Page last updated: 2024-08-16

pinacidil and 4-aminopyridine

pinacidil has been researched along with 4-aminopyridine in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19902 (9.52)18.7374
1990's8 (38.10)18.2507
2000's9 (42.86)29.6817
2010's2 (9.52)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Kamijo, T; Kido, H; Miwa, A; Nakamura, F; Sugimoto, T; Tomaru, T; Uchida, Y1
Lydrup, ML1
MacLeod, KM; Ray, A1
Baeyens, JM; Barrios, M; Del Pozo, E1
Imai, S; Ogawa, Y1
Coldwell, MC; Cooper, SM; Hamilton, TC; Howlett, DR; Wilson, C1
Ebisu, H; Eda, M; Fukaya, C; Gohda, M; Hihara, M; Matzno, S; Nakamura, N; Okada, T; Sakashita, H; Takemoto, T1
Bányász, T; Nánási, PP; Pankucsi, C; Szigligeti, P; Varró, A1
Bojić, M; Djukanović, B; Gojkoviíc Bukarica, L; Kazić, T; Panić, G; Perić, M; Sajić, Z1
Kecskeméti, V; Losonczy, G; Mucha, I; Nánási, PP; Pacher, P; Ungvári, Z1
Barrett, JE; Brandsgaard, R; Rosenzweig-Lipson, S1
Long, W; Longo, LD; Zhang, L1
Dacey, RG; Dietrich, HH; Horiuchi, T; Tsugane, S1
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI; Rosas, R; Torres-López, JE; Vidal-Cantú, GC1
Allen, T; Cole, WC; Iftinca, M; Plane, F1
El-Mahmoudy, A; Matsuyama, H; Shimizu, Y; Takewaki, T; Thapaliya, S1
Baker, PN; Fyfe, GK; Greenwood, SL; Sibley, CP; Williams, JL1
Greenwood, IA; Ohya, S; Tribe, RM; Yeung, SY1
Beleslin-Cokic, B; Gojkovic-Bukarica, L; Heinle, H; Ilic, B; Novakovic, R; Radunovic, N; Scepanovic, R1

Other Studies

21 other study(ies) available for pinacidil and 4-aminopyridine

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
[The vasospasmolytic effects of nicorandil, cromakalim and pinacidil on 3,4-diaminopyridine-induced phasic contractions in canine coronary arteries as an experimental vasospasm model].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1992, Volume: 100, Issue:4

    Topics: 4-Aminopyridine; Amifampridine; Animals; Benzopyrans; Coronary Vasospasm; Cromakalim; Disease Models, Animal; Dogs; Female; Glyburide; Guanidines; In Vitro Techniques; Ion Channel Gating; Male; Methylene Blue; Niacinamide; Nicorandil; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents

1992
Role of K+ channels in spontaneous electrical and mechanical activity of smooth muscle in the guinea-pig mesotubarium.
    The Journal of physiology, 1991, Volume: 433

    Topics: 4-Aminopyridine; Animals; Apamin; Electrophysiology; Female; Guanidines; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Pinacidil; Potassium Channels; Rubidium; Tetraethylammonium; Tetraethylammonium Compounds; Uterine Contraction; Uterus

1991
Adrenergic-cholinergic interactions in left atria: a study using K+ channel agonists, antagonist and pertussis toxin.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: 4-Aminopyridine; Animals; Benzopyrans; Carbachol; Cromakalim; Cyclic AMP; Dogs; Female; Guanidines; Heart; Isoproterenol; Male; Myocardial Contraction; Parasympathetic Nervous System; Pertussis Toxin; Phenylephrine; Pinacidil; Potassium Channels; Pyrroles; Rabbits; Sympathetic Nervous System; Virulence Factors, Bordetella

1990
Effects of potassium channel openers on pentylenetetrazole-induced seizures in mice.
    Pharmacology & toxicology, 1990, Volume: 67, Issue:2

    Topics: 4-Aminopyridine; Animals; Benzopyrans; Cromakalim; Drug Antagonism; Female; Guanidines; Mice; Pentylenetetrazole; Pinacidil; Potassium Channels; Pyrroles; Seizures

1990
[Effects of vasodilators on cyclic contraction induced by 3,4-diaminopyridine in isolated porcine coronary arteries].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1987, Volume: 89, Issue:6

    Topics: 4-Aminopyridine; Amifampridine; Aminopyridines; Angina Pectoris; Animals; Calcium; Coronary Vessels; Drug Interactions; Guanidines; In Vitro Techniques; Ion Channels; Periodicity; Pinacidil; Potassium; Swine; Vasodilator Agents

1987
Comparative effects of K+ channel blockade on the vasorelaxant activity of cromakalim, pinacidil and nicorandil.
    European journal of pharmacology, 1988, Aug-02, Volume: 152, Issue:3

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Benzopyrans; Cardiovascular Agents; Cromakalim; Guanidines; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Pinacidil; Potassium Channels; Procaine; Pyrroles; Rabbits; Rubidium Radioisotopes; Tetraethylammonium Compounds; Vasodilator Agents

1988
Novel potassium channel openers: synthesis and pharmacological evaluation of new N-(substituted-3-pyridyl)-N'-alkylthioureas and related compounds.
    Journal of medicinal chemistry, 1994, Jan-07, Volume: 37, Issue:1

    Topics: 4-Aminopyridine; Amifampridine; Animals; Antihypertensive Agents; Biomechanical Phenomena; Glyburide; Guanidines; Hypertension; Male; Molecular Structure; Norbornanes; Pinacidil; Portal Vein; Potassium Channels; Rats; Rats, Inbred SHR; Rats, Wistar; Structure-Activity Relationship

1994
Action potential duration and force-frequency relationship in isolated rabbit, guinea pig and rat cardiac muscle.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1996, Volume: 166, Issue:2

    Topics: 4-Aminopyridine; Action Potentials; Animals; Benzopyrans; Cromakalim; Cytosol; Guanidines; Guinea Pigs; Heart; In Vitro Techniques; Myocardial Contraction; Pinacidil; Potassium Channel Blockers; Potassium Channels; Pyrroles; Rabbits; Rats; Sodium; Strophanthidin; Tetraethylammonium; Tetraethylammonium Compounds

1996
The effects of levcromakalim and pinacidil on the human internal mammary artery.
    Fundamental & clinical pharmacology, 1997, Volume: 11, Issue:6

    Topics: 4-Aminopyridine; Adenosine Triphosphate; Apamin; Charybdotoxin; Coronary Artery Bypass; Coronary Disease; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Guanidines; Humans; In Vitro Techniques; Male; Mammary Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Pinacidil; Potassium Channels; Tetraethylammonium; Vasodilation; Vasodilator Agents

1997
Post-partum prolongation of the atrial repolarization in rabbit.
    Acta physiologica Scandinavica, 1999, Volume: 166, Issue:1

    Topics: 4-Aminopyridine; Action Potentials; Animals; Atrial Function; Electrophysiology; Estrogens; Female; Glyburide; Heart Atria; Heart Conduction System; Hypoglycemic Agents; Muscle Fibers, Skeletal; Myocardium; Pinacidil; Postpartum Period; Potassium Channels; Pregnancy; Rabbits; Vasodilator Agents

1999
Pharmacological characterization of the discriminative stimulus effects of the potassium channel blocker 4-aminopyridine in rats.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:1

    Topics: 4-Aminopyridine; Animals; Cholinergic Agents; Discrimination Learning; Dopamine Agents; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Pinacidil; Potassium Channel Blockers; Prazosin; Rats; Rats, Sprague-Dawley; Serotonin Agents

2000
Cerebral artery K(ATP)- and K(Ca)-channel activity and contractility: changes with development.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 279, Issue:6

    Topics: 4-Aminopyridine; Animals; Benzimidazoles; Calcium; Fetus; In Vitro Techniques; Middle Cerebral Artery; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Peptides; Pinacidil; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Sheep

2000
Role of potassium channels in regulation of brain arteriolar tone: comparison of cerebrum versus brain stem.
    Stroke, 2001, Volume: 32, Issue:1

    Topics: 4-Aminopyridine; Animals; Arterioles; Barium Compounds; Brain; Brain Stem; Chlorides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Nitric Oxide Synthase; Nitroarginine; Pinacidil; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Telencephalon; Tetraethylammonium; Vasoconstriction; Vasodilator Agents

2001
Pharmacological evidence for the activation of K(+) channels by diclofenac.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: 4-Aminopyridine; Analgesics; Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Behavior, Animal; Charybdotoxin; Diclofenac; Dose-Response Relationship, Drug; Female; Formaldehyde; Glyburide; Hindlimb; Morphine; Pain; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide

2002
Smooth muscle membrane potential modulates endothelium-dependent relaxation of rat basilar artery via myo-endothelial gap junctions.
    The Journal of physiology, 2002, 12-15, Volume: 545, Issue:3

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Basilar Artery; Endothelium, Vascular; Gap Junctions; Glycyrrhetinic Acid; In Vitro Techniques; Male; Membrane Potentials; Muscle, Smooth, Vascular; Nitric Oxide; Pinacidil; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Vasodilation; Vasodilator Agents

2002
An endothelium-derived factor modulates purinergic neurotransmission to mesenteric arterial smooth muscle of hamster.
    European journal of pharmacology, 2003, Feb-14, Volume: 461, Issue:2-3

    Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Apamin; Biological Factors; Charybdotoxin; Cricetinae; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Epoprostenol; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Male; Membrane Potentials; Mesenteric Arteries; Mesocricetus; Muscle, Smooth, Vascular; Neuromuscular Junction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Ouabain; Pinacidil; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Synaptic Transmission; Tetraethylammonium; Time Factors; Triazines; Uridine Triphosphate; Vasodilator Agents

2003
K+ channel inhibition modulates the biochemical and morphological differentiation of human placental cytotrophoblast cells in vitro.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2008, Volume: 295, Issue:4

    Topics: 4-Aminopyridine; Arachidonic Acids; Barium Compounds; Calcium Channel Blockers; Cell Differentiation; Cells, Cultured; Chlorides; Chorionic Gonadotropin; Cromakalim; Endocannabinoids; Female; Giant Cells; Humans; L-Lactate Dehydrogenase; Nifedipine; Pinacidil; Placenta; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Channels; Pregnancy; Tetraethylammonium; Trophoblasts

2008
Loss of functional K+ channels encoded by ether-à-go-go-related genes in mouse myometrium prior to labour onset.
    The Journal of physiology, 2009, May-15, Volume: 587, Issue:Pt 10

    Topics: 4-Aminopyridine; Animals; Chlorobenzenes; Cresols; Electric Stimulation; Electrophysiological Phenomena; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Female; Gene Expression; Labor, Obstetric; Mice; Mice, Inbred BALB C; Myocytes, Smooth Muscle; Myometrium; ortho-Aminobenzoates; Oxytocin; Patch-Clamp Techniques; Phenylurea Compounds; Pinacidil; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Pregnancy; Uterine Contraction

2009
The effect of resveratrol on contractility of non-pregnant rat uterus: the contribution of K(+) channels.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2013, Volume: 64, Issue:6

    Topics: 4-Aminopyridine; Animals; Benzimidazoles; Female; Glyburide; Isometric Contraction; Muscle, Smooth; Oxytocin; Peptides; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Resveratrol; Stilbenes; Tetraethylammonium; Uterus

2013