pindolol has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 132 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 25 (18.94) | 18.7374 |
1990's | 84 (63.64) | 18.2507 |
2000's | 20 (15.15) | 29.6817 |
2010's | 3 (2.27) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Glennon, RA | 1 |
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B | 1 |
Chaput, C; Millan, MJ; Newman-Tancredi, A; Verrièle, L | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Chodkowski, A; Dawidowski, M; Dybała, M; Herold, F; Izbicki, Ł; Kleps, J; Mazurek, A; Mazurek, AP; Nowak, G; Pluciński, F; Siwek, A; Stachowicz, K; Turło, J | 1 |
Shibata, S; Tominaga, K; Ueki, S; Watanabe, S | 1 |
Guan, XM; Kobilka, BK; Peroutka, SJ | 1 |
Coop, CF; McNaughton, N; Scott, DJ | 1 |
Bohmaker, K; Chalfin, M; Meller, E | 1 |
Buisson-Defferier, S; Van den Buuse, M | 1 |
Gilbert, F; Pan, L | 1 |
Jacobs, M; McRee, C; Meyer, DC | 1 |
Newman-Tancredi, A; Strange, PG; Sundaram, H | 1 |
Barrett, JE; Gleeson, S | 1 |
Blitz-Siebert, A; Helke, CJ; Thor, KB | 2 |
McEwen, BS; Mendelson, SD | 1 |
Dreteler, GH; Ramage, AG; Saxena, PR; Wouters, W | 1 |
Gradin, K | 1 |
Hjorth, S; Liu, Y; Sharp, T | 1 |
Beller, KD; Kolassa, N; Sanders, KH | 1 |
Hillegaart, V | 1 |
Cerruti, C; Marlier, L; Privat, A; Teilhac, JR | 1 |
Kostowski, W; Pałejko, W; Płaźnik, A; Stefański, R | 1 |
Schwab, EF; Zemlan, FP | 1 |
Fukuda, H; Ono, H; Ono, SS | 1 |
Ulrichsen, J | 1 |
Cowen, PJ; Gartside, SE; Hjorth, S | 1 |
Bird, ED; Crino, PB; Plager, MD; Vogt, BA | 1 |
Crino, PB; Vogt, BA; Volicer, L; Wiley, RG | 1 |
Eison, AS; Margraf, RR; Wright, RN; Yocca, FD | 1 |
Budziszewska, B; Błaszczyńska, E; Chojnacka-Wójcik, E; Ismaiel, AM; Przegaliński, E; Tatarczyńska, E | 1 |
Connor, HE; Higgins, GA | 1 |
Manaker, S; Verderame, HM | 1 |
Kalkman, HO; Soar, J | 1 |
Cherqui, C; Dabiré, H; Drouillat, M; Laubie, M; Schmitt, H | 1 |
Curzon, G; Haleem, DJ; Kennett, GA; Whitton, PS | 1 |
Ahlenius, S; Fernandez-Guasti, A; Larsson, K | 1 |
Fuller, RW; Perry, KW | 1 |
Jazayeri, A; Kent, TA; Meyer, WJ | 1 |
Dalpé, M; de Montigny, C; Lal, S; Martial, J; Olivier, A; Quirion, R | 1 |
Kellar, KJ; Stockmeier, CA | 1 |
Cornfield, LJ; Martin, AR; Nelson, DL; Taylor, EW | 1 |
Ahlenius, S; Larsson, K | 1 |
Kalkman, HO | 1 |
Fozard, JR; Kidd, EJ; Neill, J; Tricklebank, MD | 1 |
Brazell, C; Gilbert, F; Stahl, SM; Tricklebank, MD | 1 |
Murakami, H; Sano, M; Tsukimura, T; Yamazaki, A | 1 |
Baumann, PA; Bischoff, S; Neale, RF; Sills, MA; Waldmeier, PC; Williams, M | 1 |
Engel, G; Hoyer, D; Kalkman, HO | 1 |
Engel, G; Hoyer, D; Markstein, R | 1 |
Gudelsky, GA; Koenig, JI; Meltzer, HY | 2 |
Feuerstein, TJ; Hertting, G; Lupp, A | 1 |
Houston, DS; Vanhoutte, PM | 1 |
el-Yassir, N; Fleetwood-Walker, SM; Mitchell, R | 1 |
Oksenberg, D; Peroutka, SJ | 1 |
De Jonge, A; Doods, HN; Kalkman, HO; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Wilffert, B | 1 |
Cortés, R; Palacios, JM; Pazos, A | 1 |
Hirayama, T; Kikuchi, K; Morita, K; Ogawa, Y; Onodera, S; Takeda, A; Takenaka, T; Tobise, K | 1 |
Bianchetti, A; Croci, T; Landi, M; Manara, L | 1 |
Baudrie, V; Bluet-Pajot, MT; Broqua, P; Chaouloff, F; Laude, D; Schmidt, B | 1 |
Blanchard, DC; Blanchard, RJ; McEwen, BS; McKittrick, CR; Sakai, RR | 1 |
Bramwell, S; Hjorth, S; McQuade, R; Sharp, T | 1 |
Jantos, H; Monti, JM | 1 |
Bosker, FJ; Donker, MG; Klompmakers, AA; Kurata, K; Westenberg, HG | 1 |
Esposito, E; Pagannone, S; Prisco, S | 1 |
Andersson, G; Larsson, K | 1 |
Olivier, B; Slangen, JL; Ybema, CE | 1 |
Ahrens, O; Flügge, G; Fuchs, E | 1 |
Hjorth, S; Sharp, T | 1 |
Carli, M; Grondin, L; Nénonéné, EK; Radja, F; Reader, TA | 1 |
Frankfurt, M; McEwen, BS; McKittrick, CR; Mendelson, SD | 1 |
Ahlenius, S; Cortizo, L; Wadenberg, ML | 1 |
Clark, M; Post, RM; Weiss, SR | 1 |
Moore, NA; Perrett, L; Rees, G; Sanger, G | 1 |
Battaglia, G; Pinto, W | 1 |
Muck-Seler, D; Pericić, D | 1 |
Helke, CJ; Nickolaus, S; Thor, KB | 1 |
Bruinvels, AT; Hoyer, D; Palacios, JM | 1 |
Hill, RG; Kennedy, AT; Kitchen, I | 1 |
Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
Rabin, RA; Winter, JC | 1 |
Dean, RR; Edgar, DM; Heller, HC; Miller, JD; Prosser, RA | 1 |
Grignaschi, G; Mantelli, B; Samanin, R | 1 |
Crick, H; Manuel, NA; Wallis, DI | 1 |
Browning, RA; Dailey, JW; Jobe, PC; Statnick, MA | 1 |
Assie, MB; Koek, W | 1 |
Andrade, M; Caldarola-Pastuszka, M; Jackson, A; Uphouse, L | 1 |
Crews, FT; Janowsky, DS; Knapp, DJ; Overstreet, DH; Rezvani, AH | 1 |
Arnt, J; Moltzen, E; Sánchez, C | 1 |
Bourin, M; MacSweeney, CP; Redrobe, JP | 1 |
Herremans, AH; Mos, J; Olivier, B; Van Drimmelen, M; Van Hest, A | 1 |
Leander, JD; Wolff, MC | 1 |
Rosenberg, R; Smith, DF; Wegener, G | 1 |
Farde, L; Ginovart, N; Halldin, C; Ito, H; Lundkvist, C; McCarron, JA; Pike, VW | 1 |
Gur, E; Lerer, B; Newman, ME | 1 |
Baker, GB; Bourin, M; Colombel, MC; Redrobe, JP | 2 |
Cryan, JF; Leonard, BE; McGrath, C; Norman, TR | 1 |
De Leyn, P; Demedts, MG; Deneffe, G; Dupont, LJ; Pype, JL; Verleden, GM | 1 |
Barnes, NM; Stowe, RL | 1 |
Ahlenius, S; Hillegaart, V | 1 |
Bergeron, R; Blier, P; de Montigny, C; el Mansari, M; Piñeyro, G | 1 |
Braselton, J; Reynolds, L; Sprouse, J | 1 |
Carden, SE; Joyce, MP | 1 |
Dremencov, E; Gur, E; Lerer, B; Newman, ME | 1 |
Arnold, PB; Cardenas, CG; Cardenas, LM; Mar, LP; Scroggs, RS; Surmeier, DJ; Vysokanov, AV | 1 |
Moser, PC; Sanger, DJ | 1 |
Gobert, A; Millan, MJ | 1 |
Fornal, CA; Jacobs, BL; Martin, FJ; Metzler, CW | 1 |
Filipink, RA; Helsley, SE; Rabin, RA; Timineri, D; Winter, JC | 1 |
Misane, I; Ogren, SO | 1 |
Crews, T; Garcia-Rill, E; Miyazato, H; Skinner, RD; Williams, K | 1 |
Dawson, LA; Nguyen, HQ; Schechter, LE; Smith, DI | 1 |
Lejeune, F; Millan, MJ | 1 |
Ahlenius, S; Kaur, P | 1 |
Gibert-Rahola, J; Micó, JA; Ortega-Alvaro, A; Roca-Vinardell, A; Rojas-Corrales, OM | 1 |
Chaput, C; Millan, MJ; Newman-Tancredi, A; Touzard, M | 1 |
Cussac, D; Duqueyroix, D; Millan, MJ; Newman-Tancredi, A | 1 |
Ase, AR; Descarries, L; Hen, R; Reader, TA; Riad, M | 1 |
Kimura, I; Sugimoto, Y; Watanabe, Y; Yamada, J | 1 |
Yan, QS; Yan, SE | 1 |
Inoue, T; Itoh, S; Morimoto, T; Ogawa, S; Saito, M; Wakisaka, S | 1 |
Estrada-Camarena, E; López-Rubalcava, C; Martínez-Mota, L | 1 |
Chen, CF; Hung, WY; Liao, JF | 1 |
Kehr, J; Ogren, SO; Yamaguchi, M; Yoshitake, S; Yoshitake, T | 1 |
Chen, R; Hamilton, R; Jordan, S; Kikuchi, T; Koprivica, V; Tottori, K; Whitehead, RE | 1 |
Bourin, M; Chenu, F; David, DJ; Gardier, AM; Guiard, BP; Guilloux, JP; Repérant, C; Toth, M | 1 |
Marona-Lewicka, D; Nichols, DE | 1 |
Mallmann, ES; Paixão, L; Ribeiro, MF; Spritzer, PM | 1 |
Bregman, T; Diwan, M; Fletcher, PJ; Hamani, C; Nobrega, JN; Raymond, R; Scott, B; Volle, J | 1 |
2 review(s) available for pindolol and 8-hydroxy-2-(di-n-propylamino)tetralin
Article | Year |
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Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
Role of somatodendritic 5-HT autoreceptors in modulating 5-HT neurotransmission.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Dendrites; Feedback; Neurons; Pindolol; Pyrimidines; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission | 1998 |
130 other study(ies) available for pindolol and 8-hydroxy-2-(di-n-propylamino)tetralin
Article | Year |
---|---|
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes | 1996 |
Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Affinity Labels; Animals; Binding, Competitive; CHO Cells; Cricetinae; Guanine Nucleotides; Hippocampus; Humans; Male; Membranes; Piperazines; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists | 1998 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT(1A) activity. part 3.
Topics: Animals; Body Temperature; Mice; Models, Molecular; Protein Conformation; Pyrimidines; Rats; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Structure-Activity Relationship | 2011 |
Effects of 5-HT1A receptor agonists on the circadian rhythm of wheel-running activity in hamsters.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Circadian Rhythm; Cricetinae; Male; Melatonin; Mesocricetus; Motor Activity; Pindolol; Piperazines; Receptors, GABA-A; Receptors, Serotonin; Tetrahydronaphthalenes | 1992 |
Identification of a single amino acid residue responsible for the binding of a class of beta-adrenergic receptor antagonists to 5-hydroxytryptamine1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Amino Acid Sequence; Amino Acids; Binding, Competitive; Cell Line; Cross Reactions; Humans; Molecular Sequence Data; Pindolol; Receptors, Serotonin; Sequence Homology, Nucleic Acid; Tetrahydronaphthalenes | 1992 |
Pindolol antagonizes the effects on hippocampal rhythmical slow activity of clonidine, baclofen and 8-OH-DPAT, but not chlordiazepoxide and sodium amylobarbitone.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Amobarbital; Animals; Baclofen; Chlordiazepoxide; Clonidine; Electric Stimulation; Electrodes; Electroencephalography; Flumazenil; Hippocampus; Male; Pindolol; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes | 1992 |
Serotonin 5-HT1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Body Temperature; Colforsin; Drug Tolerance; Fenclonine; Hypothermia; Male; Mice; Pindolol; Piperazines; Quinolines; Receptors, Serotonin; Serotonin | 1992 |
Cardiovascular effects of the 5-HT1A receptor ligand, MDL 73005EF, in conscious spontaneously hypertensive rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Buspirone; Dioxins; Heart Rate; Hypertension; Male; Pindolol; Piperazines; Rats; Rats, Inbred SHR; Receptors, Serotonin; Serotonin Receptor Agonists; Spiro Compounds; Vasodilator Agents | 1992 |
Activation of 5-HT1A receptor subtype in the paraventricular nuclei of the hypothalamus induces CRH and ACTH release in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Animals; Buspirone; Corticotropin-Releasing Hormone; Male; Paraventricular Hypothalamic Nucleus; Pindolol; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists | 1992 |
Role of 5-hydroxytryptamine receptors on luteinizing-hormone-releasing hormone release in the ovariectomized, estradiol-treated rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Estradiol; Female; Gonadotropin-Releasing Hormone; Hypothalamus, Middle; Ketanserin; Ovariectomy; Pindolol; Preoptic Area; Quipazine; Radioimmunoassay; Rats; Receptors, Serotonin; Serotonin Antagonists; Suprachiasmatic Nucleus; Tetrahydronaphthalenes | 1992 |
Pharmacological characterisation of the 5-HT1A serotonin receptor using the agonist [3H]8-OH-DPAT, and the antagonist [3H]spiperone.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; CHO Cells; Cricetinae; Humans; Kinetics; Lisuride; Methiothepin; Pindolol; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Spiperone; Transfection; Tritium | 1992 |
Discriminative stimulus effects of 8-OH-DPAT in pigeons: antagonism studies with the putative 5-HT1A receptor antagonists BMY 7378 and NAN-190.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Indoles; Pindolol; Piperazines; Prazosin; Serotonin Antagonists | 1992 |
Autoradiographic localization of 5HT1 binding sites in the medulla oblongata of the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain; Iodine Radioisotopes; Iodocyanopindolol; Male; Medulla Oblongata; Organ Specificity; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Tritium | 1992 |
Autoradiographic localization of 5HT1 binding sites in autonomic areas of the rat dorsomedial medulla oblongata.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Iodine Radioisotopes; Iodocyanopindolol; Male; Medulla Oblongata; Organ Specificity; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Tritium; Vagotomy | 1992 |
Autoradiographic analyses of the effects of adrenalectomy and corticosterone on 5-HT1A and 5-HT1B receptors in the dorsal hippocampus and cortex of the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenalectomy; Animals; Autoradiography; Cerebral Cortex; Corticosterone; Hippocampus; Iodocyanopindolol; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1992 |
Pressor effects following microinjection of 5-HT1A receptor agonists into the raphe obscurus of the anaesthetized rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Electric Stimulation; Glutamates; Glutamic Acid; Heart Rate; Male; Methiothepin; Microinjections; Phrenic Nerve; Pindolol; Piperazines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1991 |
Interactions between substance P and serotonergic mechanisms at preganglionic sympathetic nerves in thoracic spinal cord.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Heart Rate; Injections, Spinal; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord; Substance P; Sympathetic Nervous System; Tetrahydronaphthalenes | 1990 |
cis-(+)-8-OH-1-CH3-DPAT, (+)ALK-3, a novel stereoselective pharmacological probe for characterizing 5-HT release-controlling 5-HT1A autoreceptors. An in vivo brain microdialysis study.
Topics: 3,4-Dihydroxyphenylacetic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Dialysis; Hippocampus; Hydroxyindoleacetic Acid; Male; Naphthalenes; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stereoisomerism; Tetrahydronaphthalenes | 1990 |
Involvement of 5-HT1A receptors in blood pressure reduction by 8-OH-DPAT and urapidil in cats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Cats; Dose-Response Relationship, Drug; Female; Heart Rate; Imidazoles; Male; Pindolol; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
Effects of local application of 5-HT and 8-OH-DPAT into the dorsal and median raphe nuclei on core temperature in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Injections, Intraventricular; Pindolol; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Autoradiographic mapping of 5-HT1, 5-HT1A, 5-HT1B and 5-HT2 receptors in the rat spinal cord.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Iodine Radioisotopes; Iodocyanopindolol; Ketanserin; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes; Tritium | 1991 |
Serotonergic mechanisms in the nucleus accumbens affected by chronic desipramine treatment.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Buspirone; Chromans; Desipramine; Dose-Response Relationship, Drug; Methysergide; Microinjections; Nucleus Accumbens; Pindolol; Quipazine; Rats; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Characterization of a novel serotonin receptor subtype (5-HT1S) in rat CNS: interaction with a GTP binding protein.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; GTP-Binding Proteins; Indoles; Male; Pindolol; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord; Tetrahydronaphthalenes; Tissue Distribution | 1991 |
5-HT receptor-mediated regulation of thyrotropin-releasing hormone release in rat spinal cord.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes; Thyrotropin-Releasing Hormone; Veratridine | 1991 |
Alterations in serotonin receptor subtypes in ethanol-dependent rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alcohol Withdrawal Delirium; Alcoholic Intoxication; Alcoholism; Animals; Brain; Ethanol; Ketanserin; Pindolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Effects of MDL 73005EF on central pre- and postsynaptic 5-HT1A receptor function in the rat in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Animals; Central Nervous System; Dialysis; Dioxins; Fenfluramine; Hippocampus; Male; Neurosecretory Systems; Pindolol; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiro Compounds; Synapses; Tetrahydronaphthalenes | 1990 |
Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Autoradiography; Cerebral Cortex; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Humans; Iodocyanopindolol; Ketanserin; Male; Middle Aged; Oxotremorine; Paroxetine; Pindolol; Piperidines; Pirenzepine; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1990 |
Cellular localization of serotonin 1A, 1B and uptake sites in cingulate cortex of the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cerebral Cortex; Immunotoxins; Iodocyanopindolol; Male; Paroxetine; Pindolol; Piperidines; Rats; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1990 |
8-OH-DPAT and buspirone analogs inhibit the ketanserin-sensitive quipazine-induced head shake response in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Head; Ketanserin; Male; Naphthalenes; Pindolol; Pyrimidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Stereotyped Behavior; Tetrahydronaphthalenes | 1990 |
The behavioural, but not the hypothermic or corticosterone, response to 8-hydroxy-2-(DI-n-propylamino)-tetralin, is antagonized by NAN-190 in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Body Temperature; Corticosterone; Male; Naphthalenes; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Reserpine; Serotonin Antagonists; Spiperone; Tetrahydronaphthalenes | 1990 |
Cardiovascular effects of 5-HT1A receptor agonists injected into the dorsal raphe nucleus of conscious rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antihypertensive Agents; Atropine Derivatives; Behavior, Animal; Catheterization; Hemodynamics; Injections; Injections, Intravenous; Male; Pindolol; Piperazines; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1990 |
Organization of serotonin 1A and 1B receptors in the nucleus of the solitary tract.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Chloroform; Iodocyanopindolol; Medulla Oblongata; Pindolol; Rats; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tissue Distribution | 1990 |
Determination of the 5-HT receptor subtype involved in 8-OH-DPAT-induced hyperlocomotion: potential difficulties arising from inadequate pharmacological tools.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Dioxanes; Haloperidol; Male; Motor Activity; Pindolol; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spiro Compounds; Tetrahydronaphthalenes | 1990 |
Ventrolateral medullary pressor area: site of hypotensive and sympatho-inhibitory effects of (+/-)8-OH-DPAT in anaesthetized dogs.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; alpha-Methyltyrosine; Anesthesia; Animals; Blood Pressure; Catecholamines; Cisterna Magna; Dogs; Female; Heart Rate; Male; Medulla Oblongata; Methiothepin; Methyltyrosines; Microinjections; Naphthalenes; Neurons; Pindolol; Pressoreceptors; Sympathetic Nervous System; Tetrahydronaphthalenes | 1989 |
8-OH-DPAT increases corticosterone but not other 5-HT1A receptor-dependent responses more in females.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Chloral Hydrate; Chlordiazepoxide; Corticosterone; Eating; Female; Hypothalamus, Middle; Injections; Male; Naphthalenes; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sex Factors; Stress, Psychological; Temperature; Tetrahydronaphthalenes | 1989 |
Evidence for the involvement of central 5-HT1A receptors in the mediation of lordosis behavior in the female rat.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Betaxolol; Estradiol; Female; Male; Methiothepin; Pindolol; Piperidines; Posture; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Sexual Behavior, Animal; Tetrahydronaphthalenes | 1989 |
Determination of brain concentrations of 8-hydroxy-2-(di-n-propylamino)tetralin by liquid chromatography with electrochemical detection.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Chromatography, Liquid; Male; Naphthalenes; Pindolol; Pyridines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1989 |
5-HT1B and 5-HT2 serotonin binding sites in cultured Wistar-Kyoto rat aortic smooth muscle cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Aorta, Thoracic; Cell Membrane; Cells, Cultured; Iodine Radioisotopes; Iodocyanopindolol; Kinetics; Muscle, Smooth, Vascular; Pindolol; Rats; Rats, Inbred WKY; Receptors, Serotonin; Tetrahydronaphthalenes | 1989 |
Apparent absence of serotonin1B receptors in biopsied and post-mortem human brain.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Biopsy; Brain; Female; Humans; Male; Pindolol; Postmortem Changes; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Tissue Preservation | 1989 |
Serotonin depletion unmasks serotonergic component of [3H]dihydroalprenolol binding in rat brain.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Animals; Brain; Dihydroalprenolol; Fenclonine; In Vitro Techniques; Iodocyanopindolol; Male; p-Chloroamphetamine; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1989 |
MDL 73005EF: partial agonist at the 5-HT1A receptor negatively linked to adenylate cyclase.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenosine Triphosphate; Adenylyl Cyclase Inhibitors; Animals; Buspirone; Colforsin; Cyclic AMP; Dioxins; Hippocampus; In Vitro Techniques; Male; Membranes; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiro Compounds; Tetrahydronaphthalenes; Tryptamines | 1989 |
Antagonism by pindolol, but not betaxolol, of 8-OH-DPAT-induced facilitation of male rat sexual behavior.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Betaxolol; Ejaculation; Female; Male; Naphthalenes; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Sexual Behavior, Animal; Tetrahydronaphthalenes | 1989 |
Beta-adrenoceptor blockade in rats enhances the ambulation induced by 5-HT1A receptor agonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Male; Motor Activity; Pindolol; Piperazines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1989 |
Mediation of the discriminative stimulus properties of 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT) by the putative 5-HT1A receptor.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alprenolol; Animals; Buspirone; Discrimination Learning; Dose-Response Relationship, Drug; Generalization, Psychological; Male; Naphthalenes; Pindolol; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1987 |
Activation of the 5-HT1A receptor subtype increases rat plasma ACTH concentration.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Buspirone; Male; Physostigmine; Pindolol; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1988 |
The relaxation induced by indole and nonindole 5-HT agonists in the molluscan smooth muscle.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bivalvia; Cyclic AMP; In Vitro Techniques; Indoles; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pindolol; Propranolol; Proteins; Serotonin; Spiperone; Tetrahydronaphthalenes | 1988 |
Interactions of isamoltane (CGP 361A), an anxiolytic phenoxypropanolamine derivative, with 5-HT1 receptor subtypes in the rat brain.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Brain; Cerebral Cortex; Corpus Striatum; Electric Stimulation; Hippocampus; In Vitro Techniques; Iodocyanopindolol; Male; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Reserpine; Serotonin; Stereoisomerism; Tetrahydronaphthalenes | 1988 |
Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and [3H]ketanserin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Choroid Plexus; Ergolines; In Vitro Techniques; Iodocyanopindolol; Ketanserin; Male; Membranes; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tetrahydronaphthalenes | 1985 |
5-HT1A-receptors mediate stimulation of adenylate cyclase in rat hippocampus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Cerebral Cortex; Enzyme Activation; Hippocampus; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Male; Pindolol; Rats; Receptors, Serotonin; Tetrahydronaphthalenes | 1986 |
Thermoregulatory responses to serotonin (5-HT) receptor stimulation in the rat. Evidence for opposing roles of 5-HT2 and 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature Regulation; Ketanserin; Male; Methoxydimethyltryptamines; Pindolol; Piperidines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes | 1986 |
Stimulation of corticosterone and beta-endorphin secretion in the rat by selective 5-HT receptor subtype activation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; beta-Endorphin; Corticosterone; Endorphins; Ketanserin; Male; Pindolol; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Tetrahydronaphthalenes | 1987 |
The serotonin (5-HT) autoreceptor in the hippocampus of the rabbit: role of 5-HT biophase concentration.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Hippocampus; Mathematics; Metergoline; Methiothepin; Methoxydimethyltryptamines; Methysergide; Phentolamine; Pindolol; Quipazine; Rabbits; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1987 |
Comparison of serotonergic receptor subtypes on the smooth muscle and endothelium of the canine coronary artery.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Ketanserin; Male; Metergoline; Methiothepin; Muscle, Smooth, Vascular; Pindolol; Receptors, Serotonin; Tetrahydronaphthalenes; Vasodilation | 1988 |
Heterogeneous effects of serotonin in the dorsal horn of rat: the involvement of 5-HT1 receptor subtypes.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Indoles; Ketanserin; Male; Neurons, Afferent; Pain; Physical Stimulation; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Spinal Cord; Tetrahydronaphthalenes | 1988 |
Antagonism of 5-hydroxytryptamine1A (5-HT1A) receptor-mediated modulation of adenylate cyclase activity by pindolol and propranolol isomers.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Colforsin; GTP-Binding Proteins; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Pindolol; Propranolol; Rats; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism; Tetrahydronaphthalenes | 1988 |
Differential selectivities of RU 24969 and 8-OH-DPAT for the purported 5-HT1A and 5-HT1B binding sites. Correlation between 5-HT1A affinity and hypotensive activity.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Binding Sites; Blood Pressure; In Vitro Techniques; Indoles; Male; Naphthalenes; Pentobarbital; Pindolol; Rats; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes | 1985 |
Quantitative receptor autoradiography: application to the characterization of multiple receptor subtypes.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Autoradiography; Benzodiazepinones; Binding, Competitive; Brain; Carbachol; Hippocampus; Indoles; Oxotremorine; Pindolol; Pirenzepine; Rats; Receptors, Muscarinic; Receptors, Serotonin; Superior Colliculi; Tetrahydronaphthalenes | 1984 |
Comparison of 5-hydroxytryptamine-induced contraction of rat pulmonary artery to that of aorta in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Ketanserin; Male; Pindolol; Pulmonary Artery; Quinazolines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Ritanserin; Serotonin; Vasoconstriction | 1995 |
Drug-induced defaecation in rats: role of central 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Buspirone; Colon; Defecation; Feces; Fenclonine; Male; Naphthalenes; Pindolol; Pyridines; Rats; Receptors, Serotonin; Serotonin Receptor Agonists; Time Factors | 1995 |
Are 5-HT1A autoreceptors involved in the inhibitory effect of ipsapirone on cold-elicited thyrotropin secretion?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Glucose; Cold Temperature; Corticosterone; Fenclonine; Hydroxyindoleacetic Acid; Hypothalamus; Male; Metergoline; Pindolol; Proadifen; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Thyrotropin | 1993 |
Serotonin receptor binding in a colony model of chronic social stress.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Arousal; Autoradiography; Brain; Corticosterone; Dominance-Subordination; Female; Iodocyanopindolol; Ketanserin; Male; Pindolol; Rats; Receptors, Serotonin; Social Environment; Stress, Psychological | 1995 |
Effect of acute and repeated administration of 5-HT1A receptor agonists on 5-HT release in rat brain in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Brain Chemistry; Buspirone; Dose-Response Relationship, Drug; Electrodes, Implanted; Electrophysiology; Hippocampus; Male; Microdialysis; Pindolol; Pyrimidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists | 1993 |
Stereoselective antagonism by the pindolol enantiomers of 8-OH-DPAT-induced changes of sleep and wakefulness.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Betaxolol; Electroencephalography; Electromyography; Male; Pindolol; Rats; Rats, Wistar; Sleep; Sleep, REM; Stereoisomerism; Wakefulness | 1994 |
5-Hydroxytryptamine release in dorsal hippocampus of freely moving rats: modulation by pindolol.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Hippocampus; Male; Pindolol; Potassium; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Tetrodotoxin; Time Factors | 1994 |
Serotonin-dopamine interaction in the rat ventral tegmental area: an electrophysiological study in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Ergolines; Male; Motor Activity; Pindolol; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Ventral Tegmental Area | 1994 |
Effects of FG 5893, a new compound with 5-HT1A receptor agonistic and 5-HT2 receptor antagonistic properties, on male rat sexual behavior.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ejaculation; Female; Male; Nicotinic Acids; Pindolol; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal | 1994 |
Discriminative stimulus effect of flesinoxan: effect of 5-HT1A antagonists and PCPA.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Discrimination Learning; Fenclonine; Male; Pindolol; Piperazines; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 1994 |
Monoamine receptors in the amygdaloid complex of the tree shrew (Tupaia belangeri).
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amygdala; Animals; Autoradiography; Iodocyanopindolol; Pindolol; Prazosin; Receptors, Biogenic Amine; Tupaiidae; Yohimbine | 1994 |
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism | 1993 |
Heterogeneity of cortical and hippocampal 5-HT1A receptors: a reappraisal of homogenate binding with 8-[3H]hydroxydipropylaminotetralin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Biogenic Amines; Buspirone; Cell Membrane; Cerebral Cortex; Fenclonine; Guanylyl Imidodiphosphate; Hippocampus; Kinetics; Male; Organ Specificity; p-Chloroamphetamine; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1994 |
Effect of 5,7-dihydroxytryptamine, ovariectomy and gonadal steroids on serotonin receptor binding in rat brain.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain Chemistry; Carrier Proteins; Estrogens; Female; Gonadal Steroid Hormones; Hippocampus; Iodocyanopindolol; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Orchiectomy; Ovariectomy; Paroxetine; Pindolol; Progesterone; Rats; Receptors, Serotonin; Serotonin Plasma Membrane Transport Proteins; Ventromedial Hypothalamic Nucleus | 1994 |
Evidence for specific interactions between 5-HT1A and dopamine D2 receptor mechanisms in the mediation of extrapyramidal motor functions in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Betaxolol; Catalepsy; Dopamine D2 Receptor Antagonists; Extrapyramidal Tracts; Male; Pindolol; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Serotonin; Salicylamides; Serotonin Antagonists | 1994 |
Autoradiographic analysis of serotonin receptors and transporter in kindled rat brain.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amygdala; Animals; Autoradiography; Cerebral Cortex; Hippocampus; Iodine Radioisotopes; Iodocyanopindolol; Kindling, Neurologic; Male; Paroxetine; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Receptors, Serotonin; Seizures; Tritium | 1993 |
5-HT1A-mediated lower lip retraction: effects of 5-HT1A agonists and antagonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Lip; Male; Pindolol; Piperazines; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1993 |
In vivo EEDQ dose-dependently inactivates rat brain 5-HT receptors but not 5-HT uptake sites.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Brain; Carrier Proteins; Cerebral Cortex; Dose-Response Relationship, Drug; Iodocyanopindolol; Ketanserin; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Paroxetine; Pindolol; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins | 1993 |
Possible antidepressant dihydroergosine preferentially binds to 5-HT1B receptor sites in the rat hippocampus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Binding, Competitive; Chlorpromazine; Ergotamines; Hippocampus; In Vitro Techniques; Male; Pindolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Serotonin | 1993 |
Autoradiographic localization of 5-hydroxytryptamine1A, 5-hydroxytryptamine1B and 5-hydroxytryptamine1C/2 binding sites in the rat spinal cord.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Iodocyanopindolol; Male; Motor Neurons; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Spinal Cord | 1993 |
Autoradiographic characterisation and localisation of 5-HT1D compared to 5-HT1B binding sites in rat brain.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Binding, Competitive; Brain; Cloning, Molecular; Dipeptides; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Pindolol; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin | 1993 |
Assessment of 8-OH-DPAT induced spontaneous tailflicks as an in vivo model of 5-HT1A function in young rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Animals, Newborn; Behavior, Animal; Dose-Response Relationship, Drug; Male; Pindolol; Propranolol; Rats; Rats, Wistar; Restraint, Physical; Serotonin; Tail | 1993 |
Activity of serotonin (5-HT) receptor agonists, partial agonists and antagonists at cloned human 5-HT1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HeLa cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Colforsin; Cyclic AMP; HeLa Cells; Humans; Indoles; Lysergic Acid Diethylamide; Models, Biological; Pindolol; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Transfection | 1993 |
Antagonism of the stimulus effects of yohimbine and 8-hydroxydipropylaminotetralin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Animals; Cerebral Cortex; Discrimination, Psychological; Hippocampus; Male; Pindolol; Piperazines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Adrenergic, alpha; Serotonin; Serotonin Antagonists; Yohimbine | 1993 |
Serotonin and the mammalian circadian system: I. In vitro phase shifts by serotonergic agonists and antagonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Circadian Rhythm; Dose-Response Relationship, Drug; Electrophysiology; In Vitro Techniques; Iodocyanopindolol; Lysergic Acid Diethylamide; Male; Metergoline; Neurons; Pindolol; Quipazine; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus | 1993 |
The hypophagic effect of restraint stress in rats can be mediated by 5-HT2 receptors in the paraventricular nucleus of the hypothalamus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amidines; Animals; Anorexia; Anorexia Nervosa; Disease Models, Animal; Feeding Behavior; Ketanserin; Male; Paraventricular Hypothalamic Nucleus; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Restraint, Physical; Ritanserin; Stress, Physiological | 1993 |
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan | 1995 |
Abnormalities in 5-HT1A and 5-HT1B receptor binding in severe-seizure genetically epilepsy-prone rats (GEPR-9s).
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Epilepsy; Male; Pindolol; Rats; Receptors, Serotonin; Serotonin Antagonists | 1996 |
(-)-pindolol and (+/-)-tertatolol affect rat hippocampal 5-HT levels through mechanisms involving not only 5-HT1A, but also 5-HT1B receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Betaxolol; Hippocampus; Male; Microdialysis; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Serotonin; Thiophenes | 1996 |
5-HT1A receptor antagonists and lordosis behavior.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Female; Hypothalamus, Middle; Infusions, Parenteral; Ovariectomy; Ovary; Pindolol; Piperazines; Posture; Propranolol; Rats; Rats, Inbred Strains; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal | 1996 |
Further selection of rat lines differing in 5-HT-1A receptor sensitivity: behavioral and functional correlates.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Crosses, Genetic; Ethanol; Female; Food Preferences; Male; Maze Learning; Motor Activity; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Saccharin; Selection, Genetic; Serotonin Antagonists; Serotonin Receptor Agonists; Taste | 1996 |
Assessment of relative efficacies of 5-HT1A receptor ligands by means of in vivo animal models.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Male; Models, Neurological; Pindolol; Rats; Rats, Wistar; Receptors, Serotonin; Vocalization, Animal | 1996 |
The role of 5-HT1A and 5-HT1B receptors in antidepressant drug actions in the mouse forced swimming test.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Immobilization; Indoles; Male; Mice; Pindolol; Receptors, Serotonin; Swimming | 1996 |
The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Columbidae; Discrimination Learning; Fluvoxamine; Indoles; Pindolol; Piperazines; Pyridines; Pyrimidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles | 1997 |
Differentiation of 5-HT1A receptor ligands by drug discrimination.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aminopyridines; Animals; Behavior, Animal; Buspirone; Columbidae; Cyclohexylamines; Discrimination Learning; Dose-Response Relationship, Drug; Idazoxan; Ligands; Male; Pindolol; Piperazines; Pyridines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 1997 |
5-HT1A receptors in lithium-induced conditioned taste aversion.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Feeding Behavior; Lithium; Male; Pindolol; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Saccharin; Taste | 1997 |
PET-characterization of [carbonyl-11C]WAY-100635 binding to 5-HT1A receptors in the primate brain.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Buspirone; Carbon Radioisotopes; Cerebellum; Macaca fascicularis; Male; Neocortex; Pindolol; Piperazines; Pyridines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Tomography, Emission-Computed | 1997 |
Chronic electroconvulsive shock and 5-HT autoreceptor activity in rat brain: an in vivo microdialysis study.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Electroshock; Frontal Lobe; Hippocampus; Male; Microdialysis; Pindolol; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1997 |
Dose-dependent noradrenergic and serotonergic properties of venlafaxine in animal models indicative of antidepressant activity.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Second-Generation; Cyclohexanols; Male; Mice; Motor Activity; Pindolol; Piperazines; Selective Serotonin Reuptake Inhibitors; Venlafaxine Hydrochloride | 1998 |
Combining pindolol and paroxetine in an animal model of chronic antidepressant action--can early onset of action be detected?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Antidepressive Agents; Depression; Disease Models, Animal; Drug Therapy, Combination; Exploratory Behavior; Hypothermia; Male; Olfactory Bulb; Paroxetine; Pindolol; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists | 1998 |
The effects of 8-hydroxy-2-(di-n-propylamino)tetralin on the cholinergic contraction in guinea pig and human airways in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Bronchi; Bronchoconstriction; Capsaicin; Cholinergic Fibers; Culture Techniques; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Humans; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pindolol; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Trachea; Tropisetron | 1998 |
Selective labelling of 5-HT7 receptor recognition sites in rat brain using [3H]5-carboxamidotryptamine.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Brain; Clozapine; Indoles; Kinetics; Male; Pindolol; Piperazines; Pyridines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Recombinant Proteins; Serotonin; Sulfonamides; Tritium | 1998 |
Facilitation and inhibition of male rat ejaculatory behaviour by the respective 5-HT1A and 5-HT1B receptor agonists 8-OH-DPAT and anpirtoline, as evidenced by use of the corresponding new and selective receptor antagonists NAD-299 and NAS-181.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Benzopyrans; Ejaculation; Female; Male; Morpholines; Pindolol; Piperidines; Propanolamines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal; Time Factors | 1998 |
5-HT1A agonist activity of pindolol: reversal of the inhibitory effects on cell firing in the dorsal raphe nucleus but not in the hippocampus by WAY-100,635.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Hippocampus; Neurons; Pindolol; Piperazines; Pyramidal Cells; Pyridines; Raphe Nuclei; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 1998 |
Psychopharmacological profile of the selective serotonin reuptake inhibitor, paroxetine: implication of noradrenergic and serotonergic mechanisms.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amines; Animals; Antidepressive Agents; Apomorphine; Brain; Clonidine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Hypothermia; Indoles; Male; Mice; Motor Activity; Norepinephrine; Paroxetine; Pindolol; Piperazines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming | 1998 |
The effects of 8-OH-DPAT and (+/-)-pindolol on isolation-induced ultrasonic vocalizations in 3-, 10-, and 14-day-old rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Body Temperature; Dose-Response Relationship, Drug; Female; Male; Pindolol; Rats; Rats, Wistar; Sensitivity and Specificity; Serotonin Antagonists; Serotonin Receptor Agonists; Social Isolation; Statistics, Nonparametric; Ultrasonics; Vocalization, Animal | 1999 |
Venlafaxine: acute and chronic effects on 5-hydroxytryptamine levels in rat brain in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Brain; Cyclohexanols; Dose-Response Relationship, Drug; Hippocampus; Injections, Intraperitoneal; Male; Pindolol; Prefrontal Cortex; Rats; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Venlafaxine Hydrochloride | 1999 |
Serotonergic modulation of hyperpolarization-activated current in acutely isolated rat dorsal root ganglion neurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Cell Size; Cyclic Nucleotide-Gated Cation Channels; Dopamine Antagonists; Ganglia, Spinal; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Neurons, Afferent; Patch-Clamp Techniques; Pindolol; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1999 |
5-HT1A receptor antagonists neither potentiate nor inhibit the effects of fluoxetine and befloxatone in the forced swim test in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antidepressive Agents; Antidepressive Agents, Second-Generation; Drug Interactions; Fluoxetine; Male; Monoamine Oxidase Inhibitors; Oxazoles; Pindolol; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Swimming | 1999 |
Modulation of dialysate levels of dopamine, noradrenaline, and serotonin (5-HT) in the frontal cortex of freely-moving rats by (-)-pindolol alone and in association with 5-HT reuptake inhibitors: comparative roles of beta-adrenergic, 5-HT1A, and 5-HT1B re
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Betaxolol; Dopamine; Fluoxetine; Frontal Lobe; Guinea Pigs; Humans; Male; Microdialysis; Norepinephrine; Pindolol; Piperazines; Propanolamines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, beta; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Pindolol suppresses serotonergic neuronal activity and does not block the inhibition of serotonergic neurons produced by 8-hydroxy-2-(di-n-propylamino)tetralin in awake cats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Cats; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Neurons; Pindolol; Propanolamines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes | 1999 |
The paradox of 5-methoxy-N,N-dimethyltryptamine: an indoleamine hallucinogen that induces stimulus control via 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Male; Methoxydimethyltryptamines; Pindolol; Piperazines; Pyridines; Rats; Rats, Inbred F344; Receptors, Serotonin; Receptors, Serotonin, 5-HT1 | 2000 |
Multiple 5-HT receptors in passive avoidance: comparative studies of p-chloroamphetamine and 8-OH-DPAT.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Avoidance Learning; Carrier Proteins; Male; Membrane Glycoproteins; Membrane Transport Proteins; Memory, Short-Term; Nerve Tissue Proteins; p-Chloroamphetamine; Pindolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists | 2000 |
Serotonergic modulation of the P13 midlatency auditory evoked potential in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cyclohexane Monoterpenes; Evoked Potentials, Auditory, Brain Stem; Male; Mesencephalon; Microinjections; Pindolol; Pons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Effects of chronic fluoxetine treatment in the presence and absence of (+/-)pindolol: a microdialysis study.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Fluoxetine; Frontal Lobe; Male; Microdialysis; Pindolol; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2000 |
Pindolol excites dopaminergic and adrenergic neurons, and inhibits serotonergic neurons, by activation of 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Dopamine; Dose-Response Relationship, Drug; Epinephrine; Locus Coeruleus; Male; Neurons; Pindolol; Piperazines; Pyridines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Ventral Tegmental Area | 2000 |
Non-serotonergic potentiation by (-)-pindolol of DOI-induced forward locomotion in rats: possible involvement of beta-adrenoceptors?.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Animals; Betaxolol; Biogenic Monoamines; Dihydroxyphenylalanine; Drug Synergism; Indophenol; Male; Motor Activity; Pindolol; Piperazines; Piperidines; Propanolamines; Prosencephalon; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, beta; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reserpine; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Pindolol, a beta-adrenoceptor blocker/5-hydroxytryptamine(1A/1B) antagonist, enhances the analgesic effect of tramadol.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analgesics, Opioid; Animals; Drug Synergism; Hot Temperature; Male; Pain Measurement; Pindolol; Rats; Rats, Wistar; Reaction Time; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Tramadol | 2000 |
Pindolol antagonises G-protein activation at both pre- and postsynaptic serotonin 5-HT1A receptors: a.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Binding Sites; Brain; Drug Interactions; GTP-Binding Proteins; Pindolol; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2001 |
Agonist properties of pindolol at h5-HT1A receptors coupled to mitogen-activated protein kinase.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Pindolol; Piperazines; Pyridines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 2001 |
Regional changes in density of serotonin transporter in the brain of 5-HT1A and 5-HT1B knockout mice, and of serotonin innervation in the 5-HT1B knockout.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Behavior, Animal; Brain; Carrier Proteins; Citalopram; Female; Immunohistochemistry; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons; Pindolol; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists | 2001 |
The 5-HT1A receptor agonist 8-hydroxy-2-di-n-(propylamino)tetralin (8-OH-DPAT) induces hyperglucagonemia in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenal Medulla; Adrenalectomy; Adrenergic beta-Antagonists; Animals; Blood Glucose; Dose-Response Relationship, Drug; Glucagon; Male; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists | 2001 |
Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Oxadiazoles; Pindolol; Piperazines; Potassium; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Ventral Tegmental Area | 2001 |
Involvement of 5-HT7 receptors in serotonergic effects on spike afterpotentials in presumed jaw-closing motoneurons of rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Alkaloids; Animals; Benzophenanthridines; Brain Stem; Calcium; Clozapine; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Enzyme Inhibitors; Isoquinolines; Jaw; Membrane Potentials; Motor Neurons; Phenanthridines; Pindolol; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides | 2002 |
Indorenate produces antidepressant-like actions in the rat forced swimming test via 5-HT1A receptors.
Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antidepressive Agents; Behavior, Animal; Benzamides; Buspirone; Dose-Response Relationship, Drug; Drug Interactions; Ketanserin; Male; Motor Activity; Pindolol; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming | 2002 |
Anxiolytic-like effects of baicalein and baicalin in the Vogel conflict test in mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conflict, Psychological; Dose-Response Relationship, Drug; Drinking; Drinking Behavior; Flavanones; Flavonoids; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred ICR; Pindolol; Psychological Tests; Serotonin Antagonists; Serotonin Receptor Agonists | 2003 |
Activation of 5-HT(1A) autoreceptors enhances the inhibitory effect of galanin on hippocampal 5-HT release in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Galanin; Hippocampus; Male; Microdialysis; Pindolol; Piperazines; Pyridines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2003 |
In vitro profile of the antidepressant candidate OPC-14523 at rat and human 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Autoradiography; Binding, Competitive; Buspirone; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Frontal Lobe; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Humans; Male; Middle Aged; Pindolol; Piperazines; Pyridines; Quinolones; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfur Radioisotopes | 2005 |
Blockade of 5-HT1A receptors by (+/-)-pindolol potentiates cortical 5-HT outflow, but not antidepressant-like activity of paroxetine: microdialysis and behavioral approaches in 5-HT1A receptor knockout mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Area Under Curve; Behavior, Animal; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Interactions; Immobility Response, Tonic; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Paroxetine; Pindolol; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming | 2006 |
WAY 100635 produces discriminative stimulus effects in rats mediated by dopamine D(4) receptor activation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Benzimidazoles; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Drug Therapy, Combination; Pindolol; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D4; Reinforcement Schedule; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Sulfonamides; Tryptamines | 2009 |
Serotonergic 5-HT2A/2C receptors are involved in prolactin secretion in hyperestrogenic rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Estradiol; Estrogens; Female; Pindolol; Prolactin; Pyrazines; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Serotonin Receptor Agonists | 2014 |
Deep brain stimulation and fluoxetine exert different long-term changes in the serotonergic system.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Deep Brain Stimulation; Fluoxetine; Hippocampus; Iodine Radioisotopes; Pindolol; Prefrontal Cortex; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Plasma Membrane Transport Proteins; Time Factors; Tritium | 2018 |