Page last updated: 2024-09-05

piboserod and td-5108

piboserod has been researched along with td-5108 in 37 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(td-5108)
Trials
(td-5108)
Recent Studies (post-2010) (td-5108)
11955334052216

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (21.62)29.6817
2010's22 (59.46)24.3611
2020's7 (18.92)2.80

Authors

AuthorsStudies
Ishihara, K; Sasa, M1
Kemp, A; Manahan-Vaughan, D1
Fujii, H; Katsui, R; Kojima, Y; Nakagawa, T; Nakajima, Y; Takaki, M1
Becker, DP; Flynn, DL; Gullikson, GW; Loeffler, R; Moormann, AE; Moummi, C; Nosal, R; Villamil, CI; Yang, DC1
Cachard-Chastel, M; Croes, S; Deloménie, C; Devijver, H; Dewachter, I; Gardier, AM; Langlois, M; Lezoualc'h, F; Sicsic, S; Van Leuven, F1
Han, JS; Liu, FY; Qu, XX; Wan, Y; Xing, GG; Xu, IS1
De Maeyer, JH; Lefebvre, RA; Schuurkes, JA1
Eda, H; Kimura, N; Komada, T; Mikami, T; Naganeo, R; Nakata, E; Nakatani, K; Ohmi, T; Sakakibara, M; Sugimoto, H; Suzuki, K; Toga, T1
Modica, MN; Pittalà, V; Romeo, G; Salerno, L; Siracusa, MA1
Boulouard, M; Bureau, R; Dauphin, F; Lezoualc'h, F; Rault, S1
Ajdary, S; Ataee, R; Rezayat, M; Shahriari, S; Shokrgozar, MA; Zarrindast, MR1
Back, H; Jang, Y; Jung, SW; Kim, JW; Lee, B; Oh, U; Seo, EK; Shim, CK; Shim, WS1
Hong, J; Morse, CL; Pike, VW; Xu, R1
Hayashi, SS; Kamei, J; Nakanishi, Y; Ohsawa, M1
Bockaert, J; Claeysen, S; Compan, V; Dumuis, A1
Kaneko, H; Seto, Y; Yoshida, N1
Fujinoki, M1
Andreeva, AV; Fukai, T; Hen, R; Krbanjevic, A; Profirovic, J; Strekalova, E; Urao, N; Ushio-Fukai, M; Varadarajan, S; Voyno-Yasenetskaya, TA1
Amano, T; Ariga, H; Shimizu, K; Uchida, M; Yamato, S1
Darcet, F; David, DJ; Gardier, AM; Hen, R; Kerdine-Römer, S; Mendez-David, I; Wu, MV1
Goshima, H; Ishizuka, T; Ozawa, A; Watanabe, Y1
Broad, J; Dukes, GE; Góralczyk, A; Mannur, K; Sanger, GJ1
Khakpai, F; Nasehi, M; Tabatabaie, M; Zarrindast, MR1
Chen, JH; Du, X; Hong, L; Huizinga, JD; Jiang, L; Li, H; Liao, H; Luo, H; Shi, J; Tan, S; Yang, Z; Yu, Y; Zhao, L1
De Deurwaerdère, P; Di Giovanni, G; Navailles, S1
Hagena, H; Manahan-Vaughan, D; Twarkowski, H1
Ebrahimi-Ghiri, M; Farrahizadeh, M; Nasehi, M; Zarrindast, MR1
Kozono, N; Ohtani, A; Shiga, T1
Du, CX; Guo, Y; Liu, J; Lv, SX; Wang, HS; Wang, T; Xie, W; Zhang, J; Zhang, L2
Agrawal, L; Shiga, T; Vimal, SK1
Eydipour, Z; Jamaldini, SH; Nasehi, M; Vaseghi, S; Zarrindast, MR1
Agrawal, L; Bhattacharyya, S; Korkutata, M; Shiga, T; Vimal, SK; Yadav, MK1
Claeysen, S; Dallemagne, P; Lanthier, C; Lecoutey, C; Rochais, C1
Hamada, A; Hira, T; Ohsaka, F; Okumura, M; Sonoyama, K; Tsuruta, T1
Castro-Alvarez, A; Chávez-Ángel, E; Nelson, R1
Fehse, C; Gergs, U; Hofmann, B; Marušáková, M; Neumann, J; Seidler, T1

Reviews

5 review(s) available for piboserod and td-5108

ArticleYear
Serotonin 5-HT3 and 5-HT4 ligands: an update of medicinal chemistry research in the last few years.
    Current medicinal chemistry, 2010, Volume: 17, Issue:4

    Topics: Animals; Chemistry, Pharmaceutical; Humans; Ligands; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2010
Review of 5-HT4R ligands: state of art and clinical applications.
    Current topics in medicinal chemistry, 2010, Volume: 10, Issue:5

    Topics: Humans; Ligands; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

2010
5-HT(4) receptors, a place in the sun: act two.
    Current opinion in pharmacology, 2011, Volume: 11, Issue:1

    Topics: Animals; Brain; Brain Diseases; Humans; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2011
Therapeutic potential of serotonin 4 receptor for chronic depression and its associated comorbidity in the gut.
    Neuropharmacology, 2020, Volume: 166

    Topics: Animals; Brain; Comorbidity; Depression; Gastrointestinal Diseases; Gastrointestinal Microbiome; Humans; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2020
Therapeutic modulators of the serotonin 5-HT
    Expert opinion on therapeutic patents, 2020, Volume: 30, Issue:7

    Topics: Animals; Central Nervous System Diseases; Drug Development; Gastrointestinal Diseases; Humans; Ligands; Patents as Topic; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2020

Other Studies

32 other study(ies) available for piboserod and td-5108

ArticleYear
Failure of repeated electroconvulsive shock treatment on 5-HT4-receptor-mediated depolarization due to protein kinase A system in young rat hippocampal CA1 neurons.
    Journal of pharmacological sciences, 2004, Volume: 95, Issue:3

    Topics: Aniline Compounds; Animals; Cyclic AMP-Dependent Protein Kinases; Electroshock; Hippocampus; In Vitro Techniques; Male; Neurons; Piperazines; Piperidines; Propane; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Second Messenger Systems; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2004
The 5-hydroxytryptamine4 receptor exhibits frequency-dependent properties in synaptic plasticity and behavioural metaplasticity in the hippocampal CA1 region in vivo.
    Cerebral cortex (New York, N.Y. : 1991), 2005, Volume: 15, Issue:7

    Topics: Aniline Compounds; Animals; Electric Stimulation; Excitatory Postsynaptic Potentials; Exploratory Behavior; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Motor Activity; Neuronal Plasticity; Piperidines; Propane; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2005
A 5-HT4 agonist, mosapride, enhances intrinsic rectorectal and rectoanal reflexes after removal of extrinsic nerves in guinea pigs.
    American journal of physiology. Gastrointestinal and liver physiology, 2005, Volume: 289, Issue:2

    Topics: Acute Disease; Anal Canal; Animals; Benzamides; Chronic Disease; Denervation; Disease Models, Animal; Gastrointestinal Agents; Gastrointestinal Motility; Guinea Pigs; Indoles; Male; Morpholines; Rectum; Reflex; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Spinal Cord Injuries; Sulfonamides

2005
Pyrrolizidine esters and amides as 5-HT4 receptor agonists and antagonists.
    Journal of medicinal chemistry, 2006, Feb-09, Volume: 49, Issue:3

    Topics: Amides; Animals; Benzamides; Bradycardia; Brain; Dogs; Esophagus; Esters; Female; Gastric Emptying; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Muscle Contraction; Muscle, Smooth; Pyloric Antrum; Pyrroles; Pyrrolizidine Alkaloids; Radioligand Assay; Rats; Rats, Wistar; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Structure-Activity Relationship

2006
5-HT4 receptor agonists increase sAPPalpha levels in the cortex and hippocampus of male C57BL/6j mice.
    British journal of pharmacology, 2007, Volume: 150, Issue:7

    Topics: Aminobenzoates; Amyloid beta-Protein Precursor; Animals; Benzofurans; Cerebral Cortex; Cholinesterase Inhibitors; Donepezil; Hippocampus; Indans; Indoles; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; para-Aminobenzoates; Piperidines; RNA, Messenger; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2007
Roles of 5-hydroxytryptamine (5-HT) receptor subtypes in the inhibitory effects of 5-HT on C-fiber responses of spinal wide dynamic range neurons in rats.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Action Potentials; Animals; Cholinergic Fibers; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Male; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Sciatic Nerve; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord

2007
Selective desensitization of the 5-HT4 receptor-mediated response in pig atrium but not in stomach.
    British journal of pharmacology, 2009, Volume: 156, Issue:2

    Topics: Animals; Atrial Function, Left; Benzofurans; Female; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Organ Specificity; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach; Swine; Synaptic Transmission; Tachyphylaxis

2009
In vitro and in vivo pharmacological characterization of PF-01354082, a novel partial agonist selective for the 5-HT(4) receptor.
    European journal of pharmacology, 2009, May-01, Volume: 609, Issue:1-3

    Topics: Administration, Oral; Animals; Benzimidazoles; Carbachol; Cell Line; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Esophagus; Gastrointestinal Motility; Humans; Indoles; Kidney; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Inbred Strains; Sensitivity and Specificity; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Receptor Agonists; Time Factors

2009
Study of 5HT3 and HT4 receptor expression in HT29 cell line and human colon adenocarcinoma tissues.
    Archives of Iranian medicine, 2010, Volume: 13, Issue:2

    Topics: Adenocarcinoma; Aminobenzoates; Biguanides; Blotting, Western; Bridged Bicyclo Compounds, Heterocyclic; Cell Proliferation; Cisapride; Colonic Neoplasms; HT29 Cells; Humans; Oxazines; para-Aminobenzoates; Piperidines; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2010
An aqueous extract of Poncirus fructus activates the prokinetic activity of 5-HT receptor subtype 4 without hERG interaction.
    Journal of ethnopharmacology, 2010, Oct-28, Volume: 132, Issue:1

    Topics: Animals; Astemizole; Cell Line; Cell Membrane; Cyclic AMP; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Fruit; Gastrointestinal Transit; Humans; Patch-Clamp Techniques; Plant Extracts; Poncirus; Potassium Channel Blockers; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Transfection

2010
Synthesis, structure-affinity relationships, and radiolabeling of selective high-affinity 5-HT4 receptor ligands as prospective imaging probes for positron emission tomography.
    Journal of medicinal chemistry, 2010, 10-14, Volume: 53, Issue:19

    Topics: 4-Aminobenzoic Acid; Animals; Brain; Carbon Radioisotopes; Cell Line; Cricetinae; Drug Inverse Agonism; Drug Partial Agonism; Fluorine Radioisotopes; Guinea Pigs; Humans; Isotope Labeling; Ligands; para-Aminobenzoates; Positron-Emission Tomography; Radiopharmaceuticals; Rats; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Species Specificity; Structure-Activity Relationship

2010
Effect of chronic pain on morphine-induced respiratory depression in mice.
    Neuroscience, 2011, Feb-03, Volume: 174

    Topics: Analgesics, Opioid; Animals; Benzamides; Brain Stem; Chronic Disease; Indoles; Ligation; Male; Mice; Mice, Inbred ICR; Morphine; Morpholines; Pain; Peripheral Nervous System Diseases; Receptors, Serotonin, 5-HT4; Respiration; Respiratory Insufficiency; Sciatic Nerve; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2011
Effects of mosapride citrate, a 5-HT4-receptor agonist, on gastric distension-induced visceromotor response in conscious rats.
    Journal of pharmacological sciences, 2011, Volume: 116, Issue:1

    Topics: Abdominal Pain; Analgesics, Non-Narcotic; Animals; Benzamides; Benzyl Compounds; Dose-Response Relationship, Drug; Dyspepsia; Gastric Dilatation; Gastrointestinal Agents; Gastrointestinal Motility; Granisetron; Male; Morpholines; Random Allocation; Rats; Rats, Wistar; Reflex, Abdominal; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach

2011
Serotonin-enhanced hyperactivation of hamster sperm.
    Reproduction (Cambridge, England), 2011, Volume: 142, Issue:2

    Topics: Animals; Calcium Signaling; Cricetinae; Culture Media, Serum-Free; Epididymis; Male; Mesocricetus; Osmolar Concentration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sperm Capacitation; Sperm Motility; Sperm Tail; Spermatozoa; Time Factors

2011
A novel regulator of angiogenesis in endothelial cells: 5-hydroxytriptamine 4 receptor.
    Angiogenesis, 2013, Volume: 16, Issue:1

    Topics: Aniline Compounds; Animals; Capillaries; Cell Adhesion; Cell Membrane Permeability; Cell Movement; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Female; GTP-Binding Protein alpha Subunits, G12-G13; Human Umbilical Vein Endothelial Cells; Ischemia; Mice; Muscles; Neovascularization, Physiologic; Piperidines; Propane; Receptors, Serotonin, 5-HT4; Regional Blood Flow; rhoA GTP-Binding Protein; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Wound Healing

2013
Dual role of mosapride citrate hydrate on the gastric emptying evaluated by the breath test in conscious rats.
    Journal of pharmacological sciences, 2013, Volume: 121, Issue:4

    Topics: Acetic Acid; Animals; Benzamides; Breath Tests; Carbon Radioisotopes; Depression, Chemical; Dose-Response Relationship, Drug; Gastric Emptying; Indoles; Male; Morpholines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stimulation, Chemical; Sulfonamides

2013
Rapid anxiolytic effects of a 5-HT₄ receptor agonist are mediated by a neurogenesis-independent mechanism.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:6

    Topics: Aniline Compounds; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Anxiety; Comorbidity; Corticosterone; Depressive Disorder; Disease Models, Animal; Fluoxetine; Hippocampus; Indoles; Male; Mice; Mice, Inbred C57BL; Neurogenesis; Neurons; Piperidines; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides; Time Factors

2014
Stimulation of 5-HT4 receptor enhances differentiation of mouse induced pluripotent stem cells into neural progenitor cells.
    Clinical and experimental pharmacology & physiology, 2014, Volume: 41, Issue:5

    Topics: Animals; Cell Culture Techniques; Cell Differentiation; Cell Line; CREB-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Indoles; Induced Pluripotent Stem Cells; Mice; Microscopy, Fluorescence; Neural Stem Cells; Phosphorylation; Protein Kinase Inhibitors; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2014
Drugs acting at 5-HT4 , D2 , motilin, and ghrelin receptors differ markedly in how they affect neuromuscular functions in human isolated stomach.
    Neurogastroenterology and motility, 2014, Volume: 26, Issue:6

    Topics: Dopamine D2 Receptor Antagonists; Electric Stimulation; Gastric Emptying; Humans; Muscle, Smooth; Pyloric Antrum; Receptors, Gastrointestinal Hormone; Receptors, Ghrelin; Receptors, Neuropeptide; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2014
The effects of CA1 5HT4 receptors in MK801-induced amnesia and hyperlocomotion.
    Neuroscience letters, 2015, Feb-05, Volume: 587

    Topics: Amnesia; Aniline Compounds; Animals; CA1 Region, Hippocampal; Dizocilpine Maleate; Drug Partial Agonism; Exploratory Behavior; Male; Memory; Mice; Motor Activity; para-Aminobenzoates; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2015
Involvement of 5-HT3 and 5-HT4 receptors in colonic motor patterns in rats.
    Neurogastroenterology and motility, 2015, Volume: 27, Issue:7

    Topics: Animals; Colon; Gastrointestinal Motility; Myoelectric Complex, Migrating; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2015
The 5-HT4 Agonist Prucalopride Stimulates L-DOPA-Induced Dopamine Release in Restricted Brain Regions of the Hemiparkinsonian Rat In Vivo.
    CNS neuroscience & therapeutics, 2015, Volume: 21, Issue:9

    Topics: Animals; Benzofurans; Brain; Dopamine; Dopamine Agents; Functional Laterality; Indoles; Levodopa; Microdialysis; Oxidopamine; Parkinsonian Disorders; Rats; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2015
The 5-hydroxytryptamine4 receptor enables differentiation of informational content and encoding in the hippocampus.
    Hippocampus, 2016, Volume: 26, Issue:7

    Topics: Animals; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Dentate Gyrus; Electric Stimulation; Electrodes, Implanted; Excitatory Postsynaptic Potentials; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Perforant Pathway; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Synapses

2016
Modulation of cannabinoid signaling by hippocampal 5-HT4 serotonergic system in fear conditioning.
    Journal of psychopharmacology (Oxford, England), 2016, Volume: 30, Issue:9

    Topics: Aniline Compounds; Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Cannabinoids; Conditioning, Classical; Dose-Response Relationship, Drug; Fear; Freezing Reaction, Cataleptic; Hippocampus; Male; Memory; Mice; para-Aminobenzoates; Piperidines; Receptor, Cannabinoid, CB1; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2016
Roles of the serotonin 5-HT4 receptor in dendrite formation of the rat hippocampal neurons in vitro.
    Brain research, 2017, 01-15, Volume: 1655

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzimidazoles; Brain-Derived Neurotrophic Factor; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dendrites; Enzyme Inhibitors; Hippocampus; Immunohistochemistry; Neuronal Outgrowth; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, trkB; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2017
Activation and blockade of serotonin
    Neurological research, 2019, Volume: 41, Issue:7

    Topics: Animals; Benzimidazoles; Brain; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dose-Response Relationship, Drug; Habenula; Indoles; Male; Maze Learning; Memory, Short-Term; Microinjections; Norepinephrine; Oxidopamine; Parkinsonian Disorders; Rats; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Substantia Nigra; Sulfonamides

2019
Role of serotonin 4 receptor in the growth of hippocampal neurons during the embryonic development in mice.
    Neuropharmacology, 2019, 11-01, Volume: 158

    Topics: Aniline Compounds; Animals; Axons; Brain-Derived Neurotrophic Factor; Dendrites; Embryo, Mammalian; Gene Knockdown Techniques; Hippocampus; Indoles; Intercellular Signaling Peptides and Proteins; Mice; Nerve Growth Factor; Nerve Growth Factors; Nerve Tissue Proteins; Neurogenesis; Neurons; Piperidines; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2019
The role of 5-HT4 serotonin receptors in the CA1 hippocampal region on memory acquisition impairment induced by total (TSD) and REM sleep deprivation (RSD).
    Physiology & behavior, 2020, 03-01, Volume: 215

    Topics: Aniline Compounds; Animals; Avoidance Learning; CA1 Region, Hippocampal; Male; Memory Consolidation; Memory Disorders; Microinjections; Motor Activity; Pain Perception; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sleep Deprivation

2020
Activation and Blockade of Serotonin-4 Receptors in the Lateral Habenula Produce Antidepressant Effects in the Hemiparkinsonian Rat.
    Neuropsychobiology, 2021, Volume: 80, Issue:1

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Depression; Disease Models, Animal; Dopamine; Habenula; Hippocampus; Norepinephrine; Parkinson Disease; Prefrontal Cortex; Rats; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2021
Expression of serotonin receptor HTR4 in glucagon-like peptide-1-positive enteroendocrine cells of the murine intestine.
    Pflugers Archiv : European journal of physiology, 2020, Volume: 472, Issue:10

    Topics: Animals; Cells, Cultured; Enteroendocrine Cells; Gastrointestinal Agents; Glucagon-Like Peptide 1; Indoles; Male; Mice; Mice, Inbred C57BL; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2020
Understanding the Molecular Basis of 5-HT
    International journal of molecular sciences, 2021, Mar-30, Volume: 22, Issue:7

    Topics: Humans; Models, Molecular; Molecular Docking Simulation; Quantitative Structure-Activity Relationship; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Structure-Activity Relationship

2021
Cardiovascular effects of metoclopramide and domperidone on human 5-HT
    European journal of pharmacology, 2021, Jun-15, Volume: 901

    Topics: Aged; Animals; Calcium-Binding Proteins; Cardiovascular Agents; Domperidone; Dopamine Antagonists; Heart; Humans; In Vitro Techniques; Male; Metoclopramide; Mice, Transgenic; Middle Aged; Myocardial Contraction; Myocytes, Cardiac; Phosphorylation; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists

2021