Page last updated: 2024-08-21

picolinamide and acetylene

picolinamide has been researched along with acetylene in 1 studies

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bridges, TM; Chun, A; Conn, PJ; Daniels, JS; Gogi, KK; Gogliotti, RD; Gregory, KJ; Jones, C; Lindsley, CW; Meiler, J; Nguyen, ED; Niswender, CM; Noetzel, MJ; Rook, JM; Stauffer, SR; Turlington, M; Vinson, PN; Xiang, Z; Zhou, Y1

Other Studies

1 other study(ies) available for picolinamide and acetylene

ArticleYear
Exploration of allosteric agonism structure-activity relationships within an acetylene series of metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulators (PAMs): discovery of 5-((3-fluorophenyl)ethynyl)-N-(3-methyloxetan-3-yl)picolinamide
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Acetylene; Allosteric Regulation; Amides; Animals; Binding, Competitive; Cell Membrane; Drug Discovery; Excitatory Postsynaptic Potentials; HEK293 Cells; Hippocampus; Humans; Male; Models, Chemical; Models, Molecular; Molecular Structure; Picolinic Acids; Protein Structure, Tertiary; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Structure-Activity Relationship

2013