Page last updated: 2024-09-04

phorbols and colforsin

phorbols has been researched along with colforsin in 25 studies

Compound Research Comparison

Studies
(phorbols)
Trials
(phorbols)
Recent Studies (post-2010)
(phorbols)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
2,21707213,460461,298

Protein Interaction Comparison

ProteinTaxonomyphorbols (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-199020 (80.00)18.7374
1990's3 (12.00)18.2507
2000's2 (8.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PE; Montgomery, BT; Tindall, DJ; Young, CY1
Eckhardt, L; Imamura, K; Kimura, T; Schulz, I1
Blackmore, PF; Exton, JH1
Brown, BL; Dobson, PR; Evans, DB; Russell, RG1
Niki, A; Niki, H; Tamagawa, T1
Houchi, H; Nakanishi, A; Ohuchi, T; Oka, M; Uddin, MM1
Kiss, Z; Steinberg, RA1
Ashby, B; Daniel, JL; Kowalska, MA; Rigmaiden, M; Smith, JB; Wernick, E1
Bohnet, HG; Brunswig, B; Budnik, LT; Leidenberger, FA; Mukhopadhyay, AK1
Daly, JW; Hollingsworth, EB; Ukena, D1
Goto, H; Kato, R; Uzumaki, H; Yamamoto, S1
Grubbs, RD; Maguire, ME1
Burke, G; Friedman, Y; Levasseur, S; Morgan, L1
Beinfeld, MC; Eiden, LE; Moskal, JR; Pruss, RM1
Aizawa, T; Hinkle, PM1
Mukhopadhyay, AK; Schumacher, M1
Bauer, S; Jakobs, KH; Watanabe, Y1
Dale, MM; Obianime, W1
Dannies, PS; Delbeke, D; Kojima, I; Rasmussen, H1
Forder, J; Kojima, I; Rasmussen, H; Scriabine, A1
Schorderet-Slatkine, S; Urner, F1
Ichikawa, K; Ito, M; Itoh, H; Konishi, T; Nakano, T; Okubo, S; Shimomura, A1
Amara, SG; Daniels, GM1
Dunlop, J; Hediger, MA; Peng, JB; Trotti, D1
Brueggemeier, RW; Díaz-Cruz, ES; Landini, S; Su, B1

Other Studies

25 other study(ies) available for phorbols and colforsin

ArticleYear
Tumor-promoting phorbol ester down-regulates the androgen induction of prostate-specific antigen in a human prostatic adenocarcinoma cell line.
    Cancer research, 1992, Mar-15, Volume: 52, Issue:6

    Topics: Alkaloids; Antigens, Neoplasm; Biomarkers, Tumor; Calcimycin; Colforsin; Dose-Response Relationship, Drug; Down-Regulation; Humans; Male; Nandrolone; Phorbols; Prostate-Specific Antigen; Prostatic Neoplasms; RNA, Messenger; Staurosporine; Testosterone Congeners; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured

1992
Ca2+-, phorbol ester-, and cAMP-stimulated enzyme secretion from permeabilized rat pancreatic acini.
    The American journal of physiology, 1986, Volume: 250, Issue:5 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Amylases; Animals; Calcium; Carbachol; Cell Membrane Permeability; Colforsin; Cyclic AMP; Cytoplasmic Granules; Digitonin; Egtazic Acid; Pancreas; Phorbols; Rats; Rats, Inbred Strains; Saponins; Spermine; Tetradecanoylphorbol Acetate; Trifluoperazine

1986
Studies on the hepatic calcium-mobilizing activity of aluminum fluoride and glucagon. Modulation by cAMP and phorbol myristate acetate.
    The Journal of biological chemistry, 1986, Aug-25, Volume: 261, Issue:24

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adrenergic alpha-Agonists; Aluminum; Aluminum Compounds; Angiotensin II; Calcium; Colforsin; Cyclic AMP; Drug Synergism; Fluorides; Glucagon; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Liver; Pertussis Toxin; Phorbols; Protein Kinase C; Sodium Fluoride; Tetradecanoylphorbol Acetate; Thionucleotides; Vasopressins; Virulence Factors, Bordetella

1986
Agents affecting adenylate cyclase activity modulate the stimulatory action of 1,25-dihydroxyvitamin D3 on the production of osteocalcin by human bone cells.
    Biochemical and biophysical research communications, 1989, Nov-15, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Alkaline Phosphatase; Bone and Bones; Bucladesine; Calcitriol; Cells, Cultured; Colforsin; Humans; Interleukin-1; Kinetics; Osteoblasts; Osteocalcin; Phorbols; Recombinant Proteins; Theophylline

1989
Insulin release independent of a rise in cytosolic free Ca2+ by forskolin and phorbol ester.
    FEBS letters, 1985, Apr-22, Volume: 183, Issue:2

    Topics: Animals; Calcium; Colforsin; Cyclic AMP; Digitonin; Diterpenes; Insulin; Islets of Langerhans; Male; Phorbols; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate

1985
Phorbol ester stimulates catecholamine synthesis in isolated bovine adrenal medullary cells.
    FEBS letters, 1985, Sep-02, Volume: 188, Issue:2

    Topics: Adrenal Medulla; Animals; Bucladesine; Calcium; Carbachol; Catecholamines; Cattle; Colforsin; Cyclic AMP; Diterpenes; Enzyme Activation; In Vitro Techniques; Phorbols; Protein Kinase C; Protein Kinases; Tetradecanoylphorbol Acetate; Tyrosine

1985
Interactions between cyclic AMP- and phorbol ester-dependent phosphorylation systems in S49 mouse lymphoma cells.
    Journal of cellular physiology, 1985, Volume: 125, Issue:2

    Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Drug Synergism; Lymphoma; Mice; Phorbols; Phosphorylation; Proteins; Tetradecanoylphorbol Acetate

1985
Differences in the mode of action of 1-oleoyl-2-acetyl-glycerol and phorbol ester in platelet activation.
    Journal of cyclic nucleotide and protein phosphorylation research, 1985, Volume: 10, Issue:5

    Topics: Adenylyl Cyclases; Apyrase; Blood Platelets; Blood Proteins; Colforsin; Cyclic AMP; Diglycerides; Glycerides; Humans; Kinetics; Papaverine; Phorbols; Phosphorylation; Platelet Aggregation; Tetradecanoylphorbol Acetate

1985
Phorbol ester stimulates progesterone production by isolated bovine luteal cells.
    Endocrinology, 1986, Volume: 118, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cattle; Cholera Toxin; Chorionic Gonadotropin; Colforsin; Corpus Luteum; Cyclic AMP; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Female; Kinetics; Luteal Cells; Phorbols; Progesterone; Protein Kinase C; Tetradecanoylphorbol Acetate

1986
The protein kinase C activator phorbol-12-myristate-13-acetate enhances cyclic AMP accumulation in pheochromocytoma cells.
    FEBS letters, 1986, Feb-03, Volume: 196, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Adrenal Gland Neoplasms; Animals; Cell Line; Colforsin; Cyclic AMP; Enzyme Activation; Pheochromocytoma; Phorbols; Phosphatidylinositols; Protein Kinase C; Rats; Stimulation, Chemical; Tetradecanoylphorbol Acetate

1986
Potentiation of prostaglandin E1-stimulated cAMP formation by 12-O-tetradecanoylphorbol-13-acetate in BALB/c mouse 3T3 cells.
    Biochemical pharmacology, 1986, Mar-01, Volume: 35, Issue:5

    Topics: Adenylyl Cyclases; Alprostadil; Animals; Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Kinetics; Mice; Phorbols; Tetradecanoylphorbol Acetate

1986
Regulation of magnesium but not calcium transport by phorbol ester.
    The Journal of biological chemistry, 1986, Sep-25, Volume: 261, Issue:27

    Topics: Animals; Biological Transport, Active; Calcium; Cell Line; Colforsin; Cyclic AMP; Isoproterenol; Kinetics; Lymphoma; Magnesium; Phorbols; Phosphorylation; Tetradecanoylphorbol Acetate

1986
Forskolin and 12-0-tetradecanoylphorbol-13-acetate mimic thyrotropin-stimulated protein iodination in mouse thyroid.
    Biochemical and biophysical research communications, 1985, Apr-30, Volume: 128, Issue:2

    Topics: Adenylyl Cyclases; Animals; Colforsin; Diterpenes; Female; Iodine; Mice; Phorbols; Protein Kinase C; Protein Kinases; Proteins; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin

1985
Specific regulation of vasoactive intestinal polypeptide biosynthesis by phorbol ester in bovine chromaffin cells.
    Endocrinology, 1985, Volume: 117, Issue:3

    Topics: Animals; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Colforsin; Diterpenes; Dose-Response Relationship, Drug; Enkephalin, Methionine; Enkephalins; Peptide Biosynthesis; Peptide PHI; Phorbols; Protein Precursors; RNA, Messenger; Tetradecanoylphorbol Acetate; Time Factors; Vasoactive Intestinal Peptide

1985
Differential effects of thyrotropin-releasing hormone, vasoactive intestinal peptide, phorbol ester, and depolarization in GH4C1 rat pituitary cells.
    Endocrinology, 1985, Volume: 116, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cells, Cultured; Colforsin; Diterpenes; Drug Synergism; Electrochemistry; Growth Hormone; Phorbols; Pituitary Gland; Potassium Chloride; Prolactin; Rats; Stimulation, Chemical; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Time Factors; Vasoactive Intestinal Peptide

1985
Inhibition of hCG-stimulated adenylate cyclase in purified mouse Leydig cells by the phorbol ester PMA.
    FEBS letters, 1985, Jul-22, Volume: 187, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Cholera Toxin; Chorionic Gonadotropin; Colforsin; Diterpenes; Guanylyl Imidodiphosphate; Leydig Cells; Male; Mice; Phorbols; Testosterone; Tetradecanoylphorbol Acetate

1985
Modulation of adenylate cyclase of human platelets by phorbol ester. Impairment of the hormone-sensitive inhibitory pathway.
    European journal of biochemistry, 1985, Sep-02, Volume: 151, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Alprostadil; Blood Platelets; Catalysis; Colforsin; Diterpenes; Enzyme Activation; Epinephrine; Guanosine Triphosphate; Humans; Phorbols; Prostaglandins E; Tetradecanoylphorbol Acetate; Thrombin

1985
Phorbol myristate acetate causes in guinea-pig lung parenchymal strip a maintained spasm which is relatively resistant to isoprenaline.
    FEBS letters, 1985, Oct-07, Volume: 190, Issue:1

    Topics: Aminophylline; Animals; Colforsin; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lung; Male; Muscle Contraction; Muscle, Smooth; Nitroprusside; Phorbols; Tetradecanoylphorbol Acetate

1985
Synergistic stimulation of prolactin release by phorbol ester, A23187 and forskolin.
    Biochemical and biophysical research communications, 1984, Sep-17, Volume: 123, Issue:2

    Topics: Animals; Calcimycin; Calcium; Cell Line; Colforsin; Cyclic AMP; Diterpenes; Drug Synergism; Phorbols; Pituitary Neoplasms; Prolactin; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Time Factors

1984
TPA-induced contraction of isolated rabbit vascular smooth muscle.
    Biochemical and biophysical research communications, 1984, Jul-31, Volume: 122, Issue:2

    Topics: Animals; Arteries; Calcimycin; Calcium; Colforsin; Diterpenes; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phorbols; Phosphorylation; Protein Kinases; Rabbits; Tetradecanoylphorbol Acetate

1984
Inhibition of denuded mouse oocyte meiotic maturation by tumor-promoting phorbol esters and its reversal by retinoids.
    Experimental cell research, 1984, Volume: 154, Issue:2

    Topics: Animals; Colforsin; Diterpenes; Drug Interactions; Female; Meiosis; Mice; Oocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Retinoids; Tetradecanoylphorbol Acetate

1984
Inhibition of myosin light chain phosphatase during Ca(2+)-independent vasocontraction.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 1

    Topics: Animals; Aorta, Thoracic; Calcium; Colforsin; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbols; Phosphates; Phosphoprotein Phosphatases; Phosphorus Radioisotopes; Rats; Rats, Wistar; Vasoconstriction; Vasodilator Agents

1993
Regulated trafficking of the human dopamine transporter. Clathrin-mediated internalization and lysosomal degradation in response to phorbol esters.
    The Journal of biological chemistry, 1999, Dec-10, Volume: 274, Issue:50

    Topics: Acetylcysteine; Animals; Carrier Proteins; Cell Line; Chloroquine; Clathrin; Colforsin; Cycloheximide; Dogs; Dopamine; Dopamine Plasma Membrane Transport Proteins; Endocytosis; Enzyme Activation; Humans; Kinetics; Lysosomes; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Phorbols; Protein Kinase C; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Transfection

1999
Inhibition of the glutamate transporter EAAC1 expressed in Xenopus oocytes by phorbol esters.
    Brain research, 2001, Sep-28, Volume: 914, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Amino Acid Transport System X-AG; Animals; Carcinogens; Carrier Proteins; Cell Membrane; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Transporter 3; Glutamate Plasma Membrane Transport Proteins; Glutamic Acid; Humans; Indoles; Maleimides; Membrane Potentials; Oocytes; Phorbols; Protein Kinase C; RNA, Complementary; Symporters; Tetradecanoylphorbol Acetate; Tritium; Tumor Cells, Cultured; Xenopus laevis

2001
Suppression of aromatase in human breast cells by a cyclooxygenase-2 inhibitor and its analog involves multiple mechanisms independent of cyclooxygenase-2 inhibition.
    Steroids, 2008, Volume: 73, Issue:1

    Topics: Aromatase; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Colforsin; Cyclooxygenase 2 Inhibitors; Dexamethasone; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Humans; Inhibitory Concentration 50; Microsomes; Molecular Structure; Nitrobenzenes; Phorbols; Sulfonamides; Testosterone

2008