Page last updated: 2024-09-05

piboserod and prucalopride

piboserod has been researched along with prucalopride in 6 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(prucalopride)
Trials
(prucalopride)
Recent Studies (post-2010) (prucalopride)
11955323857167

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (66.67)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fischmeister, R; Langlois, M1
Boulouard, M; Bureau, R; Butt-Gueulle, S; Dauphin, F; Daveu, C; Duchatelle, P; Dumuis, A; Lelong-Boulouard, V; Lemaître, S; Lepailleur, A; Lezoualc'h, F; Pfeiffer, B; Rault, S1
Cachard-Chastel, M; Croes, S; Deloménie, C; Devijver, H; Dewachter, I; Gardier, AM; Langlois, M; Lezoualc'h, F; Sicsic, S; Van Leuven, F1
De Maeyer, JH; Lefebvre, RA; Schuurkes, JA1
Ajjala, DR; Aleti, RR; Bhyrapuneni, G; Kandikere, V; Nirogi, R; Rasheed, MA; Saralaya, R1
De Deurwaerdère, P; Di Giovanni, G; Navailles, S1

Reviews

1 review(s) available for piboserod and prucalopride

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

5 other study(ies) available for piboserod and prucalopride

ArticleYear
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
    Bioorganic & medicinal chemistry, 2009, Mar-15, Volume: 17, Issue:6

    Topics: Animals; Chlorocebus aethiops; COS Cells; Humans; Indoles; Models, Molecular; Molecular Structure; Pyrazines; Radioligand Assay; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides

2009
5-HT4 receptor agonists increase sAPPalpha levels in the cortex and hippocampus of male C57BL/6j mice.
    British journal of pharmacology, 2007, Volume: 150, Issue:7

    Topics: Aminobenzoates; Amyloid beta-Protein Precursor; Animals; Benzofurans; Cerebral Cortex; Cholinesterase Inhibitors; Donepezil; Hippocampus; Indans; Indoles; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; para-Aminobenzoates; Piperidines; RNA, Messenger; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2007
Selective desensitization of the 5-HT4 receptor-mediated response in pig atrium but not in stomach.
    British journal of pharmacology, 2009, Volume: 156, Issue:2

    Topics: Animals; Atrial Function, Left; Benzofurans; Female; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Organ Specificity; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach; Swine; Synaptic Transmission; Tachyphylaxis

2009
In-vivo rat striatal 5-HT4 receptor occupancy using non-radiolabelled SB207145.
    The Journal of pharmacy and pharmacology, 2013, Volume: 65, Issue:5

    Topics: Aniline Compounds; Animals; Benzofurans; Binding, Competitive; Brain; Drug Discovery; Indoles; Ligands; Male; Oxazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; Serotonin Receptor Agonists; Sulfonamides; Tandem Mass Spectrometry; Tissue Distribution

2013
The 5-HT4 Agonist Prucalopride Stimulates L-DOPA-Induced Dopamine Release in Restricted Brain Regions of the Hemiparkinsonian Rat In Vivo.
    CNS neuroscience & therapeutics, 2015, Volume: 21, Issue:9

    Topics: Animals; Benzofurans; Brain; Dopamine; Dopamine Agents; Functional Laterality; Indoles; Levodopa; Microdialysis; Oxidopamine; Parkinsonian Disorders; Rats; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2015