pilocarpine has been researched along with oxotremorine in 107 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 60 (56.07) | 18.7374 |
1990's | 31 (28.97) | 18.2507 |
2000's | 15 (14.02) | 29.6817 |
2010's | 1 (0.93) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Amstutz, R; Boelsterli, J; Bolliger, G; Floersheim, P; Gammenthaler, H; Gmelin, G; Shapiro, G; Supavilai, P; Walkinshaw, M | 1 |
Fraser, CM; Lai, J; Mei, L; Roeske, WR; Venter, JC; Yamamura, HI | 1 |
Andrews, PR; Craik, DJ; Martin, JL | 1 |
Abuh, YF; Dunbar, PG; Edgar, MA; El-Assadi, AA; Fang, Z; Huzl, JJ; Liu, Y; Messer, WS; Nagy, PI; Ngur, DO; Ojo, B; Periyasamy, S; Rho, T; Roknich, S; Sbeih, S; Zhang, H | 1 |
Bacáková, L; El-Fakahany, EE; Jakubík, J; Tucek, S | 1 |
Bymaster, FP; Calligaro, DO; DeLapp, NW; Fink-Jensen, A; Jeppesen, L; Olesen, PH; Rasmussen, T; Rimvall, K; Sauerberg, P; Shannon, HE; Sheardown, MJ; Swedberg, MD; Thomsen, C; Thøgersen, H; Ward, JS | 1 |
Chen, D; Shan, L; Wang, H; Yang, R; Yun, L; Zhao, R | 1 |
Casida, JE; Honda, H; Tomizawa, M | 1 |
Dei, S; Marconi, C; Pedretti, A; Romanelli, MN; Scapecchi, S; Vistoli, G | 1 |
Bhattarai, D; Cho, NC; Huang, M; Kang, SB; Keum, G; Kim, Y; Pae, AN; Rhim, H; Suk, DH | 1 |
Lamble, AP; Lamble, JW | 1 |
Joh, TH; Lewander, T; Reis, DJ | 1 |
Birdsall, NJ; Burgen, AS; Strange, PG | 1 |
Baroody, RA; Bito, LZ | 1 |
Bentley, GA; Wong, CL | 1 |
Dulis, BH; Gordon, MA; Wilson, IB | 1 |
Hata, F; Lai, RT; Maruno, M; Takeyasu, K; Uchida, S; Wada, A; Yoshida, H | 1 |
Fuller, RW; Molloy, BB; Snoddy, HD | 1 |
Dage, RC | 1 |
Dudar, JD; Hadházy, P; Szerb, JC | 1 |
Boissier, JR; Chermat, R; Simon, P | 1 |
Biggs, DF; Yang, ZJ | 1 |
Hynie, S; Kadlec, O; Masek, K; Seferna, I; Sevcík, J | 1 |
Aksoy, S; Gibson, VA; McKinney, M; Miller, JH; Nickelson, L | 1 |
Boddeke, HW | 1 |
Ebadi, M; Govitrapong, P; Pujito, PP | 1 |
Chapman, MA; See, RE | 1 |
Schimerlik, MI; Tota, MR | 1 |
Bemis, KG; Hendrix, JC; Shannon, HE; Ward, JS | 1 |
Nezu, E; Yoneyama, T; Yoshimura, K | 1 |
Broekkamp, CL; Hagan, JJ; Jansen, JH | 1 |
Hollingsworth, PJ; Smith, CB | 1 |
Ellerbrock, B; Hoss, W; Messer, WS; Price, M | 1 |
Drews, U; Oettling, G; Schmidt, H | 2 |
Imaizumi, T; Misaki, N; Mizushima, A; Osugi, T; Tatebayashi, Y; Uchida, S; Yoshida, H; Zhou, XM | 1 |
Flynn, DD; Palermo, N; Suarez, A | 1 |
Brunner, F; Christophe, J; Gillard, M; Svoboda, M; Waelbroeck, M | 1 |
Cornfeldt, M; Fielding, S; Gorney, B; Locke, KW | 1 |
Esbenshade, TA; Gerald, MC; Kolta, MG; Ordway, GA; Wallace, LJ | 1 |
Baux, G; Fossier, P; Poulain, B; Tauc, L | 1 |
DeGeorge, JJ; Lapetina, EG; McCarthy, KD; Morell, P | 1 |
Channell, SL; Iversen, SD; Lalies, MD; Salamone, JD | 1 |
Costa, L; Jung, M; Kelly, PH; Shearman, GT | 1 |
Camus, J; Christophe, J; De Neef, P; Fourmy, D; Pradayrol, L; Robberecht, P; Scemama, JL; Tastenoy, M; Vaysse, N; Waelbroeck, M | 1 |
Löschmann, PA; Pietzuch, P; Wachtel, H | 1 |
Gies, JP; Landry, Y | 1 |
Drews, U; Oettling, G; Schmidt, H; Show-Klett, A | 1 |
Alvarado-Garcia, R; Lee, MA; Witkin, JM; Witkin, KM | 1 |
Christophe, J; Gillard, M; Waelbroeck, M | 1 |
Chrachri, A; Clarac, F | 1 |
Bartfai, T; Hedlund, B | 1 |
Kilbinger, H; Nafziger, M | 1 |
Ahlenius, S; Larsson, K | 1 |
Barker, DL; Mpitsos, GJ; Murray, TF; Siebenaller, JF | 1 |
Fujimoto, JM; Ishii, TK; Lange, DG; Quock, RM | 1 |
Konno, F; Takayanagi, I | 1 |
Higuchi, H; Kagiya, T; Matsumoto, K; Mizushima, A; Osugi, T; Uchida, S; Yoshida, H; Zhou, XM | 1 |
Snyder, SH; Yamamura, HI | 1 |
Lindström, LH | 2 |
Bhargava, AK; Bhargava, KP; Tangri, KK | 1 |
Hamilton, TC | 1 |
Leaf, RC; Wnek, DJ | 1 |
Cheng, HC; Long, JP | 1 |
Brase, DA; Loh, HH; Tseng, LF; Way, EL | 1 |
Fozard, JR; Muscholl, E | 1 |
Hauser, G; Parks, JM | 1 |
Asselin, J; Christophe, J; de Neef, P; Robberecht, P; Waelbroeck, M | 1 |
Jedrych, Z | 1 |
Bättig, K; Driscoll, P; Martin, JR; Overstreet, DH | 1 |
Huger, FP; Smith, CP | 1 |
Coppi, G; Leone, L; Lumachi, B; Rossini, L; Valsecchi, B | 1 |
Glick, SD; Guido, RA | 1 |
Klein, WL; Shifrin, GS | 1 |
Ellis, J; Hoss, W | 1 |
Birmingham, AT; Harriss, DR; Hill, SJ; Marsh, KA | 1 |
Honda, K; Kamiya, H; Takano, Y | 1 |
Bratt, AM; Cassel, JC; Greene, PL; Jeltsch, H; Kelche, C; Will, BE | 1 |
Freedman, SB; Patel, S | 1 |
Bernard, V; Bloch, B; Dumartin, B; Lamy, E | 1 |
Clement, JG | 1 |
Castoldi, AF; Costa, LG; Tang, C | 1 |
Habecker, BA; Nathanson, NM; Wang, H | 1 |
Cristi, C; Raithby, A; Snider, M; Tanner, C; Vanderwolf, CH | 1 |
De Neef, P; Domenach, V; Vandermeers, A; Vandermeers-Piret, MC; Waelbroeck, M | 1 |
Matsumoto, K; Murakami, Y; Ohta, H; Watanabe, H | 1 |
Coffin, VL; Cohen-Williams, M; Kistler, MK; Smith, RD | 1 |
Björklund, M; Jäkälä, P; Koivisto, E; Riekkinen, P | 1 |
Edwardson, JM; Koenig, JA; Szekeres, PG | 1 |
Gebauer, M; Versen, B | 1 |
Bymaster, FP; Calligaro, DO; Delapp, NW; Fink-Jensen, A; Jeppesen, L; Kristensen, P; Rasmusseen, T; Sauerberg, P; Shannon, HE; Sheardown, MJ; Thomsen, C; Ward, JS; Whitesitt, C | 1 |
Jaen, JC; Mirzadegan, T; Moreland, D; Schwarz, RD; Spencer, CJ; Tecle, H; Thomas, AJ | 1 |
Gebauer, M; Schipp, R; Versen, B | 1 |
Curtis, CA; Hulme, EC; Ward, SD | 1 |
Guarente, L; Hawdon, J; Hotez, P; Perregaux, M; Ruvkun, G; Tissenbaum, HA | 1 |
Bymaster, FP; Calligaro, DO; DeLapp, NW; Fink-Jensen, A; Jeppesen, L; Nielsen, EB; Rasmussen, T; Sauerberg, P; Shannon, HE; Sheardown, MJ; Swedberg, MD; Thomsen, C; Ward, JS; Whitesitt, C | 1 |
Shannon, HE; Womer, DE | 1 |
Anagnostaras, SG; Feigl, EO; Hamilton, SE; Hardouin, SN; Murphy, GG; Nathanson, NM; Richmond, KN; Silva, AJ | 1 |
Choppin, A; Eglen, RM | 1 |
Bymaster, FP; Calligaro, DO; Carter, PA; DeLapp, NW; Felder, CC | 1 |
Cunha, GM; Farias, PA; Viana, GS | 1 |
Goodhead, LH; Mitchell, SN; Moss, S; Sharott, A | 1 |
Bymaster, FP; Carter, PA; Felder, CC; Gomeza, J; Hamilton, SE; McKinzie, DL; Nathanson, NM; Wess, J; Yamada, M | 1 |
Luo, ZP; Wan, Q; Wang, H | 1 |
Carnicella, S; Oberling, P; Pain, L | 1 |
Aguiar, LM; Fonteles, MM; Freitas, RM; Nascimento, VS; Nogueira, CR; Oliveira, AA; Sousa, FC; Viana, GS | 1 |
1 review(s) available for pilocarpine and oxotremorine
Article | Year |
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The therapeutic use of cholinergic drugs acting on the vegetative nervous system. I - Direct, indirect and mixed agonists.
Topics: Animals; Arecoline; Bethanechol Compounds; Carbachol; Chemical Phenomena; Chemistry; Dimethylphenylpiperazinium Iodide; Ganglia; Kinetics; Lobeline; Neuroeffector Junction; Nicotine; Oxotremorine; Parasympathomimetics; Pilocarpine; Stereoisomerism | 1981 |
106 other study(ies) available for pilocarpine and oxotremorine
Article | Year |
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Muscarinic activity of the thiolactone, lactam, lactol, and thiolactol analogues of pilocarpine and a hypothetical model for the binding of agonists to the m1 receptor.
Topics: Animals; Binding, Competitive; Crystallography; Guinea Pigs; Lactams; Male; Mice; Models, Biological; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Sulfhydryl Compounds | 1992 |
Pharmacological characterization of the M1 muscarinic receptors expressed in murine fibroblast B82 cells.
Topics: Alprostadil; Animals; Carbachol; Cells, Cultured; Cyclic AMP; Fibroblasts; Inositol Phosphates; Mice; Parasympatholytics; Pertussis Toxin; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1989 |
Functional group contributions to drug-receptor interactions.
Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship | 1984 |
Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
Topics: Animals; Arecoline; Brain; Carbachol; Cell Line; Models, Molecular; Muscarinic Agonists; Phosphatidylinositols; Pyrimidines; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship | 1997 |
Positive cooperativity of acetylcholine and other agonists with allosteric ligands on muscarinic acetylcholine receptors.
Topics: Acetylcholine; Allosteric Regulation; Animals; Binding, Competitive; CHO Cells; Cricetinae; Ligands; Muscarinic Agonists; N-Methylscopolamine; Receptors, Muscarinic; Scopolamine Derivatives | 1997 |
Muscarinic agonists with antipsychotic-like activity: structure-activity relationships of 1,2,5-thiadiazole analogues with functional dopamine antagonist activity.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Brain; Dopamine Antagonists; Drug Evaluation, Preclinical; In Vitro Techniques; Injections, Subcutaneous; Male; Mice; Models, Molecular; Molecular Conformation; Motor Activity; Muscarinic Agonists; Rats; Rats, Sprague-Dawley; Salivation; Stereoisomerism; Structure-Activity Relationship; Thiadiazoles; Tremor | 1998 |
Discovering selective agonists of endothelial target for acetylcholine (ETA) via diversity-guided pharmacophore simplification and simulation.
Topics: Acetylcholine; Animals; Aorta; Endothelium, Vascular; Guinea Pigs; Muscarinic Agonists; Rabbits; Rats; Vasodilation | 2004 |
Insect muscarinic acetylcholine receptor: pharmacological and toxicological profiles of antagonists and agonists.
Topics: Animals; Brain; Drosophila; Houseflies; Insecta; Muscarinic Agonists; Muscarinic Antagonists; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tritium | 2007 |
Docking analyses on human muscarinic receptors: unveiling the subtypes peculiarities in agonists binding.
Topics: Binding Sites; Computer Simulation; Humans; Ligands; Muscarinic Agonists; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M5; Receptors, Muscarinic | 2008 |
Synthesis and biological evaluation of isoxazoline derivatives as potent M₁ muscarinic acetylcholine receptor agonists.
Topics: Dose-Response Relationship, Drug; Humans; Isoxazoles; Molecular Structure; Receptor, Muscarinic M1; Structure-Activity Relationship | 2015 |
The effect of miotics on the intraocular pressure of conscious owl monkeys.
Topics: Anesthesia, Local; Animals; Aotus trivirgatus; Carbachol; Dose-Response Relationship, Drug; Haplorhini; Intraocular Pressure; Male; Miotics; Oxotremorine; Parasympathomimetics; Pilocarpine; Quinuclidines; Spiro Compounds; Succinimides; Tonometry, Ocular | 1976 |
Tyrosine hydroxylase: delayed activation in central noradrenergic neurons and induction in adrenal medulla elicited by stimulation of central cholinergic receptors.
Topics: Adrenal Medulla; Animals; Atropine; Brain; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Male; Nicotine; Oxotremorine; Physostigmine; Pilocarpine; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Tyrosine 3-Monooxygenase | 1977 |
Occupancy of muscarinic acetylcholine receptors stimulates a guanylate cyclase in neuroblastoma cells.
Topics: Acetylcholine; Atropine; Carbachol; Cell Line; Cell Membrane; Enzyme Activation; Guanylate Cyclase; Kinetics; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic | 1977 |
Gradual changes in the sensitivity of rhesus monkey eyes to miotics and the dependence of these changes on the regimen of topical cholinesterase inhibitor treatment.
Topics: Accommodation, Ocular; Age Factors; Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Resistance; Echothiophate Iodide; Female; Haplorhini; Iris; Isoflurophate; Macaca mulatta; Miotics; Oxotremorine; Photic Stimulation; Pilocarpine; Reflex, Pupillary; Time Factors | 1979 |
Further studies on the role of cholinergic mechanisms in the development of increased naloxone potency in mice.
Topics: Abdominal Muscles; Animals; Atropine; Drug Synergism; Humans; Male; Mice; Morphine; Motor Activity; Muscle Contraction; Naloxone; Nociceptors; Oxotremorine; Pilocarpine; Substance Withdrawal Syndrome | 1979 |
Identification of muscarinic binding sites in human neutrophils by direct binding.
Topics: Atropine; Benzilates; Binding, Competitive; Humans; In Vitro Techniques; Kinetics; Neutrophils; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic | 1979 |
Experimental evidence and dynamic aspects of spare receptor.
Topics: Animals; Bethanechol Compounds; Binding Sites; Dibenzylchlorethamine; Guinea Pigs; Ileum; In Vitro Techniques; Methacholine Compounds; Mice; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Drug | 1979 |
Effect of cholinomimetic drugs in combination with amfonelic acid or spiperone on the concentration of 3,4-dihydroxyphenylacetic acid in rat brain.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain Chemistry; Butyrophenones; Drug Interactions; Male; Nalidixic Acid; Naphthyridines; Oxotremorine; Parasympathomimetics; Phenylacetates; Pilocarpine; Rats; Spiperone | 1978 |
A centrally mediated prolonged hypotension produced by oxotremorine or pilocarpine.
Topics: Animals; Arecoline; Blood Pressure; Cardiac Output; Cats; Central Nervous System; Decerebrate State; Depression, Chemical; Dogs; Female; Heart Rate; Male; Oxotremorine; Pilocarpine; Spinal Cord; Sympathetic Nervous System | 1979 |
Release of [3H]acetylcholine from rat hippocampal slices: effect of septal lesion and of graded concentrations of muscarnic agonists and antagonists.
Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Carbachol; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Mecamylamine; Oxotremorine; Pilocarpine; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Septum Pellucidum | 1977 |
Interaction of atropine or methylatropinium with four effects of two cholinergic drugs.
Topics: Animals; Atropine; Atropine Derivatives; Blepharoptosis; Drug Interactions; Ganglionic Stimulants; Male; Mice; Motor Activity; Oxotremorine; Pilocarpine; Reaction Time; Reserpine | 1976 |
Muscarinic receptors and parasympathetic neurotransmission in guinea-pig trachea.
Topics: Animals; Arecoline; Bethanidine; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Muscarinic Antagonists; Oxotremorine; Parasympathetic Nervous System; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Synaptic Transmission; Trachea | 1991 |
Non-synaptic cholinergic modulation of neurogenic twitches of the guinea-pig ileum.
Topics: Acetylcholine; Action Potentials; Adenylyl Cyclases; Animals; Atropine; Calcium; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ouabain; Oxotremorine; Parasympathetic Nervous System; Pilocarpine; Pirenzepine; Potassium; Synapses | 1991 |
Interactions of agonists with M2 and M4 muscarinic receptor subtypes mediating cyclic AMP inhibition.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Cells, Cultured; CHO Cells; Corpus Striatum; Cricetinae; Cyclic AMP; Kinetics; Male; Muscarine; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1991 |
Different effects of muscarinic agonists in rat superior cervical ganglion and hippocampal slices.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Ganglia, Sympathetic; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pilocarpine; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains | 1991 |
Inhibitory actions of muscarinic cholinergic receptor agonists on serotonin N-acetyltransferase in bovine pineal explants in culture.
Topics: Animals; Arylamine N-Acetyltransferase; Carbachol; Cattle; Kinetics; Methacholine Chloride; Organ Culture Techniques; Oxotremorine; Parasympathomimetics; Pilocarpine; Pineal Gland; Receptors, Muscarinic | 1991 |
Cholinergic modulation of oral activity in drug-naive and chronic haloperidol-treated rats.
Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Fourier Analysis; Haloperidol; Male; Mouth; Movement; Oxotremorine; Parasympathetic Nervous System; Parasympathomimetics; Physostigmine; Pilocarpine; Rats; Rats, Inbred Strains; Scopolamine | 1991 |
Partial agonist effects on the interaction between the atrial muscarinic receptor and the inhibitory guanine nucleotide-binding protein in a reconstituted system.
Topics: Animals; Carbachol; GTP Phosphohydrolases; GTP-Binding Proteins; Heart Atria; Kinetics; Oxotremorine; Phosphoric Monoester Hydrolases; Pilocarpine; Receptors, Cholinergic; Structure-Activity Relationship; Swine | 1990 |
Interactions between scopolamine and muscarinic cholinergic agonists or cholinesterase inhibitors on spatial alternation performance in rats.
Topics: Animals; Arecoline; Behavior, Animal; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Memory; Oxotremorine; Parasympathomimetics; Physostigmine; Pilocarpine; Rats; Rats, Inbred F344; Scopolamine; Spatial Behavior; Succinimides; Tacrine | 1990 |
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains | 1985 |
Hemicholinium-3 impairs spatial learning and the deficit is reversed by cholinomimetics.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Arecoline; Cholinesterase Inhibitors; Discrimination Learning; Hemicholinium 3; Learning; Male; Oxotremorine; Parasympathomimetics; Physostigmine; Pilocarpine; Rats; Space Perception; Tetrahydronaphthalenes | 1989 |
Effects of muscarinic receptor agonists and antagonists on alpha 2-adrenoceptors in rat brain.
Topics: Animals; Atropine; Atropine Derivatives; Brain; Clonidine; Male; N-Methylscopolamine; Neurons; Oxotremorine; Parasympatholytics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Scopolamine; Scopolamine Derivatives; Time Factors | 1989 |
Autoradiographic analyses of agonist binding to muscarinic receptor subtypes.
Topics: Animals; Arecoline; Autoradiography; Bethanechol; Bethanechol Compounds; Binding Sites; Brain; Oxotremorine; Parasympathomimetics; Pilocarpine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic | 1989 |
An embryonic Ca++ mobilizing muscarinic system in the chick embryo heart.
Topics: Animals; Benzofurans; Bethanechol; Bethanechol Compounds; Calcium; Carbachol; Chick Embryo; Chlortetracycline; Female; Fura-2; Heart; Heart Rate, Fetal; In Vitro Techniques; Methacholine Chloride; Methacholine Compounds; Oxotremorine; Parasympathomimetics; Pilocarpine; Pregnancy; Receptors, Muscarinic | 1989 |
The H-L subgroup of guinea-pig cardiac M2 receptors (M2 beta) regulates inositol phosphate formation.
Topics: Acetylcholine; Adenylate Cyclase Toxin; Animals; Carbachol; Guinea Pigs; Hydrolysis; In Vitro Techniques; Inositol Phosphates; Male; Myocardium; Oxotremorine; Pertussis Toxin; Pilocarpine; Receptors, Muscarinic; Virulence Factors, Bordetella | 1989 |
Agonist binding to M1 muscarinic receptors is sensitive to guanine nucleotides.
Topics: Animals; Carbachol; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Indicators and Reagents; Kinetics; Male; Methacholine Compounds; Oxotremorine; Pilocarpine; Pirenzepine; Rabbits; Receptors, Muscarinic; Second Messenger Systems | 1989 |
Bretylium tosylate binds preferentially to muscarinic receptors labelled with [3H]oxotremorine M (SH or 'high affinity' receptors) in rat heart and brain cortex.
Topics: Animals; Bretylium Compounds; Bretylium Tosylate; Cerebral Cortex; Guanosine Triphosphate; Heart; In Vitro Techniques; Male; Membranes; Myocardium; N-Methylscopolamine; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives | 1989 |
Characterization of the discriminative stimulus effects of physostigmine in the rat.
Topics: Animals; Arecoline; Avoidance Learning; Discrimination, Psychological; Male; Oxotremorine; Physostigmine; Pilocarpine; Rats; Rats, Inbred F344 | 1989 |
The muscarinic receptor of chick embryo cells: correlation between ligand binding and calcium mobilization.
Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Binding, Competitive; Calcium; Carbachol; Chick Embryo; Dose-Response Relationship, Drug; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Spectrometry, Fluorescence | 1985 |
Effect of age on cholinergic muscarinic responsiveness and receptors in the rat urinary bladder.
Topics: Acetylcholine; Aging; Animals; Atropine; Bethanechol; Bethanechol Compounds; Male; Muscle Contraction; Muscle, Smooth; Oxotremorine; Parasympathomimetics; Phenylmethylsulfonyl Fluoride; Physostigmine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred F344; Receptors, Muscarinic; Urinary Bladder | 1986 |
Both presynaptic nicotinic-like and muscarinic-like autoreceptors regulate acetylcholine release at an identified neuro-neuronal synapse of Aplysia.
Topics: Acetylcholine; Animals; Aplysia; Carbachol; Curare; Hexamethonium; Hexamethonium Compounds; Muscarine; Oxotremorine; Pilocarpine; Receptors, Muscarinic; Receptors, Nicotinic; Synapses | 1988 |
Cholinergic stimulation of arachidonic acid and phosphatidic acid metabolism in C62B glioma cells.
Topics: Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Atropine; Calcimycin; Carbachol; Cell Line; Glioma; Oxotremorine; Parasympathomimetics; Phosphatidic Acids; Pilocarpine; Rats; Time Factors; Tubocurarine | 1986 |
Behavioural and pharmacological characterization of the mouth movements induced by muscarinic agonists in the rat.
Topics: Animals; Arecoline; Brain; Carbachol; Male; Motor Activity; Mouth; Oxotremorine; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Scopolamine | 1986 |
Discriminative stimulus properties of muscarinic agonists.
Topics: Animals; Arecoline; Discrimination Learning; Male; Oxotremorine; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine | 1987 |
Characterization of muscarinic receptors in human pancreatic membranes.
Topics: Carbachol; Cell Membrane; Humans; Oxotremorine; Pancreas; Pilocarpine; Pirenzepine; Receptors, Muscarinic | 1988 |
Absence of anticholinergic activity of rolipram, an antidepressant with a novel mechanism of action, in three different animal models in vivo.
Topics: Animals; Antidepressive Agents; Body Temperature; Female; Mice; Oxotremorine; Parasympatholytics; Pilocarpine; Pyrrolidinones; Rolipram; Salivation; Tremor | 1988 |
Sialic acid is selectively involved in the interaction of agonists with M2 muscarinic acetylcholine receptors.
Topics: Animals; Atropine; Binding, Competitive; Carbachol; Cell Membrane; Kinetics; Male; Myocardium; Neuraminidase; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Sialic Acids | 1988 |
Expression of the Ca2+ mobilizing muscarinic system in the chick embryo correlates with morphogenesis.
Topics: Acetylcholine; Animals; Calcium; Chick Embryo; Ligands; Morphogenesis; Oxotremorine; Pilocarpine; Receptors, Muscarinic; Spectrometry, Fluorescence | 1988 |
Nonmuscarinic neurotoxicity of oxotremorine.
Topics: Animals; Arecoline; Atropine; Atropine Derivatives; Benactyzine; Benztropine; Crying; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Male; Mecamylamine; Nervous System; Nicotine; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Salivation; Scopolamine; Seizures; Time Factors | 1987 |
Muscarinic receptor heterogeneity in rat central nervous system. II. Brain receptors labeled by [3H]oxotremorine-M correspond to heterogeneous M2 receptors with very high affinity for agonists.
Topics: Animals; Binding, Competitive; Brain; Carbachol; Cerebral Cortex; Kinetics; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives | 1987 |
Induction of rhythmic activity in motoneurons of crayfish thoracic ganglia by cholinergic agonists.
Topics: Animals; Astacoidea; Electrophysiology; Ganglia; Membrane Potentials; Motor Neurons; Oxotremorine; Pilocarpine | 1987 |
Determination of thermodynamic constants for agonist binding to muscarinic receptors from rat cerebral cortex.
Topics: Acetylcholine; Animals; Carbachol; Cerebral Cortex; Kinetics; Male; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thermodynamics | 1987 |
Two types of neuronal muscarine receptors modulating acetylcholine release from guinea-pig myenteric plexus.
Topics: Acetylcholine; Animals; Benzodiazepinones; Guinea Pigs; Ileum; In Vitro Techniques; Muscarine; Muscle Contraction; Myenteric Plexus; Oxotremorine; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Scopolamine | 1985 |
Central muscarinic receptors and male rat sexual behavior: facilitation by oxotremorine but not arecoline or pilocarpine in methscopolamine pretreated animals.
Topics: Animals; Arecoline; Dose-Response Relationship, Drug; Female; Male; N-Methylscopolamine; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Sexual Behavior, Animal | 1985 |
Characterization of muscarinic cholinergic receptors in the crab nervous system.
Topics: Animals; Arecoline; Binding, Competitive; Brachyura; Carbachol; Decamethonium Compounds; Kinetics; Male; Mathematics; Nervous System; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Stereoisomerism; Tissue Distribution; Tubocurarine | 1986 |
Microwave facilitation of methylatropine antagonism of central cholinomimetic drug effects.
Topics: Animals; Atropine Derivatives; Blood-Brain Barrier; Male; Mice; Microwaves; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pilocarpine | 1986 |
Muscarinic acetylcholine receptors in the rabbit ciliary body smooth muscle: spare receptors and threshold phenomenon.
Topics: Animals; Arecoline; Atropine; Carbachol; Ciliary Body; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Oxotremorine; Phenoxybenzamine; Pilocarpine; Rabbits; Receptors, Muscarinic | 1985 |
Multiple agonist binding sites of muscarinic acetylcholine receptors and their relation to the negative inotropic action of agonists in guinea-pig heart.
Topics: Animals; Binding Sites; Carbachol; Depression, Chemical; Dithionitrobenzoic Acid; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Myocardial Contraction; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1985 |
Muscarinic cholinergic binding in rat brain.
Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Binding Sites; Binding, Competitive; Brain; Brompheniramine; Carbachol; Chlorpheniramine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Microsomes; Mitochondria; Oxotremorine; Pilocarpine; Quaternary Ammonium Compounds; Quinuclidines; Rats; Receptors, Cholinergic; Scopolamine; Temperature; Time Factors; Tritium | 1974 |
The effect of pilocarpine and oxotremorine on hormone-activated copulatory behavior in the ovariectomized hamster.
Topics: Animals; Atropine; Castration; Cricetinae; Estradiol; Female; Fenclonine; Lordosis; Male; Ovary; Oxotremorine; Pilocarpine; Progesterone; Rats; Reserpine; Sexual Behavior, Animal | 1972 |
Interrelation between monoaminergic and cholinergic mechanisms in the hypothalamic thermoregulatory centre of rabbits.
Topics: Acetylcholine; Animals; Atropine; Biogenic Amines; Body Temperature Regulation; Carbachol; Cerebral Ventricles; Dopamine; Dose-Response Relationship, Drug; Epinephrine; Female; Hypothalamus; Injections; Male; Norepinephrine; Oxotremorine; Parasympathetic Nervous System; Phenoxybenzamine; Physostigmine; Pilocarpine; Propranolol; Rabbits; Receptors, Cholinergic; Serotonin; Time Factors; Tubocurarine | 1974 |
Comparison of the vasodilator activity of acetylcholine, cholinomimetics and other vasodilators in two vascular beds of the cat.
Topics: Abdomen; Acetylcholine; Animals; Arecoline; Atropine; Blood Pressure; Cats; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Hindlimb; Histamine; Injections, Intra-Arterial; Isoproterenol; Male; Neostigmine; Oxotremorine; Papaverine; Parasympathomimetics; Perfusion; Pilocarpine; Regional Blood Flow; Vascular Resistance; Vasodilator Agents | 1974 |
Further studies on cholinergic mechanisms and hormone-activated copulatory behaviour in the female rat.
Topics: Adrenalectomy; Animals; Atropine; Castration; Copulation; Dexamethasone; Estradiol; Female; Hypophysectomy; Oxotremorine; Pilocarpine; Pituitary-Adrenal System; Progesterone; Rats; Scopolamine; Sexual Behavior, Animal; Stimulation, Chemical | 1973 |
Effects of cholinergic drugs on prey-killing by rodents.
Topics: Aggression; Animals; Appetitive Behavior; Arecoline; Atropine; Dose-Response Relationship, Drug; Humans; Male; Methacholine Compounds; Neostigmine; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Pilocarpine; Rats; Receptors, Cholinergic; Scopolamine | 1973 |
Dopaminergic nature of apomorphine-induced pecking in pigeons.
Topics: Animals; Apomorphine; Aporphines; Behavior, Animal; Chlorpromazine; Columbidae; Dihydroxyphenylalanine; Dioxoles; Dopamine; Haloperidol; Imipramine; Methyltyrosines; Nicotine; Oxotremorine; Phentolamine; Physostigmine; Pilocarpine; Propranolol; Receptors, Drug; Reserpine; Serotonin; Time Factors | 1974 |
Cholinergic modification of naloxone-induced jumping in morphine dependent mice.
Topics: Animals; Arecoline; Atropine; Behavior, Animal; Benztropine; Brain Chemistry; Dimethylphenylpiperazinium Iodide; Humans; Lobeline; Male; Mecamylamine; Mice; Mice, Inbred ICR; Morphine Dependence; Naloxone; Nicotine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pempidine; Physostigmine; Pilocarpine; Tremorine; Tritium | 1974 |
Effects of several muscarinic agonists on cardiac performance and the release of noradrenaline from sympathetic nerves of the perfused rabbit heart.
Topics: Acetylcholine; Animals; Atropine; Carbachol; Carbamates; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Female; Heart; Heart Rate; Hexamethonium Compounds; In Vitro Techniques; Male; Methacholine Compounds; Norepinephrine; Oxotremorine; Parasympathomimetics; Perfusion; Pilocarpine; Quaternary Ammonium Compounds; Rabbits; Sympathetic Nervous System | 1972 |
Evidence from phospholipid metabolism changes for muscarinic cholinergic receptors on rat anterior pituitary cells.
Topics: Animals; Carbachol; Culture Techniques; Male; Membrane Lipids; Oxotremorine; Phospholipids; Pilocarpine; Pituitary Gland, Anterior; Rats; Receptors, Muscarinic | 1983 |
Effect of pH on binding of agonists and antagonists to rat heart muscarinic receptors.
Topics: Animals; Atropine; Carbachol; Cell Membrane; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Models, Biological; Myocardium; Oxotremorine; Parasympathomimetics; Pilocarpine; Rats; Receptors, Muscarinic; Scopolamine; Solanaceous Alkaloids | 1983 |
Cholinolytic activity of 3-hydroxyquinuclidyl-1-phenyl-1-cyclohexyl-1-carboxylate hydrochloride (ANC-821).
Topics: Acetylcholine; Animals; Atropine; Bronchi; Electrocardiography; In Vitro Techniques; Male; Mice; Muscle Contraction; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Rats; Rats, Inbred Strains | 1983 |
Effects of scopolamine, pilocarpine, and oxotremorine on the exploratory behavior of two psychogenetically selected lines of rats in a complex maze.
Topics: Animals; Exploratory Behavior; Learning; Male; Motor Activity; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Scopolamine | 1981 |
Effect of zinc on [3H]-QNB displacement by cholinergic agonists and antagonists.
Topics: Acetylcholine; Animals; Arecoline; Atropine; Binding, Competitive; Male; Oxotremorine; Parasympatholytics; Parasympathomimetics; Physostigmine; Pilocarpine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Zinc | 1983 |
Scopolamine self-administration: cholinergic involvement in reward mechanisms.
Topics: Animals; Arecoline; Atropine; Behavior, Animal; Female; Mecamylamine; N-Methylscopolamine; Oxotremorine; Parasympathetic Nervous System; Physostigmine; Pilocarpine; Rats; Rats, Inbred Strains; Reinforcement, Psychology; Reward; Scopolamine; Scopolamine Derivatives; Self Administration | 1982 |
Regulation of muscarinic acetylcholine receptor concentration in cloned neuroblastoma cells.
Topics: Acetylcholine; Animals; Arecoline; Carbachol; Cell Line; Clone Cells; Dose-Response Relationship, Drug; Kinetics; Mice; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic | 1980 |
Analysis of regional variations in the affinities of muscarinic agonists in the rat brain.
Topics: Animals; Atropine; Binding, Competitive; Brain; Carbachol; Male; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1980 |
Expression of muscarinic M3-receptors coupled to inositol phospholipid hydrolysis in human detrusor cultured smooth muscle cells.
Topics: Carbachol; Cells, Cultured; Diamines; Humans; Hydrolysis; Inositol Phosphates; Methacholine Chloride; Muscarinic Agonists; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Urinary Bladder | 1995 |
The mechanism of muscarinic agonist-stimulated inositol phosphate formation in permeabilized ileal smooth muscle.
Topics: Acetylcholine; Animals; Calcium; Carbachol; Dose-Response Relationship, Drug; Drug Synergism; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrolysis; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Pilocarpine; Substrate Specificity; Time Factors; Type C Phospholipases | 1994 |
Differential behavioral effects of supracallosal and infracallosal lesions of the septohippocampal pathways: no ameliorative effects of oxotremorine or pilocarpine on radial-maze performance.
Topics: Afferent Pathways; Animals; Behavior, Animal; Corpus Callosum; Female; Hippocampus; Maze Learning; Neural Pathways; Oxotremorine; Pilocarpine; Rats; Septum Pellucidum | 1994 |
The muscarinic receptor agonist L-658,903 modulates the in vivo accumulation of inositol monophosphates in mouse brain.
Topics: Animals; Binding Sites; Brain; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol Phosphates; Lithium Chloride; Male; Mice; N-Methylscopolamine; Oxadiazoles; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Receptors, Muscarinic; Scopolamine; Scopolamine Derivatives | 1994 |
Fos immunoreactivity after stimulation or inhibition of muscarinic receptors indicates anatomical specificity for cholinergic control of striatal efferent neurons and cortical neurons in the rat.
Topics: Acetylcholine; Animals; Atropine; Corpus Striatum; Male; Muscarinic Antagonists; Neurons, Efferent; Oxotremorine; Pilocarpine; Prosencephalon; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic | 1993 |
Chromodacryorrhea in rats: absence following soman poisoning.
Topics: Acetylcholinesterase; Animals; Brain; Carbachol; Carboxylesterase; Carboxylic Ester Hydrolases; Harderian Gland; Lacrimal Apparatus Diseases; Male; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Pilocarpine; Rats; Rats, Sprague-Dawley; Soman | 1994 |
Effects of the muscarinic agonist oxotremorine on membrane fluidity in rat lymphocytes.
Topics: Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Fluorescence Polarization; Lymphocytes; Male; Membrane Fluidity; Oxotremorine; Pilocarpine; Rats; Rats, Sprague-Dawley; Scopolamine; Spleen | 1993 |
Multiple second-messenger pathways mediate agonist regulation of muscarinic receptor mRNA expression.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Chick Embryo; Cyclic AMP; Enzyme Activation; Gene Expression Regulation; Heart; Myocardium; Oxotremorine; Pertussis Toxin; Pilocarpine; Receptors, Muscarinic; RNA, Messenger; Second Messenger Systems; Type C Phospholipases; Virulence Factors, Bordetella | 1993 |
Effects of some cholinergic agonists on neocortical slow wave activity in rats with basal forebrain lesions.
Topics: Animals; Arecoline; Body Temperature; Brain; Cerebral Cortex; Dose-Response Relationship, Drug; Electroencephalography; Kainic Acid; Male; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pilocarpine; Prosencephalon; Rats; Scopolamine Derivatives; Tacrine | 1993 |
Binding of the labelled muscarinic toxin 125I-MT1 to rat brain muscarinic M1 receptors.
Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Elapid Venoms; Furans; Gallamine Triethiodide; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Naphthalenes; Oxotremorine; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Protein Binding; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Membranes; Tubocurarine | 1996 |
Effects of oxotremorine and pilocarpine on striatal acetylcholine release as studied by brain dialysis in anesthetized rats.
Topics: Acetylcholine; Anesthesia, General; Animals; Brain Chemistry; Choline; Dose-Response Relationship, Drug; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Oxotremorine; Pilocarpine; Pirenzepine; Rats; Rats, Wistar; Receptors, Presynaptic | 1996 |
Cholinergic improvement of a naturally-occurring memory deficit in the young rat.
Topics: Animals; Animals, Newborn; Avoidance Learning; Cholinergic Agents; Dose-Response Relationship, Drug; Male; Memory; Nicotine; Oxotremorine; Pilocarpine; Rats; Rats, Sprague-Dawley; Reaction Time; Tacrine | 1996 |
The effects of cholinergic drugs on rat neocortical high-voltage spindles in ketanserin-treated rats.
Topics: Animals; Cerebral Cortex; Electroencephalography; Ketanserin; Male; Oxotremorine; Physostigmine; Pilocarpine; Rats; Rats, Wistar | 1996 |
The relationship between agonist intrinsic activity and the rate of endocytosis of muscarinic receptors in a human neuroblastoma cell line.
Topics: Arecoline; Bethanechol; Carbachol; Endocytosis; Humans; Kinetics; Ligands; Methacholine Chloride; Muscarinic Agonists; Neuroblastoma; Oxotremorine; Pilocarpine; Receptor, Muscarinic M3; Receptors, Muscarinic; Tumor Cells, Cultured | 1998 |
Cholinergic mechanisms in the neurocontrol of the branchial heart of the cephalopod Sepia officinalis L.
Topics: Acetylcholine; Animals; Arecoline; Branchial Region; Bungarotoxins; Carbachol; Dose-Response Relationship, Drug; Heart; Hexamethonium; Mollusca; Muscarine; Nicotine; Oxotremorine; Pilocarpine; Receptors, Cholinergic; Tetraethylammonium; Tubocurarine | 1998 |
Muscarinic agonists exhibit functional dopamine antagonism in unilaterally 6-OHDA lesioned rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antibodies; Antipsychotic Agents; Brain Chemistry; Bridged Bicyclo Compounds; Cholinergic Fibers; Dopamine; Dopamine Agonists; Dopamine Antagonists; Male; Muscarinic Agonists; Oxidopamine; Oxotremorine; Parasympathomimetics; Pilocarpine; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Substantia Nigra; Succinimides; Sympatholytics; Thiadiazoles | 1998 |
Mutations of aspartate 103 in the Hm2 receptor and alterations in receptor binding properties of muscarinic agonists.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Alanine; Amino Acid Substitution; Animals; Arecoline; Asparagine; Aspartic Acid; Carbachol; COS Cells; Muscarinic Agonists; Mutagenesis, Site-Directed; Oxotremorine; Pilocarpine; Receptor, Muscarinic M2; Receptors, Muscarinic; Transfection | 1995 |
Inhibitory cholinergic effects on the autonomously contractile bulbus cordis branchialis of the cephalopod Sepia officinalis L.
Topics: Acetylcholine; Animals; Arecoline; Bungarotoxins; Carbachol; Cholinergic Agents; Cholinergic Agonists; Cholinergic Antagonists; Female; Heart; Male; Mollusca; Muscarine; Myocardial Contraction; Nicotine; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate | 1999 |
Alanine-scanning mutagenesis of transmembrane domain 6 of the M(1) muscarinic acetylcholine receptor suggests that Tyr381 plays key roles in receptor function.
Topics: Acetylcholine; Alanine; Animals; Atropine; Binding, Competitive; COS Cells; Immunohistochemistry; Ligands; Muscarinic Agonists; Muscarinic Antagonists; Mutagenesis, Site-Directed; N-Methylscopolamine; Oxotremorine; Phosphatidylinositols; Pilocarpine; Protein Structure, Tertiary; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Tyrosine | 1999 |
A common muscarinic pathway for diapause recovery in the distantly related nematode species Caenorhabditis elegans and Ancylostoma caninum.
Topics: Ancylostoma; Ancylostomatoidea; Animals; Arecoline; Atropine; Caenorhabditis elegans; Insulin; Larva; Muscarinic Agonists; Muscarinic Antagonists; Neuropeptides; Neurotransmitter Agents; Oxotremorine; Pilocarpine; Signal Transduction | 2000 |
Muscarinic receptor agonists decrease cocaine self-administration rates in drug-naive mice.
Topics: Animals; Antipsychotic Agents; Bridged Bicyclo Compounds; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mice; Muscarinic Agonists; Oxotremorine; Pilocarpine; Self Administration; Thiadiazoles | 2000 |
Reversal of pertussis toxin-induced thermal allodynia by muscarinic cholinergic agonists in mice.
Topics: Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Hot Temperature; Injections, Subcutaneous; Male; Mice; Muscarinic Agonists; Oxotremorine; Pain; Pain Measurement; Pertussis Toxin; Pilocarpine; Succinimides; Virulence Factors, Bordetella | 2000 |
Alteration of cardiovascular and neuronal function in M1 knockout mice.
Topics: Animals; Calcium Channels; Cells, Cultured; Electrophysiology; Gene Targeting; GTP-Binding Proteins; Heart; Hippocampus; Humans; Learning; Memory; Mice; Mice, Knockout; Muscarinic Agonists; Neurons; Oxotremorine; Pilocarpine; Potassium Channels; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Seizures; Signal Transduction; Telencephalon | 2001 |
Pharmacological characterization of muscarinic receptors in mouse isolated urinary bladder smooth muscle.
Topics: Acetylcholine; Animals; Carbachol; Diamines; Dioxolanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pilocarpine; Piperidines; Receptors, Muscarinic; Urinary Bladder | 2001 |
Receptor reserve of phosphoinositide-coupled muscarinic receptors in mouse hippocampus in vivo.
Topics: Acetylcholine; Alzheimer Disease; Animals; Cholinergic Fibers; Dioxolanes; Dose-Response Relationship, Drug; Drug Interactions; Hippocampus; Hydrolysis; Lithium; Male; Mice; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Phosphatidylinositols; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Synaptic Transmission | 2001 |
Evidence for the involvement of the muscarinic cholinergic system in the central actions of pentoxifylline.
Topics: Acetylcholinesterase; Animals; Anxiety; Avoidance Learning; Hippocampus; Learning Disabilities; Male; Memory Disorders; Mice; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Pentoxifylline; Pilocarpine; Rats; Rats, Wistar; Receptors, Muscarinic; Scopolamine; Seizures; Tremor | 2002 |
Role of muscarinic receptors in the activation of the ventral subiculum and the consequences for dopamine release in the nucleus accumbens.
Topics: Animals; Atropine; Bicuculline; Bridged-Ring Compounds; Carbachol; Cholinergic Agonists; Diamines; Dopamine; Hippocampus; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nucleus Accumbens; Oxotremorine; Pilocarpine; Pyridines; Rats; Receptors, Muscarinic; Spiro Compounds; Thiadiazoles; Tropanes | 2003 |
Role of specific muscarinic receptor subtypes in cholinergic parasympathomimetic responses, in vivo phosphoinositide hydrolysis, and pilocarpine-induced seizure activity.
Topics: Animals; Apomorphine; Body Temperature; Cerebral Cortex; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Genotype; Hippocampus; Hydrolysis; Hypothermia; Lithium; Mice; Mice, Knockout; Muscarinic Agonists; Oxotremorine; Parasympathetic Nervous System; Phosphatidylinositols; Pilocarpine; Pupil; Receptors, Muscarinic; Salivation; Seizures | 2003 |
Muscarinic receptor activities potentiated by desensitization of nicotinic receptors in rat superior cervical ganglia.
Topics: Animals; Cells, Cultured; Electrophysiology; Mecamylamine; Muscarinic Agonists; Neurons; Nicotine; Nicotinic Antagonists; Oxotremorine; Patch-Clamp Techniques; Pilocarpine; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Nicotinic; Superior Cervical Ganglion | 2003 |
Cholinergic effects on fear conditioning II: nicotinic and muscarinic modulations of atropine-induced disruption of the degraded contingency effect.
Topics: Animals; Atropine; Conditioning, Classical; Fear; Male; Memory; Muscarinic Antagonists; Nicotine; Nicotinic Antagonists; Oxotremorine; Parasympathetic Fibers, Postganglionic; Pilocarpine; Psychopharmacology; Pyridines; Rats; Rats, Sprague-Dawley; Thiadiazoles | 2005 |
Evaluation of levetiracetam effects on pilocarpine-induced seizures: cholinergic muscarinic system involvement.
Topics: Animals; Anticonvulsants; Convulsants; Disease Models, Animal; Hippocampus; Levetiracetam; Male; Mice; Muscarinic Agonists; Oxotremorine; Pilocarpine; Piracetam; Receptors, Muscarinic; Seizures | 2005 |