Page last updated: 2024-09-04

phorbols and propranolol

phorbols has been researched along with propranolol in 7 studies

Compound Research Comparison

Studies
(phorbols)
Trials
(phorbols)
Recent Studies (post-2010)
(phorbols)
Studies
(propranolol)
Trials
(propranolol)
Recent Studies (post-2010) (propranolol)
2,21707233,3103,4063,218

Protein Interaction Comparison

ProteinTaxonomyphorbols (IC50)propranolol (IC50)
Beta-1 adrenergic receptor Cavia porcellus (domestic guinea pig)0.0347
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.294
Cytochrome P450 1A2Homo sapiens (human)4
Beta-2 adrenergic receptorHomo sapiens (human)0.0114
Beta-1 adrenergic receptorHomo sapiens (human)0.0575
5-hydroxytryptamine receptor 1AHomo sapiens (human)3.9811
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.012
Cytochrome P450 2D6Homo sapiens (human)2.9706
Beta-3 adrenergic receptorHomo sapiens (human)0.0493
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0288
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.012
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0827
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0288
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.012
5-hydroxytryptamine receptor 2AHomo sapiens (human)1.466
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.294
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.243
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0288
Sodium-dependent serotonin transporterHomo sapiens (human)0.38
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.342
5-hydroxytryptamine receptor 6Homo sapiens (human)3.065
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.017
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0288
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)2.828
Sodium channel protein type 5 subunit alphaHomo sapiens (human)2.1
Sodium/bile acid cotransporterHomo sapiens (human)5.5
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0288
GABA theta subunitRattus norvegicus (Norway rat)0.0288
Sigma non-opioid intracellular receptor 1Homo sapiens (human)2.87
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0288

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19907 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Choi, EJ; Toscano, WA1
Blackmore, PF; Bocckino, SB; Charest, R; Exton, JH; Lynch, CJ1
García-Sáinz, JA; Hernández-Sotomayor, SM; Tussié-Luna, MI1
Corvera, S; García-Sáinz, JA1
Edwards, MC; Evans, FJ; Taylor, SE; Williamson, EM1
Blumberg, PM; Castagna, M; Jaken, S; Nagle, DS1
Boutwell, RK; Conrad, EA; Kishore, GS; Perchellet, JP1

Other Studies

7 other study(ies) available for phorbols and propranolol

ArticleYear
Modulation of adenylate cyclase in human keratinocytes by protein kinase C.
    The Journal of biological chemistry, 1988, Nov-15, Volume: 263, Issue:32

    Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Cell Line; Epidermis; Humans; Isoproterenol; Keratins; Pertussis Toxin; Phorbol Esters; Phorbols; Propranolol; Protein Kinase C; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella

1988
Inhibition of hepatic alpha 1-adrenergic effects and binding by phorbol myristate acetate.
    The Journal of biological chemistry, 1985, Mar-10, Volume: 260, Issue:5

    Topics: Animals; Calcimycin; Calcium; Cyclic AMP; Dose-Response Relationship, Drug; Epinephrine; Glucagon; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Liver; Phentolamine; Phorbols; Phosphorylase a; Propranolol; Protein Kinase C; Protein Kinases; Rats; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate; Time Factors; Vasopressins

1985
Phorbol esters, vasopressin and angiotensin II block alpha 1-adrenergic action in rat hepatocytes. Possible role of protein kinase C.
    Biochimica et biophysica acta, 1986, Jun-16, Volume: 887, Issue:1

    Topics: Angiotensin II; Animals; Egtazic Acid; Epinephrine; Female; Gluconeogenesis; In Vitro Techniques; Kinetics; Liver; Liver Glycogen; Phorbols; Propranolol; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate; Urea; Vasopressins

1986
Phorbol esters inhibit alpha 1 adrenergic stimulation of glycogenolysis in isolated rat hepatocytes.
    Biochemical and biophysical research communications, 1984, Mar-30, Volume: 119, Issue:3

    Topics: Angiotensin II; Animals; Calcimycin; Epinephrine; Female; In Vitro Techniques; Kinetics; Liver; Liver Glycogen; Phorbols; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate; Urea; Vasopressins

1984
New phorbol and deoxyphorbol esters: isolation and relative potencies in inducing platelet aggregation and erythema of skin.
    Acta pharmacologica et toxicologica, 1983, Volume: 53, Issue:3

    Topics: Animals; Chemical Phenomena; Chemistry; Erythema; Female; Humans; Imipramine; Male; Mice; Phorbol Esters; Phorbols; Plants; Platelet Aggregation; Promethazine; Propranolol; Rabbits; Trifluoperazine

1983
Variation with embryonic development and regional localization of specific [3H]phorbol 12,13-dibutyrate binding to brain.
    Cancer research, 1981, Volume: 41, Issue:1

    Topics: Animals; Brain; Brain Mapping; Caenorhabditis elegans Proteins; Carrier Proteins; Cattle; Chick Embryo; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Propranolol; Protein Kinase C; Receptors, Drug

1981
Effects of cell surface receptor-altering agents on the binding and biological activity of 12-O-tetradecanoylphorbol-13-acetate in isolated epidermal cells.
    Carcinogenesis, 1982, Volume: 3, Issue:10

    Topics: alpha-L-Fucosidase; Animals; Atropine; Binding Sites; Binding, Competitive; Carboxy-Lyases; Cell Membrane; Cholera Toxin; G(M1) Ganglioside; Galactose Oxidase; Kinetics; Mice; Neuraminidase; Ornithine Decarboxylase; Phentolamine; Phorbols; Phospholipases; Propranolol; Skin; Tetradecanoylphorbol Acetate; Tretinoin

1982