Page last updated: 2024-09-05

piboserod and alosetron

piboserod has been researched along with alosetron in 2 studies

Compound Research Comparison

Studies
(piboserod)
Trials
(piboserod)
Recent Studies (post-2010)
(piboserod)
Studies
(alosetron)
Trials
(alosetron)
Recent Studies (post-2010) (alosetron)
1195532263733

Protein Interaction Comparison

ProteinTaxonomypiboserod (IC50)alosetron (IC50)
Cytochrome P450 1A2Homo sapiens (human)5.3024
Cytochrome P450 3A4Homo sapiens (human)0.6
Cytochrome P450 2D6Homo sapiens (human)10
Cytochrome P450 2C9 Homo sapiens (human)10
Cytochrome P450 2B6Homo sapiens (human)10
Cytochrome P450 2C19Homo sapiens (human)10
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.1
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.068

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Axelsson, LG; Gillberg, PG; Hellström, PM; Sjöberg, B; Söderberg, C; Wallin, B1
Holzer, P; Painsipp, E; Shahbazian, A1

Other Studies

2 other study(ies) available for piboserod and alosetron

ArticleYear
Regulatory role of 5-HT and muscarinic receptor antagonists on the migrating myoelectric complex in rats.
    European journal of pharmacology, 2003, Apr-25, Volume: 467, Issue:1-3

    Topics: Animals; Atropine; Carbolines; Carboxylic Acids; Cyclopropanes; Dose-Response Relationship, Drug; Electromyography; Esters; Indoles; Intestine, Small; Muscarinic Antagonists; Myoelectric Complex, Migrating; Oxazines; Rats; Receptors, Muscarinic; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists

2003
Alosetron, cilansetron and tegaserod modify mesenteric but not colonic blood flow in rats.
    British journal of pharmacology, 2009, Volume: 158, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Carbazoles; Carbolines; Clonidine; Colitis; Colon; Fasting; Female; Heart Rate; Indoles; Mesenteric Artery, Superior; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pyridines; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Splanchnic Circulation; Vasoconstrictor Agents; Vasodilator Agents

2009