piboserod has been researched along with mdl 100907 in 8 studies
Studies (piboserod) | Trials (piboserod) | Recent Studies (post-2010) (piboserod) | Studies (mdl 100907) | Trials (mdl 100907) | Recent Studies (post-2010) (mdl 100907) |
---|---|---|---|---|---|
119 | 5 | 53 | 1,241 | 65 | 539 |
Protein | Taxonomy | piboserod (IC50) | mdl 100907 (IC50) |
---|---|---|---|
5-hydroxytryptamine receptor 2A | Homo sapiens (human) | 0.0048 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 4 (50.00) | 29.6817 |
2010's | 4 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Andrade, R; Béïque, JC; Chapin-Penick, EM; Mladenovic, L | 1 |
Abrahamsson, PA; Bjartell, A; Dizeyi, N; Gadaleanu, V; Hedlund, P; Taskén, KA | 1 |
Han, JS; Liu, FY; Qu, XX; Wan, Y; Xing, GG; Xu, IS | 1 |
Birkeland, JA; Enger, U; Levy, FO; Lunde, PK; Qvigstad, E; Sejersted, OM; Sjaastad, I; Swift, F; Tovsrud, N | 1 |
Argibay, JA; Bourmeyster, N; Bozon, V; Defamie, N; Derangeon, M; Hervé, JC; Peineau, N; Sarrouilhe, D | 1 |
Arreola, JL; Campos-Bedolla, P; Chávez, J; Córdoba-Rodríguez, G; García-Hernández, LM; Méndez, C; Montaño, LM; Ruiz, V; Segura, P; Vargas, MH | 1 |
Fujinoki, M | 1 |
Asao, T; Fujii, T; Kawamura, K; Kuwano, H; Mochiki, E; Morita, H; Ogata, K; Ogawa, A; Ohno, T; Sutou, T; Takahashi, N; Tsutsumi, S; Watanabe, A; Yanai, M | 1 |
8 other study(ies) available for piboserod and mdl 100907
Article | Year |
---|---|
Serotonergic facilitation of synaptic activity in the developing rat prefrontal cortex.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amphetamines; Animals; Bicuculline; Fluorobenzenes; GABA-A Receptor Antagonists; Glutamic Acid; Indoles; Lidocaine; Male; Patch-Clamp Techniques; Phenols; Pindolol; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sodium Channel Blockers; Sulfonamides; Synapses; Tetrodotoxin; Time Factors | 2004 |
Expression of serotonin receptors 2B and 4 in human prostate cancer tissue and effects of their antagonists on prostate cancer cell lines.
Topics: Biomarkers, Tumor; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Enzyme-Linked Immunosorbent Assay; Flow Cytometry; Humans; Immunohistochemistry; In Vitro Techniques; Male; Prostatic Neoplasms; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists | 2005 |
Roles of 5-hydroxytryptamine (5-HT) receptor subtypes in the inhibitory effects of 5-HT on C-fiber responses of spinal wide dynamic range neurons in rats.
Topics: Action Potentials; Animals; Cholinergic Fibers; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Male; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Sciatic Nerve; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord | 2007 |
Serotonin increases L-type Ca2+ current and SR Ca2+ content through 5-HT4 receptors in failing rat ventricular cardiomyocytes.
Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Calcium Channels, L-Type; Calcium Signaling; Calcium-Binding Proteins; Cardiac Myosins; Cardiotonic Agents; Coronary Vessels; Disease Models, Animal; Heart Failure; Indoles; Isoproterenol; Ketanserin; Ligation; Male; Myocardial Contraction; Myocardial Infarction; Myocytes, Cardiac; Myosin Light Chains; Phosphorylation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT4; Sarcoplasmic Reticulum; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides; Time Factors; Troponin I; Ventricular Function | 2007 |
5-HT4 and 5-HT2 receptors antagonistically influence gap junctional coupling between rat auricular myocytes.
Topics: Adenylyl Cyclases; Aminobenzoates; Animals; Animals, Newborn; Blotting, Western; Cells, Cultured; Connexins; Gap Junctions; Heart Atria; In Vitro Techniques; Indoles; Myocytes, Cardiac; para-Aminobenzoates; Patch-Clamp Techniques; Phosphorylation; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Agents; Serotonin Antagonists; Sulfonamides | 2010 |
Role of 5-HT2A, 5-HT4 and 5-HT7 receptors in the antigen-induced airway hyperresponsiveness in guinea-pigs.
Topics: Animals; Bronchial Hyperreactivity; Chromatography, High Pressure Liquid; Disease Models, Animal; Dose-Response Relationship, Drug; Guinea Pigs; Male; Ovalbumin; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sensitivity and Specificity; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists | 2010 |
Serotonin-enhanced hyperactivation of hamster sperm.
Topics: Animals; Calcium Signaling; Cricetinae; Culture Media, Serum-Free; Epididymis; Male; Mesocricetus; Osmolar Concentration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sperm Capacitation; Sperm Motility; Sperm Tail; Spermatozoa; Time Factors | 2011 |
Effects of 5-HT2B, 5-HT3 and 5-HT4 receptor antagonists on gastrointestinal motor activity in dogs.
Topics: Animals; Colon; Dogs; Dose-Response Relationship, Drug; Female; Gastric Mucosa; Gastrointestinal Motility; Gastrointestinal Tract; Ileum; Male; Models, Animal; Myoelectric Complex, Migrating; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Stomach; Time Factors; Transducers, Pressure | 2013 |