands; Molecular Sequence Data; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1995
Atypical beta-adrenoceptor- (beta 3-adrenoceptor) mediated relaxation of canine isolated bronchial smooth muscle.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 74, Issue:1

    Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bronchi; Cyclic AMP; Dogs; Ethanolamines; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1993
Transcriptional modulation by n-butyric acid of beta 1-, beta 2-, and beta 3-adrenergic receptor balance in 3T3-F442A adipocytes.
    The Journal of biological chemistry, 1994, Mar-04, Volume: 269, Issue:9

    Topics: 3T3 Cells; Adenylyl Cyclase Inhibitors; Adipocytes; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Base Sequence; Butyrates; Butyric Acid; DNA Primers; DNA, Complementary; Ethanolamines; Gene Expression Regulation; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Molecular Sequence Data; Oligonucleotides, Antisense; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Transcription, Genetic

1994
Different atypical beta-adrenoceptors mediate isoprenaline-induced relaxation in vascular and non-vascular smooth muscles.
    Life sciences, 1995, Mar-03, Volume: 56, Issue:15

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Pindolol; Rats; Receptors, Adrenergic, beta

1995
Regulation of heat production of brown adipocytes via typical and atypical beta-adrenoceptors in the rat.
    The Japanese journal of physiology, 1995, Volume: 45, Issue:6

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Calorimetry; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Phenoxyacetates; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1995
Pharmacological study of atypical beta-adrenoceptors in rat esophageal smooth muscle.
    European journal of pharmacology, 1996, Jul-11, Volume: 308, Issue:1

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Carbachol; Clenbuterol; Cyclohexane Monoterpenes; Esophagus; Ethanolamines; Female; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Phenoxyacetates; Phenoxypropanolamines; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Serotonin Antagonists; Trachea; Tretoquinol

1996
Characteristics of cyanopindolol analogues active at the beta 3-adrenoceptor in rat ileum.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Ethanolamines; Female; Ileum; Iodocyanopindolol; Linear Models; Male; Muscle Relaxation; Pindolol; Rats

1996
Beta 3-adrenoceptors mediating relaxation of the oesophageal tunica muscularis mucosae and distal colon in the rat: comparative pharmacology and their desensitization by BRL 37344.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Esophagus; Ethanolamines; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1996
Atypical adrenoceptor-mediated relaxation of canine pulmonary artery through a cAMP-dependent pathway.
    Biochemical and biophysical research communications, 1998, Jul-30, Volume: 248, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dioxoles; Dogs; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Pulmonary Artery; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3

1998
Characterisation of the atypical beta-adrenoceptor in rabbit isolated jejunum using BRL 37344, cyanopindolol and SR 59230A.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Isoproterenol; Jejunum; Male; Pindolol; Propanolamines; Propranolol; Rabbits; Receptors, Adrenergic, beta

1999
Beta1- and beta3-adrenoceptors mediate relaxation in ovine trachealis smooth muscle.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Ethanolamines; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; Sheep; Trachea

1999
(+/-)-Pindolol acts as a partial agonist at atypical beta-adrenoceptors in the guinea pig duodenum.
    Japanese journal of pharmacology, 2001, Volume: 85, Issue:1

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Duodenum; Ethanolamines; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta

2001
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
    European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism

2001
Studies on the expression and function of beta-3-adrenoceptors in the colon of rats with acetic acid-induced colitis.
    Pharmacology, 2002, Volume: 64, Issue:2

    Topics: Acetic Acid; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colitis, Ulcerative; Colon; Dose-Response Relationship, Drug; Ethanolamines; Female; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Peroxidase; Pindolol; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-3; RNA, Messenger

2002
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Evidence for the presence of beta-3-adrenoceptors mediating relaxation in the human oviduct.
    Pharmacology, 2005, Volume: 74, Issue:3

    Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adult; Dose-Response Relationship, Drug; Ethanolamines; Fallopian Tubes; Female; Humans; In Vitro Techniques; Isoproterenol; Middle Aged; Muscle Relaxation; Pindolol; Propranolol; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2005