piboserod has been researched along with arecoline in 1 studies
Studies (piboserod) | Trials (piboserod) | Recent Studies (post-2010) (piboserod) | Studies (arecoline) | Trials (arecoline) | Recent Studies (post-2010) (arecoline) |
---|---|---|---|---|---|
119 | 5 | 53 | 1,110 | 20 | 271 |
Protein | Taxonomy | piboserod (IC50) | arecoline (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 3.6 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 1.011 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 0.963 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 0.963 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 0.963 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 0.9163 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 0.115 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Boulouard, M; Bureau, R; Butt-Gueulle, S; Dauphin, F; Daveu, C; Duchatelle, P; Dumuis, A; Lelong-Boulouard, V; LemaƮtre, S; Lepailleur, A; Lezoualc'h, F; Pfeiffer, B; Rault, S | 1 |
1 other study(ies) available for piboserod and arecoline
Article | Year |
---|---|
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
Topics: Animals; Chlorocebus aethiops; COS Cells; Humans; Indoles; Models, Molecular; Molecular Structure; Pyrazines; Radioligand Assay; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides | 2009 |