Page last updated: 2024-09-05

piboserod and mdl 100907

piboserod has been researched along with mdl 100907 in 8 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(mdl 100907)
Trials
(mdl 100907)
Recent Studies (post-2010) (mdl 100907)
1195531,24165539

Protein Interaction Comparison

ProteinTaxonomypiboserod (IC50)mdl 100907 (IC50)
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0048

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (50.00)29.6817
2010's4 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrade, R; Béïque, JC; Chapin-Penick, EM; Mladenovic, L1
Abrahamsson, PA; Bjartell, A; Dizeyi, N; Gadaleanu, V; Hedlund, P; Taskén, KA1
Han, JS; Liu, FY; Qu, XX; Wan, Y; Xing, GG; Xu, IS1
Birkeland, JA; Enger, U; Levy, FO; Lunde, PK; Qvigstad, E; Sejersted, OM; Sjaastad, I; Swift, F; Tovsrud, N1
Argibay, JA; Bourmeyster, N; Bozon, V; Defamie, N; Derangeon, M; Hervé, JC; Peineau, N; Sarrouilhe, D1
Arreola, JL; Campos-Bedolla, P; Chávez, J; Córdoba-Rodríguez, G; García-Hernández, LM; Méndez, C; Montaño, LM; Ruiz, V; Segura, P; Vargas, MH1
Fujinoki, M1
Asao, T; Fujii, T; Kawamura, K; Kuwano, H; Mochiki, E; Morita, H; Ogata, K; Ogawa, A; Ohno, T; Sutou, T; Takahashi, N; Tsutsumi, S; Watanabe, A; Yanai, M1

Other Studies

8 other study(ies) available for piboserod and mdl 100907

ArticleYear
Serotonergic facilitation of synaptic activity in the developing rat prefrontal cortex.
    The Journal of physiology, 2004, May-01, Volume: 556, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amphetamines; Animals; Bicuculline; Fluorobenzenes; GABA-A Receptor Antagonists; Glutamic Acid; Indoles; Lidocaine; Male; Patch-Clamp Techniques; Phenols; Pindolol; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sodium Channel Blockers; Sulfonamides; Synapses; Tetrodotoxin; Time Factors

2004
Expression of serotonin receptors 2B and 4 in human prostate cancer tissue and effects of their antagonists on prostate cancer cell lines.
    European urology, 2005, Volume: 47, Issue:6

    Topics: Biomarkers, Tumor; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Enzyme-Linked Immunosorbent Assay; Flow Cytometry; Humans; Immunohistochemistry; In Vitro Techniques; Male; Prostatic Neoplasms; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists

2005
Roles of 5-hydroxytryptamine (5-HT) receptor subtypes in the inhibitory effects of 5-HT on C-fiber responses of spinal wide dynamic range neurons in rats.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Action Potentials; Animals; Cholinergic Fibers; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Male; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Sciatic Nerve; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord

2007
Serotonin increases L-type Ca2+ current and SR Ca2+ content through 5-HT4 receptors in failing rat ventricular cardiomyocytes.
    American journal of physiology. Heart and circulatory physiology, 2007, Volume: 293, Issue:4

    Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Calcium Channels, L-Type; Calcium Signaling; Calcium-Binding Proteins; Cardiac Myosins; Cardiotonic Agents; Coronary Vessels; Disease Models, Animal; Heart Failure; Indoles; Isoproterenol; Ketanserin; Ligation; Male; Myocardial Contraction; Myocardial Infarction; Myocytes, Cardiac; Myosin Light Chains; Phosphorylation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT4; Sarcoplasmic Reticulum; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides; Time Factors; Troponin I; Ventricular Function

2007
5-HT4 and 5-HT2 receptors antagonistically influence gap junctional coupling between rat auricular myocytes.
    Journal of molecular and cellular cardiology, 2010, Volume: 48, Issue:1

    Topics: Adenylyl Cyclases; Aminobenzoates; Animals; Animals, Newborn; Blotting, Western; Cells, Cultured; Connexins; Gap Junctions; Heart Atria; In Vitro Techniques; Indoles; Myocytes, Cardiac; para-Aminobenzoates; Patch-Clamp Techniques; Phosphorylation; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Agents; Serotonin Antagonists; Sulfonamides

2010
Role of 5-HT2A, 5-HT4 and 5-HT7 receptors in the antigen-induced airway hyperresponsiveness in guinea-pigs.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2010, Volume: 40, Issue:2

    Topics: Animals; Bronchial Hyperreactivity; Chromatography, High Pressure Liquid; Disease Models, Animal; Dose-Response Relationship, Drug; Guinea Pigs; Male; Ovalbumin; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sensitivity and Specificity; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists

2010
Serotonin-enhanced hyperactivation of hamster sperm.
    Reproduction (Cambridge, England), 2011, Volume: 142, Issue:2

    Topics: Animals; Calcium Signaling; Cricetinae; Culture Media, Serum-Free; Epididymis; Male; Mesocricetus; Osmolar Concentration; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Sperm Capacitation; Sperm Motility; Sperm Tail; Spermatozoa; Time Factors

2011
Effects of 5-HT2B, 5-HT3 and 5-HT4 receptor antagonists on gastrointestinal motor activity in dogs.
    World journal of gastroenterology, 2013, Oct-21, Volume: 19, Issue:39

    Topics: Animals; Colon; Dogs; Dose-Response Relationship, Drug; Female; Gastric Mucosa; Gastrointestinal Motility; Gastrointestinal Tract; Ileum; Male; Models, Animal; Myoelectric Complex, Migrating; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Stomach; Time Factors; Transducers, Pressure

2013