Page last updated: 2024-09-05

piboserod and mosapride

piboserod has been researched along with mosapride in 5 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(mosapride)
Trials
(mosapride)
Recent Studies (post-2010) (mosapride)
11955328690142

Protein Interaction Comparison

ProteinTaxonomypiboserod (IC50)mosapride (IC50)
hepatocyte nuclear factor 4-alpha isoform 2Homo sapiens (human)4.18
perilipin-5Homo sapiens (human)1.315
perilipin-1Homo sapiens (human)1.196
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform aHomo sapiens (human)1.2753
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.3966
Cytochrome P450 1A2Homo sapiens (human)0.4
Cytochrome P450 3A4Homo sapiens (human)0.7
Alpha-2A adrenergic receptorHomo sapiens (human)3.6794
Cytochrome P450 2C9 Homo sapiens (human)1
Alpha-2B adrenergic receptorHomo sapiens (human)1.908
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.3966
Sodium-dependent serotonin transporterHomo sapiens (human)3.8117
Cytochrome P450 2C19Homo sapiens (human)1
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.2959
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)4.7932
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.3056

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fischmeister, R; Langlois, M1
Fujii, H; Katsui, R; Kojima, Y; Nakagawa, T; Nakajima, Y; Takaki, M1
Hayashi, SS; Kamei, J; Nakanishi, Y; Ohsawa, M1
Kaneko, H; Seto, Y; Yoshida, N1
Amano, T; Ariga, H; Shimizu, K; Uchida, M; Yamato, S1

Reviews

1 review(s) available for piboserod and mosapride

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

4 other study(ies) available for piboserod and mosapride

ArticleYear
A 5-HT4 agonist, mosapride, enhances intrinsic rectorectal and rectoanal reflexes after removal of extrinsic nerves in guinea pigs.
    American journal of physiology. Gastrointestinal and liver physiology, 2005, Volume: 289, Issue:2

    Topics: Acute Disease; Anal Canal; Animals; Benzamides; Chronic Disease; Denervation; Disease Models, Animal; Gastrointestinal Agents; Gastrointestinal Motility; Guinea Pigs; Indoles; Male; Morpholines; Rectum; Reflex; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Spinal Cord Injuries; Sulfonamides

2005
Effect of chronic pain on morphine-induced respiratory depression in mice.
    Neuroscience, 2011, Feb-03, Volume: 174

    Topics: Analgesics, Opioid; Animals; Benzamides; Brain Stem; Chronic Disease; Indoles; Ligation; Male; Mice; Mice, Inbred ICR; Morphine; Morpholines; Pain; Peripheral Nervous System Diseases; Receptors, Serotonin, 5-HT4; Respiration; Respiratory Insufficiency; Sciatic Nerve; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sulfonamides

2011
Effects of mosapride citrate, a 5-HT4-receptor agonist, on gastric distension-induced visceromotor response in conscious rats.
    Journal of pharmacological sciences, 2011, Volume: 116, Issue:1

    Topics: Abdominal Pain; Analgesics, Non-Narcotic; Animals; Benzamides; Benzyl Compounds; Dose-Response Relationship, Drug; Dyspepsia; Gastric Dilatation; Gastrointestinal Agents; Gastrointestinal Motility; Granisetron; Male; Morpholines; Random Allocation; Rats; Rats, Wistar; Reflex, Abdominal; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach

2011
Dual role of mosapride citrate hydrate on the gastric emptying evaluated by the breath test in conscious rats.
    Journal of pharmacological sciences, 2013, Volume: 121, Issue:4

    Topics: Acetic Acid; Animals; Benzamides; Breath Tests; Carbon Radioisotopes; Depression, Chemical; Dose-Response Relationship, Drug; Gastric Emptying; Indoles; Male; Morpholines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stimulation, Chemical; Sulfonamides

2013