piboserod has been researched along with td-5108 in 37 studies
Studies (piboserod) | Trials (piboserod) | Recent Studies (post-2010) (piboserod) | Studies (td-5108) | Trials (td-5108) | Recent Studies (post-2010) (td-5108) |
---|---|---|---|---|---|
119 | 5 | 53 | 340 | 52 | 216 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 8 (21.62) | 29.6817 |
2010's | 22 (59.46) | 24.3611 |
2020's | 7 (18.92) | 2.80 |
Authors | Studies |
---|---|
Ishihara, K; Sasa, M | 1 |
Kemp, A; Manahan-Vaughan, D | 1 |
Fujii, H; Katsui, R; Kojima, Y; Nakagawa, T; Nakajima, Y; Takaki, M | 1 |
Becker, DP; Flynn, DL; Gullikson, GW; Loeffler, R; Moormann, AE; Moummi, C; Nosal, R; Villamil, CI; Yang, DC | 1 |
Cachard-Chastel, M; Croes, S; Deloménie, C; Devijver, H; Dewachter, I; Gardier, AM; Langlois, M; Lezoualc'h, F; Sicsic, S; Van Leuven, F | 1 |
Han, JS; Liu, FY; Qu, XX; Wan, Y; Xing, GG; Xu, IS | 1 |
De Maeyer, JH; Lefebvre, RA; Schuurkes, JA | 1 |
Eda, H; Kimura, N; Komada, T; Mikami, T; Naganeo, R; Nakata, E; Nakatani, K; Ohmi, T; Sakakibara, M; Sugimoto, H; Suzuki, K; Toga, T | 1 |
Modica, MN; Pittalà, V; Romeo, G; Salerno, L; Siracusa, MA | 1 |
Boulouard, M; Bureau, R; Dauphin, F; Lezoualc'h, F; Rault, S | 1 |
Ajdary, S; Ataee, R; Rezayat, M; Shahriari, S; Shokrgozar, MA; Zarrindast, MR | 1 |
Back, H; Jang, Y; Jung, SW; Kim, JW; Lee, B; Oh, U; Seo, EK; Shim, CK; Shim, WS | 1 |
Hong, J; Morse, CL; Pike, VW; Xu, R | 1 |
Hayashi, SS; Kamei, J; Nakanishi, Y; Ohsawa, M | 1 |
Bockaert, J; Claeysen, S; Compan, V; Dumuis, A | 1 |
Kaneko, H; Seto, Y; Yoshida, N | 1 |
Fujinoki, M | 1 |
Andreeva, AV; Fukai, T; Hen, R; Krbanjevic, A; Profirovic, J; Strekalova, E; Urao, N; Ushio-Fukai, M; Varadarajan, S; Voyno-Yasenetskaya, TA | 1 |
Amano, T; Ariga, H; Shimizu, K; Uchida, M; Yamato, S | 1 |
Darcet, F; David, DJ; Gardier, AM; Hen, R; Kerdine-Römer, S; Mendez-David, I; Wu, MV | 1 |
Goshima, H; Ishizuka, T; Ozawa, A; Watanabe, Y | 1 |
Broad, J; Dukes, GE; Góralczyk, A; Mannur, K; Sanger, GJ | 1 |
Khakpai, F; Nasehi, M; Tabatabaie, M; Zarrindast, MR | 1 |
Chen, JH; Du, X; Hong, L; Huizinga, JD; Jiang, L; Li, H; Liao, H; Luo, H; Shi, J; Tan, S; Yang, Z; Yu, Y; Zhao, L | 1 |
De Deurwaerdère, P; Di Giovanni, G; Navailles, S | 1 |
Hagena, H; Manahan-Vaughan, D; Twarkowski, H | 1 |
Ebrahimi-Ghiri, M; Farrahizadeh, M; Nasehi, M; Zarrindast, MR | 1 |
Kozono, N; Ohtani, A; Shiga, T | 1 |
Du, CX; Guo, Y; Liu, J; Lv, SX; Wang, HS; Wang, T; Xie, W; Zhang, J; Zhang, L | 2 |
Agrawal, L; Shiga, T; Vimal, SK | 1 |
Eydipour, Z; Jamaldini, SH; Nasehi, M; Vaseghi, S; Zarrindast, MR | 1 |
Agrawal, L; Bhattacharyya, S; Korkutata, M; Shiga, T; Vimal, SK; Yadav, MK | 1 |
Claeysen, S; Dallemagne, P; Lanthier, C; Lecoutey, C; Rochais, C | 1 |
Hamada, A; Hira, T; Ohsaka, F; Okumura, M; Sonoyama, K; Tsuruta, T | 1 |
Castro-Alvarez, A; Chávez-Ángel, E; Nelson, R | 1 |
Fehse, C; Gergs, U; Hofmann, B; Marušáková, M; Neumann, J; Seidler, T | 1 |
5 review(s) available for piboserod and td-5108
Article | Year |
---|---|
Serotonin 5-HT3 and 5-HT4 ligands: an update of medicinal chemistry research in the last few years.
Topics: Animals; Chemistry, Pharmaceutical; Humans; Ligands; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2010 |
Review of 5-HT4R ligands: state of art and clinical applications.
Topics: Humans; Ligands; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship | 2010 |
5-HT(4) receptors, a place in the sun: act two.
Topics: Animals; Brain; Brain Diseases; Humans; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2011 |
Therapeutic potential of serotonin 4 receptor for chronic depression and its associated comorbidity in the gut.
Topics: Animals; Brain; Comorbidity; Depression; Gastrointestinal Diseases; Gastrointestinal Microbiome; Humans; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2020 |
Therapeutic modulators of the serotonin 5-HT
Topics: Animals; Central Nervous System Diseases; Drug Development; Gastrointestinal Diseases; Humans; Ligands; Patents as Topic; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2020 |
32 other study(ies) available for piboserod and td-5108
Article | Year |
---|---|
Failure of repeated electroconvulsive shock treatment on 5-HT4-receptor-mediated depolarization due to protein kinase A system in young rat hippocampal CA1 neurons.
Topics: Aniline Compounds; Animals; Cyclic AMP-Dependent Protein Kinases; Electroshock; Hippocampus; In Vitro Techniques; Male; Neurons; Piperazines; Piperidines; Propane; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Second Messenger Systems; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides | 2004 |
The 5-hydroxytryptamine4 receptor exhibits frequency-dependent properties in synaptic plasticity and behavioural metaplasticity in the hippocampal CA1 region in vivo.
Topics: Aniline Compounds; Animals; Electric Stimulation; Excitatory Postsynaptic Potentials; Exploratory Behavior; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Motor Activity; Neuronal Plasticity; Piperidines; Propane; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2005 |
A 5-HT4 agonist, mosapride, enhances intrinsic rectorectal and rectoanal reflexes after removal of extrinsic nerves in guinea pigs.
Topics: Acute Disease; Anal Canal; Animals; Benzamides; Chronic Disease; Denervation; Disease Models, Animal; Gastrointestinal Agents; Gastrointestinal Motility; Guinea Pigs; Indoles; Male; Morpholines; Rectum; Reflex; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Spinal Cord Injuries; Sulfonamides | 2005 |
Pyrrolizidine esters and amides as 5-HT4 receptor agonists and antagonists.
Topics: Amides; Animals; Benzamides; Bradycardia; Brain; Dogs; Esophagus; Esters; Female; Gastric Emptying; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Muscle Contraction; Muscle, Smooth; Pyloric Antrum; Pyrroles; Pyrrolizidine Alkaloids; Radioligand Assay; Rats; Rats, Wistar; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Structure-Activity Relationship | 2006 |
5-HT4 receptor agonists increase sAPPalpha levels in the cortex and hippocampus of male C57BL/6j mice.
Topics: Aminobenzoates; Amyloid beta-Protein Precursor; Animals; Benzofurans; Cerebral Cortex; Cholinesterase Inhibitors; Donepezil; Hippocampus; Indans; Indoles; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; para-Aminobenzoates; Piperidines; RNA, Messenger; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides | 2007 |
Roles of 5-hydroxytryptamine (5-HT) receptor subtypes in the inhibitory effects of 5-HT on C-fiber responses of spinal wide dynamic range neurons in rats.
Topics: Action Potentials; Animals; Cholinergic Fibers; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Male; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Sciatic Nerve; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord | 2007 |
Selective desensitization of the 5-HT4 receptor-mediated response in pig atrium but not in stomach.
Topics: Animals; Atrial Function, Left; Benzofurans; Female; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Organ Specificity; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach; Swine; Synaptic Transmission; Tachyphylaxis | 2009 |
In vitro and in vivo pharmacological characterization of PF-01354082, a novel partial agonist selective for the 5-HT(4) receptor.
Topics: Administration, Oral; Animals; Benzimidazoles; Carbachol; Cell Line; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Esophagus; Gastrointestinal Motility; Humans; Indoles; Kidney; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Inbred Strains; Sensitivity and Specificity; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Receptor Agonists; Time Factors | 2009 |
Study of 5HT3 and HT4 receptor expression in HT29 cell line and human colon adenocarcinoma tissues.
Topics: Adenocarcinoma; Aminobenzoates; Biguanides; Blotting, Western; Bridged Bicyclo Compounds, Heterocyclic; Cell Proliferation; Cisapride; Colonic Neoplasms; HT29 Cells; Humans; Oxazines; para-Aminobenzoates; Piperidines; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2010 |
An aqueous extract of Poncirus fructus activates the prokinetic activity of 5-HT receptor subtype 4 without hERG interaction.
Topics: Animals; Astemizole; Cell Line; Cell Membrane; Cyclic AMP; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Fruit; Gastrointestinal Transit; Humans; Patch-Clamp Techniques; Plant Extracts; Poncirus; Potassium Channel Blockers; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Transfection | 2010 |
Synthesis, structure-affinity relationships, and radiolabeling of selective high-affinity 5-HT4 receptor ligands as prospective imaging probes for positron emission tomography.
Topics: 4-Aminobenzoic Acid; Animals; Brain; Carbon Radioisotopes; Cell Line; Cricetinae; Drug Inverse Agonism; Drug Partial Agonism; Fluorine Radioisotopes; Guinea Pigs; Humans; Isotope Labeling; Ligands; para-Aminobenzoates; Positron-Emission Tomography; Radiopharmaceuticals; Rats; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Species Specificity; Structure-Activity Relationship | 2010 |
Effect of chronic pain on morphine-induced respiratory depression in mice.
Topics: Analgesics, Opioid; Animals; Benzamides; Brain Stem; Chronic Disease; Indoles; Ligation; Male; Mice; Mice, Inbred ICR; Morphine; Morpholines; Pain; Peripheral Nervous System Diseases; Receptors, Serotonin, 5-HT4; Respiration; Respiratory Insufficiency; Sciatic Nerve; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides | 2011 |
Effects of mosapride citrate, a 5-HT4-receptor agonist, on gastric distension-induced visceromotor response in conscious rats.
Topics: Abdominal Pain; Analgesics, Non-Narcotic; Animals; Benzamides; Benzyl Compounds; Dose-Response Relationship, Drug; Dyspepsia; Gastric Dilatation; Gastrointestinal Agents; Gastrointestinal Motility; Granisetron; Male; Morpholines; Random Allocation; Rats; Rats, Wistar; Reflex, Abdominal; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach | 2011 |
Serotonin-enhanced hyperactivation of hamster sperm.
Topics: Animals; Calcium Signaling; Cricetinae; Culture Media, Serum-Free; Epididymis; Male; Mesocricetus; Osmolar Concentration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sperm Capacitation; Sperm Motility; Sperm Tail; Spermatozoa; Time Factors | 2011 |
A novel regulator of angiogenesis in endothelial cells: 5-hydroxytriptamine 4 receptor.
Topics: Aniline Compounds; Animals; Capillaries; Cell Adhesion; Cell Membrane Permeability; Cell Movement; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Female; GTP-Binding Protein alpha Subunits, G12-G13; Human Umbilical Vein Endothelial Cells; Ischemia; Mice; Muscles; Neovascularization, Physiologic; Piperidines; Propane; Receptors, Serotonin, 5-HT4; Regional Blood Flow; rhoA GTP-Binding Protein; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Wound Healing | 2013 |
Dual role of mosapride citrate hydrate on the gastric emptying evaluated by the breath test in conscious rats.
Topics: Acetic Acid; Animals; Benzamides; Breath Tests; Carbon Radioisotopes; Depression, Chemical; Dose-Response Relationship, Drug; Gastric Emptying; Indoles; Male; Morpholines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stimulation, Chemical; Sulfonamides | 2013 |
Rapid anxiolytic effects of a 5-HT₄ receptor agonist are mediated by a neurogenesis-independent mechanism.
Topics: Aniline Compounds; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Anxiety; Comorbidity; Corticosterone; Depressive Disorder; Disease Models, Animal; Fluoxetine; Hippocampus; Indoles; Male; Mice; Mice, Inbred C57BL; Neurogenesis; Neurons; Piperidines; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides; Time Factors | 2014 |
Stimulation of 5-HT4 receptor enhances differentiation of mouse induced pluripotent stem cells into neural progenitor cells.
Topics: Animals; Cell Culture Techniques; Cell Differentiation; Cell Line; CREB-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Indoles; Induced Pluripotent Stem Cells; Mice; Microscopy, Fluorescence; Neural Stem Cells; Phosphorylation; Protein Kinase Inhibitors; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides | 2014 |
Drugs acting at 5-HT4 , D2 , motilin, and ghrelin receptors differ markedly in how they affect neuromuscular functions in human isolated stomach.
Topics: Dopamine D2 Receptor Antagonists; Electric Stimulation; Gastric Emptying; Humans; Muscle, Smooth; Pyloric Antrum; Receptors, Gastrointestinal Hormone; Receptors, Ghrelin; Receptors, Neuropeptide; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2014 |
The effects of CA1 5HT4 receptors in MK801-induced amnesia and hyperlocomotion.
Topics: Amnesia; Aniline Compounds; Animals; CA1 Region, Hippocampal; Dizocilpine Maleate; Drug Partial Agonism; Exploratory Behavior; Male; Memory; Mice; Motor Activity; para-Aminobenzoates; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2015 |
Involvement of 5-HT3 and 5-HT4 receptors in colonic motor patterns in rats.
Topics: Animals; Colon; Gastrointestinal Motility; Myoelectric Complex, Migrating; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2015 |
The 5-HT4 Agonist Prucalopride Stimulates L-DOPA-Induced Dopamine Release in Restricted Brain Regions of the Hemiparkinsonian Rat In Vivo.
Topics: Animals; Benzofurans; Brain; Dopamine; Dopamine Agents; Functional Laterality; Indoles; Levodopa; Microdialysis; Oxidopamine; Parkinsonian Disorders; Rats; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides | 2015 |
The 5-hydroxytryptamine4 receptor enables differentiation of informational content and encoding in the hippocampus.
Topics: Animals; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Dentate Gyrus; Electric Stimulation; Electrodes, Implanted; Excitatory Postsynaptic Potentials; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Perforant Pathway; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Synapses | 2016 |
Modulation of cannabinoid signaling by hippocampal 5-HT4 serotonergic system in fear conditioning.
Topics: Aniline Compounds; Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Cannabinoids; Conditioning, Classical; Dose-Response Relationship, Drug; Fear; Freezing Reaction, Cataleptic; Hippocampus; Male; Memory; Mice; para-Aminobenzoates; Piperidines; Receptor, Cannabinoid, CB1; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2016 |
Roles of the serotonin 5-HT4 receptor in dendrite formation of the rat hippocampal neurons in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzimidazoles; Brain-Derived Neurotrophic Factor; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dendrites; Enzyme Inhibitors; Hippocampus; Immunohistochemistry; Neuronal Outgrowth; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, trkB; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2017 |
Activation and blockade of serotonin
Topics: Animals; Benzimidazoles; Brain; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dose-Response Relationship, Drug; Habenula; Indoles; Male; Maze Learning; Memory, Short-Term; Microinjections; Norepinephrine; Oxidopamine; Parkinsonian Disorders; Rats; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Substantia Nigra; Sulfonamides | 2019 |
Role of serotonin 4 receptor in the growth of hippocampal neurons during the embryonic development in mice.
Topics: Aniline Compounds; Animals; Axons; Brain-Derived Neurotrophic Factor; Dendrites; Embryo, Mammalian; Gene Knockdown Techniques; Hippocampus; Indoles; Intercellular Signaling Peptides and Proteins; Mice; Nerve Growth Factor; Nerve Growth Factors; Nerve Tissue Proteins; Neurogenesis; Neurons; Piperidines; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides | 2019 |
The role of 5-HT4 serotonin receptors in the CA1 hippocampal region on memory acquisition impairment induced by total (TSD) and REM sleep deprivation (RSD).
Topics: Aniline Compounds; Animals; Avoidance Learning; CA1 Region, Hippocampal; Male; Memory Consolidation; Memory Disorders; Microinjections; Motor Activity; Pain Perception; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sleep Deprivation | 2020 |
Activation and Blockade of Serotonin-4 Receptors in the Lateral Habenula Produce Antidepressant Effects in the Hemiparkinsonian Rat.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Depression; Disease Models, Animal; Dopamine; Habenula; Hippocampus; Norepinephrine; Parkinson Disease; Prefrontal Cortex; Rats; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2021 |
Expression of serotonin receptor HTR4 in glucagon-like peptide-1-positive enteroendocrine cells of the murine intestine.
Topics: Animals; Cells, Cultured; Enteroendocrine Cells; Gastrointestinal Agents; Glucagon-Like Peptide 1; Indoles; Male; Mice; Mice, Inbred C57BL; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2020 |
Understanding the Molecular Basis of 5-HT
Topics: Humans; Models, Molecular; Molecular Docking Simulation; Quantitative Structure-Activity Relationship; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Structure-Activity Relationship | 2021 |
Cardiovascular effects of metoclopramide and domperidone on human 5-HT
Topics: Aged; Animals; Calcium-Binding Proteins; Cardiovascular Agents; Domperidone; Dopamine Antagonists; Heart; Humans; In Vitro Techniques; Male; Metoclopramide; Mice, Transgenic; Middle Aged; Myocardial Contraction; Myocytes, Cardiac; Phosphorylation; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists | 2021 |