Page last updated: 2024-09-05

piboserod and ondansetron

piboserod has been researched along with ondansetron in 4 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(ondansetron)
Trials
(ondansetron)
Recent Studies (post-2010) (ondansetron)
1195533,3801,216994

Protein Interaction Comparison

ProteinTaxonomypiboserod (IC50)ondansetron (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)10
Solute carrier family 22 member 2Homo sapiens (human)1.295
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)10
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.0136
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.717
5-hydroxytryptamine receptor 3AHomo sapiens (human)0.0001
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)10
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.7303
Multidrug and toxin extrusion protein 2Homo sapiens (human)2.4533
GABA theta subunitRattus norvegicus (Norway rat)10
Multidrug and toxin extrusion protein 1Homo sapiens (human)0.0875
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)10
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.0181

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Endo, T; Hamaue, N; Hirafuji, M; Minami, M1
Nylander, O; Pihl, L1
Amano, T; Ariga, H; Ishida, T; Kimura, T; Matsueda, K; Tajiri, H; Torii, A; Uehara, H; Yamato, S1
Gribovskaja-Rupp, I; Kosinski, L; Ludwig, K; Ridolfi, T; Takahashi, T1

Reviews

1 review(s) available for piboserod and ondansetron

ArticleYear
[Serotonin and anticancer drug-induced emesis].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2004, Volume: 124, Issue:8

    Topics: Animals; Antiemetics; Antineoplastic Agents; Cisplatin; Enterochromaffin Cells; Granisetron; Humans; Indoles; Ondansetron; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Tropisetron; Vagus Nerve; Vomiting

2004

Other Studies

3 other study(ies) available for piboserod and ondansetron

ArticleYear
Luminal hypotonicity increases duodenal mucosal permeability by a mechanism involving 5-hydroxytryptamine.
    Acta physiologica (Oxford, England), 2006, Volume: 186, Issue:1

    Topics: Anesthetics, Local; Animals; Cyclooxygenase Inhibitors; Duodenum; Granisetron; Indoles; Indomethacin; Intestinal Mucosa; Lidocaine; Male; Ondansetron; Osmotic Pressure; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Agents; Serotonin Antagonists; Tetrodotoxin; Tropisetron

2006
Urocortin I is present in the enteric nervous system and exerts an excitatory effect via cholinergic and serotonergic pathways in the rat colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 293, Issue:4

    Topics: Animals; Atropine; Colon; Corticotropin-Releasing Hormone; Dioxanes; Electric Stimulation; Enteric Nervous System; Gastrointestinal Motility; Hexamethonium; Immunohistochemistry; Male; NG-Nitroarginine Methyl Ester; Ondansetron; Peptide Fragments; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Tetrodotoxin; Urocortins

2007
Upregulation of mucosal 5-HT3 receptors is involved in restoration of colonic transit after pelvic nerve transection.
    Neurogastroenterology and motility, 2012, Volume: 24, Issue:5

    Topics: Animals; Blotting, Western; Chromium Radioisotopes; Colon; Denervation; Dose-Response Relationship, Drug; Enteric Nervous System; Gastrointestinal Transit; In Vitro Techniques; Indoles; Intestinal Mucosa; Male; Ondansetron; Pelvis; Peripheral Nerves; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides; Up-Regulation

2012