Page last updated: 2024-08-23

picrotoxin and bilobalide

picrotoxin has been researched along with bilobalide in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (71.43)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chebib, M; Duke, RK; Huang, SH; Johnston, GA; Sasaki, K; Wada, K2
Hawthorne, R; Lynch, JW1
Hartmann, J; Hildmann, O; Kiewert, C; Klein, J; Kumar, V; Naik, RS; Rueda, M1
Buckley, F; Sacks, B1
Duke, RK; Lummis, SC; Thompson, AJ1
Duke, RK; Hinton, T; Johnston, GAR; Ng, CC1

Other Studies

7 other study(ies) available for picrotoxin and bilobalide

ArticleYear
Bilobalide, a sesquiterpene trilactone from Ginkgo biloba, is an antagonist at recombinant alpha1beta2gamma2L GABA(A) receptors.
    European journal of pharmacology, 2003, Mar-07, Volume: 464, Issue:1

    Topics: Animals; Bicuculline; Cyclopentanes; Diterpenes; Dose-Response Relationship, Drug; Furans; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ginkgo biloba; Ginkgolides; Humans; Membrane Potentials; Oocytes; Picrotoxin; Receptors, GABA-A; Recombinant Proteins; Sesterterpenes; Xenopus laevis

2003
A picrotoxin-specific conformational change in the glycine receptor M2-M3 loop.
    The Journal of biological chemistry, 2005, Oct-28, Volume: 280, Issue:43

    Topics: Allosteric Site; Cyclopentanes; Cysteine; Dimerization; Diterpenes; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Furans; Ginkgolides; Glycine; Humans; Inhibitory Concentration 50; Kinetics; Mesylates; Mutagenesis, Site-Directed; Mutation; Picrotoxin; Protein Binding; Protein Conformation; Protein Structure, Secondary; Protein Structure, Tertiary; Receptors, Glycine; Time Factors

2005
Mixed antagonistic effects of bilobalide at rho1 GABAC receptor.
    Neuroscience, 2006, Volume: 137, Issue:2

    Topics: Animals; Chloride Channels; Cyclopentanes; Diterpenes; Dose-Response Relationship, Drug; Female; Furans; GABA Antagonists; gamma-Aminobutyric Acid; Gene Transfer Techniques; Ginkgolides; Humans; Neural Inhibition; Oocytes; Patch-Clamp Techniques; Picrotoxin; Plant Extracts; Protein Subunits; Receptors, GABA; Recombinant Fusion Proteins; Xenopus laevis

2006
Role of GABAergic antagonism in the neuroprotective effects of bilobalide.
    Brain research, 2007, Jan-12, Volume: 1128, Issue:1

    Topics: Animals; Area Under Curve; Bicuculline; Brain Edema; Bridged Bicyclo Compounds, Heterocyclic; Choline; Cyclopentanes; Drug Interactions; Excitatory Amino Acid Agonists; Furans; GABA Antagonists; gamma-Aminobutyric Acid; Ginkgolides; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Neuroprotective Agents; Nonlinear Dynamics; Picrotoxin; Rats; Rats, Sprague-Dawley; Synaptosomes

2007
Drug treatment improves memory in mice.
    Down's syndrome, research and practice : the journal of the Sarah Duffen Centre, 2007, Volume: 12, Issue:1

    Topics: Animals; Central Nervous System Stimulants; Chromosomes, Human, Pair 21; Cyclopentanes; Disease Models, Animal; Down Syndrome; Furans; GABA Antagonists; Ginkgolides; Humans; Maze Learning; Memory; Mice; Mice, Transgenic; Neuropsychological Tests; Pentylenetetrazole; Picrotoxin

2007
Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor.
    Molecular pharmacology, 2011, Volume: 80, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding Sites; Cyclopentanes; Diltiazem; Female; Furans; Ginkgolides; Humans; Molecular Sequence Data; Picrotoxin; Radioligand Assay; Receptors, Serotonin, 5-HT3; Sequence Homology, Amino Acid; Sesterterpenes; Xenopus laevis

2011
Effects of bilobalide, ginkgolide B and picrotoxinin on GABA
    European journal of pharmacology, 2017, Jul-05, Volume: 806

    Topics: Animals; Cyclopentanes; Dose-Response Relationship, Drug; Electrophysiological Phenomena; Furans; GABA Modulators; Ginkgo biloba; Ginkgolides; Humans; Lactones; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Terpenes; Xenopus laevis

2017