Page last updated: 2024-08-17

pilocarpine and carbamazepine

pilocarpine has been researched along with carbamazepine in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19902 (6.90)18.7374
1990's2 (6.90)18.2507
2000's11 (37.93)29.6817
2010's14 (48.28)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Goncikowska, M1
Ebinger, G; Michotte, Y; Smolders, I; Van Belle, K1
George, B; Kulkarni, SK1
Capella, HM; Lemos, T1
Clinckers, R; Ebinger, G; Meurs, A; Michotte, Y; Smolders, I1
Bentivoglio, M; Chakir, A; Fabene, PF; Ouazzani, R1
Bogo, MR; Bonan, CD; Bruno, AN; Cognato, Gde P; da Silva, RS; Sarkis, JJ1
Beck, H; Schaub, C; Uebachs, M1
Cunha, AO; dos Santos, WF; Liberato, JL; Mortari, MR1
Abraham, PM; Krishnakumar, A; Paul, J; Paulose, CS1
Krishnakumar, A; Nandhu, MS; Paulose, CS1
Mathew, J; Nandhu, MS; Paul, J; Paulose, CS1
Khan, RS; Mathew, J; Paulose, CS; Peeyush Kumar, T1
Mathew, J; Paulose, CS; Sadanandan, J; Soman, S1
Citraro, R; De Fazio, S; De Sarro, G; Mainardi, P; Perucca, E; Raggio, R; Russo, E; Scicchitano, F1
Anju, TR; Antony, S; Jayanarayanan, S; Paulose, CS; Soman, S1
Averkin, RG; Beck, H; Bellistri, E; Menendez de la Prida, L; Miklitz, C; Müller, C; Pothmann, L; Remy, S; Uebachs, M1
Kaminski, RM; Leclercq, K1
Blanco, MM; Cinini, SM; Lima, TZ; Mello, LE; Pontes, JC; Queiroz, CM1
Gulec Suyen, G; Isbil-Buyukcoskun, N; Kahveci, N; Ozluk, K; Sengun, E1
Adongo, DW; Mante, PK; Woode, E1

Reviews

1 review(s) available for pilocarpine and carbamazepine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for pilocarpine and carbamazepine

ArticleYear
[Treatment of Horton's headache with small doses of pilocarpine and carbamazepine].
    Wiadomosci lekarskie (Warsaw, Poland : 1960), 1984, Jul-15, Volume: 37, Issue:14

    Topics: Adult; Carbamazepine; Clinical Trials as Topic; Cluster Headache; Double-Blind Method; Drug Therapy, Combination; Humans; Male; Middle Aged; Pilocarpine; Vascular Headaches

1984

Other Studies

27 other study(ies) available for pilocarpine and carbamazepine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Hippocampal and cerebellar extracellular amino acids during pilocarpine-induced seizures in freely moving rats.
    European journal of pharmacology, 1997, Jan-14, Volume: 319, Issue:1

    Topics: Amino Acids; Animals; Aspartic Acid; Carbamazepine; Cerebellum; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Male; Microdialysis; Phenobarbital; Pilocarpine; Rats; Rats, Wistar; Seizures

1997
Modulation of lithium-pilocarpine-induced status epilepticus by adenosinergic agents.
    Methods and findings in experimental and clinical pharmacology, 1997, Volume: 19, Issue:5

    Topics: 2-Chloroadenosine; Adenosine; Animals; Anticonvulsants; Carbamazepine; Dipyridamole; Disease Models, Animal; Dose-Response Relationship, Drug; Lithium; Male; Pilocarpine; Rats; Rats, Wistar; Status Epilepticus; Theophylline; Vasodilator Agents

1997
Effect on epileptogenesis of carbamazepine treatment during the silent period of the pilocarpine model of epilepsy.
    Epilepsia, 2002, Volume: 43 Suppl 5

    Topics: Animals; Anticonvulsants; Carbamazepine; Convulsants; Epilepsy; Hippocampus; Male; Pilocarpine; Rats; Rats, Wistar

2002
Quantitative in vivo microdialysis study on the influence of multidrug transporters on the blood-brain barrier passage of oxcarbazepine: concomitant use of hippocampal monoamines as pharmacodynamic markers for the anticonvulsant activity.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: Animals; Anticonvulsants; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biogenic Monoamines; Biomarkers; Blood-Brain Barrier; Carbamazepine; Chromatography, Liquid; Convulsants; Dose-Response Relationship, Drug; Hippocampus; Kinetics; Microdialysis; Oxcarbazepine; Pilocarpine; Rats; Seizures; Spectrophotometry, Ultraviolet

2005
Drug resistance and hippocampal damage after delayed treatment of pilocarpine-induced epilepsy in the rat.
    Brain research bulletin, 2006, Dec-11, Volume: 71, Issue:1-3

    Topics: Animals; Anticonvulsants; Brain Damage, Chronic; Carbamazepine; Convulsants; Disease Models, Animal; Down-Regulation; Drug Administration Schedule; Drug Resistance; Epilepsy; Epilepsy, Temporal Lobe; Gliosis; Hippocampus; Male; Nerve Degeneration; Neurons; Parvalbumins; Pilocarpine; Rats; Status Epilepticus; Time Factors

2006
Antiepileptic drugs prevent changes induced by pilocarpine model of epilepsy in brain ecto-nucleotidases.
    Neurochemical research, 2007, Volume: 32, Issue:6

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Anticonvulsants; Brain; Carbamazepine; Cerebral Cortex; Epilepsy; Hippocampus; Male; Muscarinic Agonists; Phenytoin; Pilocarpine; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Synaptosomes; Valproic Acid

2007
Diminished response of CA1 neurons to antiepileptic drugs in chronic epilepsy.
    Epilepsia, 2007, Volume: 48, Issue:7

    Topics: Action Potentials; Animals; Anticonvulsants; Carbamazepine; Chronic Disease; Dentate Gyrus; Disease Models, Animal; Drug Resistance; Epilepsy; Hippocampus; Humans; Neurons; Patch-Clamp Techniques; Phenytoin; Pilocarpine; Pyramidal Cells; Rats; Sodium Channels; Synaptic Transmission

2007
Neuroprotective effects of diazepam, carbamazepine, phenytoin and ketamine after pilocarpine-induced status epilepticus.
    Basic & clinical pharmacology & toxicology, 2009, Volume: 104, Issue:6

    Topics: Animals; Anticonvulsants; Carbamazepine; Dentate Gyrus; Diazepam; Drug Administration Schedule; Glial Fibrillary Acidic Protein; Hippocampus; Ketamine; Male; Maze Learning; Neuroprotective Agents; Phenytoin; Pilocarpine; Rats; Rats, Wistar; Status Epilepticus

2009
Down-regulation of cerebellar 5-HT(2C) receptors in pilocarpine-induced epilepsy in rats: therapeutic role of Bacopa monnieri extract.
    Journal of the neurological sciences, 2009, Sep-15, Volume: 284, Issue:1-2

    Topics: Animals; Anticonvulsants; Ataxia; Bacopa; Carbamazepine; Cerebellum; Down-Regulation; Drug Evaluation, Preclinical; Epilepsy; Male; Neuroprotective Agents; Phytotherapy; Pilocarpine; Plant Extracts; Protein Binding; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin Receptor Agonists

2009
Upregulation of 5-HT2C receptors in hippocampus of pilocarpine-induced epileptic rats: antagonism by Bacopa monnieri.
    Epilepsy & behavior : E&B, 2009, Volume: 16, Issue:2

    Topics: Animals; Anticonvulsants; Bacopa; Carbamazepine; Disease Models, Animal; Epilepsy; Ergolines; Hippocampus; Inositol 1,4,5-Trisphosphate; Male; Pilocarpine; Plant Preparations; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Statistics, Nonparametric; Swimming; Tritium; Up-Regulation

2009
Increased excitability and metabolism in pilocarpine induced epileptic rats: effect of Bacopa monnieri.
    Fitoterapia, 2010, Volume: 81, Issue:6

    Topics: Acetylcholinesterase; Animals; Anticonvulsants; Bacopa; Carbamazepine; Epilepsy; Epinephrine; Insulin; Malate Dehydrogenase; Male; Muscarinic Agonists; Myocardium; Norepinephrine; Phytotherapy; Pilocarpine; Plant Extracts; Rats; Rats, Wistar; Saponins; Triiodothyronine; Triterpenes

2010
Behavioral deficit and decreased GABA receptor functional regulation in the cerebellum of epileptic rats: effect of Bacopa monnieri and bacoside A.
    Epilepsy & behavior : E&B, 2010, Volume: 17, Issue:4

    Topics: Animals; Anticonvulsants; Behavioral Symptoms; Bicuculline; Carbamazepine; Cerebellum; Disease Models, Animal; Epilepsy; GABA Antagonists; gamma-Aminobutyric Acid; Male; Maze Learning; Phytotherapy; Pilocarpine; Plant Preparations; Protein Binding; Rats; Rats, Wistar; Receptors, GABA; Saponins; Triterpenes; Tritium

2010
Decreased GABA receptor in the striatum and spatial recognition memory deficit in epileptic rats: effect of Bacopa monnieri and bacoside-A.
    Journal of ethnopharmacology, 2010, Jul-20, Volume: 130, Issue:2

    Topics: Animals; Anticonvulsants; Bacopa; Basal Ganglia; Behavior, Animal; Bicuculline; Binding, Competitive; Carbamazepine; Disease Models, Animal; Down-Regulation; GABA Antagonists; gamma-Aminobutyric Acid; Male; Maze Learning; Motor Activity; Pilocarpine; Rats; Rats, Wistar; Receptors, GABA-A; Recognition, Psychology; RNA, Messenger; Saponins; Status Epilepticus; Triterpenes

2010
Preclinical activity profile of α-lactoalbumin, a whey protein rich in tryptophan, in rodent models of seizures and epilepsy.
    Epilepsy research, 2011, Volume: 95, Issue:1-2

    Topics: Amino Acids; Animals; Carbamazepine; Convulsants; Drug Evaluation, Preclinical; Electroshock; Epilepsy; Epilepsy, Reflex; Female; Lactalbumin; Male; Mice; Mice, Inbred C57BL; Models, Animal; Pilocarpine; Rats; Rats, Mutant Strains; Rats, Wistar; Seizures; Serotonin; Tryptophan

2011
Impaired motor learning attributed to altered AMPA receptor function in the cerebellum of rats with temporal lobe epilepsy: ameliorating effects of Withania somnifera and withanolide A.
    Epilepsy & behavior : E&B, 2013, Volume: 27, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Carbamazepine; Cerebellum; Disease Models, Animal; Epilepsy, Temporal Lobe; Excitatory Amino Acid Transporter 1; Gene Expression Regulation; Glutamate Decarboxylase; Glutamic Acid; Inositol 1,4,5-Trisphosphate; Learning Disabilities; Linear Models; Locomotion; Male; Motor Activity; Phytotherapy; Pilocarpine; Protein Binding; Psychomotor Performance; Rats; Rats, Wistar; Receptors, AMPA; RNA, Messenger; Time Factors; Tritium; Withania; Withanolides

2013
Function of inhibitory micronetworks is spared by Na+ channel-acting anticonvulsant drugs.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Jul-16, Volume: 34, Issue:29

    Topics: Animals; Anticonvulsants; Biophysics; Carbamazepine; Convulsants; Disease Models, Animal; Electric Stimulation; Epilepsy; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Kainic Acid; Membrane Potentials; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Pilocarpine; Rats; Rats, Wistar; Sodium Channels

2014
Status epilepticus induction has prolonged effects on the efficacy of antiepileptic drugs in the 6-Hz seizure model.
    Epilepsy & behavior : E&B, 2015, Volume: 49

    Topics: Animals; Anticonvulsants; Carbamazepine; Diazepam; Disease Models, Animal; Levetiracetam; Male; Mice; Phenytoin; Pilocarpine; Piracetam; Seizures; Status Epilepticus; Treatment Outcome

2015
Seizures triggered by pentylenetetrazol in marmosets made chronically epileptic with pilocarpine show greater refractoriness to treatment.
    Epilepsy research, 2016, Volume: 126

    Topics: Animals; Anticonvulsants; Brain; Callithrix; Carbamazepine; Chronic Disease; Disease Models, Animal; Electrocorticography; Epilepsy; Female; Immunohistochemistry; Male; Neuropeptide Y; Pentylenetetrazole; Phenobarbital; Pilocarpine; Proto-Oncogene Proteins c-fos; Seizures; Valproic Acid

2016
Immediate and delayed treatment with gabapentin, carbamazepine and CNQX have almost similar impact on cognitive functions and behavior in the lithium-pilocarpine model in rats.
    Pharmacology, biochemistry, and behavior, 2016, Volume: 148

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amines; Animals; Behavior, Animal; Carbamazepine; Cognition; Cyclohexanecarboxylic Acids; Disease Models, Animal; Gabapentin; gamma-Aminobutyric Acid; Lithium; Male; Maze Learning; Motor Activity; Pilocarpine; Rats; Rats, Wistar; Status Epilepticus

2016
Anticonvulsant effects of antiaris toxicaria aqueous extract: investigation using animal models of temporal lobe epilepsy.
    BMC research notes, 2017, Apr-26, Volume: 10, Issue:1

    Topics: Animals; Antiaris; Anticonvulsants; Carbamazepine; Diazepam; Disease Models, Animal; Drug Administration Schedule; Epilepsy, Temporal Lobe; Hippocampus; Kainic Acid; Male; Mice; Mice, Inbred ICR; Nifedipine; Pentylenetetrazole; Pilocarpine; Plant Extracts; Rats; Rats, Sprague-Dawley

2017