piboserod has been researched along with alosetron in 2 studies
Studies (piboserod) | Trials (piboserod) | Recent Studies (post-2010) (piboserod) | Studies (alosetron) | Trials (alosetron) | Recent Studies (post-2010) (alosetron) |
---|---|---|---|---|---|
119 | 5 | 53 | 226 | 37 | 33 |
Protein | Taxonomy | piboserod (IC50) | alosetron (IC50) |
---|---|---|---|
Cytochrome P450 1A2 | Homo sapiens (human) | 5.3024 | |
Cytochrome P450 3A4 | Homo sapiens (human) | 0.6 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 10 | |
Cytochrome P450 2C9 | Homo sapiens (human) | 10 | |
Cytochrome P450 2B6 | Homo sapiens (human) | 10 | |
Cytochrome P450 2C19 | Homo sapiens (human) | 10 | |
5-hydroxytryptamine receptor 2B | Homo sapiens (human) | 0.1 | |
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 3.068 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Axelsson, LG; Gillberg, PG; Hellström, PM; Sjöberg, B; Söderberg, C; Wallin, B | 1 |
Holzer, P; Painsipp, E; Shahbazian, A | 1 |
2 other study(ies) available for piboserod and alosetron
Article | Year |
---|---|
Regulatory role of 5-HT and muscarinic receptor antagonists on the migrating myoelectric complex in rats.
Topics: Animals; Atropine; Carbolines; Carboxylic Acids; Cyclopropanes; Dose-Response Relationship, Drug; Electromyography; Esters; Indoles; Intestine, Small; Muscarinic Antagonists; Myoelectric Complex, Migrating; Oxazines; Rats; Receptors, Muscarinic; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists | 2003 |
Alosetron, cilansetron and tegaserod modify mesenteric but not colonic blood flow in rats.
Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Carbazoles; Carbolines; Clonidine; Colitis; Colon; Fasting; Female; Heart Rate; Indoles; Mesenteric Artery, Superior; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pyridines; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Splanchnic Circulation; Vasoconstrictor Agents; Vasodilator Agents | 2009 |