Page last updated: 2024-09-05

piboserod and sdz 205-557

piboserod has been researched along with sdz 205-557 in 2 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(sdz 205-557)
Trials
(sdz 205-557)
Recent Studies (post-2010) (sdz 205-557)
1195535609

Protein Interaction Comparison

ProteinTaxonomypiboserod (IC50)sdz 205-557 (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.2512
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.2512

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fischmeister, R; Langlois, M1
Boulouard, M; Bureau, R; Butt-Gueulle, S; Dauphin, F; Daveu, C; Duchatelle, P; Dumuis, A; Lelong-Boulouard, V; LemaƮtre, S; Lepailleur, A; Lezoualc'h, F; Pfeiffer, B; Rault, S1

Reviews

1 review(s) available for piboserod and sdz 205-557

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

1 other study(ies) available for piboserod and sdz 205-557

ArticleYear
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
    Bioorganic & medicinal chemistry, 2009, Mar-15, Volume: 17, Issue:6

    Topics: Animals; Chlorocebus aethiops; COS Cells; Humans; Indoles; Models, Molecular; Molecular Structure; Pyrazines; Radioligand Assay; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides

2009