Page last updated: 2024-08-17

pilocarpine and quinuclidines

pilocarpine has been researched along with quinuclidines in 84 studies

Research

Studies (84)

TimeframeStudies, this research(%)All Research%
pre-199035 (41.67)18.7374
1990's11 (13.10)18.2507
2000's26 (30.95)29.6817
2010's11 (13.10)24.3611
2020's1 (1.19)2.80

Authors

AuthorsStudies
Lamble, AP; Lamble, JW1
Birdsall, NJ; Burgen, AS; Strange, PG1
François, J; Goes, F3
Dengler, G; Mayer, U1
Ober, M; Scharrer, A1
Dulis, BH; Gordon, MA; Wilson, IB1
Fechner, PU; Teichmann, KD; Weyrauch, W1
Lepple-Wienhues, A; Stahl, F; Wiederholt, M1
Erickson-Lamy, K; Schroeder, A1
Brandeis, R; Fisher, A; Gurwitz, D; Haring, R; Heldman, E; Karton, I; Levy, A; Pittel, Z; Sapir, M1
Dwyer, TM; Farley, JM; Yang, CM1
Snyder, SH; Yamamura, HI1
Roger, MJ1
Holland, MG1
Mashkovsky, MD; Yakhontov, LN1
Braun, H; Dausch, D; Meythaler, H1
Lommatzsch, P; Pilz, A; Ulrich, WD1
Romano, JH1
Drance, SM; Fairclough, M; Schulzer, M1
Samoĭlovich, IM1
Iuglio, N1
Meythaler, H; Ruppert, W1
Collignon, J; Lennes, G; Luyckx, J; Weekers, R1
Verraz, R1
Collignon-Brach, J; Prijot, E; Weekers, R1
Lepri, G; Tota, G1
Bastide, P; Rouher, F; Tronche, P1
Nud'ga, LI; Sharts, SE; Shul'pina, NB1
Smith, SA; Smith, SE1
Keren, G; Treister, G1
Ciracì, G; Giummarra, C; Reibaldi, A1
Fedorov, VI1
Jedrych, Z1
Huger, FP; Smith, CP1
Giorgi, O; Rubio, MC1
Ehlert, FJ; Fairhurst, AS; Kokka, N1
Iwabuchi, Y; Masuhara, T1
Freedman, SB; Patel, S1
Fisher, A; Fraser, CM; Gurwitz, D; Haring, R; Heldman, E; Manor, D1
Hubbard, WC; Kaufman, PL; Kee, C1
Masunaga, H; Ogawa, H; Takeshita, Y; Tomizuka, T; Uematsu, Y; Yasuda, H1
Bymaster, FP; Calligaro, DO; Carter, PA; DeLapp, N; Fink-Jensen, A; Jeppesen, L; Mitch, CH; Peters, SC; Rimvall, K; Sauerberg, P; Shannon, HE; Sheardown, MJ; Ward, JS; Whitesitt, CA; Zhang, W1
Belmonte, KE; Costello, RW; Fryer, AD; Jacoby, DB1
Anaya, JM; Talal, N1
Erickson, KA; Schroeder, A1
Elwood, T; Fryer, AD; Jacoby, DB; Yost, BL1
Fox, RI; Michelson, P1
al-Hashimi, I; Taylor, SE1
Atkinson, JC; Baum, BJ1
Fisher, A; Fox, RI; Konttinen, Y1
Muzyka, BC1
Gu, Y; Peng, D; Wu, Y; Zeng, S1
Iida, H; Inoue, N; Ishida, H; Ishikawa, Y; Yuan, Z1
Nieuw Amerongen, AV; Veerman, EC1
Asari, T; Kojima, M; Kusama, H; Maruyama, K; Omori, Y; Shibata, N1
Bruce, SD1
Aframian, DJ; Nahlieli, O; Palmon, A1
Shetty, K1
Atkinson, JC; Grisius, M; Massey, W1
Chen, HZ; Cui, YY; Feng, JM; Wu, XJ; Zhu, L1
Al-Hashimi, I1
Johnstone, PA; Kahn, ST1
Gause, A1
Brennan, MT; Carrozzo, M; Daniels, T; Fox, PC; Fujibayashi, T; Gandera, B; Jonsson, R; Lockhart, PB; Navazesh, M; Rhodus, NL; Schiødt, M; Sollecito, TP; von Bültzingslöwen, I; Wray, D1
Wick, JY1
Akamatsu, T; Azlina, A; Hasegawa, T; Hosoi, K; Karabasil, MR; Li, X; Purwanti, N; Yao, C1
Andrade, ED; Bergamaschi, CC; Braga, MA; Groppo, FC; Santos, FA; Tarzia, O1
Hosokawa, R; Iida, T; Inagaki, T; Inenaga, K; Ono, K1
Adyanthaya, RS; Akpek, EK; Baer, AN; Lindsley, KB; McDonnell, PJ; Swamy, R1
Hosokawa, R; Iida, T; Inagaki, T; Inenaga, K; Ono, K; Wakasugi-Sato, N1
Chimenos Küstner, E; Jané Salas, E; López-López, J1
Kawakami, A; Nakamura, H; Nakamura, T; Sato, S; Sumi, M; Takagi, Y1
Asbell, PA; Kuklinski, E1
Barbe, AG1
Forbes, B; Garcia, CMA; Malallah, OS; Proctor, GB; Royall, PG1
Cherubini, K; Figueiredo, MAZ; Medella-Junior, FAC; Salum, FG1
B E, S; Badam, RK; Boringi, M; Garlapati, K; Kammari, A; Soni, P1
Chen, CH; Chou, YC; Huang, WY; Ju, UH; Kao, CH; Lin, CL; Lin, CS; Lin, KT; Lin, TY; Liu, FC; Shen, CH; Yang, TY1
Cimmino, J; Farag, AM; Holliday, C; Papas, A; Roomian, T1
Graue-Hernandez, EO; Kahuam-López, N; Navas, A; Pérez Vázquez, AK; Ramirez-Miranda, A; Serrano-Robles, JG1

Reviews

18 review(s) available for pilocarpine and quinuclidines

ArticleYear
Autonomic drugs in ophthalmology: some problems and promises. I. Directly and indirectly acting parasympathomimetic drugs.
    Annals of ophthalmology, 1974, Volume: 6, Issue:5

    Topics: Administration, Topical; Animals; Carbachol; Cataract; Cholinesterase Inhibitors; Contact Lenses, Hydrophilic; Echothiophate Iodide; Eye; Eye Diseases; Glaucoma; Haplorhini; Humans; Intraocular Pressure; Isoflurophate; Parasympathomimetics; Pharmaceutical Vehicles; Pilocarpine; Pralidoxime Compounds; Quaternary Ammonium Compounds; Quinuclidines; Rabbits

1974
Relationships between the chemical structure and pharmacological activity in a series of synthetic quinuclidine derivatives.
    Progress in drug research. Fortschritte der Arzneimittelforschung. Progres des recherches pharmaceutiques, 1969, Volume: 13

    Topics: Animals; Benactyzine; Carbamates; Cats; Chemical Phenomena; Chemistry; Esters; Ganglionic Blockers; Iodides; Mice; Parasympatholytics; Pilocarpine; Piperidines; Prochlorperazine; Pupil; Quinuclidines; Rabbits; Rats; Salicylates; Tubocurarine

1969
Sjögren's syndrome comes of age.
    Seminars in arthritis and rheumatism, 1999, Volume: 28, Issue:6

    Topics: Apoptosis; Humans; Lymphocytosis; Muscarinic Agonists; Pilocarpine; Quinuclidines; Receptors, Muscarinic; Salivary Glands; Sjogren's Syndrome; Thiophenes

1999
Approaches to the treatment of Sjögren's syndrome.
    The Journal of rheumatology. Supplement, 2000, Volume: 61

    Topics: Humans; Muscarinic Agonists; Pilocarpine; Quinuclidines; Sjogren's Syndrome; Thiophenes

2000
Use of muscarinic agonists in the treatment of Sjögren's syndrome.
    Clinical immunology (Orlando, Fla.), 2001, Volume: 101, Issue:3

    Topics: Humans; Muscarinic Agonists; Neuroimmunomodulation; Neurosecretory Systems; Pilocarpine; Quinuclidines; Receptors, Muscarinic; Sjogren's Syndrome; Thiophenes

2001
Current therapies for xerostomia and salivary gland hypofunction associated with cancer therapies.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 2003, Volume: 11, Issue:4

    Topics: Acupuncture Therapy; Antineoplastic Agents; Chewing Gum; Diet; Flavoring Agents; Humans; Muscarinic Agonists; Neoplasms; Oral Hygiene; Palliative Care; Parasympathomimetics; Pilocarpine; Quinuclidines; Radiotherapy; Saliva; Salivary Glands; Thiophenes; Xerostomia

2003
Radiation-induced xerostomia: how dry is your patient?
    Clinical journal of oncology nursing, 2004, Volume: 8, Issue:1

    Topics: Acupuncture Therapy; Head and Neck Neoplasms; Humans; Muscarinic Agonists; Nurse's Role; Nursing Assessment; Oncology Nursing; Oral Hygiene; Pilocarpine; Quality of Life; Quinuclidines; Radiotherapy; Radiotherapy Dosage; Salivation; Thiophenes; Xerostomia

2004
Salivary hypofunction and xerostomia: diagnosis and treatment.
    Dental clinics of North America, 2005, Volume: 49, Issue:2

    Topics: Aged; Aged, 80 and over; Cariostatic Agents; Fluorides; Humans; Pilocarpine; Polypharmacy; Quinuclidines; Radiotherapy; Salivation; Sjogren's Syndrome; Thiophenes; Xerostomia

2005
Xerostomia secondary to Sjögren's syndrome in the elderly: recognition and management.
    Drugs & aging, 2005, Volume: 22, Issue:11

    Topics: Aged; Aged, 80 and over; Diagnosis, Differential; Humans; Muscarinic Agonists; Pilocarpine; Quinuclidines; Sjogren's Syndrome; Thiophenes; Xerostomia

2005
Management of xerostomia related to radiotherapy for head and neck cancer.
    Oncology (Williston Park, N.Y.), 2005, Volume: 19, Issue:14

    Topics: Acupuncture Therapy; Amifostine; Clinical Trials as Topic; Head and Neck Neoplasms; Humans; Muscarinic Agonists; Palliative Care; Pilocarpine; Quinuclidines; Radiation-Protective Agents; Radiotherapy; Submandibular Gland; Thiophenes; Xerostomia

2005
Salivary dysfunction associated with systemic diseases: systematic review and clinical management recommendations.
    Oral surgery, oral medicine, oral pathology, oral radiology, and endodontics, 2007, Volume: 103 Suppl

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Murine-Derived; Antiviral Agents; Diabetes Complications; HIV Infections; Humans; Interferon-alpha; Muscarinic Agonists; Pilocarpine; Quinuclidines; Rituximab; Salivation; Sjogren's Syndrome; Thiophenes; Xerostomia

2007
Xerostomia: causes and treatment.
    The Consultant pharmacist : the journal of the American Society of Consultant Pharmacists, 2007, Volume: 22, Issue:12

    Topics: Autoimmune Diseases; Bone Marrow Transplantation; Drug-Related Side Effects and Adverse Reactions; Humans; Pilocarpine; Quinuclidines; Saliva; Thiophenes; Xerostomia

2007
Treatment of Sjögren's syndrome-associated dry eye an evidence-based review.
    Ophthalmology, 2011, Volume: 118, Issue:7

    Topics: Administration, Oral; Administration, Topical; Anti-Inflammatory Agents; Dry Eye Syndromes; Evidence-Based Medicine; Humans; Hydroxychloroquine; Immunosuppressive Agents; Lubricants; Pilocarpine; Quinuclidines; Sjogren's Syndrome; Thiophenes

2011
[Prognosis and treatment of dry mouth. Systematic review].
    Medicina clinica, 2014, Feb-04, Volume: 142, Issue:3

    Topics: Cholinergic Antagonists; Clinical Trials as Topic; Dental Caries; Disease Susceptibility; Double-Blind Method; Fluid Therapy; Humans; Meta-Analysis as Topic; Mouthwashes; Observational Studies as Topic; Pilocarpine; Prognosis; Quinuclidines; Radiation Injuries; Radiotherapy; Saliva, Artificial; Salivation; Sjogren's Syndrome; Thiophenes; Xerostomia

2014
Sjogren's syndrome from the perspective of ophthalmology.
    Clinical immunology (Orlando, Fla.), 2017, Volume: 182

    Topics: Administration, Ophthalmic; Cyclosporine; Dry Eye Syndromes; Fatty Acids, Omega-3; Glucocorticoids; Humans; Immunosuppressive Agents; Lubricant Eye Drops; Muscarinic Agonists; Ophthalmology; Phenylalanine; Pilocarpine; Punctal Plugs; Quinuclidines; Sjogren's Syndrome; Sulfones; Thiophenes

2017
Buccal drug delivery technologies for patient-centred treatment of radiation-induced xerostomia (dry mouth).
    International journal of pharmaceutics, 2018, Apr-25, Volume: 541, Issue:1-2

    Topics: Drug Delivery Systems; Head and Neck Neoplasms; Humans; Mouth Mucosa; Muscarinic Agonists; Pilocarpine; Quinuclidines; Radiation Injuries; Saliva; Thiophenes; Time Factors; Xerostomia

2018
Salivary hypofunction: An update on therapeutic strategies.
    Gerodontology, 2018, Volume: 35, Issue:4

    Topics: Acupuncture Therapy; Bethanechol; Chewing Gum; Humans; Hyperbaric Oxygenation; Muscarinic Agonists; Pilocarpine; Quinuclidines; Thiophenes; Xerostomia

2018
Meta-analysis on pharmacological therapies in the management of xerostomia in patients with Sjogren's syndrome.
    Immunopharmacology and immunotoxicology, 2019, Volume: 41, Issue:2

    Topics: Female; Humans; Interferon-alpha; Male; Pilocarpine; Quinuclidines; Saliva; Sjogren's Syndrome; Thiophenes

2019

Trials

3 trial(s) available for pilocarpine and quinuclidines

ArticleYear
Double-blind cross-over comparison of aceclidine and pilocarpine in open-angle glaucoma.
    The British journal of ophthalmology, 1970, Volume: 54, Issue:8

    Topics: Aqueous Humor; Clinical Trials as Topic; Female; Glaucoma; Humans; Intraocular Pressure; Male; Miotics; Parasympathomimetics; Pilocarpine; Placebos; Quinuclidines; Tonometry, Ocular

1970
[The myopic and miotic effect of pilocarpin and glaucostat].
    Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie. Albrecht von Graefe's archive for clinical and experimental ophthalmology, 1971, Volume: 181, Issue:3

    Topics: Accommodation, Ocular; Adolescent; Adult; Child; Cocaine; Color; Eye; Humans; Hyperemia; Iris; Miotics; Mydriatics; Myopia; Phenylephrine; Pilocarpine; Pupil; Quinuclidines

1971
Comparison of the effects of pilocarpine and cevimeline on salivary flow.
    International journal of dental hygiene, 2009, Volume: 7, Issue:2

    Topics: Administration, Oral; Adult; Cross-Over Studies; Humans; Male; Muscarinic Agonists; Physical Stimulation; Pilocarpine; Quinuclidines; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Saliva; Salivary Glands; Secretory Rate; Single-Blind Method; Thiophenes; Time Factors; Young Adult

2009

Other Studies

63 other study(ies) available for pilocarpine and quinuclidines

ArticleYear
The effect of miotics on the intraocular pressure of conscious owl monkeys.
    Investigative ophthalmology, 1976, Volume: 15, Issue:10

    Topics: Anesthesia, Local; Animals; Aotus trivirgatus; Carbachol; Dose-Response Relationship, Drug; Haplorhini; Intraocular Pressure; Male; Miotics; Oxotremorine; Parasympathomimetics; Pilocarpine; Quinuclidines; Spiro Compounds; Succinimides; Tonometry, Ocular

1976
Occupancy of muscarinic acetylcholine receptors stimulates a guanylate cyclase in neuroblastoma cells.
    Biochemical Society transactions, 1977, Volume: 5, Issue:1

    Topics: Acetylcholine; Atropine; Carbachol; Cell Line; Cell Membrane; Enzyme Activation; Guanylate Cyclase; Kinetics; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic

1977
Ultrasonographic study of the effect of different miotics on the eye components.
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 1977, Volume: 175, Issue:6

    Topics: Administration, Topical; Adult; Anterior Chamber; Carbachol; Epinephrine; Eye; Humans; Lens, Crystalline; Middle Aged; Miotics; Myopia; Pain; Pilocarpine; Pupil; Quinuclidines; Refraction, Ocular; Ultrasonography; Vitreous Body

1977
[Comparative investigations concerning the influence of pilocarpine and aceclidine on the glucose consumption of surviving ocular tissues (author's transl)].
    Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie. Albrecht von Graefe's archive for clinical and experimental ophthalmology, 1978, Jan-31, Volume: 205, Issue:2

    Topics: Animals; Cattle; Cell Survival; Eye; Glucose; Iris; Lens, Crystalline; Pilocarpine; Quinuclidines; Tissue Preservation

1978
[The effect of timolol and parasympathicomimetica in the treatment of the elevated intraocular pressure (author's transl)].
    Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie. Albrecht von Graefe's archive for clinical and experimental ophthalmology, 1979, Jul-02, Volume: 211, Issue:1

    Topics: Carbachol; Drug Administration Schedule; Glaucoma; Humans; Intraocular Pressure; Parasympathomimetics; Pilocarpine; Propanolamines; Quinuclidines; Timolol

1979
Identification of muscarinic binding sites in human neutrophils by direct binding.
    Molecular pharmacology, 1979, Volume: 15, Issue:1

    Topics: Atropine; Benzilates; Binding, Competitive; Humans; In Vitro Techniques; Kinetics; Neutrophils; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic

1979
Accommodative effects of aceclidine in the treatment of glaucoma.
    American journal of ophthalmology, 1975, Volume: 79, Issue:1

    Topics: Accommodation, Ocular; Adult; Age Factors; Amides; Glaucoma; Humans; Intraocular Pressure; Middle Aged; Myopia; Ophthalmic Solutions; Pilocarpine; Pyridines; Quinuclidines

1975
Ultrasonographic comparative study of the effect of pilocarpine and aceclidine on the eye components.
    Bibliotheca ophthalmologica : supplementa ad ophthalmologica, 1975, Issue:83

    Topics: Accommodation, Ocular; Adolescent; Adult; Age Factors; Aged; Anterior Chamber; Eye; Glaucoma; Humans; Lens, Crystalline; Middle Aged; Ophthalmic Solutions; Pilocarpine; Quinuclidines; Ultrasonography

1975
Differential smooth muscle-like contractile properties of trabecular meshwork and ciliary muscle.
    Experimental eye research, 1991, Volume: 53, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Cattle; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Isometric Contraction; Muscle, Smooth; Pilocarpine; Potassium; Quinuclidines; Trabecular Meshwork

1991
Dissociation between the effect of aceclidine on outflow facility and accommodation.
    Experimental eye research, 1990, Volume: 50, Issue:2

    Topics: Accommodation, Ocular; Animals; Aqueous Humor; Dose-Response Relationship, Drug; Macaca fascicularis; Pilocarpine; Quinuclidines

1990
(+-)-cis-2-methyl-spiro(1,3-oxathiolane-5,3')quinuclidine, an M1 selective cholinergic agonist, attenuates cognitive dysfunctions in an animal model of Alzheimer's disease.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Alzheimer Disease; Animals; Avoidance Learning; Binding, Competitive; Cognition Disorders; Copper; Disease Models, Animal; Male; Memory; Mice; Motor Activity; Parasympathomimetics; Pilocarpine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Thiophenes

1991
Biochemical characteristics of muscarinic cholinoreceptors in swine tracheal smooth muscle.
    Journal of autonomic pharmacology, 1986, Volume: 6, Issue:1

    Topics: Animals; Atropine; Binding Sites; Carbachol; Epithelium; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Muscle, Smooth; Pilocarpine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Scopolamine; Swine; Temperature; Trachea; Tritium

1986
Muscarinic cholinergic binding in rat brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1974, Volume: 71, Issue:5

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Binding Sites; Binding, Competitive; Brain; Brompheniramine; Carbachol; Chlorpheniramine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Microsomes; Mitochondria; Oxotremorine; Pilocarpine; Quaternary Ammonium Compounds; Quinuclidines; Rats; Receptors, Cholinergic; Scopolamine; Temperature; Time Factors; Tritium

1974
[Use of drug solutions on hydrophylic lenses].
    Bulletin des societes d'ophtalmologie de France, 1974, Volume: 74, Issue:3

    Topics: Adrenal Cortex Hormones; Anti-Bacterial Agents; Anti-Infective Agents, Local; Contact Lenses, Hydrophilic; Eye Diseases; Humans; Mydriatics; Ophthalmic Solutions; Pilocarpine; Quinuclidines

1974
[Tonographical examination on the effect of glaucadrine in the treatment of open-angle glaucoma (author's transl)].
    Klinische Monatsblatter fur Augenheilkunde, 1973, Volume: 163, Issue:6

    Topics: Aqueous Humor; Drug Combinations; Epinephrine; Glaucoma; Humans; Intraocular Pressure; Myopia; Pilocarpine; Quinuclidines; Tonometry, Ocular

1973
[Experimental and clinical studies with aceclidine (Glaucostat)].
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 1974, Volume: 168, Issue:5

    Topics: Accommodation, Ocular; Adolescent; Adult; Age Factors; Child; Ciliary Body; Glaucoma; Humans; In Vitro Techniques; Intraocular Pressure; Iris; Middle Aged; Muscle, Smooth; Ophthalmic Solutions; Pilocarpine; Pupil; Quinuclidines; Refraction, Ocular; Visual Acuity

1974
Ultrasonographic comparative study of the effect of pilocarpine and aceclidine on the eye components.
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 1974, Volume: 168, Issue:4

    Topics: Accommodation, Ocular; Adult; Aged; Anterior Chamber; Depression, Chemical; Evaluation Studies as Topic; Glaucoma; Humans; Lens, Crystalline; Middle Aged; Pilocarpine; Quinuclidines; Refraction, Ocular; Stimulation, Chemical; Ultrasonography

1974
Dose response of human intraocular pressure to aceclidine.
    Archives of ophthalmology (Chicago, Ill. : 1960), 1972, Volume: 88, Issue:4

    Topics: Acetates; Aged; Dose-Response Relationship, Drug; Glaucoma; Humans; Intraocular Pressure; Middle Aged; Ophthalmic Solutions; Parasympathomimetics; Pilocarpine; Quinuclidines; Time Factors; Tonometry, Ocular

1972
[Relation between internal activity and magnitude of the maximal effect].
    Biulleten' eksperimental'noi biologii i meditsiny, 1971, Volume: 71, Issue:6

    Topics: Acetylcholine; Animals; Carbachol; In Vitro Techniques; Miotics; Muscle, Smooth; Nicotinic Acids; Parasympathomimetics; Pilocarpine; Quinuclidines; Rats; Receptors, Drug; Stomach

1971
[Comparative evaluation of the action of aceclidine and pilocarpine on the peripheral anterior chamber depth of the normal human eye].
    Bollettino della Societa italiana di biologia sperimentale, 1971, Oct-15, Volume: 47, Issue:19

    Topics: Anterior Chamber; Humans; Intraocular Pressure; Pilocarpine; Quinuclidines

1971
[The mode of action of aceclidine on ocular pressure].
    Documenta ophthalmologica. Advances in ophthalmology, 1969, Volume: 26

    Topics: Aqueous Humor; Glaucoma; Humans; Intraocular Pressure; Pilocarpine; Quinuclidines

1969
[On the value of aceclidine in the treatment of chronic simple glaucoma as compared with pilocarpine].
    Annali di ottalmologia e clinica oculistica, 1969, Volume: 95, Issue:4

    Topics: Adult; Chronic Disease; Female; Glaucoma; Humans; Male; Middle Aged; Pilocarpine; Quinuclidines

1969
[Treatment of open-angle glaucoma with an association of aceclidine and adrenaline (glaucadrine)].
    Bulletin de la Societe belge d'ophtalmologie, 1970, Volume: 155

    Topics: Aqueous Humor; Blood Pressure; Epinephrine; Glaucoma; Humans; Injections, Intravenous; Intraocular Pressure; Pilocarpine; Quinuclidines

1970
[The action of aceclydine in ocular hypertension].
    Annali di ottalmologia e clinica oculistica, 1967, Volume: 93, Issue:6

    Topics: Adult; Aged; Female; Glaucoma; Humans; Male; Middle Aged; Pilocarpine; Quinuclidines

1967
[Aceclidine, a new pressure descreasing miotic. Pharmacological and Clinical studies].
    Arzneimittel-Forschung, 1968, Volume: 18, Issue:3

    Topics: Animals; Aqueous Humor; Blood Pressure; Depression, Chemical; Drug Tolerance; Eye; Glaucoma; Humans; Intraocular Pressure; Mice; Miotics; Parasympatholytics; Pilocarpine; Quinuclidines; Rabbits; Rats; Respiration

1968
[On the effect of aceclidine on the size of the blind spot].
    Oftalmologicheskii zhurnal, 1966, Volume: 21, Issue:2

    Topics: Glaucoma; Humans; Miotics; Pilocarpine; Quinuclidines; Visual Field Tests

1966
Subsensitivity to cholinoceptor stimulation of the human iris sphincter in situ following acute and chronic administration of cholinomimetic miotic drugs.
    British journal of pharmacology, 1980, Volume: 69, Issue:3

    Topics: Adult; Arecoline; Glaucoma; Humans; Iris; Light; Miotics; Parasympathomimetics; Physostigmine; Pilocarpine; Pupil; Quinuclidines; Receptors, Cholinergic; Time Factors

1980
Effect of aceclidine(+) isomer and pilocarpine on the intraocular pressure decrease and the miosis in glaucomatous eyes. Effect on accommodation in normal eyes of young subjects.
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 1980, Volume: 180, Issue:4

    Topics: Accommodation, Ocular; Adult; Aqueous Humor; Glaucoma; Humans; Intraocular Pressure; Middle Aged; Parasympathomimetics; Pilocarpine; Pupil; Quinuclidines; Stereoisomerism

1980
[The effect of antiglaucoma drugs on the depth of the anterior chamber (I)].
    Bollettino della Societa italiana di biologia sperimentale, 1982, Aug-15, Volume: 58, Issue:15

    Topics: Adult; Anterior Chamber; Carbachol; Clonidine; Glaucoma; Humans; Middle Aged; Miotics; Moxisylyte; Pilocarpine; Propranolol; Quinuclidines; Timolol

1982
[Effect of parasympathetic agents on renin secretion in vitro].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 97, Issue:3

    Topics: Animals; Atropine; Diphenylacetic Acids; Galantamine; Ganglionic Blockers; Hexamethonium Compounds; In Vitro Techniques; Kidney Cortex; Neostigmine; Parasympatholytics; Parasympathomimetics; Pilocarpine; Pyrrolizidine Alkaloids; Quaternary Ammonium Compounds; Quinuclidines; Rats; Renin

1984
Cholinolytic activity of 3-hydroxyquinuclidyl-1-phenyl-1-cyclohexyl-1-carboxylate hydrochloride (ANC-821).
    Polish journal of pharmacology and pharmacy, 1983, Volume: 35, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Bronchi; Electrocardiography; In Vitro Techniques; Male; Mice; Muscle Contraction; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Rats; Rats, Inbred Strains

1983
Effect of zinc on [3H]-QNB displacement by cholinergic agonists and antagonists.
    Biochemical pharmacology, 1983, Jan-15, Volume: 32, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Binding, Competitive; Male; Oxotremorine; Parasympatholytics; Parasympathomimetics; Physostigmine; Pilocarpine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Zinc

1983
Decreased 3H-L-quinuclidinyl benzilate binding and muscarine receptor subsensitivity after chronic gamma-butyrolactone treatment.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 318, Issue:1

    Topics: 4-Butyrolactone; Animals; Behavior, Animal; Choline O-Acetyltransferase; Corpus Striatum; Furans; Male; Membranes; Pilocarpine; Postural Balance; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic

1981
Altered [3H]quinuclidinyl benzilate binding in the striatum of rats following chronic cholinesterase inhibition with diisopropylfluorophosphate.
    Molecular pharmacology, 1980, Volume: 17, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Cholinesterase Inhibitors; Corpus Striatum; In Vitro Techniques; Isoflurophate; Male; Pilocarpine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic

1980
Sialogogic activities of SNI-2011 compared with those of pilocarpine and McN-A-343 in rat salivary glands: identification of a potential therapeutic agent for treatment of Sjörgen's syndrome.
    General pharmacology, 1994, Volume: 25, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adrenergic Antagonists; Animals; Cholinergic Antagonists; Male; Pilocarpine; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Salivary Glands; Salivation; Sjogren's Syndrome; Thiophenes

1994
The muscarinic receptor agonist L-658,903 modulates the in vivo accumulation of inositol monophosphates in mouse brain.
    European journal of pharmacology, 1994, May-17, Volume: 267, Issue:3

    Topics: Animals; Binding Sites; Brain; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol Phosphates; Lithium Chloride; Male; Mice; N-Methylscopolamine; Oxadiazoles; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Receptors, Muscarinic; Scopolamine; Scopolamine Derivatives

1994
Discrete activation of transduction pathways associated with acetylcholine m1 receptor by several muscarinic ligands.
    European journal of pharmacology, 1994, Mar-15, Volume: 267, Issue:1

    Topics: Adenylyl Cyclases; Animals; Arachidonic Acid; Calcium; Carbachol; Cells, Cultured; CHO Cells; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Hydrolysis; Phosphatidylinositols; Pilocarpine; Protein Binding; Quinuclidines; Receptors, Cholinergic; Signal Transduction; Thiophenes; Transfection

1994
Aceclidine effects on outflow facility after ciliary muscle disinsertion.
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 1996, Volume: 210, Issue:5

    Topics: Accommodation, Ocular; Animals; Aqueous Humor; Carbachol; Ciliary Body; Cytochalasin B; Dose-Response Relationship, Drug; Gonioscopy; Macaca mulatta; Male; Muscarinic Agonists; Muscle, Smooth; Pilocarpine; Quinuclidines; Trabecular Meshwork

1996
Long-lasting salivation induced by a novel muscarinic receptor agonist SNI-2011 in rats and dogs.
    European journal of pharmacology, 1997, Nov-19, Volume: 339, Issue:1

    Topics: Animals; Dogs; Female; Male; Muscarinic Agonists; Pilocarpine; Quinuclidines; Rats; Rats, Wistar; Salivation; Secretory Rate; Thiophenes; Time Factors

1997
Xanomeline compared to other muscarinic agents on stimulation of phosphoinositide hydrolysis in vivo and other cholinomimetic effects.
    Brain research, 1998, Jun-08, Volume: 795, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain Chemistry; Bridged Bicyclo Compounds, Heterocyclic; Cholinergic Agents; Cholinesterase Inhibitors; Dihydropyridines; Dose-Response Relationship, Drug; Hydrolysis; Hypothermia; Imines; Lithium; Male; Mice; Mice, Inbred Strains; Muscarinic Agonists; Oximes; Parasympathomimetics; Phosphatidylinositols; Physostigmine; Pilocarpine; Pyridines; Quinuclidines; Radioligand Assay; Salivation; Tacrine; Tetrazoles; Thiadiazoles; Tremor

1998
Effects of tachykinin NK1 receptor antagonists on vagal hyperreactivity and neuronal M2 muscarinic receptor function in antigen challenged guinea-pigs.
    British journal of pharmacology, 1998, Volume: 124, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biphenyl Compounds; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Electric Stimulation; Eosinophilia; Guinea Pigs; Lung; Neurokinin A; Neurokinin-1 Receptor Antagonists; Ovalbumin; Peptide Fragments; Pilocarpine; Piperidines; Quinuclidines; Receptor, Muscarinic M2; Receptors, Muscarinic; Receptors, Tachykinin; Specific Pathogen-Free Organisms; Substance P; Trachea; Vagus Nerve

1998
Direct effects of muscarinic agents on the outflow pathways in human eyes.
    Investigative ophthalmology & visual science, 2000, Volume: 41, Issue:7

    Topics: Aged; Anterior Eye Segment; Aqueous Humor; Atropine; Carbachol; Dose-Response Relationship, Drug; Humans; Muscarinic Agonists; Muscarinic Antagonists; Pilocarpine; Quinuclidines; Receptors, Muscarinic

2000
Effects of neurokinin receptor antagonists in virus-infected airways.
    American journal of physiology. Lung cellular and molecular physiology, 2000, Volume: 279, Issue:1

    Topics: Animals; Benzamides; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Electric Stimulation; Female; Guinea Pigs; Leukocyte Count; Leukocytes; Lung; Muscarinic Agonists; Neurokinin-1 Receptor Antagonists; Pilocarpine; Piperidines; Quinuclidines; Receptors, Muscarinic; Receptors, Neurokinin-2; Respirovirus; Respirovirus Infections; Vagus Nerve

2000
Cevimeline (Evoxac) for dry mouth.
    The Medical letter on drugs and therapeutics, 2000, Aug-07, Volume: 42, Issue:1084

    Topics: Acetylcholine; Clinical Trials as Topic; Contraindications; Humans; Intestinal Absorption; Muscarinic Agonists; Nausea; Pilocarpine; Quinuclidines; Thiophenes; Xerostomia

2000
A new medication for treatment of dry mouth in Sjögren's syndrome.
    Texas dental journal, 2001, Volume: 118, Issue:3

    Topics: Contraindications; Humans; Muscarinic Agonists; Pilocarpine; Quinuclidines; Receptors, Muscarinic; Salivary Glands; Salivation; Sjogren's Syndrome; Thiophenes; Xerostomia

2001
Salivary enhancement: current status and future therapies.
    Journal of dental education, 2001, Volume: 65, Issue:10

    Topics: Animals; Aquaporin 1; Aquaporins; Blood Group Antigens; Cholinergic Agents; Cranial Irradiation; Dental Caries; Genetic Therapy; Humans; Parasympathomimetics; Pilocarpine; Quinuclidines; Salivary Glands; Sjogren's Syndrome; Thiophenes; Xerostomia

2001
Assessing salivary gland hypofunction--Part two.
    Practical procedures & aesthetic dentistry : PPAD, 2002, Volume: 14, Issue:3

    Topics: Anti-Infective Agents, Local; Candidiasis, Oral; Dental Caries; Humans; Maltose; Mastication; Muscarinic Agonists; Pilocarpine; Quinuclidines; Saliva; Thiophenes; Xerostomia

2002
[The muscarinic receptor subtype study of the action on lowering IOP of cholinomimetic drugs].
    Yan ke xue bao = Eye science, 2000, Volume: 16, Issue:4

    Topics: Animals; Cholinergic Agents; Female; Intraocular Pressure; Male; Miotics; Muscarinic Agonists; Pilocarpine; Quinuclidines; Rabbits; Receptors, Muscarinic

2000
Effect of SNI-2011 on amylase secretion from parotid tissue in rats and in neuronal nitric oxide synthase knockout mice.
    European journal of pharmacology, 2003, Mar-19, Volume: 464, Issue:2-3

    Topics: Alkaloids; Amylases; Animals; Azepines; Benzoates; Benzylamines; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbazoles; Chelating Agents; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Gallic Acid; Genotype; Guanylate Cyclase; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Mice, Knockout; Molsidomine; Muscarinic Agonists; Myosin-Light-Chain Kinase; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxadiazoles; Parotid Gland; Penicillamine; Phosphodiesterase Inhibitors; Pilocarpine; Protein Kinase Inhibitors; Pyrroles; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Wistar; Sulfonamides; Thiophenes; Type C Phospholipases

2003
Effects of pilocarpine hydrochloride and cevimeline on submandibular/sublingual salivation in rat xerostomia model produced by X-ray irradiation.
    Arzneimittel-Forschung, 2003, Volume: 53, Issue:5

    Topics: Animals; Antipsychotic Agents; Body Temperature; Cardiovascular System; Central Nervous System; Chlorpromazine; Dose-Response Relationship, Drug; Male; Muscarinic Agonists; Pilocarpine; Quinuclidines; Radiation Injuries, Experimental; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Respiratory System; Salivary Proteins and Peptides; Salivation; Submandibular Gland; Thiophenes; Xerostomia

2003
[Future therapy strategies for salivary gland impairment].
    Refu'at ha-peh veha-shinayim (1993), 2004, Volume: 21, Issue:3

    Topics: Amifostine; Cranial Irradiation; Head and Neck Neoplasms; Humans; Muscarinic Agonists; Pilocarpine; Quinuclidines; Radiation Injuries; Radiation-Protective Agents; Regeneration; Saliva; Salivary Glands; Thiophenes

2004
Dentistry. Implications and management of xerostomia in the HIV patient.
    HIV clinician, 2005,Winter, Volume: 17, Issue:1

    Topics: Antiretroviral Therapy, Highly Active; Cholinergic Agents; HIV Infections; HIV Protease Inhibitors; Humans; Pilocarpine; Quinuclidines; Reverse Transcriptase Inhibitors; Thiophenes; Xerostomia

2005
Aceclidine and pilocarpine interact differently with muscarinic receptor in isolated rabbit iris muscle.
    Life sciences, 2006, Feb-28, Volume: 78, Issue:14

    Topics: Animals; Carbachol; Iris; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Pilocarpine; Quinuclidines; Rabbits; Receptors, Muscarinic

2006
New approaches to preventing xerostomia.
    The journal of supportive oncology, 2006, Volume: 4, Issue:2

    Topics: Amifostine; Cytoprotection; Humans; Muscarinic Agonists; Neoplasms; Pilocarpine; Quinuclidines; Radiation Injuries; Radiation-Protective Agents; Radiotherapy Dosage; Radiotherapy, Intensity-Modulated; Salivary Glands; Thiophenes; Xerostomia

2006
[Revision of the recommendations of the Commission on Pharmacotherapy of the German Society for Rheumatology. Recommendations for supportive therapy for Sjögren's syndrome].
    Zeitschrift fur Rheumatologie, 2007, Volume: 66, Issue:1

    Topics: Bromhexine; Cyclosporine; Dry Eye Syndromes; Electric Stimulation Therapy; Expectorants; Humans; Muscarinic Antagonists; Ophthalmic Solutions; Pilocarpine; Quinuclidines; Sjogren's Syndrome; Thiophenes; Xerostomia

2007
Degradation of submandibular gland AQP5 by parasympathetic denervation of chorda tympani and its recovery by cevimeline, an M3 muscarinic receptor agonist.
    American journal of physiology. Gastrointestinal and liver physiology, 2008, Volume: 295, Issue:1

    Topics: Animals; Aquaporin 1; Aquaporin 5; Chorda Tympani Nerve; Gene Expression Regulation; Lysosomes; Male; Muscarinic Agonists; Parasympathectomy; Pilocarpine; Quinuclidines; Rats; Rats, Sprague-Dawley; RNA, Messenger; Submandibular Gland; Sympathectomy; Thiophenes; Time Factors

2008
Effects of pilocarpine and cevimeline on Ca2+ mobilization in rat parotid acini and ducts.
    The journal of medical investigation : JMI, 2009, Volume: 56 Suppl

    Topics: Animals; Calcium; Calcium Signaling; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Pilocarpine; Piperidines; Quinuclidines; Rats; Receptors, Muscarinic; Thiophenes

2009
Distinct effects of cevimeline and pilocarpine on salivary mechanisms, cardiovascular response and thirst sensation in rats.
    Archives of oral biology, 2012, Volume: 57, Issue:4

    Topics: Analysis of Variance; Animals; Cardiovascular System; Drinking; Muscarinic Agonists; Parotid Gland; Pilocarpine; Quinuclidines; Rats; Rats, Wistar; Salivation; Sensitivity and Specificity; Subfornical Organ; Thiophenes; Thirst

2012
Salivary gland ultrasonography as a primary imaging tool for predicting efficacy of xerostomia treatment in patients with Sjögren's syndrome.
    Rheumatology (Oxford, England), 2016, Volume: 55, Issue:2

    Topics: Administration, Oral; Aged; Dose-Response Relationship, Drug; Female; Follow-Up Studies; Glucocorticoids; Humans; Male; Middle Aged; Muscarinic Agonists; Parasympathomimetics; Pilocarpine; Prednisolone; Prognosis; Quinuclidines; Retrospective Studies; Salivary Glands; Severity of Illness Index; Sjogren's Syndrome; Therapeutic Irrigation; Thiophenes; Treatment Outcome; Ultrasonography; Xerostomia

2016
Long-term Use of the Sialogogue Medications Pilocarpine and Cevimeline Can Reduce Xerostomia Symptoms and Increase Salivary Flow in Head and Neck Cancer Survivors After Radiotherapy.
    The journal of evidence-based dental practice, 2017, Volume: 17, Issue:3

    Topics: Head and Neck Neoplasms; Humans; Pilocarpine; Quinuclidines; Survivors; Thiophenes; Xerostomia

2017
Risk of Parkinson disease in Sjögren syndrome administered ineffective immunosuppressant therapies: A nationwide population-based study.
    Medicine, 2019, Volume: 98, Issue:14

    Topics: Adult; Aged; Anti-Inflammatory Agents; Antirheumatic Agents; Comorbidity; Female; Humans; Hydroxychloroquine; Immunosuppression Therapy; Incidence; Male; Methylprednisolone; Middle Aged; Muscarinic Agonists; National Health Programs; Parkinson Disease; Pilocarpine; Quinuclidines; Retrospective Studies; Risk Factors; Sjogren's Syndrome; Taiwan; Thiophenes

2019
Comparing the effectiveness and adverse effects of pilocarpine and cevimeline in patients with hyposalivation.
    Oral diseases, 2019, Volume: 25, Issue:8

    Topics: Adult; Aged; Female; Follow-Up Studies; Humans; Middle Aged; Muscarinic Agonists; Pilocarpine; Quinuclidines; Retrospective Studies; Thiophenes; Time Factors; Xerostomia

2019
Safety and efficacy of pilocarpine, cevimeline, and diquafosol compared to artificial tears for the treatment of dry eye: protocol for a systematic review.
    Systematic reviews, 2022, 05-28, Volume: 11, Issue:1

    Topics: Dry Eye Syndromes; Humans; Lubricant Eye Drops; Meta-Analysis as Topic; Pilocarpine; Polyphosphates; Quinuclidines; Secretagogues; Systematic Reviews as Topic; Thiophenes; Uracil Nucleotides

2022