picrotoxin has been researched along with bilobalide in 7 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 5 (71.43) | 29.6817 |
2010's | 2 (28.57) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chebib, M; Duke, RK; Huang, SH; Johnston, GA; Sasaki, K; Wada, K | 2 |
Hawthorne, R; Lynch, JW | 1 |
Hartmann, J; Hildmann, O; Kiewert, C; Klein, J; Kumar, V; Naik, RS; Rueda, M | 1 |
Buckley, F; Sacks, B | 1 |
Duke, RK; Lummis, SC; Thompson, AJ | 1 |
Duke, RK; Hinton, T; Johnston, GAR; Ng, CC | 1 |
7 other study(ies) available for picrotoxin and bilobalide
Article | Year |
---|---|
Bilobalide, a sesquiterpene trilactone from Ginkgo biloba, is an antagonist at recombinant alpha1beta2gamma2L GABA(A) receptors.
Topics: Animals; Bicuculline; Cyclopentanes; Diterpenes; Dose-Response Relationship, Drug; Furans; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ginkgo biloba; Ginkgolides; Humans; Membrane Potentials; Oocytes; Picrotoxin; Receptors, GABA-A; Recombinant Proteins; Sesterterpenes; Xenopus laevis | 2003 |
A picrotoxin-specific conformational change in the glycine receptor M2-M3 loop.
Topics: Allosteric Site; Cyclopentanes; Cysteine; Dimerization; Diterpenes; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Furans; Ginkgolides; Glycine; Humans; Inhibitory Concentration 50; Kinetics; Mesylates; Mutagenesis, Site-Directed; Mutation; Picrotoxin; Protein Binding; Protein Conformation; Protein Structure, Secondary; Protein Structure, Tertiary; Receptors, Glycine; Time Factors | 2005 |
Mixed antagonistic effects of bilobalide at rho1 GABAC receptor.
Topics: Animals; Chloride Channels; Cyclopentanes; Diterpenes; Dose-Response Relationship, Drug; Female; Furans; GABA Antagonists; gamma-Aminobutyric Acid; Gene Transfer Techniques; Ginkgolides; Humans; Neural Inhibition; Oocytes; Patch-Clamp Techniques; Picrotoxin; Plant Extracts; Protein Subunits; Receptors, GABA; Recombinant Fusion Proteins; Xenopus laevis | 2006 |
Role of GABAergic antagonism in the neuroprotective effects of bilobalide.
Topics: Animals; Area Under Curve; Bicuculline; Brain Edema; Bridged Bicyclo Compounds, Heterocyclic; Choline; Cyclopentanes; Drug Interactions; Excitatory Amino Acid Agonists; Furans; GABA Antagonists; gamma-Aminobutyric Acid; Ginkgolides; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Neuroprotective Agents; Nonlinear Dynamics; Picrotoxin; Rats; Rats, Sprague-Dawley; Synaptosomes | 2007 |
Drug treatment improves memory in mice.
Topics: Animals; Central Nervous System Stimulants; Chromosomes, Human, Pair 21; Cyclopentanes; Disease Models, Animal; Down Syndrome; Furans; GABA Antagonists; Ginkgolides; Humans; Maze Learning; Memory; Mice; Mice, Transgenic; Neuropsychological Tests; Pentylenetetrazole; Picrotoxin | 2007 |
Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor.
Topics: Amino Acid Sequence; Animals; Binding Sites; Cyclopentanes; Diltiazem; Female; Furans; Ginkgolides; Humans; Molecular Sequence Data; Picrotoxin; Radioligand Assay; Receptors, Serotonin, 5-HT3; Sequence Homology, Amino Acid; Sesterterpenes; Xenopus laevis | 2011 |
Effects of bilobalide, ginkgolide B and picrotoxinin on GABA
Topics: Animals; Cyclopentanes; Dose-Response Relationship, Drug; Electrophysiological Phenomena; Furans; GABA Modulators; Ginkgo biloba; Ginkgolides; Humans; Lactones; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Terpenes; Xenopus laevis | 2017 |