Page last updated: 2024-09-04

phorbols and trifluoperazine

phorbols has been researched along with trifluoperazine in 13 studies

Compound Research Comparison

Studies
(phorbols)
Trials
(phorbols)
Recent Studies (post-2010)
(phorbols)
Studies
(trifluoperazine)
Trials
(trifluoperazine)
Recent Studies (post-2010) (trifluoperazine)
2,2170723,696157198

Protein Interaction Comparison

ProteinTaxonomyphorbols (IC50)trifluoperazine (IC50)
Genome polyprotein 0.7
Ubiquitin carboxyl-terminal hydrolase 1Homo sapiens (human)8
Bile salt export pumpHomo sapiens (human)10
Lysozyme C-1Rattus norvegicus (Norway rat)9
Beta-glucuronidaseRattus norvegicus (Norway rat)7.8
ATP-dependent translocase ABCB1Homo sapiens (human)6.75
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)6.226
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.35
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.35
Pleiotropic ABC efflux transporter of multiple drugsSaccharomyces cerevisiae S288C1.4
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.35
D(2) dopamine receptorRattus norvegicus (Norway rat)0.016
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)6.226
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)6.226
WD repeat-containing protein 48Homo sapiens (human)8

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-199013 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Eckhardt, L; Imamura, K; Kimura, T; Schulz, I1
Cohen, S; Goetz, JD; Grinstein, S; Rothstein, A1
Hagiwara, M; Hidaka, H; Inagaki, M; Saitoh, M1
Hebbert, D; Morgan, EH1
Abe, K; Adachi, I; Fujiki, H; Kimura, S; Nagasaki, K; Yamaguchi, K1
Murakami, H; Ohmura, E; Shizume, K; Tsushima, T; Wakai, K1
Smolen, JE; Weissmann, G1
Brostrom, CO; Brostrom, MA; Brotman, LA; Geller, HM; Lee, C; Wolff, DJ1
Becker, EL; Hill, JM; Huang, CK; Naccache, PH; Sha'afi, RI; White, JR1
Edwards, MC; Evans, FJ; Taylor, SE; Williamson, EM1
Iwashima, A; Nishino, H; Yamanishi, K1
Fujimura, S; Hiwasa, T; Sakiyama, S1
Froscio, M; Guy, GR; Murray, AW1

Other Studies

13 other study(ies) available for phorbols and trifluoperazine

ArticleYear
Ca2+-, phorbol ester-, and cAMP-stimulated enzyme secretion from permeabilized rat pancreatic acini.
    The American journal of physiology, 1986, Volume: 250, Issue:5 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Amylases; Animals; Calcium; Carbachol; Cell Membrane Permeability; Colforsin; Cyclic AMP; Cytoplasmic Granules; Digitonin; Egtazic Acid; Pancreas; Phorbols; Rats; Rats, Inbred Strains; Saponins; Spermine; Tetradecanoylphorbol Acetate; Trifluoperazine

1986
Osmotic and phorbol ester-induced activation of Na+/H+ exchange: possible role of protein phosphorylation in lymphocyte volume regulation.
    The Journal of cell biology, 1985, Volume: 101, Issue:1

    Topics: Adenosine Triphosphate; Amiloride; Animals; Calcium; Carrier Proteins; Cytoplasm; Diglycerides; Enzyme Activation; Lymphocytes; Male; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Rats; Rats, Inbred Strains; Sodium-Hydrogen Exchangers; Trifluoperazine; Water-Electrolyte Balance

1985
Protein kinase C negatively modulated by phorbol ester.
    FEBS letters, 1986, Jul-07, Volume: 202, Issue:2

    Topics: Adenosine Triphosphate; Animals; Calcium; Chlorpromazine; Diglycerides; Electrophoresis, Polyacrylamide Gel; Liver; Phorbols; Phospholipids; Phosphotransferases; Protein Kinase C; Protein Kinases; Swine; Tetradecanoylphorbol Acetate; Trifluoperazine

1986
Calmodulin antagonists inhibit and phorbol esters enhance transferrin endocytosis and iron uptake by immature erythroid cells.
    Blood, 1985, Volume: 65, Issue:3

    Topics: Adenosine Triphosphate; Animals; Calmodulin; Endocytosis; Exocytosis; Fetus; Iron; Liver; Phorbol Esters; Phorbols; Rabbits; Rats; Reticulocytes; Transferrin; Trifluoperazine

1985
Stimulation of hepatic glycogenolysis by 12-O-tetradecanoylphorbol-13-acetate (TPA) via a calcium requiring process.
    Biochemical and biophysical research communications, 1984, Aug-16, Volume: 122, Issue:3

    Topics: Animals; Calcimycin; Calcium Chloride; Cyclic AMP; Cyclic GMP; Diltiazem; Glucose; Kinetics; Liver; Liver Glycogen; Male; Phorbols; Proteins; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Trifluoperazine; Verapamil

1984
Effect of phorbol esters on the release of growth hormone and prolactin from rat pituitary cells cultured in monolayer.
    Acta endocrinologica, 1984, Volume: 107, Issue:2

    Topics: Animals; Calcium; Cells, Cultured; Growth Hormone; Hyaluronoglucosaminidase; Indomethacin; Male; Phorbol Esters; Phorbols; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Somatostatin; Trifluoperazine; Verapamil

1984
The effect of various stimuli and calcium antagonists on the fluorescence response of chlorotetracycline-loaded human neutrophils.
    Biochimica et biophysica acta, 1982, Apr-29, Volume: 720, Issue:2

    Topics: Calcium; Chlortetracycline; Concanavalin A; Egtazic Acid; Gallic Acid; Glucuronidase; Humans; Lysosomes; Muramidase; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oligopeptides; Phorbols; Spectrometry, Fluorescence; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate; Trifluoperazine; Vasodilator Agents

1982
Alterations of glial tumor cell Ca2+ metabolism and Ca2+-dependent cAMP accumulation by phorbol myristate acetate.
    The Journal of biological chemistry, 1982, Jun-25, Volume: 257, Issue:12

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Biological Transport, Active; Calcium; Cell Line; Cholera Toxin; Cyclic AMP; Glioma; Kinetics; Neoplasms, Experimental; Norepinephrine; Phorbols; Rats; Tetradecanoylphorbol Acetate; Trifluoperazine

1982
Effect of phorbol 12-myristate 13-acetate and its analogue 4 alpha-phorbol 12,13-didecanoate on protein phosphorylation and lysosomal enzyme release in rabbit neutrophils.
    The Journal of biological chemistry, 1984, Jul-10, Volume: 259, Issue:13

    Topics: Animals; Blood Proteins; Calcimycin; Carcinogens; Cytochalasin B; Kinetics; Lysosomes; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phorbol Esters; Phorbols; Phosphorylation; Protein Kinases; Rabbits; Tetradecanoylphorbol Acetate; Trifluoperazine

1984
New phorbol and deoxyphorbol esters: isolation and relative potencies in inducing platelet aggregation and erythema of skin.
    Acta pharmacologica et toxicologica, 1983, Volume: 53, Issue:3

    Topics: Animals; Chemical Phenomena; Chemistry; Erythema; Female; Humans; Imipramine; Male; Mice; Phorbol Esters; Phorbols; Plants; Platelet Aggregation; Promethazine; Propranolol; Rabbits; Trifluoperazine

1983
Possible role of calmodulin in stimulation of hexose transport by 12-O-tetradecanoylphorbol-13-acetate, a tumor promoter.
    Experientia, 1983, Sep-15, Volume: 39, Issue:9

    Topics: Animals; Biological Transport, Active; Calcium; Calcium-Binding Proteins; Calmodulin; Chick Embryo; Deoxy Sugars; Deoxyglucose; Fibroblasts; Kinetics; Phorbols; Tetradecanoylphorbol Acetate; Trifluoperazine

1983
Tumor promoters increase the synthesis of a 32,000-dalton protein in BALB/c 3T3 cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1982, Volume: 79, Issue:6

    Topics: Animals; Cell Line; Gene Expression Regulation; Mice; Molecular Weight; Phorbols; Protein Biosynthesis; Proteins; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic; Trifluoperazine

1982
Calmodulin inhibitors modify cell surface changes triggered by a tumor promoter.
    Biochemical and biophysical research communications, 1981, Feb-12, Volume: 98, Issue:3

    Topics: Animals; Calcium-Binding Proteins; Calmodulin; Cell Line; Cell Membrane; Choline; Epidermal Growth Factor; Epidermis; HeLa Cells; Humans; Membrane Lipids; Mice; Phorbols; Phospholipids; Tetradecanoylphorbol Acetate; Trifluoperazine

1981