Page last updated: 2024-08-16

pinacidil and aprikalim

pinacidil has been researched along with aprikalim in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19904 (20.00)18.7374
1990's15 (75.00)18.2507
2000's0 (0.00)29.6817
2010's1 (5.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berry, JL; Foster, RW; Small, RC1
Hood, JS; Kadowitz, PJ; McMahon, TJ1
Downing, SJ; Hollingsworth, M; Minshall, E; Piper, I; Sadraei, H1
Dunne, MJ1
Neumcke, B; Weik, R1
Cavero, I; Courteix, J; Escande, D; Laville, M; Le Guern, S; Thuringer, D1
Hollingsworth, M; Piper, I1
Eltze, M1
Grafe, P; Lehmann-Horn, F; Quasthoff, S; Spuler, A1
Advenier, C; Dumas, JP; Dumas, M; Giudicelli, JF; Sgro, C1
Atwal, KS1
Grover, GJ2
Cavero, I; Premmereur, J1
Advenier, C; Dumas, JP; Dumas, M; Giudicelli, JF1
Allen, CT; Damiano, RJ; Hsia, PW; Lawton, JS; Sepic, JD1
Guo, ZG; Shi, DH1
Kwan, YW; Lau, WM; To, KW; Tsang, SH1
Chambers, DJ; Hearse, DJ1
Breschi, MC; Calderone, V; Cecchetti, V; Martelli, A; Sabatini, S; Testai, L1

Reviews

4 review(s) available for pinacidil and aprikalim

ArticleYear
Pharmacology and structure-activity relationships for KATP modulators: tissue-selective KATP openers.
    Journal of cardiovascular pharmacology, 1994, Volume: 24 Suppl 4

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Antihypertensive Agents; Benzopyrans; Cardiovascular Diseases; Cromakalim; Diazoxide; Guanidines; Guinea Pigs; Minoxidil; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Radioligand Assay; Rats; Structure-Activity Relationship; Vasodilator Agents

1994
Protective effects of ATP-sensitive potassium-channel openers in experimental myocardial ischemia.
    Journal of cardiovascular pharmacology, 1994, Volume: 24 Suppl 4

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Dihydropyridines; Disease Models, Animal; Dogs; Guanidines; Guinea Pigs; Myocardial Contraction; Myocardial Infarction; Myocardial Ischemia; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Rats; Vasodilator Agents

1994
Pharmacology of ATP-sensitive potassium channel (KATP) openers in models of myocardial ischemia and reperfusion.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:4

    Topics: Animals; ATP-Binding Cassette Transporters; Benzopyrans; Cromakalim; Guanidines; Humans; Ischemic Preconditioning, Myocardial; KATP Channels; Mitochondria, Heart; Models, Cardiovascular; Myocardial Ischemia; Myocardial Reperfusion; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyrans; Pyrroles; Rats

1997
Developments in cardioprotection: "polarized" arrest as an alternative to "depolarized" arrest.
    The Annals of thoracic surgery, 1999, Volume: 68, Issue:5

    Topics: Adenosine; Animals; Cardioplegic Solutions; Electrocardiography; Heart Arrest, Induced; Humans; Myocardial Reperfusion Injury; Organ Preservation; Picolines; Pinacidil; Potassium Channels; Pyrans; Sodium Channel Blockers; Vasodilator Agents

1999

Other Studies

16 other study(ies) available for pinacidil and aprikalim

ArticleYear
Tracheal relaxation induced by potassium channel opening drugs: its antagonism by adrenergic neurone blocking agents.
    British journal of pharmacology, 1992, Volume: 106, Issue:4

    Topics: Adrenergic Antagonists; Animals; Benzopyrans; Cromakalim; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Parasympatholytics; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Rubidium Radioisotopes; Stereoisomerism; Theophylline; Trachea

1992
Pulmonary vasodilator responses to RP 52891 are mediated by activation of a glibenclamide-sensitive K+ATP channel.
    European journal of pharmacology, 1991, Sep-04, Volume: 202, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Adenosine Triphosphate; Animals; Benzopyrans; Blood Gas Analysis; Blood Pressure; Cats; Cromakalim; Female; Glyburide; Guanidines; Hydrogen-Ion Concentration; Isoproterenol; Male; Nitroprusside; Picolines; Pinacidil; Potassium Channels; Prostaglandin Endoperoxides, Synthetic; Pulmonary Circulation; Pyrans; Pyrroles; Vasodilation; Vasodilator Agents

1991
Effects of several potassium channel openers and glibenclamide on the uterus of the rat.
    British journal of pharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Benzopyrans; Blood Pressure; Cromakalim; Female; Glyburide; Guanidines; Heart Rate; Hemodynamics; In Vitro Techniques; Oxytocin; Parasympatholytics; Picolines; Pinacidil; Potassium Channels; Potassium Chloride; Pregnancy; Pyrans; Pyrroles; Rats; Rats, Inbred Strains; Uterus; Vasodilator Agents

1990
Effects of pinacidil, RP 49356 and nicorandil on ATP-sensitive potassium channels in insulin-secreting cells.
    British journal of pharmacology, 1990, Volume: 99, Issue:3

    Topics: Adenoma, Islet Cell; Adenosine Triphosphate; Diazoxide; Glucose; Guanidines; Humans; Insulin; Insulinoma; Islets of Langerhans; Membrane Potentials; Niacinamide; Nicorandil; Pancreatic Neoplasms; Picolines; Pinacidil; Potassium Channels; Pyrans; Rubidium Radioisotopes; Tumor Cells, Cultured

1990
Effects of potassium channel openers on single potassium channels in mouse skeletal muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:3

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Calcium; Cromakalim; Female; Guanidines; In Vitro Techniques; Membrane Potentials; Mice; Muscles; Organ Specificity; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles

1990
Potassium channel openers act through an activation of ATP-sensitive K+ channels in guinea-pig cardiac myocytes.
    Pflugers Archiv : European journal of physiology, 1989, Volume: 414, Issue:6

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Electrophysiology; Glyburide; Guanidines; Guinea Pigs; Heart; In Vitro Techniques; Ion Channel Gating; Muscle, Smooth, Vascular; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Subtraction Technique

1989
Cromakalim, RP49356, pinacidil and minoxidil sulphate in the rat uterus and their antagonism by glibenclamide. Smooth Muscle Research Group.
    British journal of pharmacology, 1989, Volume: 98 Suppl

    Topics: Animals; Benzopyrans; Cromakalim; Female; Glyburide; Guanidines; In Vitro Techniques; Minoxidil; Parasympatholytics; Picolines; Pinacidil; Pyrans; Pyrroles; Rats; Rats, Inbred Strains; Uterine Contraction

1989
Glibenclamide is a competitive antagonist of cromakalim, pinacidil and RP 49356 in guinea-pig pulmonary artery.
    European journal of pharmacology, 1989, Jun-20, Volume: 165, Issue:2-3

    Topics: Animals; Benzopyrans; Cromakalim; Glyburide; Guanidines; Guinea Pigs; In Vitro Techniques; Male; Methylene Blue; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Potassium Chloride; Pulmonary Artery; Purinones; Pyrans; Pyrroles; Tetraethylammonium Compounds

1989
Cromakalim, pinacidil and RP 49356 activate a tolbutamide-sensitive K+ conductance in human skeletal muscle fibres.
    Pflugers Archiv : European journal of physiology, 1989, Volume: 414 Suppl 1

    Topics: Benzopyrans; Cromakalim; Guanidines; Humans; In Vitro Techniques; Membrane Potentials; Muscles; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Tolbutamide; Vasodilator Agents

1989
Effects of two K+ channel openers, aprikalim and pinacidil, on hypoxic pulmonary vasoconstriction.
    European journal of pharmacology, 1994, Sep-22, Volume: 263, Issue:1-2

    Topics: Animals; Antihypertensive Agents; Arginine; Guanidines; Hypoxia; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Picolines; Pinacidil; Potassium Channels; Pyrans; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasodilator Agents

1994
ATP sensitive potassium channel openers are of potential benefit in ischaemic heart disease.
    Cardiovascular research, 1994, Volume: 28, Issue:1

    Topics: Benzopyrans; Cromakalim; Dihydropyridines; Guanidines; Humans; Myocardial Ischemia; Myocardium; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Sodium-Potassium-Exchanging ATPase; Vasodilator Agents

1994
Effects of three K+ channel openers on airways and pulmonary circulation in the isolated guinea-pig lung.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Animals; Benzopyrans; Bronchoconstriction; Cromakalim; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; In Vitro Techniques; Lung; Male; Muscle Contraction; Muscle, Smooth, Vascular; Picolines; Pinacidil; Potassium; Potassium Channels; Pulmonary Circulation; Pyrans; Pyrroles

1993
Myocardial protection with potassium-channel openers is as effective as St. Thomas' solution in the rabbit heart.
    The Annals of thoracic surgery, 1996, Volume: 62, Issue:1

    Topics: Adenosine Triphosphate; Animals; Bicarbonates; Calcium Chloride; Cardioplegic Solutions; Coronary Circulation; Female; Guanidines; Heart Arrest, Induced; Magnesium; Male; Myocardial Contraction; Myocardial Reperfusion; Myocardial Reperfusion Injury; Picolines; Pinacidil; Potassium Channels; Potassium Chloride; Pyrans; Rabbits; Sodium Chloride; Stereoisomerism; Time Factors; Ventricular Fibrillation

1996
Inhibitory effect of potassium channel openers on proliferation of cultured rabbit aortic smooth muscle cells.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1996, Volume: 17, Issue:6

    Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Cell Division; Cells, Cultured; Cromakalim; Muscle, Smooth, Vascular; Nicorandil; Picolines; Pinacidil; Potassium Channels; Pyrans; Rabbits

1996
Comparison of the vascular relaxant effects of ATP-dependent K+ channel openers on aorta and pulmonary artery isolated from spontaneously hypertensive and Wistar-Kyoto rats.
    European journal of pharmacology, 1999, Jan-22, Volume: 365, Issue:2-3

    Topics: Adenosine Triphosphate; Aminoquinolines; Animals; Aorta, Thoracic; Apamin; Benzopyrans; Charybdotoxin; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Hypertension; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nicorandil; Nitroprusside; Norepinephrine; Picolines; Pinacidil; Potassium; Potassium Channels; Pulmonary Artery; Pyrans; Pyrrolidinones; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Vasodilator Agents

1999
Effects of K openers on the QT prolongation induced by HERG-blocking drugs in guinea-pigs.
    The Journal of pharmacy and pharmacology, 2010, Volume: 62, Issue:7

    Topics: Animals; Benzothiadiazines; Cromakalim; Decanoic Acids; Ether-A-Go-Go Potassium Channels; Glyburide; Guinea Pigs; Heart; Humans; Hydroxy Acids; Intracellular Membranes; KATP Channels; Long QT Syndrome; Male; Membrane Transport Modulators; Mitochondrial Membranes; Picolines; Pinacidil; Potassium Channel Blockers; Pyrans; Sarcolemma; Tolbutamide

2010