phorbol 12,13-dibutyrate has been researched along with tetradecanoylphorbol acetate in 510 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 225 (44.12) | 18.7374 |
1990's | 250 (49.02) | 18.2507 |
2000's | 28 (5.49) | 29.6817 |
2010's | 7 (1.37) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Irie, K; Kamachi, H; Murakami, A; Nagai, H; Nakagawa, Y; Tanaka, K; Tokuda, H; Yanagita, RC | 1 |
Imoto, M; Irie, K; Kawamura, T; Matsubara, K; Otaka, H; Shindo, K; Tashiro, E; Yanagita, RC | 1 |
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P | 1 |
Blumberg, PM; Comin, MJ; Donadío, LG; Esch, TE; Garcia, LC; Hill, CS; Jelinek, R; Kedei, N; Kelley, JA; Kelsey, JS; Kolusheva, S; Lewin, NE; Mann, E; Marquez, VE; Peach, ML; Santos, M; Yang, J | 1 |
Costa, J; Delang, L; Leyssen, P; Litaudon, M; Neyts, J; Nothias-Scaglia, LF; Pannecouque, C; Paolini, J; Renucci, F; Roussi, F | 1 |
Boscá, L; Genaro, AM; Hortelano, S | 1 |
Miwa, J; Sassa, T | 1 |
el Benna, J; Hakim, J; Labro, MT | 1 |
Ansari, NA; Wu, MC | 1 |
Akhtar, RA; Wilmoth, TL | 1 |
Croatto, M; Hamilton, JA; Phillips, WA; Veis, N | 1 |
Davis, JS | 1 |
Chen, CC | 1 |
Brownsey, RW; Olivier, M; Reiner, NE | 1 |
Bourinet, E; Charnet, P; Fournier, F; Lory, P; Nargeot, J | 1 |
Horio, T; Kohno, M; Murakawa, K; Takeda, T; Yasunari, K; Yokokawa, K | 1 |
Herrero, I; Miras-Portugal, MT; Sánchez-Prieto, J | 1 |
Myers, CL; Parks, T; Schembri-King, J; Wallace, RW; Wertheimer, SJ | 1 |
Gibson, IC; Logan, SD | 1 |
Huebert, C; Kuszynski, C; Rizzino, A; Wilder, PJ | 1 |
Jentel, JJ; Lacson, RG; Oehler, DT; Unterman, TG | 1 |
Kapus, A; Ligeti, E; Szászi, K | 1 |
Brooks, G; Goss, MW; Hart, IR | 1 |
Cook, PP; Garris, TO; Messer, BR; Parker, PJ; Qin, W; Ways, DK | 1 |
Herembert, T; Marche, P; Zhu, DL | 1 |
Blumberg, PM; Kazanietz, MG; Krausz, KW | 1 |
Bajnath, RB; de Jonge, HR; Groot, JA; van Hoeve, MH | 1 |
Asano, S; Harigaya, K; Takahashi, S; Uchimaru, K; Yamashita, T | 1 |
Nakashima, T; Satoh, H; Tsuchida, K | 1 |
Byrne, JH; Critz, SD | 1 |
Moffat, MP; Ward, CA | 1 |
Hazama, K; Igarashi, K; Kikkawa, U; Nishizuka, Y; Ogita, K; Ono, Y; Taniyama, Y; Watanabe, T | 1 |
Alkhalaf, B; Gong, Y; Murphy, LC; Murphy, LJ | 1 |
Chen, ZH; Gopalakrishna, R; Gundimeda, U | 4 |
Alkon, DL; Etcheberrigaray, R; Lederhendler, II; Matzel, LD | 1 |
Meldrum, BS; Smith, SE | 1 |
Cook, PP; Parker, PJ; Ways, DK; Webster, C | 1 |
Chuang, LF; Chuang, RY; Israel, M; Kung, HF | 1 |
Bittman, R; Davenport, R; Dryden, P; Howard, S; Jones, K; Salari, H | 1 |
Elsas, LJ; Griffin, LD; Langley, SD; Longo, N | 1 |
Giridhar, G; Hayakawa, H; Kucera, L; Myrvik, QN | 1 |
Basu, A; Kozikowski, AP; Lazo, JS | 1 |
Raufman, JP | 1 |
Basu, A; Lazo, JS | 1 |
Azula, FJ; Font, J; Macarulla, JM; Marino, A; Nieva, N; Trueba, M | 1 |
Davis, PD; Nixon, JS; Sedgwick, AD; Wadsworth, J; Westmacott, D; Wilkinson, SE | 1 |
Logan, A; Logan, SD | 1 |
Walsh, KB | 1 |
Canessa, ML; Conlin, PR; Williams, GH | 1 |
Feldman, D; Krishnan, AV | 1 |
Bervig, T; Braden, TD; Conn, PM | 1 |
Ransjö, M | 1 |
Lerner, UH; Ransjö, M | 1 |
Suen, CS; Wilk, S | 2 |
Blanchard, LM; Larose, L; Morisset, J; Paquette, B | 1 |
Sekino, H; Suzuki-Nishimura, T; Uchida, MK | 1 |
Fuller, BB; Hoganson, GE; Niekrasz, I | 1 |
Malamed, S; Perez, FM; Scanes, CG | 1 |
Armstrong, L; Molony, L | 1 |
Crow, MT; Schwartz, RJ; Zhu, YY | 1 |
Alberola-Ila, J; Lozano, F; Places, L; Vives, J | 1 |
Henrich, CJ; Messing, RO; Petersen, PJ | 1 |
Casillas, T; Delicado, EG; Miras-Portugal, MT; Sen, RP | 1 |
Higuchi, H; Hiraoka, N; Ito, M; Itoh, H; Konishi, T; Lederis, K; Nakano, T | 1 |
Janik, P; Miłoszewska, J; Szaniawska, B | 1 |
Arita, H; Hanasaki, K; Kishi, M | 1 |
Hess, AD; Levine, BL; May, WS; Tyler, PG | 1 |
Albers, FJ; Caron, MG; Dennis, VW; Lefkowitz, RJ; Middleton, JP; Obeid, LM; Raymond, JR | 1 |
Endou, M; Hattori, Y; Kanno, M; Tohse, N | 1 |
Banks, P; Monk, PN | 1 |
Doré, M; Neilsen, NR; Slauson, DO | 1 |
O'Brian, CA; Ward, NE | 1 |
Kato, H; Ozawa, J; Takata, Y | 1 |
Brostrom, CO; Brostrom, MA; Gmitter-Yellen, D; Grandison, LJ; Kuznetsov, G; Prostko, CR; Wong, WL | 1 |
Alexander, RW; Clark, M; Griendling, KK; Lassègue, B | 1 |
Chang, JP; de Leeuw, R; Jobin, RM | 1 |
Baumann, D; Lester, DS | 1 |
Lauwerys, R; Lison, D; Raguzzi, F | 1 |
Bertrand, F; Capeau, J; Cherqui, G; Garcia, I; Hermelin, B; Paul, A; Picard, J | 1 |
Fabbro, D; Imber, R | 1 |
Dempsey, EC; McMurtry, IF; O'Brien, RF | 1 |
Braquet, P; Ferber, E; Fischer, G; Harell, T; Her, E; Naor, Z; Reiss, N; Zor, U | 1 |
Harmody, D; Longley, RE | 1 |
Ramsdell, JS | 1 |
Holian, O; Kumar, R | 1 |
Butler, AP; Mar, PK; McDonald, FF; Ramsay, RL | 1 |
Dong, ZY; Fan, D; Gupta, KP; O'Brian, CA; Ward, NE | 1 |
Gonzalez, FA; Heppel, LA; Huang, NN; Wang, DJ | 1 |
Brooks, G; Dooley, TP; Goss, MW; Hart, IR; Wilson, RE | 1 |
Burch, RM; Connor, JR; Shearer, BG; Sullivan, JP; Tiffany, C | 1 |
Malcolm, AR; Mills, LJ; Robson, DL | 1 |
Alkon, DL; Etcheberrigaray, R; Lederhendler, II; Matzel, LD; Yamoah, EN | 1 |
Olianas, MC; Onali, P | 1 |
Anderson, DJ; Naor, Z; Sigmund, O; Stein, R | 1 |
Goode, NT; Hart, IR; Moore, JP | 1 |
Johnson, JD; Walters, JD | 1 |
de Feijter, AW; de Haan, LH; Homan, EC; Jongen, WM; Spaaij, C; van Aelst, AC; van der Zandt, PT | 1 |
Buxbaum, JD; Cicchetti, P; Czernik, AJ; Ehrlich, ME; Fracasso, RP; Gandy, SE; Greengard, P; Ramabhadran, TV; Unterbeck, AJ | 1 |
Gross, JL; Horuk, R | 1 |
Dösemeci, A; Gaa, ST; Massey, C; Rogers, TB | 1 |
Hirst, JJ; Jenkin, G; Rice, GE; Thorburn, GD | 1 |
el-Fakahany, EE; Lai, WS; Rogers, TB | 1 |
Huang, CL; Ives, HE; Lowe, JH | 1 |
de Boland, AR; Norman, A | 1 |
Pfeffer, LM; Saltiel, AR; Strulovici, B | 1 |
Chao, W; Hanahan, DJ; Liu, H; Olson, MS | 1 |
Harnett, MM; Klaus, GG | 1 |
Burstein, DE; Lacal, JC; Pellicer, A; Thomson, TM; Trotta, RJ | 1 |
Parker, PJ; Schaap, D | 1 |
Brunsing, D; Hensel, G; Krönke, M; Meichle, A; Schütze, S | 1 |
Choladze, MA; Kondratyev, AD; Popova, ON; Posypanova, GA; Severin, ES; Severin, SE; Shmyrev, II; Tubasheva, IA; Zotova, EE | 1 |
Bhat, NK; Fisher, RJ; Fujiwara, S; June, CH; Koizumi, S; Lindsten, T; Papas, TS; Thompson, CB | 1 |
Abel, KC; Clark, MG; Cleland, PJ; Rattigan, S | 1 |
Duronio, V; Jacobs, S | 1 |
McCann, JA; Messina, JL | 1 |
Bayard, F; Darbon, JM; Issandou, M; Jozan, S; Valette, A | 1 |
Clark, JC; Fink, I; Hull, WM; O'Reilly, MA; Pryhuber, GS; Whitsett, JA | 1 |
Foucart, S; Majewski, H; Musgrave, IF | 2 |
Bishop, JF; Gehlert, DR; Patel, J; Vyas, S | 1 |
Buckley, NE; Gibson, K; Spiegel, S; Zhang, H | 1 |
Hannun, YA; Karolak, LA; Obeid, LM; Okazaki, T | 1 |
Fredholm, B; Gullberg, M; Jondal, M; Kvanta, A; Nordstedt, C | 1 |
Huang, FL; Huang, KP; Labourdette, G; Malviya, AN; Masmoudi, A; Rogue, P; Vincendon, G; Yoshida, Y; Zwiller, J | 1 |
Imaizumi, S; McGinn, MT; Mullin, JM; Snock, KV | 1 |
Goode, NT; Hart, IR | 1 |
Ahluwalia, M; Bazan, E; Garver, D; Gruenstein, E; Johnson, CG; Johnson, CL | 1 |
Leissner, J; Lindmar, R; Löffelholz, K; Sandmann, J | 1 |
Akita, Y; Konno, Y; Ohno, S; Suzuki, K; Yano, A | 1 |
Heffner, CH; Long, MW; Peters, C; Prochownik, EV; Williams, JL | 1 |
Larsen, CS | 1 |
Baglioni, C; Johnson, SE | 1 |
Kalberg, CJ; Sumners, C | 1 |
Akerlind, G; Akerman, KE; Heikkilä, J; Jalava, AM; Pettit, GR | 1 |
Godson, C; Insel, PA; Weiss, BA | 1 |
Basu, A; Lazo, JS; Teicher, BA | 1 |
Alterman, RL; Kornblith, PL; Maleci, A; Moskal, JR; Sundstrom, D | 1 |
Ikebuchi, H; Saito, Y; Suzuki, K; Suzuki, S; Terao, T | 1 |
Guitart, X; Marsal, J; Solsona, C | 1 |
Ashendel, CL; Beltran, L; Davis, MM; DiGiovanni, J; Hirabayashi, N; Petersen-Marht, S; Wang, XJ; Warren, BS | 1 |
Klein, B; Parant, MR; Vial, H | 1 |
García-Sáinz, JA; Hong, E; Ransanz, V; Torres-Márquez, ME; Villalobos-Molina, R | 1 |
Cronin, MJ; Perkins, SN; Summers, ST | 1 |
Hall, RE; Leftwich, JA | 1 |
Chida, K; Kato, N; Kuroki, T | 1 |
Pines, M; Santora, A; Spiegel, A | 1 |
Macdonald, RL; Werz, MA | 1 |
Boonstra, J; de Laat, SW; Ponec, M; Snoek, GT | 1 |
Brunden, KR; Poduslo, JF | 1 |
Chambaut-Guerin, AM; Thomopoulos, P | 1 |
Lebenthal, E; Lee, PC; Shimizu, K | 1 |
Emoto, T; Hiraiwa, M; Kasai, K; Shimoda, S | 1 |
Dale, MM; Hirst, SJ; Obianime, AW | 1 |
Obie, JF; Putney, JW; Sugiya, H | 1 |
Goto, Y; Sugamura, K; Takeshita, T | 1 |
Akai, H; Larner, AC | 1 |
Prives, J; Rapuano, M; Ross, AF | 1 |
Alonso, M; Cárdenas, L; Carrera, AC; de Landázuri, MO; Sánchez-Madrid, F; Tugores, A | 1 |
Billah, MM; Egan, RW; Mullmann, TJ; Pai, JK; Siegel, MI | 1 |
Judd, AM; Login, IS; MacLeod, RM | 1 |
Hartzell, P; Jondal, M; McConkey, DJ; Orrenius, S | 1 |
Anderson, WB; Gopalakrishna, R | 1 |
Kitajima, Y; Sheu, HM; Yaoita, H | 1 |
Chuang, DM; Dillon-Carter, O | 1 |
Cabot, MC; Cao, HT; Welsh, CJ; Zhang, ZC | 1 |
Ailhaud, G; Gaillard, D; Lagarde, M; Négrel, R | 1 |
Gillies, RJ; Hoyer, PB; Martinez, R; Sneider, JM | 1 |
Baur, U; Bühler, FR; Bürgin, M; Resink, TJ; Scott-Burden, T | 1 |
Badwey, JA; Curnutte, JT; Heyworth, PG; Robinson, JM | 1 |
Duddy, SK; Flodström, S; Hemming, H; Kass, GE; Wärngård, L | 1 |
Hagiwara, M; Hiai, H; Hidaka, H; Ito, M; Nishizuka, Y; Nunoki, K; Ohkubo, S; Ohta, H; Onoda, K; Tanaka, T | 1 |
Bazzi, MD; Nelsestuen, GL | 1 |
Folks, TM; Griffin, GE; Kunkel, S; Leung, K; Nabel, GJ | 1 |
Alexander, RW; Griendling, KK; Tsuda, T | 1 |
Conn, PM; McArdle, CA | 1 |
Long, MW | 1 |
Spiegel, S | 1 |
Fuller, SJ; Sugden, PH | 1 |
Inoue, Y; Rebois, RV | 1 |
Asou, H; Ikarashi, Y; Itoh, K; Maruyama, Y | 1 |
Aboolian, A; Nord, EP; Vander Molen, M | 1 |
Gautron, J; Martelly, I; Moraczewski, J | 1 |
Mauduit, P; Rossignol, B; Zoukhri, D | 1 |
Akerman, KE; Heikkilä, J | 1 |
Apovo, M; Beuzard, Y; Gascard, P; Giraud, F; Rhoda, MD | 1 |
Deaciuc, IV; Hermiller, JB; Mehegan, JP; Rodriguez de Turco, EB; Roth, BL; Spitzer, JA | 1 |
Alcantara, O; Boldt, DH; Denham, CA; Phillips, JL | 1 |
Alesse, E; Di Eugenio, R; Grazia Cifone, M; Morrone, S; Paolini, R; Procopio, A; Santoni, A; Santoni, G | 1 |
Flores-Romo, L; Foster, D; Gordon, J; Guy, GR | 1 |
Gárdos, G; Görög, G; Sarkadi, B; Tordai, A | 1 |
Malik, KU; Sehic, E | 1 |
Grove, DS; Mastro, AM | 1 |
Conn, PM; Huckle, WR; McArdle, CA | 1 |
Benedict, SH; Gelfand, EW; Lau, A; Mills, GB; Petsche, D; Schaffer, FM; Williams, BR | 1 |
Cronin, MJ; Sando, JJ; Summers, ST; Walker, JM | 1 |
Huhtaniemi, I; Nikula, H | 1 |
Fukumoto, Y; Hamamori, Y; Takai, Y; Tsuda, T; Yamashita, T | 1 |
Hirata, Y | 1 |
Akita, H; Fukuzaki, H; Go, M; Yokoyama, M | 1 |
Downer, RG; Gole, JW; Gupta, J; Orr, GL | 1 |
Allgaier, C; Hertting, G | 1 |
Araki, S; Fukuzaki, H; Kariya, K; Kawahara, Y; Takai, Y | 1 |
Fredholm, BB; Kvanta, A; Nordstedt, C | 1 |
Berlingieri, MT; Chiosi, E; Fusco, A; Grieco, M; Illiano, G; Spina, A | 1 |
Fondacaro, JD | 1 |
Jones, MJ; Murray, AW | 1 |
Cronin, MJ; Hewlett, EL; Sortino, MA; Summers, ST | 1 |
Janowsky, A; Labarca, R; Paul, SM | 1 |
Blumberg, PM; Herald, CL; Pettit, GR; Sako, T; Yuspa, SH | 1 |
Canonico, PL; Catania, MV; Favit, A; Nicoletti, F | 1 |
Andersson, T; Fällman, M; Stendahl, O | 1 |
Bauer, KD; Dunn, MM; Kamp, DW; Rubin, DB | 1 |
Bolard, J; Castagna, M; Frézard, F; Garnier-Suillerot, A | 1 |
Adams, JC; Gullick, WJ | 1 |
Chuang, LF; Chuang, RY; Israel, M; Zhao, FK | 1 |
Hurley, DJ; Mastro, AM | 1 |
Drummond, AH; MacIntyre, DE; McNicol, A | 1 |
Bell, RM; Czech, MP; Davis, RJ; Ganong, BR | 1 |
Civan, MM; Mauro, T; O'Brien, TG; Rubenstein, D | 1 |
Benveniste, R; Ilekis, J | 1 |
Patel, J; Rebois, RV | 1 |
Madshus, IH; Olsnes, S; Sandvig, K | 1 |
Fukuzaki, H; Kaibuchi, K; Kawahara, Y; Takai, Y; Tsuda, T | 1 |
Strnad, CF; Wong, K | 1 |
Chuang, DM | 1 |
Hamamori, Y; Kaibuchi, K; Kikuchi, A; Kozawa, O; Takai, Y | 1 |
Gainer, HS; Murray, AW | 1 |
Jetten, AM; Shirley, JE | 1 |
Bell, RM; Lambeth, JD; Merrill, AH; Olcott, MC; Wilson, E | 1 |
Adams, DO; Hamilton, TA; Johnston, PA | 1 |
Ginsberg, J; Murray, PG | 1 |
Beatty, PG; Gahmberg, CG; Nilsson, K; Patarroyo, M | 1 |
Enna, SJ; Karbon, EW; Shenolikar, S | 1 |
Ferber, E; Flesch, I | 1 |
Bonser, RW; Dawson, J; Garland, LG; Hodson, HF; Thompson, NT | 1 |
el-Fakahany, EE; Lai, WS | 1 |
Fishman, PH; Patel, J; Sullivan, M | 1 |
Cech, P; Cohen, LE; Lehrer, RI; Szklarek, D | 1 |
Kanno, Y; Sasaki, Y; Sastrodihardjo, S; Shiba, Y | 1 |
Acero, R; Erroi, A; Ghezzi, P; Mantovani, A; Salmona, M | 1 |
Cheng, YC; Grill, SP; Li, JS; Nutter, LM; Tan, RS | 1 |
Blumberg, PM; Bressler, JP; Frost, MM; Leach, KL | 1 |
Hamamori, Y; Nishimura, N; Takai, Y; Tsuda, T; Yamamoto, T | 1 |
Kaibuchi, K; Kikuchi, A; Takai, Y; Tanimoto, T; Tsuda, T; Yamashita, T | 1 |
Hunter, DD; Liles, WC; Meier, KE; Nathanson, NM | 1 |
Cavender, D; Haskard, D; Ziff, M | 1 |
Gerthoffer, WT | 1 |
Czech, MP; Davis, RJ | 1 |
Demers, LM; Veldhuis, JD | 1 |
Chadarevian, A; Pellegrini, M; Yamamoto, K | 1 |
Fink, G; Johnson, MS; Mitchell, R | 1 |
Hogans, BB; Spivak, JL | 1 |
Liskamp, RM; O'Brian, CA; Solomon, DH; Weinstein, IB | 1 |
Häring, HU; Kirsch, D; Obermaier, B | 1 |
Brown, EJ; Frank, MM; Gaither, TA; O'Shea, JJ; Takahashi, T | 1 |
Fernyhough, P; Hall, FL; Ishii, DN; Vulliet, PR | 1 |
Lytton, FD; Mitchell, MD | 1 |
Bell, RM; Davis, RJ; Faucher, M; Gironès, N; Hannun, YA | 1 |
Forsbeck, K; Ingelman-Sundberg, M; Nilsson, K; Patarroyo, M; Skoglund, G | 1 |
Allard, LR; Beinfeld, MC | 1 |
Anderson, D; Dewdney, RS; Soper, CJ | 1 |
Bogdanovic, RP; Brandes, LJ; Gerrard, JM; LaBella, FS; Lint, DW; Reid, RE | 1 |
Bennett, JL; Blair, KL; Pax, RA | 2 |
DiCorleto, PE; Uratsuji, Y | 1 |
Horiuchi, T; Kusaba, T; Mayumi, T; Nagasawa, K | 1 |
Consalvey, SD; Dexter, TM; Downes, CP; Huang, SJ; Monk, PN; Whetton, AD | 1 |
Bijsterbosch, MK; Holman, M; Klaus, GG; McLaughlin, JB | 1 |
Fujii, M; Goto, Y; Hinuma, Y; Iwami, M; Nakamura, M; Sugamura, K; Takeshita, T | 1 |
Bertrand, J; Capeau, J; Caron, M; Cherqui, G; Picard, J; Wicek, D | 1 |
Del Vecchio, PJ; Gudewicz, PW; Odekon, LE; Saba, TM | 1 |
Niedel, JE; Salehi, Z; Taylor, JD | 1 |
Barsky, SH; Gopalakrishna, R | 1 |
de Laat, SW; Mummery, CL; Snoek, GT; van den Brink, CE; van der Saag, PT | 1 |
Bayard, F; Darbon, JM; Valette, A | 1 |
Bell, RM; Hannun, YA; Kinkade, JM; Merrill, AH; Sereni, AM; Stevens, VL | 1 |
Balazovich, KJ; Boxer, LA; Smolen, JE | 1 |
Chatterjee, M; Tejada, M | 1 |
Hawkins, DJ; Miller, JR; Wells, JN | 1 |
Mullin, JM; O'Brien, TG | 1 |
Anderson, WB; Barsky, SH; Gopalakrishna, R; Thomas, TP | 1 |
Pettit, GR; Ramsdell, JS; Tashjian, AH | 1 |
Fukuzaki, H; Kariya, KI; Kawahara, Y; Takai, Y; Tsuda, T | 1 |
Hirning, LD; Matthies, HJ; Miller, RJ; Palfrey, HC | 1 |
Veldhuis, JD; Wheeler, MB | 1 |
Chobanian, MC; Hammerman, MR | 1 |
Aitken, A; Ellis, CA; Qureshi, N; Takayama, K | 1 |
Kariya, K; Takai, Y | 1 |
Hoult, JR; Nourshargh, S | 1 |
Bayard, F; Clamens, S; Darbon, JM; Oury, F | 1 |
Atherton, SE; Sando, JJ; Speizer, LA | 1 |
Abraham, I; Burnett, BA; Groppi, VE; Leach, KL; Mayo, JK; Powers, EA | 1 |
Dale, MM; Obianime, AW | 1 |
Fisher, GJ; Harris, VA; Voorhees, JJ | 1 |
Kolesnick, RN | 1 |
Cobbold, PH; Cuthbertson, KS; Woods, NM | 1 |
Blumberg, PM; Sharkey, NA | 1 |
McCulley, DE; Russell, JH; Taylor, AS | 1 |
Borner, C; Conscience, JF; Eppenberger, U; Erne, P; Fabbro, D; Mazurek, N; Regazzi, R; Wyss, R | 1 |
Fukumoto, Y; Fukuzaki, H; Kariya, K; Kawahara, Y; Takai, Y; Tsuda, T; Yamamoto, T | 1 |
de Groot, PG; Reinders, JH; van Mourik, JA; Vervoorn, RC; Verweij, CL | 1 |
Gordon, J; Guy, GR; Ledbetter, JA; Millsum, MJ | 1 |
Meldolesi, J; Pandiella, A; Vicentini, LM | 1 |
Gavin, JR; Hammerman, MR; Morrissey, JJ; Rogers, S | 1 |
Parker, PJ; Rodriguez-Pena, A; Rozengurt, E; Stabel, S; Young, S | 1 |
Tauber, AI | 1 |
Baylin, SB; Berger, CL; de Bustros, A; Leong, SS; Nelkin, BD; Roos, BA | 1 |
Aguelon-Pegouries, AM; Enomoto, T; Furstenberger, G; Marks, F; Martel, N; Yamasaki, H | 1 |
Gescher, A; Reed, DJ | 1 |
Bressler, JP; Kornblith, PL; Weingarten, D | 1 |
Degen, JL; Estensen, RD; Nagamine, Y; Reich, E | 1 |
Arcoleo, JP; Brothman, AR; Liskamp, RM; Miller, OJ; Weinstein, IB | 1 |
Stedman, DB; Welsch, F | 1 |
Finlay, TH; Kadner, SS; Katz, J; Levitz, M | 1 |
Chen, BD; Wilkins, KL | 1 |
Lefkowitz, RJ; Nambi, P; Sibley, DR | 1 |
Pettit, GR; Smith, JB; Smith, L | 1 |
Malcolm, AR; McKenna, EJ; Mills, LJ | 1 |
Carchman, RA; Lane, RW; Smith, BM; Sturm, RJ | 1 |
Adams, DO; Hamilton, TA; Rigsbee, JE; Scott, WA | 1 |
Blumberg, PM; Jeng, AY; Lichti, U; Strickland, JE | 1 |
Enomoto, T; Kanno, Y; Martel, N; Yamasaki, H | 1 |
Arcoleo, J; Backer, J; Gattoni-Celli, S; Hsiao, WL; Jeffrey, A; Kirschmeier, P; Okin, E; Weinstein, IB | 1 |
Blumberg, PM; Chritton, S; Lew, KK | 1 |
Enomoto, T; Kanno, Y; Martel, N; Shiba, Y; Yamasaki, H | 1 |
Kaibuchi, K; Kikkawa, U; Miyake, R; Nishizuka, Y; Tanaka, Y; Tsuda, T | 1 |
Dicker, P; Rozengurt, E | 1 |
Salomon, DS | 1 |
De Larco, JE; Shoyab, M; Todaro, GJ | 1 |
Dulbecco, R; Okada, S; Sonnenberg, A | 1 |
Jaken, S; Phillips, MA | 1 |
Fürstenberger, G; Marks, F; Sachs, L; Simantov, R | 1 |
Eisinger, M; Greenebaum, E; Nicolaides, M; Vogel, RH; Weinstein, IB | 1 |
Chang, J | 1 |
Colburn, NH; Dalal, B; Gindhart, TD; Hegamyer, GA | 1 |
Collins, M; McKay, I; Rozengurt, E; Taylor-Papadimitriou, J | 1 |
Chen, BD; Hsu, S; Lin, HS | 1 |
Carchman, RA; Harris, LS; Lane, RW; Laskin, DL; Smith, BM; Sturm, RJ | 1 |
Misukonis, MA; Weinberg, JB | 1 |
Fox, CF; Iwashita, S | 1 |
Kuhn, LJ; Niedel, JE; Vandenbark, GR | 1 |
Pastan, I; Werth, DK | 1 |
Craigmyle, LS; Licht, MR; Silverstein, SC; Wright, SD | 1 |
Besterman, JM; Cuatrecasas, P | 1 |
Estensen, RD; Mascioli, DW | 1 |
Isakson, PC; Simpson, L | 1 |
Peterfreund, RA; Vale, WW | 1 |
Baba, Y; Fujita, T; Ito, Y; Kobayashi, N; Matsuda, S; Morikawa, S; Nakao, Y; Saida, T; Watanabe, S | 1 |
Chida, K; Kuroki, T | 1 |
Anderson, NL; Callaham, MF; Gemmell, MA; Huberman, E; Murao, S | 1 |
Burczak, JD; Fairley, JL; Moskal, JR; Sweeley, CC; Trosko, JE | 1 |
Gahmberg, CG; Patarroyo, M | 1 |
Schorderet-Slatkine, S; Urner, F | 1 |
Janowsky, A; Labarca, R; Patel, J; Paul, SM | 1 |
Honikman-Leban, E; Moulé, Y | 1 |
Dawson, G; Golomb, HM; Lockney, MW | 1 |
Blumberg, PM; Jaken, S; Shupnik, MA; Tashjian, AH | 1 |
Bejarano, MT; Klein, E; Masucci, MG; Ramos, OF | 1 |
Hoffman, DR; Huberman, E | 1 |
Callaham, M; Huberman, E; Slaga, TJ; Solanki, V | 1 |
Cogan, U; Fisher, PB; Horowitz, AD; Schachter, D; Weinstein, IB | 1 |
Blumberg, PM; Butler-Gralla, E; Herschman, HR | 1 |
Callaham, M; Huberman, E; Slaga, T; Solanki, V; Weeks, C | 1 |
Guy, GR; Murray, AW | 1 |
Drevon, C; Martel, N; Yamasaki, H | 1 |
Farrar, JJ; Hilfiker, ML; Salomon, DS; Sando, JJ | 1 |
Blumberg, PM; Delclos, KB; Dunphy, WG; Jaken, S | 1 |
de Prost, D; Hakim, J; Khechai, F; Ollivier, V; Ramani, M; Ternisien, C; Vu, T | 1 |
Altman, A; Baier, G; Baier-Bitterlich, G; Bonnefoy-Berard, N; Burn, P; Coggeshall, KM; Gulbins, E; Langlet, C; Telford, D; Wittinghofer, A | 1 |
Mühl, H; Pfeilschifter, J | 1 |
Cano, C; Malik, KU; Slavik, KJ | 1 |
Nakamura, S; Nishizuka, Y; Ogita, K; Yamaguchi, K | 1 |
Fukao, M; Hattori, Y; Kanno, M; Kawasaki, H | 1 |
Arkhammar, P; Berggren, PO; Bertorello, AM; Efendić, S; Zaitsev, SV | 1 |
Snutch, TP; Soong, TW; Stea, A | 1 |
Mosior, M; Newton, AC | 1 |
Satoh, H | 2 |
Amon, U; Ramachers, U; von Stebut, E; Wolff, HH | 1 |
Daniel, EE; Kwan, CY; Shimamoto, H; Shimamoto, Y | 1 |
Haist, JV; Karmazyn, M | 1 |
Moallem, E; Naveh-Many, T; Silver, J | 1 |
Furukawa, Y; Kim, HN; Kubo, T | 1 |
Boulla, G; Gourdji, D; Passegue, E; Richard, JL | 1 |
Kunz, SS; Miller, KR; Wiest, PM | 1 |
Aharon, A; Kraiem, Z; Sadeh, O; Yosef, M | 1 |
Pan, M; Stevens, BR | 1 |
Akompong, T; Schonhorn, JE; Wessling-Resnick, M | 1 |
Godson, C; Li, SL; Prentki, M; Roche, E; Schlegel, W; Zhao, SJ | 1 |
Brunello, N; Perez, J; Racagni, G; Rovescalli, AC; Steardo, L; Vitali, S | 1 |
Cross, KM; Dunning, PM; Garland, CJ; Murphy, TV | 1 |
Schwartz, JH; Sossin, WS | 1 |
Smith, RD | 1 |
Hundle, B; Messing, RO; Roivainen, R | 1 |
Anderson, WB; Lehel, C; Mischak, H; Mushinski, JF; Olah, Z | 1 |
Chaki, S; Muramatsu, M; Otomo, S | 1 |
Hirano, T; Kitajima, K; Oda, T; Shimizu, N; Utiyama, H | 1 |
Brooks, G; East, JA; Goss, MW; Hart, IR | 1 |
Martin, J; Meenakshi, T; Ross, FP; Teitelbaum, SL | 1 |
Awtrey, CS; Hecht, G; Madara, JL; Matthews, JB; Tally, KJ; Thompson, RS | 1 |
Kuo, ML; Lee, KC; Lin, JK; Wu, WS | 1 |
Darcy, KM; Guan, X; Ip, MM; Wada, T | 1 |
Bazan, E; Campbell, AK; Rapoport, RM | 1 |
Fragio, C; Roldan, ER | 1 |
Bond, J; Dawson, T; Eccles, N; Wynford-Thomas, D | 1 |
Colucci, WS; Izzo, NJ; Tulenko, TN | 1 |
Fujishima, M; Hirata, M; Kosaka, C; Masuda, J; Ogata, J; Sasaguri, T; Shimokado, K | 1 |
Bean, BP; Lovinger, DM; Merritt, A; Swartz, KJ | 1 |
Fantus, IG; Nower, P; Schwartz, T; Torossian, K | 1 |
Cooper, DM; Yoshimura, M | 1 |
Hangai, K; Karibe, A; Keitoku, M; Takishima, T; Watanabe, J | 1 |
Detimary, P; Gao, ZY; Gembal, M; Gilon, P; Henquin, JC | 1 |
Rossignol, B; Sergheraert, C; Zoukhri, D | 1 |
McCabe, MJ; Orrenius, S | 1 |
Huber, G; Löffler, J | 1 |
Ching, KN; Nicholson, WE; Orth, DN; Won, JG | 1 |
Ashby, CR; Edwards, E; Wang, RY | 1 |
Nakano, R; Shimamoto, T; Yamoto, M | 1 |
Bullock, WW; Creamer, HR; Gabler, WL | 1 |
Celis, JE; Rasmussen, HH | 1 |
Craven, PA; DeRubertis, FR; Studer, RK | 1 |
Autrup, H; Christensen, B; Kieler, J; Skouv, J | 1 |
Hansen, H; Parissenti, AM; Riedel, H; Shieh, HL; Su, L | 1 |
Fredholm, BB; Lerner, UH; Ljunggren, O; Ljunghall, S; Nordstedt, C | 1 |
Chambers, TC; Chiou, SH; Kuo, JF; Raynor, RL; Zheng, B | 1 |
Kitamura, Y; Miyazaki, A; Nomura, Y | 1 |
Kruger, H; Shanley, BC; Wilce, PA | 1 |
Erusalimsky, JD; Hong, Y; Martin, JF; Vainchenker, W | 1 |
Birch, KA; Dell, C; Heath, WF; Hermeling, RN; Johnston, CM; Reifel-Miller, A; Smith, C; Stramm, L; Williamson, JR | 1 |
Benz, D; Möller, K; Perrin, D; Söling, HD | 1 |
Groen, AK; Klinkspoor, JH; Lee, SP; Tytgat, GN | 1 |
Galea-Lauri, J; Katz, DR; Latchman, DS | 1 |
Gong, MC; Jensen, PE; Somlyo, AP; Somlyo, AV | 1 |
Mills, J; Reiner, PB | 1 |
Kotsonis, P; Majewski, H | 1 |
Hori, M; Ikuhara, T; Isogai, Y; Matsuzaki, K; Nakamura, I; Suda, T; Suzuki, H; Takahashi, N | 1 |
Gaudette, GR; Kirvaitis, RJ; Krukenkamp, IB; Levitsky, S; Miyatake, T | 1 |
Boneh, A; Turgeman, D | 1 |
Kan, H; Malik, KU; Ruan, Y | 1 |
Bevan, JA; Laher, I; Xie, H | 1 |
Ball, SG; Goodall, AR; Turner, NA; Vaughan, PF; Walker, JH | 1 |
Acs, P; Blumberg, PM; Giese, T; Goodnight, J; Mischak, H; Mushinski, JF; Wang, QJ | 1 |
Haak, LL; Heller, HC; van den Pol, AN | 1 |
Bellamy, F; Nicolas, V; Riffaud, JP; Yablonsky, F | 1 |
Hsu, MF; Lin, CN; Raung, SL; Tsao, LT; Wang, JP | 1 |
Fu, WM; Lee, KF; Tang, YB | 1 |
Matthews, SA; Pettit, GR; Rozengurt, E | 1 |
Daniele, E; Lograno, MD; Villani, G | 1 |
Linde, C; Löffler, C; Quast, U | 1 |
Chelliah, J; Freemerman, AJ; Grant, S; Jarvis, WD; Wu-Pong, S | 1 |
Lin, CN; Raung, SL; Tsao, LT; Wang, JP | 1 |
Almazan, G; Larocca, JN | 1 |
Dent, G; Leff, AR; Magnussen, H; Muñoz, NM; Rabe, KF; Rühlmann, E; Zhu, X | 1 |
Han, Z; Patil, RV; Wax, MB | 1 |
Cox, A; Findlay, JB; Law, NM | 1 |
Locniskar, MF; Mouat, MF | 1 |
Garzaro, D; Kalvatchev, Z; Walder, R | 1 |
Compton, MM; Waldrip, HM | 1 |
Cubillos, S; Lima, L | 1 |
Ciereszko, RE; Guan, Z; Ottobre, AC; Ottobre, JS; Petroff, BK; Stokes, BT | 1 |
Groen, AK; Klinkspoor, JH; Lee, SP; Mok, KS; Tytgat, GN; Van Klinken, BJ | 1 |
Ezumi, Y; Takayama, H; Uchiyama, T | 1 |
Bełtowski, J; Górny, D; Marciniak, A | 1 |
Emiliozzi, C; Mograbi, B; Rochet, N; Rossi, B | 1 |
Dugué, B; Titievsky, A; Törnquist, K; Tuominen, R; Vainio, P | 1 |
Dessauer, CW; Hume, JR; Keef, KD; Zhong, J | 1 |
Walaas, SI | 1 |
Borowski, P; Kühl, R; Laufs, R; Medem, S; Roloff, S | 1 |
Alvarez, LJ; Candia, OA; Turner, HC; Zamudio, AC | 1 |
Belury, MA; Nickel, KP | 1 |
Dietz, R; Haller, H; Li, PF; Maasch, C; von Harsdorf, R | 1 |
Barbazuk, SM; Gold, MR | 1 |
Ford, BD; Ivy, MT; Mtshali, CP; Townsel, JG | 1 |
Kobayashi, H; Nakayama, T; Takami, Y; Wada, A; Yamamoto, R; Yanagita, T; Yokoo, H; Yuhi, T | 1 |
Iannazzo, L; Kotsonis, P; Majewski, H; Murphy, TV; Prountzos, C | 1 |
Inoue, T; Koono, M; Nabeshima, K; Shimao, Y | 1 |
Bienfait, B; Blumberg, PM; Fang, TW; Fenick, D; Garfield, S; Marquez, VE; Wang, QJ | 1 |
Oleskevich, S; Walmsley, B | 1 |
Checler, F; Frobert, Y; Grassi, J; Lehmann, S; Paitel, E; Vincent, B | 1 |
Brown, PD; Kajita, H; Whitwell, C | 1 |
Dartt, DA; Hodges, RR; Kanno, H; Ralda, N; Rawe, IM; Rios, JD; Rios, JR; Zieske, JD; Zoukhri, D | 1 |
Franceschi, RT; McCauley, LK; Ouyang, H; Somerman, MJ; Wang, D | 1 |
Asghar, M; Hussain, T; Lokhandwala, MF | 1 |
Charli, JL; Cisneros, M; Joseph-Bravo, P; Vargas, MA | 1 |
Checler, F; Creemers, J; Frank, SJ; Lopez-Perez, E; Seidah, N; Zhang, Y | 1 |
Ahmed, IS; Alderton, F; Darroch, P; McKie, A; Pyne, N; Pyne, S; Sambi, B | 1 |
Fujitani, K; Fukazawa, Y; Fukuda, T; Inokuchi, K; Isojima, Y; Kato, A; Sugiyama, H | 1 |
Balla, Z; Edes, I; Ferdinandy, P; Flameng, W; Mubagwa, K; Pongo, E; Szilvassy, Z | 1 |
Blumberg, PM; Fujii, T; Garcia-Bermejo, ML; Han, KC; Kazanietz, MG; Kuroki, T; Lee, J; Leskow, FC; Marquez, VE; Ohba, M; Wang, Q | 1 |
Chung, KH; Gye, MH; Shin, HJ; Yoo, BS | 1 |
Clark, JH; Glazer, RI; Haridasse, V | 1 |
Ciereszko, RE; Dusza, L; Kaminska, B; Opalka, M | 1 |
Iijima, T; Satoh, E; Xu, F | 1 |
Griese, A; Iakubov, R; Mischak, H; Riepenhausen, G; Schaefer, M; Schnell, S; Schöfl, C | 1 |
Korf, HW; Laedtke, E; Schomerus, C | 1 |
Bełtowski, J; Borkowska, E; Jamroz-Wiśniewska, A; Marciniak, A; Wójcicka, G | 1 |
Blumberg, PM; Braun, DC; Cao, Y; Garfield, SH; Hur, GM; Wang, S | 1 |
Anderson, G; Chen, J; Wang, QJ | 1 |
Basu, A; Huang, J; Mohanty, S | 1 |
Illsley, NP; You, G; Zhou, F | 1 |
Isacke, CM; Thorne, RF; Tzircotis, G | 1 |
Bond, JA; Errington, R; Gescher, AJ; Lemoine, NR; Smith, PJ; Verschoyle, RD; Wiltshire, M; Wynford-Thomas, D | 1 |
Förstermann, U; Goettsch, C; Horke, S; Li, H; Morawietz, H; Xia, N; Xu, H | 1 |
Anderson, SJ; Bashari, E; Benos, DJ; Fuller, CM; Kapoor, N; Meltzer, RH; Qadri, YJ; Zhou, ZH | 1 |
Arttamangkul, S; Birdsong, W; Williams, JT | 1 |
Boydens, C; Pauwels, B; Van de Voorde, J; Vanden Daele, L | 1 |
5 review(s) available for phorbol 12,13-dibutyrate and tetradecanoylphorbol acetate
Article | Year |
---|---|
Intestinal ion transport and diarrheal disease.
Topics: Acid-Base Equilibrium; Adrenergic alpha-Agonists; Animals; Arachidonic Acids; Carbachol; Chlorides; Cholera Toxin; Cyclic AMP; Cyclic GMP; Diarrhea; Electric Stimulation; Electrolytes; Hydroxyeicosatetraenoic Acids; Intestinal Absorption; Intestinal Mucosa; Intestine, Small; Leukotrienes; Models, Biological; Narcotics; Phenothiazines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Protein Kinase C; Receptors, Cholinergic; Receptors, Muscarinic; Renin-Angiotensin System; Sodium; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate | 1986 |
Protein kinase C and the activation of the human neutrophil NADPH-oxidase.
Topics: Arachidonic Acids; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Diglycerides; Enzyme Activation; Membrane Proteins; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate | 1987 |
Molecular mechanisms of tumor promotion and multistage carcinogenesis.
Topics: Adenosine Triphosphate; Animals; Base Sequence; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Transformation, Neoplastic; ErbB Receptors; Humans; Lyngbya Toxins; Molecular Conformation; Neoplasms; Oncogenes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1983 |
Epidermal growth factor receptors interact with transforming growth factors produced by certain human tumor cells and are distinct from specific membrane receptors for phorbol and ingenol esters.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Adhesion; Cell Line; Cell Transformation, Neoplastic; Cell Transformation, Viral; Cocarcinogenesis; ErbB Receptors; Humans; Neoplasms; Peptides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Transforming Growth Factors | 1982 |
Specific binding of phorbol ester tumor promoters to mouse tissues and cultured cells.
Topics: Animals; Biological Evolution; Brain; Caenorhabditis elegans Proteins; Calcium; Carcinogens; Carrier Proteins; Cell Membrane; Cells, Cultured; Humans; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Skin; Spleen; Structure-Activity Relationship; Temperature; Tetradecanoylphorbol Acetate; Thermodynamics | 1982 |
505 other study(ies) available for phorbol 12,13-dibutyrate and tetradecanoylphorbol acetate
Article | Year |
---|---|
Role of the phenolic hydroxyl group in the biological activities of simplified analogue of aplysiatoxin with antiproliferative activity.
Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Humans; Hydroxyl Radical; Lyngbya Toxins; Neoplasms; Protein Kinase C | 2010 |
Generation of 'Unnatural Natural Product' library and identification of a small molecule inhibitor of XIAP.
Topics: Antineoplastic Agents; Apoptosis; Biological Products; Caspase 3; Caspase Inhibitors; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Enzyme Activation; HeLa Cells; Humans; Imides; Indole Alkaloids; Lyngbya Toxins; Magnetic Resonance Spectroscopy; Molecular Structure; Protein Binding; Small Molecule Libraries; Stereoisomerism; Structure-Activity Relationship; X-Linked Inhibitor of Apoptosis Protein | 2011 |
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship | 2012 |
Synthesis, biological, and biophysical studies of DAG-indololactones designed as selective activators of RasGRP.
Topics: Animals; Cell Membrane; Cells, Cultured; CHO Cells; Cricetulus; Diglycerides; DNA-Binding Proteins; Fluorescence Polarization; Fluorescence Resonance Energy Transfer; Guanine Nucleotide Exchange Factors; HEK293 Cells; Humans; Indoles; Lactones; Male; Models, Molecular; Prostatic Neoplasms; Protein Isoforms; Protein Kinase C | 2014 |
Antiviral Activity of Diterpene Esters on Chikungunya Virus and HIV Replication.
Topics: Anti-HIV Agents; Antiviral Agents; Chikungunya virus; Diterpenes; DNA Replication; Esters; Euphorbiaceae; HIV Infections; HIV-1; HIV-2; Molecular Structure; Phorbol Esters; Tetradecanoylphorbol Acetate; Virus Replication | 2015 |
Phorbol esters induce nitric oxide synthase activity in rat hepatocytes. Antagonism with the induction elicited by lipopolysaccharide.
Topics: Amino Acid Oxidoreductases; Animals; Arginine; Calcimycin; Carcinogens; Cells, Cultured; Cyclic GMP; Diglycerides; Enzyme Induction; Kinetics; Lipopolysaccharides; Liver; Nitric Oxide Synthase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Rats; Tetradecanoylphorbol Acetate | 1992 |
Purification and characterization of protein kinase C from the nematode Caenorhabditis elegans.
Topics: Animals; Caenorhabditis; Calcium Chloride; Chromatography; Chromatography, Affinity; Chromatography, Ion Exchange; Diglycerides; Durapatite; Hydroxyapatites; Kinetics; Molecular Weight; Phorbol 12,13-Dibutyrate; Protein Kinase C; Substrate Specificity; Tetradecanoylphorbol Acetate | 1992 |
Inhibition of human neutrophil protein kinase C activity by the antimalarial drug mefloquine.
Topics: Dose-Response Relationship, Drug; Humans; Kinetics; Mefloquine; Neutrophils; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Respiratory Burst; Superoxides; Tetradecanoylphorbol Acetate | 1992 |
A phorbol diester resistant monocytic leukemia cell line is PKC deficient.
Topics: Animals; Blotting, Northern; Blotting, Western; Cell Division; Drug Resistance; Leukemia, Monocytic, Acute; Phorbol 12,13-Dibutyrate; Protein Kinase C; Proto-Oncogene Mas; Proto-Oncogene Proteins c-fos; Rats; Receptors, Cell Surface; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1992 |
Phorbol esters inhibit ionomycin-induced hydrolysis of phosphoinositides and phosphatidylcholine in bovine corneal epithelial cells.
Topics: Animals; Cattle; Chromatography, Ion Exchange; Chromatography, Thin Layer; Cornea; Enzyme Activation; Epithelium; Hydrolysis; Ionomycin; Phorbol 12,13-Dibutyrate; Phosphatidylcholines; Phosphatidylinositols; Protein Kinase C; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1992 |
Protein kinase C has both stimulatory and suppressive effects on macrophage superoxide production.
Topics: Alkaloids; Animals; Biological Transport; Bone Marrow Cells; Cells, Cultured; Cytokines; Dose-Response Relationship, Drug; Endotoxins; Granulocyte-Macrophage Colony-Stimulating Factor; Inositol Phosphates; Iodine Radioisotopes; Macrophages; Mice; Mice, Inbred CBA; Phorbol 12,13-Dibutyrate; Protein Kinase C; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate; Time Factors; Tumor Necrosis Factor-alpha; Zymosan | 1992 |
Modulation of luteinizing hormone-stimulated inositol phosphate accumulation by phorbol esters in bovine luteal cells.
Topics: Animals; Calcium; Cattle; Cyclic AMP; Dinoprost; Female; Inositol; Inositol Phosphates; Kinetics; Luteal Cells; Luteinizing Hormone; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Pregnancy; Progesterone; Sodium Fluoride; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1992 |
Differentiation of renal Na(+)-K(+)-ATPase in control and streptozotocin-induced diabetic mice by G-protein acting toxins and phorbol esters.
Topics: Adenylate Cyclase Toxin; Animals; Bucladesine; Cholera Toxin; Diabetes Mellitus, Experimental; Enzyme Activation; Kidney Cortex; Kidney Medulla; Male; Mice; Mice, Inbred ICR; Nicardipine; Ouabain; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1992 |
Defective stimulus-response coupling in human monocytes infected with Leishmania donovani is associated with altered activation and translocation of protein kinase C.
Topics: Animals; Blotting, Western; Caenorhabditis elegans Proteins; Carrier Proteins; Diglycerides; Enzyme Activation; Humans; Hydrogen Peroxide; In Vitro Techniques; Kinetics; Leishmania donovani; Monocytes; Oxygen Consumption; Phorbol 12,13-Dibutyrate; Phosphates; Phosphoproteins; Protein Kinase C; Receptors, Drug; Superoxides; Tetradecanoylphorbol Acetate | 1992 |
Protein kinase C regulation of cardiac calcium channels expressed in Xenopus oocytes.
Topics: Animals; Calcium Channels; Cyclic AMP; Diglycerides; Down-Regulation; Electrophysiology; Enzyme Activation; Myocardium; Oocytes; Phorbol 12,13-Dibutyrate; Protein Kinase C; RNA, Messenger; Tetradecanoylphorbol Acetate; Xenopus | 1992 |
Phorbol ester and atrial natriuretic peptide receptor response on vascular smooth muscle.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Atrial Natriuretic Factor; Cyclic GMP; Dose-Response Relationship, Drug; Down-Regulation; Guanylate Cyclase; Isoquinolines; Muscle, Smooth, Vascular; Natriuretic Peptide, Brain; Nerve Tissue Proteins; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Atrial Natriuretic Factor; Receptors, Cell Surface; Tetradecanoylphorbol Acetate | 1992 |
Activation of protein kinase C by phorbol esters and arachidonic acid required for the optimal potentiation of glutamate exocytosis.
Topics: 4-Aminopyridine; Animals; Arachidonic Acid; Cell Membrane; Drug Synergism; Electrophysiology; Enzyme Activation; Exocytosis; Glutamates; Glutamic Acid; Male; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1992 |
Induction of ICAM-1 by TNF-alpha, IL-1 beta, and LPS in human endothelial cells after downregulation of PKC.
Topics: Cell Adhesion Molecules; Cytokines; Endothelium, Vascular; Humans; Intercellular Adhesion Molecule-1; Interleukin-1; Lipopolysaccharides; Phorbol 12,13-Dibutyrate; Protein Kinase C; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1992 |
The actions of phorbol esters upon isolated calcium currents of Helix aspersa neurones.
Topics: Animals; Calcium; Calcium Channels; Helix, Snails; Membrane Potentials; Neurons; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1992 |
Effects of cell density and phorbol esters on the expression of epidermal growth factor receptors.
Topics: Cell Count; Cell Division; Cell Line; Epidermal Growth Factor; ErbB Receptors; Humans; KB Cells; Kinetics; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1991 |
Divergent effects of phorbol esters and insulin on insulin-like growth factor binding protein-1 (IGFBP-1) production and mRNA in rat H4IIE hepatoma cells.
Topics: Animals; Blotting, Northern; Carrier Proteins; DNA Probes; Insulin; Insulin-Like Growth Factor Binding Proteins; Insulin-Like Growth Factor I; Kinetics; Liver Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Phorbol 12-myristate 13-acetate activates an electrogenic H(+)-conducting pathway in the membrane of neutrophils.
Topics: Animals; Biological Transport; Cadmium; Cell Membrane; Cell Membrane Permeability; Chloromercuribenzoates; Hydrogen-Ion Concentration; Ion Channels; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; p-Chloromercuribenzoic Acid; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protons; Swine; Tetradecanoylphorbol Acetate; Valinomycin | 1992 |
Differential induction of 12-O-tetradecanoylphorbol-13-acetate sequence gene expression in murine melanocytes and melanoma cells.
Topics: 3T3 Cells; Animals; Blotting, Northern; Bucladesine; Cell Line, Transformed; Cells, Cultured; Cycloheximide; Gene Expression; Genes, fos; Melanocytes; Melanoma, Experimental; Mice; Molecular Weight; Phorbol 12,13-Dibutyrate; RNA; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1992 |
Modulation of protein kinase C-epsilon by phorbol esters in the monoblastoid U937 cell.
Topics: Cell Differentiation; Enzyme Activation; Enzyme Induction; Humans; Leukemia, Myeloid; Leukemia, Promyelocytic, Acute; Monocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Protein kinase C and cell proliferation in spontaneously hypertensive rats.
Topics: Animals; Aorta; Cell Division; Cells, Cultured; Dose-Response Relationship, Drug; Fibroblasts; Hypertension; Male; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Tetradecanoylphorbol Acetate; Thymidine | 1992 |
Differential irreversible insertion of protein kinase C into phospholipid vesicles by phorbol esters and related activators.
Topics: Animals; Binding Sites; Brain; Calcium; Enzyme Activation; Kinetics; Liposomes; Models, Structural; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phospholipids; Protein Binding; Protein Kinase C; Rats; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1992 |
Regulation of apical Cl- conductance and basolateral K+ conductances by phorbol esters in HT-29cl.19A cells.
Topics: Calcium; Carcinoma; Cell Membrane; Chlorides; Colforsin; Colonic Neoplasms; Electric Conductivity; Humans; Phorbol 12,13-Dibutyrate; Potassium; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Tumor necrosis factor and interleukin-1 induce activin A gene expression in a human bone marrow stromal cell line.
Topics: Activins; Blotting, Northern; Bone Marrow; Bone Marrow Cells; Cell Line; Culture Media, Conditioned; Cycloheximide; DNA; Gene Expression; Growth Substances; Humans; Inhibins; Interleukin-1; Macromolecular Substances; Phorbol 12,13-Dibutyrate; Protein Kinase C; Recombinant Proteins; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1992 |
The responses to phorbol esters which stimulated protein kinase C in canine Purkinje fibers.
Topics: Action Potentials; Animals; Calcium; Carcinogens; Dogs; Homeostasis; Microelectrodes; Myocardial Contraction; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Purkinje Fibers; Tetradecanoylphorbol Acetate | 1992 |
Modulation of IK,Ca by phorbol ester-mediated activation of PKC in pleural sensory neurons of Aplysia.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aplysia; Calcium; Dose-Response Relationship, Drug; Enzyme Activation; Ganglia; In Vitro Techniques; Isoquinolines; Kinetics; Membrane Potentials; Neurons, Afferent; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Piperazines; Potassium Channels; Protein Kinase C; Protein Kinase Inhibitors; Second Messenger Systems; Tetradecanoylphorbol Acetate; Tetraethylammonium; Tetraethylammonium Compounds | 1992 |
Positive and negative inotropic effects of phorbol 12-myristate 13-acetate: relationship to PKC-dependence and changes in [Ca2+]i.
Topics: Animals; Calcium; Enzyme Activation; Guinea Pigs; Heart; In Vitro Techniques; Intracellular Fluid; Male; Myocardial Contraction; Myocardium; Perfusion; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1992 |
Cell division arrest induced by phorbol ester in CHO cells overexpressing protein kinase C-delta subspecies.
Topics: Animals; Cell Cycle; Cell Division; CHO Cells; Cricetinae; DNA; Gene Amplification; Isoenzymes; Kinetics; Phorbol 12,13-Dibutyrate; Protein Binding; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Transfection | 1992 |
Differential effects of phorbol esters on proliferation and calcyclin expression in human endometrial carcinoma cells.
Topics: Adenocarcinoma; Alkaloids; Calcimycin; Calcium-Binding Proteins; Cell Cycle Proteins; Cell Division; Cycloheximide; Enzyme Activation; Female; Gene Expression Regulation, Neoplastic; Humans; Neoplasm Proteins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; RNA, Messenger; RNA, Neoplasm; S100 Calcium Binding Protein A6; S100 Proteins; Signal Transduction; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Uterine Neoplasms | 1992 |
Nonphorbol tumor promoters okadaic acid and calyculin-A induce membrane translocation of protein kinase C.
Topics: Animals; Carcinogens; Cell Line; Cell Membrane; Cytosol; Ethers, Cyclic; Immunoblotting; Kidney; Kinetics; Marine Toxins; Okadaic Acid; Oxazoles; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate | 1992 |
Classical conditioning and protein kinase C activation regulate the same single potassium channel in Hermissenda crassicornis photoreceptors.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Conditioning, Classical; Enzyme Activation; In Vitro Techniques; Isoquinolines; Membrane Potentials; Phorbol 12,13-Dibutyrate; Photoreceptor Cells; Piperazines; Potassium Channels; Protein Kinase C; Snails; Tetradecanoylphorbol Acetate | 1992 |
The protein kinase C activators, phorbol 12-myristate,13-acetate and phorbol 12,13-dibutyrate, are convulsant in the pico-nanomolar range in mice.
Topics: Alkaloids; Animals; Behavior, Animal; Convulsants; Enzyme Activation; Injections, Intraventricular; Male; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Seizures; Staurosporine; Tetradecanoylphorbol Acetate | 1992 |
Effect of phorbol esters on protein kinase C-zeta.
Topics: Amino Acid Sequence; Blotting, Western; Cell Line; Diglycerides; Down-Regulation; Electrophoresis, Polyacrylamide Gel; HeLa Cells; Humans; Isoenzymes; Molecular Sequence Data; Multigene Family; Phorbol 12,13-Dibutyrate; Protein Kinase C; Substrate Specificity; Tetradecanoylphorbol Acetate; Transfection | 1992 |
Activation of human leukemia protein kinase C by tumor promoters and its inhibition by N-trifluoroacetyladriamycin-14-valerate (AD 32).
Topics: Binding, Competitive; Cell Membrane; Doxorubicin; Drug Interactions; Enzyme Activation; Humans; Kinetics; Leukemia; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Binding; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Inhibition of protein kinase C by ether-linked lipids is not correlated with their antineoplastic activity on WEHI-3B and R6X-B15 cells.
Topics: Antineoplastic Agents; Cell Compartmentation; Cell Division; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Phorbol 12,13-Dibutyrate; Phospholipid Ethers; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Glucose transport by cultured human fibroblasts: regulation by phorbol esters and insulin.
Topics: 3-O-Methylglucose; Biological Transport; Cells, Cultured; Cycloheximide; Dactinomycin; Fibroblasts; Humans; Insulin; Kinetics; Methylglucosides; Phorbol 12,13-Dibutyrate; Protein Synthesis Inhibitors; Tetradecanoylphorbol Acetate | 1992 |
Pulmonary surfactant phospholipids modulate priming of rabbit alveolar macrophages for oxidative responses.
Topics: Animals; Fatty Acids; Female; Glycerylphosphorylcholine; Macrophage-Activating Factors; Macrophages, Alveolar; Male; Phagocytosis; Phorbol 12,13-Dibutyrate; Phospholipids; Pulmonary Surfactants; Rabbits; Respiratory Burst; Serum Albumin, Bovine; Tetradecanoylphorbol Acetate; Zymosan | 1992 |
Structural requirements of lyngbyatoxin A for activation and downregulation of protein kinase C.
Topics: Animals; Blotting, Western; Cattle; Down-Regulation; Enzyme Activation; HeLa Cells; Humans; Isoenzymes; Lyngbya Toxins; Marine Toxins; Phorbol 12,13-Dibutyrate; Protein Kinase C; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1992 |
Actions of phorbol esters on levels of cAMP in cholera toxin-treated chief cells from guinea pig stomach.
Topics: Animals; Calcimycin; Calmodulin; Carbachol; Cholera Toxin; Gastric Mucosa; Guinea Pigs; Imidazoles; In Vitro Techniques; Kinetics; Male; Phorbol 12,13-Dibutyrate; Phorbols; Signal Transduction; Sincalide; Tetradecanoylphorbol Acetate | 1992 |
Sensitization of human cervical carcinoma cells to cis-diamminedichloroplatinum(II) by bryostatin 1.
Topics: Antineoplastic Agents; Biological Transport; Bryostatins; Cell Division; Cell Line; Cisplatin; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Head and Neck Neoplasms; HeLa Cells; Humans; Isoenzymes; Kinetics; Lactones; Macrolides; Organoplatinum Compounds; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors | 1992 |
Intracellular Ca2+ mobilization and not calcium influx promotes phorbol ester-stimulated thromboxane A2 synthesis in human platelets.
Topics: Alkaloids; Blood Platelets; Calcimycin; Calcium; Chromatography, High Pressure Liquid; Cytosol; Drug Synergism; Humans; Membrane Lipids; Phorbol 12,13-Dibutyrate; Phospholipids; Platelet Aggregation; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Thromboxane A2 | 1992 |
Modulation of cellular processes by H7, a non-selective inhibitor of protein kinases.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Brain; CD4 Antigens; Cyclic AMP; Down-Regulation; Interleukin-2; Isoquinolines; Lymphocyte Activation; Mice; Molecular Weight; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Piperazines; Protein Kinase C; Protein Kinase Inhibitors; Rats; Receptors, Antigen, T-Cell; Staurosporine; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1991 |
Studies on the mechanisms of signalling and inhibition by pertussis toxin of fibroblast growth factor-stimulated mitogenesis in Balb/c 3T3 cells.
Topics: Adenylate Cyclase Toxin; Animals; Cells, Cultured; Cyclic AMP; Dexamethasone; DNA; Enzyme Activation; Fibroblast Growth Factors; Inositol Phosphates; Mice; Mice, Inbred BALB C; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1991 |
Activation of a heart chloride current during stimulation of protein kinase C.
Topics: Animals; Chloride Channels; Guinea Pigs; In Vitro Techniques; Membrane Proteins; Myocardium; Norepinephrine; Phorbol 12,13-Dibutyrate; Propranolol; Protein Kinase C; Tetradecanoylphorbol Acetate | 1991 |
Angiotensin II-induced activation of Na(+)-H+ exchange in adrenal glomerulosa cells is mediated by protein kinase C.
Topics: Aldosterone; Angiotensin II; Animals; Carrier Proteins; Cells, Cultured; Enzyme Activation; Kinetics; Phorbol 12,13-Dibutyrate; Protein Kinase C; Sodium-Hydrogen Exchangers; Tetradecanoylphorbol Acetate; Zona Glomerulosa | 1991 |
Activation of protein kinase-C inhibits vitamin D receptor gene expression.
Topics: Alkaloids; Animals; Blotting, Northern; Blotting, Southern; Calcimycin; Cell Division; Cells, Cultured; Diglycerides; Dose-Response Relationship, Drug; Down-Regulation; Fibroblast Growth Factor 2; Gene Expression Regulation, Enzymologic; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Calcitriol; Receptors, Steroid; RNA, Messenger; Staurosporine; Tetradecanoylphorbol Acetate | 1991 |
Protein kinase-C activation stimulates synthesis of gonadotropin-releasing hormone (GnRH) receptors, but does not mediate GnRH-stimulated receptor synthesis.
Topics: Amino Acids; Animals; Cells, Cultured; Enzyme Activation; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Cell Surface; Tetradecanoylphorbol Acetate | 1991 |
Protein kinase C activating phorbolesters enhance the cyclic AMP response to parathyroid hormone, forskolin and choleratoxin in mouse calvarial bones and rat osteosarcoma cells.
Topics: Adenylyl Cyclases; Animals; Bone and Bones; Cattle; Cholera Toxin; Colforsin; Culture Techniques; Cyclic AMP; Enzyme Activation; Mice; Osteosarcoma; Parathyroid Hormone; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1991 |
Effects of phorbol esters and pertussis toxin on calcitonin-stimulated accumulation of cyclic AMP in neonatal mouse calvarial bones.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Bone Resorption; Calcitonin; Cyclic AMP; Dinoprostone; GTP-Binding Proteins; Indomethacin; Mice; Osteoclasts; Parathyroid Hormone; Peptide Fragments; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1991 |
Inhibition of pyroglutamyl peptidase II synthesis by phorbol ester in the Y-79 retinoblastoma cell.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Cell Membrane; Humans; Immunoblotting; Isoquinolines; Kinetics; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Pyroglutamyl-Peptidase I; Retinoblastoma; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1991 |
Carbamylcholine and phorbol esters desensitize muscarinic receptors by different mechanisms in rat pancreatic acini.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amylases; Animals; Calcimycin; Carbachol; Dose-Response Relationship, Drug; Down-Regulation; Gallic Acid; Isoquinolines; Male; Pancreas; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Secretory Rate; Tetradecanoylphorbol Acetate | 1990 |
The modulatory effects of phorbol esters on histamine release from mast cells induced by a polyethylenimine and a polyallylamine.
Topics: Animals; Histamine Release; In Vitro Techniques; Male; Mast Cells; Molecular Weight; Phorbol 12,13-Dibutyrate; Phorbol Esters; Polyamines; Polyethyleneimine; Polyethylenes; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1990 |
Down-regulation of tyrosinase mRNA levels in melanoma cells by tumor promoters and by insulin.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Enzyme Induction; Gene Expression Regulation, Neoplastic; Insulin; Melanocyte-Stimulating Hormones; Melanoma, Experimental; Mice; Monophenol Monooxygenase; Phorbol 12,13-Dibutyrate; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Stimulation of chicken growth hormone release by phorbol esters.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Drug Interactions; Enzyme Activation; Growth Hormone; Growth Hormone-Releasing Hormone; Pancreas; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland, Anterior; Protein Kinase C; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone | 1990 |
Cytoskeletal reorganizations in human umbilical vein endothelial cells as a result of cytokine exposure.
Topics: Cell Adhesion Molecules; Cell Communication; Cysteine; Cytokines; Cytoskeletal Proteins; Cytoskeleton; Endothelium, Vascular; Fluorescent Antibody Technique; Humans; Immunoblotting; Interferon-gamma; Interleukin-1; Microtubules; Phorbol 12,13-Dibutyrate; Receptors, Immunologic; Receptors, Vitronectin; Sulfur Radioisotopes; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1991 |
Phorbol esters selectively downregulate contractile protein gene expression in terminally differentiated myotubes through transcriptional repression and message destabilization.
Topics: Animals; Cell Differentiation; Cell Nucleus; Cells, Cultured; Chick Embryo; Contractile Proteins; DNA Probes; Kinetics; Muscles; Phorbol 12,13-Dibutyrate; Protein Kinase C; RNA; RNA, Messenger; Tetradecanoylphorbol Acetate; Time Factors; Transcription, Genetic | 1991 |
Effect of protein kinase C activators on the phosphorylation and the surface expression of the CDw50 leukocyte antigen.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Antigens, CD; Antigens, Differentiation; Cell Adhesion Molecules; Concanavalin A; Cross-Linking Reagents; Diterpenes; Down-Regulation; Electrophoresis, Gel, Two-Dimensional; Enzyme Activation; Flow Cytometry; Fluorescent Antibody Technique; Humans; Isoquinolines; Kinetics; Lymphocytes; Phorbol 12,13-Dibutyrate; Phosphorylation; Phytohemagglutinins; Piperazines; Precipitin Tests; Protein Kinase C; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate | 1992 |
Chronic ethanol exposure increases levels of protein kinase C delta and epsilon and protein kinase C-mediated phosphorylation in cultured neural cells.
Topics: Amino Acid Sequence; Animals; Antibody Specificity; Diglycerides; Enzyme Activation; Ethanol; Immunoblotting; Kinetics; Molecular Sequence Data; Neurons; PC12 Cells; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate | 1991 |
Control of nucleoside transport in neural cells. Effect of protein kinase C activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine; Adrenal Medulla; Animals; Biological Transport; Calcimycin; Caprylates; Cells, Cultured; Diglycerides; Dinucleoside Phosphates; Enzyme Activation; Ethers, Cyclic; Isoquinolines; Kinetics; Okadaic Acid; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate; Triglycerides | 1991 |
Contraction of rat thoracic aorta strips by endothelin-1 in the absence of extracellular Ca2+.
Topics: Animals; Aorta, Thoracic; Caffeine; Calcium; Endothelins; In Vitro Techniques; Indicators and Reagents; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Phorbol 12,13-Dibutyrate; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Urotensins; Vasoconstrictor Agents | 1991 |
Phorbol binding and enzymatic activity of protein kinase C from C3H 10T1/2 cells and relation to contact inhibition.
Topics: Animals; Cells, Cultured; Contact Inhibition; Fibroblasts; Inositol Phosphates; Mice; Mice, Inbred C3H; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1991 |
Phorbol ester-induced expression of the common, low-affinity binding site for primary prostanoids in vascular smooth muscle cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aorta, Thoracic; Cells, Cultured; Enzyme Activation; Gene Expression Regulation; Isoquinolines; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Prostaglandin; Receptors, Thromboxane; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1991 |
Response of Jurkat T cells to phorbol ester and bryostatin. Development of sublines with distinct functional responses and changes in protein kinase C activity.
Topics: Antigens, CD; Antigens, Differentiation, T-Lymphocyte; Bryostatins; CD3 Complex; Clone Cells; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Activation; Humans; In Vitro Techniques; Lactones; Lymphocyte Activation; Macrolides; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Antigen, T-Cell; Receptors, Transferrin; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1991 |
5-HT1A and histamine H1 receptors in HeLa cells stimulate phosphoinositide hydrolysis and phosphate uptake via distinct G protein pools.
Topics: Biological Transport; Blotting, Northern; Down-Regulation; GTP-Binding Proteins; HeLa Cells; Histamine; Humans; Hydrolysis; Kinetics; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phosphates; Phosphatidylinositols; Phosphorylation; Protein Kinase C; Pyrilamine; Receptors, Histamine H1; Receptors, Serotonin; RNA, Messenger; Serotonin; Tetradecanoylphorbol Acetate; Transfection; Virulence Factors, Bordetella | 1991 |
Protein kinase C is not involved in alpha 1-adrenoceptor-mediated positive inotropic effect.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Electric Conductivity; Hydrolysis; Isoquinolines; Male; Membrane Potentials; Myocardial Contraction; Papillary Muscles; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Piperazines; Protein Kinase C; Protein Kinase Inhibitors; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Staurosporine; Stimulation, Chemical; Tetradecanoylphorbol Acetate | 1991 |
The role of protein kinase C activation and inositol phosphate production in the regulation of cell-surface expression of Mac-1 by complement fragment C5a.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium; Cell Line; Complement C5a; Cytoplasm; Enzyme Activation; Humans; Inositol Phosphates; Isoquinolines; Kinetics; Macrophage-1 Antigen; Oxygen; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Signal Transduction; Superoxides; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1991 |
Decreased respiratory burst activity in neonatal bovine neutrophils stimulated by protein kinase C agonists.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Animals, Newborn; Cattle; Cells, Cultured; Diglycerides; Dose-Response Relationship, Drug; Female; Isoquinolines; Neutrophils; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 1991 |
Distinct patterns of phorbol ester-induced downregulation of protein kinase C activity in adriamycin-selected multidrug resistant and parental murine fibrosarcoma cells.
Topics: Animals; Down-Regulation; Doxorubicin; Drug Resistance; Fibrosarcoma; In Vitro Techniques; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured | 1991 |
Presynaptic sites of isolated canine saphenous veins are more sensitive to protein kinase C than postsynaptic ones.
Topics: Animals; Dogs; Enzyme Activation; Female; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Phorbol 12,13-Dibutyrate; Polymyxin B; Potassium Chloride; Protein Kinase C; Saphenous Vein; Tetradecanoylphorbol Acetate; Tritium; Vasoconstriction | 1991 |
Inhibition of translational initiation by metalloendoprotease antagonists. Evidence for involvement of sequestered Ca2+ stores.
Topics: Amino Acid Sequence; Animals; Calcimycin; Calcium; Carrier Proteins; Cell Line; Cycloheximide; Dactinomycin; Dipeptides; Endoplasmic Reticulum Chaperone BiP; Heat-Shock Proteins; Immunoglobulin Heavy Chains; Inositol Phosphates; Kinetics; Leucine; Leupeptins; Metalloendopeptidases; Molecular Chaperones; Molecular Sequence Data; Oligopeptides; Peptide Chain Initiation, Translational; Phorbol 12,13-Dibutyrate; RNA, Messenger; Serine Endopeptidases; Tetradecanoylphorbol Acetate | 1991 |
Angiotensin II-induced phosphatidylcholine hydrolysis in cultured vascular smooth-muscle cells. Regulation and localization.
Topics: Angiotensin II; Animals; Aorta, Thoracic; Arsenicals; Cells, Cultured; Choline; Egtazic Acid; Hydrolysis; Kinetics; Male; Muscle, Smooth, Vascular; Myristic Acid; Myristic Acids; Phorbol 12,13-Dibutyrate; Phosphatidic Acids; Phosphatidylcholines; Phosphatidylethanolamines; Protein Kinases; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1991 |
Possible involvement of protein kinase C in gonadotropin and growth hormone release from dispersed goldfish pituitary cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Diglycerides; Egtazic Acid; Enzyme Activation; Goldfish; Gonadotropin-Releasing Hormone; Gonadotropins, Pituitary; Growth Hormone; Isoquinolines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Pituitary Gland; Protein Kinase C; Tetradecanoylphorbol Acetate; Verapamil | 1991 |
Action of organic solvents on protein kinase C.
Topics: Animals; Binding, Competitive; Diglycerides; Enzyme Activation; Histones; Lipid Bilayers; Male; Membrane Fluidity; Membranes, Artificial; Phorbol 12,13-Dibutyrate; Phosphatidylcholines; Phosphatidylserines; Phosphorylation; Protein Kinase C; Rats; Rats, Inbred Strains; Solvents; Tetradecanoylphorbol Acetate | 1991 |
Induction of macrophage plasminogen activator by asbestos is independent of PKC activation.
Topics: Animals; Asbestos; Auranofin; Cells, Cultured; Down-Regulation; Enzyme Activation; Macrophages; Mice; Phorbol 12,13-Dibutyrate; Plasminogen Activators; Protein Kinase C; Tetradecanoylphorbol Acetate | 1991 |
Further evidence for abnormal protein kinase C regulation of macromolecule secretion in fibroblasts from cystic fibrosis patients.
Topics: Binding Sites; Bucladesine; Calcimycin; Cells, Cultured; Colforsin; Cystic Fibrosis; Dose-Response Relationship, Drug; Fibroblasts; Glycoconjugates; Humans; Isoproterenol; Phorbol 12,13-Dibutyrate; Protein Kinase C; Skin; Tetradecanoylphorbol Acetate | 1990 |
Rapid inactivation and phosphorylation of pyroglutamyl peptidase II in Y-79 human retinoblastoma cells after exposure to phorbol ester.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Cell Line; Epinephrine; Eye Neoplasms; Humans; Immune Sera; Immunoblotting; Isoquinolines; Kinetics; Molecular Weight; Phorbol 12,13-Dibutyrate; Phosphorylation; Piperazines; Protein Kinase C; Pyroglutamyl-Peptidase I; Retinoblastoma; Sphingosine; Tetradecanoylphorbol Acetate | 1990 |
Tumor-promoting phorbol ester and activated Ha-ras synergistically reduce the interleukin 3 requirement in a mast cell line.
Topics: Animals; Blotting, Northern; Cell Division; Cell Line; Cell Transformation, Neoplastic; Genes, ras; Genetic Vectors; Interleukin-3; Mast Cells; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Restriction Mapping; Tetradecanoylphorbol Acetate; Transfection | 1991 |
Protein kinase C activation allows pulmonary artery smooth muscle cells to proliferate to hypoxia.
Topics: Aerobiosis; Anaerobiosis; Animals; Cattle; Cell Division; Cells, Cultured; Dimethyl Sulfoxide; DNA Replication; Enzyme Activation; Hypoxia; Kinetics; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Protein Kinase C; Pulmonary Artery; Tetradecanoylphorbol Acetate; Thymidine | 1991 |
Arachidonic acid release by basophilic leukemia cells and macrophages stimulated by Ca2+ ionophores, antigen and diacylglycerol: essential role for protein kinase C and prevention by glucocorticosteroids.
Topics: Alkaloids; Animals; Antigens; Arachidonic Acids; Calcimycin; Carbazoles; Cell Line; Cell Membrane; Cells, Cultured; Dexamethasone; Immunoglobulin E; Indole Alkaloids; Ionomycin; Kinetics; Leukemia, Basophilic, Acute; Leukemia, Experimental; Macrophages; Phorbol 12,13-Dibutyrate; Phospholipases A; Phospholipases A2; Protein Kinase C; Rats; Serum Albumin, Bovine; Staurosporine; Tetradecanoylphorbol Acetate | 1991 |
A rapid colorimetric microassay to detect agonists/antagonists of protein kinase C based on adherence of EL-4.IL-2 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Carcinogens; Cell Adhesion; Colorimetry; Diterpenes; Dose-Response Relationship, Drug; Enzyme Activation; Indoles; Isoquinolines; Lactams; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Reproducibility of Results; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate; Thymoma; Tumor Cells, Cultured | 1991 |
Transforming growth factor-alpha and -beta are potent and effective inhibitors of GH4 pituitary tumor cell proliferation.
Topics: Activins; Animals; Cell Adhesion; Cell Count; Cell Division; DNA; Inhibins; Interphase; Mitosis; Phorbol 12,13-Dibutyrate; Pituitary Neoplasms; Prolactin; Protein Kinase C; Rats; Recombinant Proteins; S Phase; Tetradecanoylphorbol Acetate; Transforming Growth Factor alpha; Transforming Growth Factor beta; Tumor Cells, Cultured | 1991 |
Inhibition of mouse skin protein kinase C by benzoyl peroxide.
Topics: Animals; Benzoyl Peroxide; Calcium; Enzyme Activation; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Skin; Tetradecanoylphorbol Acetate | 1991 |
Involvement of protein kinase C in the regulation of ornithine decarboxylase mRNA by phorbol esters in rat hepatoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Diglycerides; Down-Regulation; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Isoquinolines; Liver Neoplasms, Experimental; Ornithine Decarboxylase; Palmitoylcarnitine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Protein Kinase Inhibitors; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1991 |
In vitro model for intrinsic drug resistance: effects of protein kinase C activators on the chemosensitivity of cultured human colon cancer cells.
Topics: Antineoplastic Agents; Colonic Neoplasms; Diglycerides; Doxorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Enzyme Activation; Humans; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Vincristine | 1991 |
Multiple signal transduction pathways lead to extracellular ATP-stimulated mitogenesis in mammalian cells: I. Involvement of protein kinase C-dependent and -independent pathways.
Topics: Adenosine Triphosphate; Animals; Bombesin; Carcinoma, Squamous Cell; Cell Line; Diglycerides; DNA; Down-Regulation; Drug Synergism; Enzyme Activation; Fibroblasts; Glycerides; Humans; Mice; Mitosis; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylcholines; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Vasopressins; Virulence Factors, Bordetella | 1991 |
Protein kinase C down-regulation, and not transient activation, correlates with melanocyte growth.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Division; Cell Line; Enzyme Activation; Kinetics; Melanocytes; Melanoma, Experimental; Mice; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1991 |
NPC 15437 interacts with the C1 domain of protein kinase C. An analysis using mutant PKC constructs.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amino Acid Sequence; Animals; Binding Sites; Cell Line; DNA Mutational Analysis; Isoquinolines; Macromolecular Substances; Molecular Sequence Data; Mutation; Phorbol 12,13-Dibutyrate; Piperazines; Piperidines; Protein Conformation; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1991 |
Interactive effects of aldrin, cyclohexylamine, 2,4-diaminotoluene and two phorbol esters on metabolic cooperation between V79 cells.
Topics: Aldrin; Cell Communication; Cells, Cultured; Cyclohexylamines; Drug Synergism; Phenylenediamines; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1991 |
Outgrowths from Hermissenda photoreceptor somata are associated with activation of protein kinase C.
Topics: Animals; Calcium; Cell Membrane; Enzyme Activation; In Vitro Techniques; Learning; Mollusca; Phorbol 12,13-Dibutyrate; Photoreceptor Cells; Potassium Channels; Protein Kinase C; Tetradecanoylphorbol Acetate | 1990 |
Alteration of the GTP-dependent inhibitory pathway of rat striatal adenylate cyclase by phorbol esters.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Corpus Striatum; GTP Phosphohydrolases; Guanosine Triphosphate; Hydrolysis; Male; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1990 |
Effect of nerve growth factor and fibroblast growth factor on SCG10 and c-fos expression and neurite outgrowth in protein kinase C-depleted PC12 cells.
Topics: Adrenal Gland Neoplasms; Animals; Axons; Cell Line; Diglycerides; Fibroblast Growth Factors; Gene Expression Regulation; Nerve Growth Factors; Pheochromocytoma; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Proto-Oncogenes; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1990 |
Selection and preliminary characterization of variant lines of a murine macrophage tumor resistant to the antiproliferative effects of phorbol esters.
Topics: Animals; Cell Division; Dimethyl Sulfoxide; Drug Resistance; Enzyme Activation; Macrophages; Molecular Weight; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Terbium as a luminescent probe of metal-binding sites in protein kinase C.
Topics: Binding Sites; Binding, Competitive; Egtazic Acid; Energy Transfer; Humans; Luminescent Measurements; Metals; Phorbol 12,13-Dibutyrate; Phosphatidylserines; Protein Kinase C; Spectrophotometry; Terbium; Tetradecanoylphorbol Acetate | 1990 |
Effects of cigarette smoke condensate and 12-O-tetradecanoylphorbol-13-acetate on gap junction structure and function in cultured cells.
Topics: Animals; Caenorhabditis elegans Proteins; Calcium Chloride; Carrier Proteins; Cells, Cultured; Chick Embryo; Diglycerides; Egtazic Acid; Freeze Fracturing; Intercellular Junctions; Kinetics; Liver; Microscopy, Electron; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Drug; Smoke; Smoking; Tetradecanoylphorbol Acetate | 1990 |
Processing of Alzheimer beta/A4 amyloid precursor protein: modulation by agents that regulate protein phosphorylation.
Topics: Adrenal Gland Neoplasms; Alzheimer Disease; Amyloid; Amyloid beta-Protein Precursor; Animals; Cell Line; Ethers, Cyclic; Humans; Kinetics; Methionine; Molecular Weight; Okadaic Acid; Pheochromocytoma; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Biosynthesis; Protein Kinase C; Protein Precursors; Protein Processing, Post-Translational; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1990 |
Protein kinase C-linked inactivation of the interleukin-1 receptor in a human transformed B-cell line.
Topics: B-Lymphocytes; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Cell Membrane; Enzyme Activation; Humans; Interleukin-1; Kinetics; Lymphoma; Phorbol 12,13-Dibutyrate; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Receptors, Interleukin-1; Recombinant Proteins; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Protein kinase C inhibits Ca2+ accumulation in cardiac sarcoplasmic reticulum.
Topics: Animals; Animals, Newborn; Biological Transport; Calcium; Calcium Radioisotopes; Cells, Cultured; Cyclic AMP; Myocardial Contraction; Myocardium; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred Strains; Ryanodine; Sarcoplasmic Reticulum; Tetradecanoylphorbol Acetate | 1990 |
Regulation of oxytocin secretion by the ovine corpus luteum: effect of activators of protein kinase C.
Topics: Animals; Bucladesine; Calcimycin; Corpus Luteum; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Female; In Vitro Techniques; Oxytocin; Phorbol 12,13-Dibutyrate; Platelet Activating Factor; Protein Kinase C; Pyrimidinones; Sheep; Tetradecanoylphorbol Acetate; Thiazoles; Type C Phospholipases | 1990 |
Protein kinase C is involved in desensitization of muscarinic receptors induced by phorbol esters but not by receptor agonists.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Carbachol; Cyclic GMP; Down-Regulation; Isoquinolines; Mice; N-Methylscopolamine; Neuroblastoma; Parasympathomimetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Receptors, Muscarinic; Scopolamine Derivatives; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Sphingosine differentially inhibits activation of the Na+/H+ exchanger by phorbol esters and growth factors.
Topics: Animals; Animals, Newborn; Biological Transport; Carrier Proteins; Cells, Cultured; Detergents; Diglycerides; Hydrogen-Ion Concentration; Kinetics; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Platelet-Derived Growth Factor; Rats; Sodium-Hydrogen Exchangers; Sphingosine; Tetradecanoylphorbol Acetate; Thrombin | 1990 |
Evidence for involvement of protein kinase C and cyclic adenosine 3',5' monophosphate-dependent protein kinase in the 1,25-dihydroxy-vitamin D3-mediated rapid stimulation of intestinal calcium transport, (transcaltachia).
Topics: Alkaloids; Animals; Biological Transport; Calcitriol; Calcium; Chickens; Colforsin; Cyclic AMP; Duodenum; Intestinal Mucosa; Intestines; Kinetics; Male; Nifedipine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinases; Staurosporine; Tetradecanoylphorbol Acetate; Verapamil; Vitamin D Deficiency | 1990 |
Interferon-alpha selectively activates the beta isoform of protein kinase C through phosphatidylcholine hydrolysis.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cytosol; Diglycerides; Enzyme Activation; HeLa Cells; Humans; Hydrolysis; Interferon Type I; Isoenzymes; Kinetics; Phorbol 12,13-Dibutyrate; Phosphatidylcholines; Protein Kinase C; Receptors, Drug; Recombinant Proteins; Tetradecanoylphorbol Acetate; Vesicular stomatitis Indiana virus | 1990 |
Regulation of platelet-activating factor receptor and PAF receptor-mediated arachidonic acid release by protein kinase C activation in rat Kupffer cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cells, Cultured; Dimethyl Sulfoxide; Down-Regulation; Enzyme Activation; Kinetics; Kupffer Cells; Phorbol 12,13-Dibutyrate; Platelet Activating Factor; Platelet Membrane Glycoproteins; Protein Kinase C; Rats; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Tetradecanoylphorbol Acetate | 1990 |
Cross-talk between B cell surface immunoglobulin and interleukin 4 receptors: the role of protein kinase C and Ca2(+)-mediated signals.
Topics: Animals; Antibodies, Monoclonal; B-Lymphocytes; Calcium; DNA; Flow Cytometry; Lymphocyte Activation; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Protein Kinase C; Receptors, Antigen, B-Cell; Receptors, Interleukin-4; Receptors, Mitogen; Signal Transduction; Tetradecanoylphorbol Acetate | 1990 |
Potentiation of oncogenic N-ras-induced neurite outgrowth and ornithine decarboxylase activity by phorbol dibutyrate and protein kinase inhibitor H-8.
Topics: Animals; Cell Differentiation; Cell Transformation, Neoplastic; Colforsin; Dexamethasone; Epidermal Growth Factor; Isoquinolines; Nerve Growth Factors; Neurons; Oncogene Protein p21(ras); Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinase Inhibitors; Rats; Tetradecanoylphorbol Acetate; Tretinoin; Tumor Cells, Cultured | 1990 |
Expression, purification, and characterization of protein kinase C-epsilon.
Topics: Alkaloids; Animals; Cell Line; Chromatography, Affinity; Chromatography, Gel; Chromatography, Ion Exchange; Diglycerides; DNA; Enzyme Activation; Insect Viruses; Insecta; Isoenzymes; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Plasmids; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate | 1990 |
Protein kinase C-independent activation of nuclear factor kappa B by tumor necrosis factor.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Base Sequence; Binding Sites; Cell Line; DNA-Binding Proteins; DNA, Viral; Down-Regulation; Enhancer Elements, Genetic; Enzyme Activation; H-2 Antigens; HIV-1; Humans; Isoquinolines; Leukemia; Molecular Sequence Data; NF-kappa B; Phorbol 12,13-Dibutyrate; Piperazines; Promoter Regions, Genetic; Protein Kinase C; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Transcription Factors; Tumor Necrosis Factor-alpha | 1990 |
Nerve growth factor stimulates protein kinase C translocation in PC12 cells.
Topics: Adrenal Gland Neoplasms; Animals; Cell Line; Fluorescent Antibody Technique; Immunoblotting; Nerve Growth Factors; Pheochromocytoma; Phorbol 12,13-Dibutyrate; Protein Binding; Protein Kinase C; Subcellular Fractions; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Reciprocal expression of human ETS1 and ETS2 genes during T-cell activation: regulatory role for the protooncogene ETS1.
Topics: Calcium; Cells, Cultured; DNA Probes; DNA-Binding Proteins; Enzyme Activation; Gene Expression Regulation; Genes, Regulator; Humans; Ionomycin; Lymphocyte Activation; Models, Biological; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein-Tyrosine Kinases; Proto-Oncogene Protein c-ets-1; Proto-Oncogene Protein c-ets-2; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-ets; Proto-Oncogenes; Repressor Proteins; RNA, Messenger; T-Lymphocytes; Tetradecanoylphorbol Acetate; Trans-Activators; Transcription Factors; Transcription, Genetic | 1990 |
Long-term treatment of isolated rat soleus muscle with phorbol ester leads to loss of contraction-induced glucose transport.
Topics: Animals; Biological Transport; Female; Glucose; Glycogen; In Vitro Techniques; Insulin; Muscle Contraction; Muscles; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1990 |
The effect of protein kinase-C inhibition on insulin receptor phosphorylation.
Topics: Alkaloids; Cell Line; Down-Regulation; Electrophoresis, Gel, Two-Dimensional; Insulin; Peptide Mapping; Phorbol 12,13-Dibutyrate; Phosphorylation; Phosphoserine; Phosphothreonine; Protein Kinase C; Receptor, Insulin; Staurosporine; Tetradecanoylphorbol Acetate; Trypsin | 1990 |
Interaction of insulin and phorbol esters on the regulation of DNA synthesis in rat hepatoma cells.
Topics: Animals; Cell Line; DNA Replication; DNA, Neoplasm; Insulin; Kinetics; Liver Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Rats; Tetradecanoylphorbol Acetate; Thymidine | 1990 |
Dissociation between protein kinase C content and biological responsiveness to phorbol esters in tumor promoter-sensitive (MCF-7) and resistant (RPh-4) cells.
Topics: Animals; Cell Division; Cell Line; Cell Separation; Drug Resistance; Flow Cytometry; Models, Biological; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Subcellular Fractions; Tetradecanoylphorbol Acetate | 1990 |
Phorbol ester inhibits surfactant protein SP-A and SP-B expression.
Topics: Adenocarcinoma; Cell Line; Dactinomycin; Enzyme-Linked Immunosorbent Assay; Glycoproteins; Humans; Kinetics; L-Lactate Dehydrogenase; Lung Neoplasms; Methionine; Phorbol 12,13-Dibutyrate; Protein Binding; Proteolipids; Pulmonary Surfactant-Associated Protein A; Pulmonary Surfactant-Associated Proteins; Pulmonary Surfactants; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1990 |
Inhibition of noradrenaline release by neuropeptide Y does not involve protein kinase C in mouse atria.
Topics: Animals; Carbazoles; Electric Stimulation; Enzyme Activation; Female; Heart; Heart Atria; In Vitro Techniques; Indole Alkaloids; Mice; Neuropeptide Y; Norepinephrine; Phorbol 12,13-Dibutyrate; Polymyxin B; Protein Kinase C; Tetradecanoylphorbol Acetate; Tritium | 1990 |
Effects of protein kinase C down-regulation on secretory events and proopiomelanocortin gene expression in anterior pituitary tumor (AtT-20) cells.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Cell Membrane; Cytosol; Gene Expression Regulation; Genes; Homeostasis; Kinetics; Phorbol 12,13-Dibutyrate; Phosphorylation; Pituitary Neoplasms; Pro-Opiomelanocortin; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Sphingosine stimulates cellular proliferation via a protein kinase C-independent pathway.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Cell Division; Cell Line; DNA; Down-Regulation; Drug Synergism; Fibroblasts; Growth Substances; Isoquinolines; Phorbol 12,13-Dibutyrate; Phosphorylation; Piperazines; Protein Kinase C; Sphingosine; Tetradecanoylphorbol Acetate | 1990 |
Transcriptional regulation of protein kinase C by 1,25-dihydroxyvitamin D3 in HL-60 cells.
Topics: Caenorhabditis elegans Proteins; Calcitriol; Carrier Proteins; Cell Line; Gene Expression Regulation, Enzymologic; Genes; Humans; Kinetics; Leukemia, Promyelocytic, Acute; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Drug; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1990 |
Evidence that protein kinase C activation is essential for killing by IL-2-activated lymphocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Chromium Radioisotopes; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Humans; Interleukin-2; Isoquinolines; Killer Cells, Lymphokine-Activated; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Piperazines; Protein Kinase C; Recombinant Proteins; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Rat liver nuclei protein kinase C is the isozyme type II.
Topics: Animals; Cell Nucleus; Chromatography, DEAE-Cellulose; Chromatography, Ion Exchange; Electrophoresis, Polyacrylamide Gel; Immunoblotting; Isoenzymes; Kinetics; Liver; Molecular Weight; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate | 1990 |
The effects of teleocidin and aplysiatoxin tumor promoters on epithelial tight junctions and transepithelial permeability: comparison to phorbol esters.
Topics: Carcinogens; Cells, Cultured; Dose-Response Relationship, Drug; Epithelium; Intercellular Junctions; Lyngbya Toxins; Permeability; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1990 |
Protein kinase C levels and protein phosphorylation associated with inhibition of proliferation in a murine macrophage tumor.
Topics: Animals; Cell Division; Diglycerides; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Activation; Isoelectric Point; Macrophages; Mice; Molecular Weight; Phorbol 12,13-Dibutyrate; Phosphoproteins; Protein Kinase C; Sarcoma, Experimental; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured | 1990 |
Histamine receptors in human fibroblasts: inositol phosphates, Ca2+, and cell growth.
Topics: Aminopyridines; Calcium; Cell Division; Cell Line; DNA Replication; Fibroblasts; Fluorescent Dyes; Histamine; Humans; Inositol Phosphates; Kinetics; Phorbol 12,13-Dibutyrate; Pyrilamine; Receptors, Histamine; Skin; Tetradecanoylphorbol Acetate; Thymidine | 1990 |
The effects of phorbol esters on choline phospholipid hydrolysis in heart and brain.
Topics: Animals; Brain Chemistry; Chickens; Heart; Hydrolysis; In Vitro Techniques; Male; Myocardium; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylcholines; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1990 |
A point mutation at the putative ATP-binding site of protein kinase C alpha abolishes the kinase activity and renders it down-regulation-insensitive. A molecular link between autophosphorylation and down-regulation.
Topics: Adenosine Triphosphate; Animals; Base Sequence; Cell Line; Cytosol; DNA; Genetic Vectors; Homeostasis; Molecular Sequence Data; Mutation; Oligonucleotide Probes; Phorbol 12,13-Dibutyrate; Phosphorylation; Plasmids; Protein Kinase C; Rats; Subcellular Fractions; Tetradecanoylphorbol Acetate | 1990 |
Regulation of megakaryocyte phenotype in human erythroleukemia cells.
Topics: Antigens; Cell Differentiation; Cell Division; Cell Fusion; Humans; Interphase; Leukemia, Erythroblastic, Acute; Megakaryocytes; Phenotype; Phorbol 12,13-Dibutyrate; Protein Kinase C; Proto-Oncogene Mas; Proto-Oncogenes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Activation of human T lymphocytes by phorbol-12,13-dibutyrate and ionomycin.
Topics: Antibodies, Monoclonal; Calcium; Drug Synergism; Humans; Ionomycin; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Phytohemagglutinins; Protein Kinase C; Receptors, Interleukin-2; T-Lymphocytes; Tetradecanoylphorbol Acetate; Time Factors | 1990 |
Positive and negative regulation of a tumor necrosis factor response in melanoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cell Line; DNA Probes; Female; Humans; Isoquinolines; Kinetics; Melanoma; Phorbol 12,13-Dibutyrate; Piperazines; Plasminogen Activators; Plasminogen Inactivators; Pregnancy; Protein Kinase Inhibitors; Recombinant Proteins; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1990 |
Regulation of angiotensin II binding sites in neuronal cultures by protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Angiotensin II; Animals; Animals, Newborn; Brain Stem; Cells, Cultured; Homeostasis; Hypothalamus; Isoquinolines; Kinetics; Neurons; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetradecanoylphorbol Acetate | 1990 |
Effects of bryostatins 1 and 2 on morphological and functional differentiation of SH-SY5Y human neuroblastoma cells.
Topics: Antineoplastic Agents; Bryostatins; DNA, Neoplasm; Down-Regulation; Enzyme Induction; Humans; Lactones; Macrolides; Neuroblastoma; Norepinephrine; Oncogenes; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Muscarinic; RNA, Messenger; RNA, Neoplasm; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Differential activation of protein kinase C alpha is associated with arachidonate release in Madin-Darby canine kidney cells.
Topics: Animals; Arachidonic Acids; Bradykinin; Cell Line; Diglycerides; Dogs; Enzyme Activation; Kidney; Kinetics; Phorbol 12,13-Dibutyrate; Phospholipids; Protein Kinase C; Tetradecanoylphorbol Acetate | 1990 |
Involvement of protein kinase C in phorbol ester-induced sensitization of HeLa cells to cis-diamminedichloroplatinum(II).
Topics: Cell Division; Cell Line; Cell Survival; Cisplatin; HeLa Cells; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Effect of phorbol esters on the susceptibility of a glioma cell line to lymphokine-activated killer cell activity.
Topics: Cell Division; Glioma; Humans; Killer Cells, Lymphokine-Activated; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Tetradecanoylphorbol Acetate; Thymidine; Tumor Cells, Cultured | 1990 |
Human growth hormone-stimulated growth of human cultured lymphocytes (IM-9) and its inhibition by phorbol diesters through down-regulation of the hormone receptors. Possible involvement of phosphorylation of a 55,000 molecular weight protein associated wi
Topics: Alkaloids; Blood; Cell Division; Cell Line; Down-Regulation; Enzyme Activation; Growth Hormone; Humans; Kinetics; Lymphocytes; Molecular Weight; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphoproteins; Phosphorylation; Protein Kinase C; Receptors, Somatotropin; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate | 1990 |
Phorbol esters induce neurotransmitter release in cholinergic synaptosomes from Torpedo electric organ.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetylcholine; Animals; Botulinum Toxins; Dose-Response Relationship, Drug; Electric Organ; Isoquinolines; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Potassium Chloride; Protein Kinase C; Synaptosomes; Tetradecanoylphorbol Acetate; Torpedo | 1990 |
Partial characterization of epidermal protein kinase C in mice sensitive or resistant to phorbol ester.
Topics: Animals; Binding Sites; Biological Transport; Down-Regulation; Drug Resistance; Female; Isoenzymes; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Protein Kinase C; Skin; Species Specificity; Tetradecanoylphorbol Acetate | 1990 |
Abnormal behavior of protein kinase C in the human myeloma cell line, RPMI 8226.
Topics: Animals; Brain; Cell Fractionation; Cell Line; Cell Membrane; Chromatography, DEAE-Cellulose; Cytosol; Humans; Kinetics; Multiple Myeloma; Phorbol 12,13-Dibutyrate; Protein Binding; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Time Factors | 1990 |
Contrasting effects of phorbol dibutyrate and phorbol myristate acetate in rabbit aorta.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aorta; Cells, Cultured; Epinephrine; In Vitro Techniques; Isoquinolines; Liver; Muscle Contraction; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phosphates; Phosphatidylinositols; Piperazines; Protein Kinase Inhibitors; Rabbits; Tetradecanoylphorbol Acetate | 1990 |
Beta-adrenergic stimulation of anterior pituitary cyclic AMP is enhanced by tumor promoters.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland, Anterior; Protein Kinase C; Rats; Receptors, Adrenergic, beta; Tetradecanoylphorbol Acetate | 1985 |
Enhancement of phorbol diester-induced HL-60-mediated cytotoxicity by retinoic acid, dimethyl sulfoxide, and 5-azacytidine.
Topics: Azacitidine; Cell Differentiation; Cell Line; Cytotoxicity, Immunologic; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Leukemia, Myeloid, Acute; Macrophages; Monocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate; Tretinoin | 1986 |
Down regulation of phorbol diester receptors by proteolytic degradation of protein kinase C in a cultured cell line of fetal rat skin keratinocytes.
Topics: Animals; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Cell Line; Chromatography, Gel; Cytosol; Diglycerides; Female; Keratins; Leupeptins; Molecular Weight; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Pregnancy; Protein Kinase C; Rats; Receptors, Drug; Receptors, Immunologic; Skin; Tetradecanoylphorbol Acetate; Tosyllysine Chloromethyl Ketone; Tosylphenylalanyl Chloromethyl Ketone | 1986 |
Effects of phorbol esters and pertussis toxin on agonist-stimulated cyclic AMP production in rat osteosarcoma cells.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Line; Cyclic AMP; Drug Synergism; Interphase; Osteosarcoma; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Rats; Tetradecanoylphorbol Acetate; Time Factors; Virulence Factors, Bordetella | 1986 |
Dual actions of phorbol esters to decrease calcium and potassium conductances of mouse neurons.
Topics: Animals; Calcium; Cells, Cultured; Enzyme Activation; Ganglia, Spinal; Ion Channels; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Potassium; Protein Kinase C; Spinal Cord; Telencephalon; Tetradecanoylphorbol Acetate | 1987 |
Phorbol ester binding and protein kinase C activity in normal and transformed human keratinocytes.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Cell Transformation, Viral; Cells, Cultured; Epidermal Cells; Epidermis; ErbB Receptors; Humans; Keratins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Drug; Simian virus 40; Tetradecanoylphorbol Acetate | 1987 |
A phorbol ester-sensitive kinase catalyzes the phosphorylation of P0 glycoprotein in myelin.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cyclic AMP; Cycloheximide; Enzyme Activation; Male; Molecular Weight; Myelin P0 Protein; Myelin Proteins; Myelin Sheath; Nerve Crush; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphates; Phosphorylation; Protein Kinase C; Protein Kinases; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1987 |
Protein kinase C potentiates isoproterenol-mediated cyclic AMP production without modifying the homologous desensitization process in J774 cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Carcinogens; Cell Line; Cell Membrane; Cyclic AMP; Isoproterenol; Kinetics; Macrophages; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Adrenergic, beta; Tetradecanoylphorbol Acetate | 1987 |
Immature stimulus-secretion coupling in the developing exocrine pancreas and ontogenic changes of protein kinase C.
Topics: Amylases; Animals; Animals, Newborn; Bucladesine; Calcimycin; Cytosol; Fetus; Pancreas; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Rats, Inbred Strains; Secretory Rate; Sincalide; Tetradecanoylphorbol Acetate | 1988 |
Phorbol esters modulate cyclic AMP accumulation in porcine thyroid cells.
Topics: 1-Methyl-3-isobutylxanthine; Alprostadil; Animals; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Phorbol 12,13-Dibutyrate; Phorbol Esters; Prostaglandins E; Swine; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin | 1988 |
Interactions between phorbol esters and agents which increase cytosolic calcium in the guinea pig parenchymal strip: direct and indirect effects on the contractile response.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Cytosol; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Lung; Male; Muscle Contraction; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Vanadates | 1988 |
Two modes of regulation of the phospholipase C-linked substance-P receptor in rat parotid acinar cells.
Topics: Animals; Binding Sites; Calcium; Enzyme Activation; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Parotid Gland; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Substance P; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1988 |
Adenosine 3',5'-cyclic monophosphate (cAMP) inhibits phorbol ester-induced growth of an IL-2-dependent T cell line.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Bucladesine; Cell Division; Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; DNA Replication; Humans; Interleukin-2; Kinetics; Phorbol 12,13-Dibutyrate; Recombinant Proteins; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1988 |
Phorbol ester-mediated down-regulation of an interferon-inducible gene.
Topics: Cycloheximide; Fibroblasts; Gene Expression Regulation; Humans; Interferon Type I; Melanoma; Phorbol 12,13-Dibutyrate; Recombinant Proteins; RNA; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1989 |
Opposing effects of calcium entry and phorbol esters on fusion of chick muscle cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium Channel Blockers; Cell Fusion; Cells, Cultured; Chick Embryo; Egtazic Acid; Gallopamil; Kinetics; Muscles; Myosin Subfragments; Myosin-Light-Chain Kinase; Myosins; Nitrendipine; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Tetradecanoylphorbol Acetate | 1989 |
Activators of protein kinase C up-regulate the cell surface expression of CD2 and CD5 T cell glycoproteins.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antibodies, Monoclonal; Antigens, Differentiation; Antigens, Differentiation, T-Lymphocyte; Calcium Channel Blockers; CD2 Antigens; CD5 Antigens; Cell Membrane; Cells, Cultured; Cycloheximide; Diglycerides; Dinoprostone; Enzyme Activation; Flow Cytometry; Humans; Isoquinolines; Membrane Glycoproteins; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Receptors, Immunologic; RNA, Messenger; Sulfonamides; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1989 |
Regulation of phospholipase D in HL-60 granulocytes. Activation by phorbol esters, diglyceride, and calcium ionophore via protein kinase- independent mechanisms.
Topics: Calcimycin; Cell Line; Diglycerides; Enzyme Activation; Glycerides; Granulocytes; Humans; Kinetics; Leukemia, Promyelocytic, Acute; Phorbol 12,13-Dibutyrate; Phospholipase D; Phospholipases; Protein Kinase C; Tetradecanoylphorbol Acetate | 1989 |
Evidence that phorbol diester-sensitive protein kinase-C(s) may not be directly involved in secretagogue-stimulated prolactin release and arachidonate liberation.
Topics: Angiotensin II; Animals; Arachidonic Acid; Arachidonic Acids; Cell Line; Cells, Cultured; Female; Kinetics; Marine Toxins; Neurotensin; Oxocins; Phorbol 12,13-Dibutyrate; Pituitary Gland, Anterior; Prolactin; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone | 1989 |
Inhibition of DNA fragmentation in thymocytes and isolated thymocyte nuclei by agents that stimulate protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcium; Cell Nucleus; Cells, Cultured; Cytosol; DNA; Isoquinolines; Kinetics; Male; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thymus Gland | 1989 |
Ca2+- and phospholipid-independent activation of protein kinase C by selective oxidative modification of the regulatory domain.
Topics: Animals; Brain; Calcium; Cattle; Cell Line; Egtazic Acid; Enzyme Activation; Glioma; Hydrogen Peroxide; Kinetics; Phorbol 12,13-Dibutyrate; Phosphatidylserines; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate | 1989 |
Involvement of protein kinase C in translocation of desmoplakins from cytosol to plasma membrane during desmosome formation in human squamous cell carcinoma cells grown in low to normal calcium concentration.
Topics: Calcimycin; Calcium; Carcinoma, Squamous Cell; Cell Membrane; Cytoskeletal Proteins; Cytosol; Desmoplakins; Desmosomes; Diglycerides; Dose-Response Relationship, Drug; Humans; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Homologous desensitization of muscarinic cholinergic, histaminergic, adrenergic, and serotonergic receptors coupled to phospholipase C in cerebellar granule cells.
Topics: Animals; Carbachol; Cells, Cultured; Cerebellum; Cytoplasmic Granules; Histamine; Inositol Phosphates; Norepinephrine; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Histamine; Receptors, Muscarinic; Receptors, Serotonin; Serotonin; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1989 |
Evidence for a protein kinase C-directed mechanism in the phorbol diester-induced phospholipase D pathway of diacylglycerol generation from phosphatidylcholine.
Topics: Alkaloids; Animals; Bucladesine; Cell Line; Choline; Colforsin; Diglycerides; Embryo, Mammalian; Fibroblasts; Glycerides; Glycerophospholipids; Hydrolysis; Myristic Acid; Myristic Acids; Phorbol 12,13-Dibutyrate; Phosphatidic Acids; Phosphatidylcholines; Phospholipase D; Phospholipases; Protein Kinase C; Rats; Staurosporine; Tetradecanoylphorbol Acetate | 1989 |
Requirement and role of arachidonic acid in the differentiation of pre-adipose cells.
Topics: Adipose Tissue; Animals; Arachidonic Acid; Arachidonic Acids; Cell Differentiation; Cell Line; Cyclic AMP; Cyclic GMP; Ethers; Inositol; Ionomycin; Mice; Mice, Inbred C57BL; Mitosis; Phorbol 12,13-Dibutyrate; Phospholipids; Rats; Tetradecanoylphorbol Acetate | 1989 |
Sphingosine inhibits phorbol 12-myristate 13-acetate-, but not serum-induced, activation of Na+/H+ exchange in mammalian cells.
Topics: Animals; Blood Physiological Phenomena; Carrier Proteins; Cell Line; Diglycerides; Enzyme Activation; Humans; Hydrogen-Ion Concentration; Phorbol 12,13-Dibutyrate; Protein Kinase C; Sodium-Hydrogen Exchangers; Sphingosine; Tetradecanoylphorbol Acetate | 1989 |
Enhanced responsiveness to angiotensin II in vascular smooth muscle cells from spontaneously hypertensive rats is not associated with alterations in protein kinase C.
Topics: Angiotensin II; Animals; Cells, Cultured; Enzyme Activation; Hydrogen-Ion Concentration; Hypertension; Intracellular Membranes; Male; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Protein Kinase C; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Tetradecanoylphorbol Acetate | 1989 |
1,2-dioctanoyl-sn-glycerol can stimulate neutrophils by different mechanisms. Evidence for a pathway that does not involve phosphorylation of the 47-kDa protein.
Topics: Alkaloids; Animals; Diglycerides; Diterpenes; Glycerides; Guinea Pigs; Humans; Kinetics; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Proteins; Staurosporine; Superoxides; Terpenes; Tetradecanoylphorbol Acetate | 1989 |
Mechanistic studies on the DDT-induced inhibition of intercellular communication.
Topics: Animals; Cell Communication; Cells, Cultured; Cricetinae; DDT; gamma-Glutamyltransferase; Liver; Phorbol 12,13-Dibutyrate; Protein Kinase C; Quercetin; Tetradecanoylphorbol Acetate | 1989 |
Selective low level of protein kinase C isozyme in a tumor promoter-dependent mouse leukemia cell line.
Topics: Animals; Antibodies, Monoclonal; Caenorhabditis elegans Proteins; Carrier Proteins; Isoenzymes; Leukemia, Experimental; Mice; Mutation; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinases; Receptors, Drug; Tetradecanoylphorbol Acetate | 1989 |
Differences in the effects of phorbol esters and diacylglycerols on protein kinase C.
Topics: Animals; Calcium; Cattle; Diglycerides; Enzyme Activation; Glycerides; Kinetics; Membrane Proteins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1989 |
Do phorbol myristate and phorbol dibutyrate enhance noradrenaline release by the same mechanisms?
Topics: Animals; Electric Stimulation; Heart; In Vitro Techniques; Mice; Muscle, Smooth, Vascular; Norepinephrine; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1989 |
Activation of HIV gene expression during monocyte differentiation by induction of NF-kappa B.
Topics: Cell Differentiation; Chloramphenicol O-Acetyltransferase; DNA, Viral; Enhancer Elements, Genetic; Gene Expression Regulation; HIV; Leukemia; Monocytes; NF-kappa B; Phorbol 12,13-Dibutyrate; Plasmids; Tetradecanoylphorbol Acetate; Transcription Factors; Transfection; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1989 |
Endothelin stimulates diacylglycerol accumulation and activates protein kinase C in cultured vascular smooth muscle cells.
Topics: Animals; Aorta, Thoracic; Cells, Cultured; Diglycerides; Endothelins; Endothelium, Vascular; Enzyme Activation; Ethers; Glycerides; Ionomycin; Kinetics; Molecular Weight; Muscle, Smooth, Vascular; Peptides; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate | 1989 |
Use of protein kinase C-depleted cells for investigation of the role of protein kinase C in stimulus-response coupling in the pituitary.
Topics: Animals; Cells, Cultured; Culture Techniques; Female; Kinetics; Luteinizing Hormone; Phorbol 12,13-Dibutyrate; Phosphorus Radioisotopes; Pituitary Gland; Protein Kinase C; Radioisotope Dilution Technique; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Tritium | 1989 |
Regulation of human megakaryocytopoiesis.
Topics: Bone Marrow Cells; Cell Division; Cell Line; Colony-Stimulating Factors; Culture Media; Granulocyte-Macrophage Colony-Stimulating Factor; Growth Substances; Hematopoietic Stem Cells; Humans; Interleukin-3; Megakaryocytes; Phorbol 12,13-Dibutyrate; Radioimmunoassay; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Inhibition of protein kinase C-dependent cellular proliferation by interaction of endogenous ganglioside GM1 with the B subunit of cholera toxin.
Topics: Animals; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Cell Division; Cells, Cultured; Cholera Toxin; Cytoplasm; DNA; DNA Replication; G(M1) Ganglioside; Insulin; Mice; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Protein Binding; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1989 |
Protein synthesis in rat cardiac myocytes is stimulated at the level of translation by phorbol esters.
Topics: Animals; Dactinomycin; Kinetics; Male; Myocardium; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Biosynthesis; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1989 |
Protein kinase C activity can desensitize the gonadotropin-responsive adenylate cyclase in Leydig tumor cells. But hCG-induced desensitization does not involve protein kinase C activation.
Topics: Adenylyl Cyclases; Animals; Binding Sites; Cell Line; Chorionic Gonadotropin; Diglycerides; Enzyme Activation; Inositol; Kinetics; Leydig Cell Tumor; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1989 |
Morphological changes and neural cell adhesion molecule expression in mouse cerebrum primary cultures following long-term exposure to phorbol ester.
Topics: Animals; Antigens, Surface; Astrocytes; Cell Adhesion Molecules; Cell Differentiation; Cells, Cultured; Cerebral Cortex; Glial Fibrillary Acidic Protein; Hippocampus; Mice; Mice, Inbred ICR; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate; Time Factors | 1989 |
Differential effects of phorbol esters on PGE2 and bradykinin-induced elevation of [Cai2+] in MDCK cells.
Topics: Animals; Benzofurans; Bradykinin; Calcium; Cell Line; Dinoprostone; Fluorescent Dyes; Fura-2; Kidney; Kinetics; Phorbol 12,13-Dibutyrate; Prostaglandins; Tetradecanoylphorbol Acetate | 1989 |
Protein kinase C activity and phorbol ester binding to rat myogenic cells during growth and differentiation.
Topics: Animals; Cell Differentiation; Cell Division; Cell Line; Cells, Cultured; Muscles; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1989 |
Direct activation of a protein kinase activity from rat lacrimal gland by PMA in a phospholipid-free system.
Topics: Animals; Chromatography, DEAE-Cellulose; Enzyme Activation; Lacrimal Apparatus; Male; Phorbol 12,13-Dibutyrate; Phospholipids; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1989 |
(-)-Indolactam V activates protein kinase C and induces changes in muscarinic receptor functions in SH-SY5Y human neuroblastoma cells.
Topics: Calcium; Cell Compartmentation; Cell Differentiation; Cell Membrane; Enzyme Activation; Humans; Indoles; Lactams; Neuroblastoma; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Muscarinic; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Alteration in protein kinase C activity and subcellular distribution in sickle erythrocytes.
Topics: Anemia, Sickle Cell; Cytosol; Erythrocytes; Humans; Membrane Proteins; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Reticulocytes; Tetradecanoylphorbol Acetate | 1989 |
Modification of protein kinase C (PKC) activity and diacylglycerol (DAG) accumulation in hepatocytes in continuous endotoxemia.
Topics: Animals; Biological Transport; Cytosol; Diglycerides; Endotoxins; Glycerides; Kinetics; Liver; Male; Phenylephrine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Vasopressins | 1989 |
Transcriptional regulation of transferrin receptor expression by cultured lymphoblastoid T cells treated with phorbol diesters.
Topics: Antigens, Surface; Cell Line; Humans; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Protein Processing, Post-Translational; Receptors, Transferrin; RNA, Messenger; T-Lymphocytes; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1989 |
Effects of cadmium on lymphocyte activation.
Topics: Adult; Cadmium; Cadmium Chloride; Cadmium Radioisotopes; Calcium; Cell Division; Cell Membrane; Dose-Response Relationship, Drug; Humans; Interleukins; Kinetics; Lymphocyte Activation; Lymphocytes; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Phospholipids; Phytohemagglutinins; Protein Kinases; Receptors, Interleukin-2; Tetradecanoylphorbol Acetate | 1989 |
Phorbol ester and calcium ionophore are sufficient to promote cell replication in cultures of quiescent human B lymphocytes.
Topics: B-Lymphocytes; Cell Division; Cells, Cultured; Ethers; Humans; Ionomycin; Ionophores; Leukocyte Count; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1989 |
Inhibition of the CD3-mediated calcium signal by protein kinase C activators in human T (Jurkat) lymphoblastoid cells.
Topics: Antigens, Differentiation, T-Lymphocyte; Calcium; Cell Line; Depression, Chemical; Diglycerides; Enzyme Activation; Glycerides; Humans; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Antigen, T-Cell; Signal Transduction; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Influence of protein kinase C activators on vascular tone and adrenergic neuroeffector events in the isolated rat kidney.
Topics: Animals; Calcium; Enzyme Activation; In Vitro Techniques; Kidney; Male; Nifedipine; Norepinephrine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Vasoconstriction | 1989 |
Changes in protein kinase C and cAMP-dependent kinase in lymphocytes after treatment with 12-O-tetradecanoylphorbol-13-acetate or concanavalin A: quantitation of activities with an in situ gel assay.
Topics: Affinity Labels; Animals; Azides; Cattle; Chromatography, Affinity; Concanavalin A; Cyclic AMP; Isoenzymes; Lymphocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Protein Kinases; Tetradecanoylphorbol Acetate; Time Factors | 1987 |
Differential sensitivity of agonist- and antagonist-occupied gonadotropin-releasing hormone receptors to protein kinase C activators. A marker for receptor activation.
Topics: Animals; Buserelin; Cell Membrane; Cells, Cultured; Diglycerides; Enzyme Activation; Female; Glycerides; Gonadotropin-Releasing Hormone; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland; Protein Kinase C; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, LHRH; Tetradecanoylphorbol Acetate | 1988 |
Interferon and phorbol esters down-regulate sIgM expression by independent pathways.
Topics: 2',5'-Oligoadenylate Synthetase; Carrier Proteins; Cell Cycle; Cell Division; Cell Line; Cycloheximide; Enzyme Activation; Immunoglobulin M; Interferon Type I; Lymphocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Biosynthesis; Receptors, Antigen, B-Cell; Sodium-Hydrogen Exchangers; Tetradecanoylphorbol Acetate; Thymidine | 1988 |
Phorbol esters increase adenylate cyclase activity and stability in pituitary membranes.
Topics: Adenylyl Cyclases; Calcium; Cell Membrane; Cyclic AMP; Humans; Kinetics; Models, Biological; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1988 |
Gonadotropin-releasing hormone agonist activates protein kinase C in rat Leydig cells.
Topics: Animals; Buserelin; Cell Membrane; Cyclic AMP; Enzyme Activation; In Vitro Techniques; Leydig Cells; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Rats, Inbred Strains; Testosterone; Tetradecanoylphorbol Acetate | 1988 |
Involvement of two intracellular messenger systems, protein kinase C and cyclic AMP, in the regulation of c-fos gene expression in human promyelocytic leukemia (HL-60) cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Cyclic AMP; Diglycerides; Dinoprostone; Gene Expression Regulation; Humans; Kinetics; Leukemia, Myeloid; Phorbol 12,13-Dibutyrate; Phorbol Esters; Prostaglandins E; Protein Kinase C; Proto-Oncogenes; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1987 |
Heterologous down-regulation of vascular atrial natriuretic peptide receptors by phorbol esters.
Topics: Animals; Dose-Response Relationship, Drug; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Atrial Natriuretic Factor; Receptors, Cell Surface; Temperature; Tetradecanoylphorbol Acetate; Time Factors | 1988 |
Phorbol ester modulates serotonin-stimulated phosphoinositide breakdown in cultured vascular smooth muscle cells.
Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; GTP-Binding Proteins; Kinetics; Male; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositols; Phosphorylation; Rabbits; Receptors, Serotonin; Serotonin; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1988 |
Modulation of octopamine-mediated production of cyclic AMP by phorbol-ester-sensitive protein kinase C in an insect cell line.
Topics: Animals; Cell Line; Cholera Toxin; Cyclic AMP; Dose-Response Relationship, Drug; Lepidoptera; Octopamine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1988 |
Participation of protein kinase C and regulatory G proteins in modulation of the evoked noradrenaline release in brain.
Topics: Adenylyl Cyclases; Animals; Electric Stimulation; GTP-Binding Proteins; Hippocampus; In Vitro Techniques; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate | 1988 |
Platelet-derived growth factor (PDGF)-induced phospholipase C-mediated hydrolysis of phosphoinositides in vascular smooth muscle cells--different sensitivity of PDGF- and angiotensin II-induced phospholipase C reactions to protein kinase C-activating phor
Topics: Angiotensin II; Animals; Cells, Cultured; DNA; Enzyme Activation; Hydrolysis; Inositol; Inositol Phosphates; Kinetics; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositols; Platelet-Derived Growth Factor; Protein Kinase C; Rabbits; Recombinant Proteins; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1988 |
Agonist but not phorbol ester induced desensitization of human lymphocyte prostaglandin receptor is dependent on tubulin polymerization.
Topics: Benzimidazoles; Binding, Competitive; Carcinogens; Colchicine; Cyclic AMP; Dinoprostone; Humans; Leukemia, T-Cell; Nocodazole; Phorbol 12,13-Dibutyrate; Phorbol Esters; Receptors, Prostaglandin; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tubulin; Tumor Cells, Cultured | 1988 |
Protein kinase C activities are increased in rat thyroid epithelial cells expressing v-ras genes.
Topics: Animals; Biological Transport; Calcium; Cell Membrane; Cell Transformation, Viral; Chromatography; Cytoplasm; Diglycerides; Enzyme Activation; Epithelium; Genes, ras; Harvey murine sarcoma virus; Mutation; Phorbol 12,13-Dibutyrate; Phosphatidylserines; Phosphorylation; Protein Kinase C; Rats; Sarcoma Viruses, Murine; Tetradecanoylphorbol Acetate; Thyroid Gland | 1988 |
Effect of membrane perturbation on protein kinase C activation: treatment with exogenous phospholipase C decreases translocation of enzyme to cellular membranes.
Topics: Animals; Cell Line; Cell Membrane; Clostridium perfringens; Diglycerides; Enzyme Activation; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors; Type C Phospholipases | 1986 |
Protein kinase C enhances growth hormone releasing factor (1-40)-stimulated cyclic AMP levels in anterior pituitary. Actions of somatostatin and pertussis toxin.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Cells, Cultured; Cyclic AMP; Drug Synergism; Female; Growth Hormone-Releasing Hormone; Male; Peptide Fragments; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland, Anterior; Protein Kinase C; Rats; Somatostatin; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1986 |
Neurotransmitter-stimulated inositol phosphate accumulation in hippocampal slices.
Topics: Animals; Carbachol; Hippocampus; In Vitro Techniques; Inositol; Inositol Phosphates; Kinetics; Manganese; Neurotransmitter Agents; Phorbol 12,13-Dibutyrate; Phorbol Esters; Radioisotope Dilution Technique; Sugar Phosphates; Tetradecanoylphorbol Acetate; Tritium | 1987 |
Partial parallelism and partial blockade by bryostatin 1 of effects of phorbol ester tumor promoters on primary mouse epidermal cells.
Topics: Animals; Bryostatins; Cells, Cultured; Cycloheximide; Dactinomycin; Enzyme Activation; Epidermal Growth Factor; Epidermis; Lactones; Macrolides; Mice; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Skin Neoplasms; Tetradecanoylphorbol Acetate; Transglutaminases | 1987 |
Phorbol esters attenuate glutamate-stimulated inositol phospholipid hydrolysis in neuronal cultures.
Topics: Animals; Aspartic Acid; Carbachol; Cerebellum; Diglycerides; Glutamates; Glutamic Acid; Hydrolysis; Inositol Phosphates; N-Methylaspartate; Neurons; Oxadiazoles; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositols; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Glutamate; Receptors, Neurotransmitter; Sphingosine; Tetradecanoylphorbol Acetate | 1988 |
Phorbol ester-induced activation of protein kinase C leads to increased formation of diacylglycerol in human neutrophils.
Topics: Calcium; Diglycerides; Enzyme Activation; Glycerides; Humans; Neutrophils; Phorbol 12,13-Dibutyrate; Phosphatidylcholines; Phosphatidylinositols; Protein Kinase C; Tetradecanoylphorbol Acetate | 1989 |
Tumor-promoting phorbol esters inhibit monocyte adherence to endothelial cells.
Topics: Animals; Aorta; Carcinogens; Cell Adhesion; Cells, Cultured; Endothelium, Vascular; Male; Monocytes; Phorbol 12,13-Dibutyrate; Phorbols; Tetradecanoylphorbol Acetate | 1989 |
Membrane-phorbol ester interactions monitored by circular dichroism.
Topics: Circular Dichroism; Enzyme Activation; Erythrocyte Membrane; Humans; Liposomes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Protein Kinase C; Spectrum Analysis; Tetradecanoylphorbol Acetate | 1989 |
Differences in phorbol-ester-induced down-regulation of protein kinase C between cell lines.
Topics: Animals; Binding Sites; Cell Line; Cricetinae; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Cremophor EL, a widely used parenteral vehicle, is a potent inhibitor of protein kinase C.
Topics: Binding, Competitive; Cell Line; DNA Polymerase II; Drug Carriers; Glycerol; Humans; Kinetics; Leukemia; Phorbol 12,13-Dibutyrate; Protein Binding; Protein Kinase C; Protein Kinases; RNA Polymerase II; Solvents; Tetradecanoylphorbol Acetate | 1989 |
Differentiation of peanut lectin positive suppressor T-cells from peanut lectin negative precursors in bovine cells by 12-O-tetradecanoylphorbol-13-acetate.
Topics: Animals; Cattle; Cell Differentiation; Cell Separation; Dose-Response Relationship, Drug; Drug Synergism; Lectins; Macrophages; Peanut Agglutinin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Rosette Formation; T-Lymphocytes, Regulatory; Tetradecanoylphorbol Acetate | 1987 |
Tumour-promoting phorbol esters inhibit agonist-induced phosphatidate formation and Ca2+ flux in human platelets.
Topics: Blood Platelets; Calcium; Carcinogens; Enzyme Activation; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylinositols; Platelet Activating Factor; Protein Kinase C; Protein Kinases; Tetradecanoylphorbol Acetate; Thrombin; Vasopressins | 1985 |
Structural requirements for diacylglycerols to mimic tumor-promoting phobol diester action on the epidermal growth factor receptor.
Topics: Animals; Carcinogens; Cell Line; Diglycerides; ErbB Receptors; Glycerides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1985 |
Effects of tumor promoters on sodium ion transport across frog skin.
Topics: Amiloride; Animals; Biological Transport, Active; Carcinogens; Cyclic AMP; Indomethacin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rana pipiens; Skin; Sodium; Tetradecanoylphorbol Acetate | 1985 |
Effects of epidermal growth factor, phorbol myristate acetate, and arachidonic acid on choriogonadotropin secretion by cultured human choriocarcinoma cells.
Topics: Arachidonic Acid; Arachidonic Acids; Caenorhabditis elegans Proteins; Carrier Proteins; Catechols; Cells, Cultured; Choriocarcinoma; Chorionic Gonadotropin; Dose-Response Relationship, Drug; Epidermal Growth Factor; ErbB Receptors; Female; Humans; Indomethacin; Masoprocol; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pregnancy; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Uterine Neoplasms | 1985 |
Phorbol ester causes desensitization of gonadotropin-responsive adenylate cyclase in a murine Leydig tumor cell line.
Topics: Adenylyl Cyclases; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Chorionic Gonadotropin; Diglycerides; Dose-Response Relationship, Drug; Kinetics; Leydig Cell Tumor; Male; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Receptors, LH; Testicular Neoplasms; Tetradecanoylphorbol Acetate | 1985 |
Tumor-promoting phorbol esters and vanadate alter the sensitivity of HeLa S3 cells to poliovirus type 1.
Topics: Cell Membrane; HeLa Cells; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Poliovirus; Tetradecanoylphorbol Acetate; Vanadates; Vanadium | 1985 |
Induction of protein kinase C activation and Ca2+ mobilization by fibroblast growth factor in Swiss 3T3 cells.
Topics: Animals; Calcium; Cell Line; Diglycerides; DNA; Enzyme Activation; Fibroblast Growth Factors; Insulin; Mice; Mice, Inbred BALB C; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositols; Protein Kinase C; Tetradecanoylphorbol Acetate | 1985 |
Effect of the calcium ionophore A23187 on superoxide generation in phorbol ester stimulated human neutrophils.
Topics: Calcimycin; Calcium; Humans; In Vitro Techniques; Kinetics; L-Lactate Dehydrogenase; Lysosomes; Neutrophils; Oxygen Consumption; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Superoxides; Tetradecanoylphorbol Acetate | 1985 |
Carbachol-induced accumulation of inositol-1-phosphate in neurohybridoma NCB-20 cells: effects of lithium and phorbol esters.
Topics: Animals; Atropine; Benzodiazepinones; Brain; Carbachol; Cell Line; Chlorides; Cricetinae; Cricetulus; Embryo, Mammalian; Hybridomas; Inositol Phosphates; Lithium; Lithium Chloride; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pirenzepine; Sugar Phosphates; Tetradecanoylphorbol Acetate | 1986 |
Inhibition of chemotactic peptide-induced phosphoinositide hydrolysis by phorbol esters through the activation of protein kinase C in differentiated human leukemia (HL-60) cells.
Topics: Cell Differentiation; Cell Line; Enzyme Activation; Humans; Inositol Phosphates; Leukemia, Experimental; N-Formylmethionine Leucyl-Phenylalanine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositols; Protein Kinase C; Sugar Phosphates; Tetradecanoylphorbol Acetate | 1986 |
The effect of cAMP on tumour promoter responses mediated by C-kinase.
Topics: Aminophylline; Animals; Bucladesine; Carcinogens; Cell Communication; Cell Line; Cyclic AMP; Diglycerides; Epidermal Growth Factor; Glycerides; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylcholines; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Action of retinoic acid on the diacylglycerol-induced ornithine decarboxylase activity, reduction in EGF binding and protein kinase C activation in rat tracheal epithelial 2C5 cells.
Topics: Animals; Cell Line; Diglycerides; Enzyme Activation; Enzyme Induction; Epidermal Growth Factor; ErbB Receptors; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Receptors, Cell Surface; Tetradecanoylphorbol Acetate; Trachea; Tretinoin | 1986 |
Inhibition of the oxidative burst in human neutrophils by sphingoid long-chain bases. Role of protein kinase C in activation of the burst.
Topics: Arachidonic Acid; Arachidonic Acids; Calcium; Cell Membrane; Cell Survival; Cytochrome c Group; Dose-Response Relationship, Drug; Humans; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Oxygen Consumption; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Sphingosine; Tetradecanoylphorbol Acetate; Zymosan | 1986 |
Regulation of respiratory burst in murine peritoneal macrophages: differential sensitivity to phorbol diesters by macrophages in different states of functional activation.
Topics: Animals; BCG Vaccine; Diglycerides; Dose-Response Relationship, Drug; Hydrogen Peroxide; Macrophage Activation; Macrophages; Mice; Mice, Inbred C57BL; Oxygen Consumption; Phorbol 12,13-Dibutyrate; Phorbol Esters; Superoxides; Tetradecanoylphorbol Acetate; Zymosan | 1986 |
Protein kinase C activators modulate differentiated thyroid function in vitro.
Topics: Animals; Bucladesine; Carcinogens; Enzyme Activation; Iodine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Swine; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin | 1986 |
Identification of a cell-surface glycoprotein mediating cell adhesion in EBV-immortalized normal B cells.
Topics: Animals; Antibodies, Monoclonal; B-Lymphocytes; Cell Adhesion; Cell Aggregation; Cell Line; Fluorescent Antibody Technique; Glycoproteins; Herpesvirus 4, Human; Immunoglobulin Fab Fragments; Kinetics; Molecular Weight; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate | 1986 |
Phorbol esters down-regulate protein kinase C in rat brain cerebral cortical slices.
Topics: Animals; Cerebral Cortex; Cholera Toxin; Cyclic AMP; In Vitro Techniques; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate | 1986 |
Effect of cellular fatty acid composition on the phospholipase A2 activity of bone marrow-derived macrophages, and their ability to induce lucigenin-dependent chemiluminescence.
Topics: Acridines; Animals; Bone Marrow Cells; Fatty Acids; Female; Luminescent Measurements; Macrophages; Membrane Lipids; Mice; Mice, Inbred C57BL; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phospholipases; Phospholipases A; Phospholipases A2; Superoxides; Tetradecanoylphorbol Acetate; Zymosan | 1986 |
Inhibition of phorbol ester stimulated superoxide production by 1-oleoyl-2-acetyl-sn-glycerol (OAG); fact or artefact?
Topics: Animals; Brain; Cell Line; Cytosol; Diglycerides; Glycerides; Granulocytes; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Superoxides; Tetradecanoylphorbol Acetate | 1986 |
Phorbol ester-induced inhibition of cyclic GMP formation mediated by muscarinic receptors in murine neuroblastoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Carbachol; Cell Line; Cyclic GMP; Dose-Response Relationship, Drug; Histamine; Isoquinolines; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Piperazines; Receptors, Muscarinic; Tetradecanoylphorbol Acetate | 1987 |
Down-regulation of protein kinase C in rat glioma C6 cells: effects on the beta-adrenergic receptor-coupled adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Glioma; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Receptors, Adrenergic, beta; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate | 1987 |
High- and low-affinity receptors regulate platelet responses to phorbol diesters and teleocidin.
Topics: beta-Thromboglobulin; Binding, Competitive; Blood Platelets; Caenorhabditis elegans Proteins; Carrier Proteins; Chromatography, Gel; Humans; Lyngbya Toxins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Serotonin; Tetradecanoylphorbol Acetate | 1987 |
Possible involvement of reorganization of actin filaments, induced by tumor-promoting phorbol esters, in changes in colony shape and enhancement of proliferation of cultured epithelial cells.
Topics: Actins; Animals; Cell Division; Cyclic AMP; Diterpenes; Dogs; Epithelial Cells; Epithelium; Kidney; Microscopy, Fluorescence; Phorbol 12,13-Dibutyrate; Phorbol Esters; Terpenes; Tetradecanoylphorbol Acetate; Time Factors | 1987 |
Defective production of reactive oxygen intermediates by tumor-associated macrophages exposed to phorbol ester.
Topics: Animals; Macrophages; Male; Mice; Mice, Inbred C57BL; NADPH-Ferrihemoprotein Reductase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Sarcoma, Experimental; Superoxides; Tetradecanoylphorbol Acetate; Zymosan | 1987 |
Induction of virus enzymes by phorbol esters and n-butyrate in Epstein-Barr virus genome-carrying Raji cells.
Topics: Burkitt Lymphoma; Butyrates; Butyric Acid; Cells, Cultured; Deoxyribonucleases; DNA-Directed DNA Polymerase; DNA, Viral; Enzyme Induction; Genes, Viral; Herpesvirus 4, Human; Humans; Methylation; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Sphingosine; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1987 |
Second stage tumor promoters: differences in biological potency and phorbol ester receptor affinity in C6 cells.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Cyclic AMP; Diterpenes; Glioma; Glycerolphosphate Dehydrogenase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Receptors, Drug; Receptors, Immunologic; Terpenes; Tetradecanoylphorbol Acetate | 1987 |
Inhibition of DNA synthesis by protein kinase C-activating phorbol esters in NIH/3T3 cells.
Topics: Animals; Cells, Cultured; DNA Replication; Enzyme Activation; Fibroblast Growth Factors; Insulin; Kinetics; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1988 |
Possible involvement of protein kinase C and calcium ion in growth factor-induced expression of c-myc oncogene in Swiss 3T3 fibroblasts.
Topics: Animals; Calcimycin; Calcium; Cell Line; Diglycerides; Enzyme Activation; Ethers; Fibroblast Growth Factors; Fibroblasts; Gene Expression Regulation; Ionomycin; Mice; Oncogenes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Platelet-Derived Growth Factor; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Activation of protein kinase C induces rapid internalization and subsequent degradation of muscarinic acetylcholine receptors in neuroblastoma cells.
Topics: Animals; Calcimycin; Calcium; Carbachol; Cell Line; Diglycerides; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Kinetics; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Protein Kinase C; Quinuclidinyl Benzilate; Receptors, Cholinergic; Tetradecanoylphorbol Acetate; Time Factors | 1986 |
Phorbol ester-stimulated T lymphocytes show enhanced adhesion to human endothelial cell monolayers.
Topics: Cell Adhesion; Cells, Cultured; Endothelium; Fibroblasts; Gelatin; Humans; Interferon-gamma; Interleukin-1; Lipopolysaccharides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; T-Lymphocytes; Tetradecanoylphorbol Acetate; Umbilical Veins | 1986 |
Dissociation of myosin phosphorylation and active tension during muscarinic stimulation of tracheal smooth muscle.
Topics: Atropine; Calcium; Calcium Chloride; Carbachol; Dose-Response Relationship, Drug; Egtazic Acid; Muscle Contraction; Muscle, Smooth; Myosins; Nifedipine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Potassium; Serotonin; Tetradecanoylphorbol Acetate; Trachea | 1987 |
Stimulation of epidermal growth factor receptor threonine 654 phosphorylation by platelet-derived growth factor in protein kinase C-deficient human fibroblasts.
Topics: Carcinogens; Cell Line; ErbB Receptors; Fibroblasts; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Platelet-Derived Growth Factor; Protein Kinase C; Tetradecanoylphorbol Acetate; Threonine | 1987 |
Activation of protein kinase C is coupled to prostaglandin E2 synthesis in swine granulosa cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Cells, Cultured; Chromatography, High Pressure Liquid; Diglycerides; Dinoprostone; Drug Synergism; Enzyme Activation; Female; Follicle Stimulating Hormone; Gas Chromatography-Mass Spectrometry; Granulosa Cells; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Prostaglandins E; Protein Kinase C; Swine; Tetradecanoylphorbol Acetate | 1987 |
Juvenile hormone action mediated in male accessory glands of Drosophila by calcium and kinase C.
Topics: Animals; Calcium; Drosophila melanogaster; Enzyme Activation; Genitalia, Male; Juvenile Hormones; Male; Membrane Proteins; Mutation; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Biosynthesis; Protein Kinase C; Sesquiterpenes; Tetradecanoylphorbol Acetate | 1988 |
The role of protein kinase C in LHRH-induced LH and FSH release and LHRH self-priming in rat anterior pituitary glands in vitro.
Topics: Animals; Enzyme Activation; Female; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; In Vitro Techniques; Luteinizing Hormone; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland, Anterior; Protein Kinase C; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1988 |
Tumor-promoting phorbol esters stimulate the proliferation of interleukin-3 dependent cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Cell Division; Cell Survival; Colony-Stimulating Factors; Enzyme Activation; Granulocyte-Macrophage Colony-Stimulating Factor; Growth Substances; Interleukin-3; Isoquinolines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate | 1988 |
Inhibition of protein kinase C by tamoxifen.
Topics: Animals; Brain; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phospholipids; Protein Kinase C; Protein Kinase Inhibitors; Rats; Tamoxifen; Tetradecanoylphorbol Acetate | 1985 |
Phorbolesters enhance basal D-glucose transport but inhibit insulin stimulation of D-glucose transport and insulin binding in isolated rat adipocytes.
Topics: Adipose Tissue; Animals; Biological Transport, Active; Glucose; Insulin; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Protein-Tyrosine Kinases; Rats; Rats, Inbred Strains; Receptor, Insulin; Tetradecanoylphorbol Acetate | 1985 |
Tumor-promoting phorbol esters induce rapid internalization of the C3b receptor via a cytoskeleton-dependent mechanism.
Topics: Antibodies, Monoclonal; Binding, Competitive; Cytochalasin B; Cytoskeleton; Fibronectins; Humans; Immunoglobulin Fab Fragments; Neutrophils; Phagocytosis; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Receptors, Complement; Receptors, Complement 3b; Temperature; Tetradecanoylphorbol Acetate | 1985 |
Suppression of nerve growth factor-directed neurite outgrowth in PC12 cells by sphingosine, an inhibitor of protein kinase C.
Topics: Adrenal Gland Neoplasms; Animals; Cell Survival; Dose-Response Relationship, Drug; Nerve Growth Factors; Neurons; Pheochromocytoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; RNA, Messenger; Sphingosine; Tetradecanoylphorbol Acetate; Tubulin; Tumor Cells, Cultured | 1988 |
Phorbol ester-induced stimulation of prostaglandin biosynthesis in human amnion cells.
Topics: Amnion; Dinoprostone; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Prostaglandins E; Tetradecanoylphorbol Acetate | 1988 |
Regulation of the epidermal growth factor receptor phosphorylation state by sphingosine in A431 human epidermoid carcinoma cells.
Topics: Carcinoma, Squamous Cell; Dose-Response Relationship, Drug; ErbB Receptors; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Protein Kinase C; Sphingosine; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured | 1988 |
Evidence for separate control by phorbol esters of CD18-dependent adhesion and translocation of protein kinase C in U-937 cells.
Topics: Cell Adhesion; Cell Line; Choline; DNA Replication; Humans; Kinetics; Lipids; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Protein Processing, Post-Translational; Tetradecanoylphorbol Acetate | 1988 |
Phorbol esters stimulate the potassium-induced release of cholecystokinin from slices of cerebral cortex, caudato-putamen and hippocampus incubated in vitro.
Topics: Animals; Caudate Nucleus; Cerebral Cortex; Cholecystokinin; Hippocampus; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Potassium; Putamen; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1988 |
Characterization of lymphocyte stimulation by phorbol related compounds.
Topics: Adolescent; Adult; Animals; Humans; Irritants; Lymphocyte Activation; Male; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phytohemagglutinins; Skin Tests; Tetradecanoylphorbol Acetate | 1988 |
Correlation of the antiproliferative action of diphenylmethane-derivative antiestrogen binding site ligands with antagonism of histamine binding but not of protein kinase C-mediated phosphorylation.
Topics: Animals; Benzhydryl Compounds; Cell Line; Cerebral Cortex; Dose-Response Relationship, Drug; Estrogen Antagonists; Histamine; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylethanolamines; Phosphorylation; Platelet Aggregation; Protein Kinase C; Rats; Receptors, Drug; Receptors, Estrogen; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1988 |
Schistosoma mansoni: evidence for protein kinase-C-like modulation of muscle activity.
Topics: Animals; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Enzyme Activation; Male; Movement; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Schistosoma mansoni; Tetradecanoylphorbol Acetate | 1988 |
Growth-dependent subcellular redistribution of protein kinase C in cultured porcine aortic endothelial cells.
Topics: Animals; Cell Division; Cells, Cultured; Endothelium, Vascular; Enzyme Activation; Phorbol 12,13-Dibutyrate; Protein Kinase C; Subcellular Fractions; Swine; Tetradecanoylphorbol Acetate | 1988 |
Phorbol ester receptors and the induction of differentiation in the human T lymphoblastic cell line MOLT-3.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Differentiation; Cell Line, Transformed; Cell Transformation, Neoplastic; Drug Resistance; Humans; Leukemia-Lymphoma, Adult T-Cell; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Drug; Statistics as Topic; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1988 |
Interleukin 3 stimulates proliferation via protein kinase C activation without increasing inositol lipid turnover.
Topics: Caenorhabditis elegans Proteins; Calcium; Carcinogens; Carrier Proteins; Cell Line; Cell Survival; DNA Replication; Enzyme Activation; Inositol; Interleukin-3; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositols; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1988 |
Activation and proliferation signals in mouse B cells. IX. Protein kinase C activators synergize with non-mitogenic anti-immunoglobulin antibodies to drive B cells into G1.
Topics: Animals; Antibodies, Anti-Idiotypic; B-Lymphocytes; Calcium; Cyclosporins; Enzyme Activation; Immunoglobulin Fab Fragments; Immunoglobulin G; Interphase; Lymphocyte Activation; Male; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1988 |
Phorbol esters can persistently replace interleukin-2 (IL-2) for the growth of a human IL-2-dependent T-cell line.
Topics: Cell Line; Humans; Interleukin-2; Nucleic Acid Hybridization; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; RNA, Messenger; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1988 |
Effect of protein kinase C activation and depletion on insulin stimulation of glycogen synthesis in cultured hepatoma cells.
Topics: Animals; Enzyme Activation; Glycogen; Insulin; Liver Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1988 |
Generation of neutrophil chemotactic activity by phorbol ester-stimulated calf pulmonary artery endothelial cells.
Topics: Animals; Cattle; Cells, Cultured; Chemotactic Factors; Culture Media; Dactinomycin; Endothelium, Vascular; Interleukin-8; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pulmonary Artery; Tetradecanoylphorbol Acetate | 1988 |
Dioctanoylglycerol and phorbol esters regulate transcription of c-myc in human promyelocytic leukemia cells.
Topics: Diglycerides; Enzyme Activation; Glycerides; Humans; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Proto-Oncogenes; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1988 |
Tumor promoter-induced membrane-bound protein kinase C regulates hematogenous metastasis.
Topics: Animals; Carcinogens; Cell Line; Cell Membrane; Cytosol; Enzyme Induction; Kinetics; Lung Neoplasms; Melanoma, Experimental; Mice; Mice, Inbred C57BL; Neoplasm Metastasis; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1988 |
Protein kinase C and phorbol ester receptor expression related to growth and differentiation of nullipotent and pluripotent embryonal carcinoma cells.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Differentiation; Cell Division; Cell Line; DNA Replication; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Teratoma; Tetradecanoylphorbol Acetate; Thymidine | 1986 |
Phorbol esters inhibit the proliferation of MCF-7 cells. Possible implication of protein kinase C.
Topics: Breast Neoplasms; Cell Division; Cell Line; Dose-Response Relationship, Drug; Female; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Inhibition of phorbol ester-dependent differentiation of human promyelocytic leukemic (HL-60) cells by sphinganine and other long-chain bases.
Topics: Acid Phosphatase; Binding, Competitive; Cell Adhesion; Cell Differentiation; Cell Line; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Sphingosine; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1986 |
Endogenous inhibitor of protein kinase C: association with human peripheral blood neutrophils but not with specific granule-deficient neutrophils or cytoplasts.
Topics: Cytoplasmic Granules; Diglycerides; Humans; Intracellular Membranes; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Phorbol ester-induced contraction in chemically skinned vascular smooth muscle.
Topics: Animals; Calcium; Carotid Arteries; Enzyme Activation; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Myosins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Potassium; Protein Kinase C; Skin Physiological Phenomena; Swine; Tetradecanoylphorbol Acetate | 1986 |
Phorbol diesters alter the contractile responses of porcine coronary artery.
Topics: Animals; Calcium; Drug Synergism; Histamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Polymyxin B; Potassium; Protein Kinase C; Swine; Tetradecanoylphorbol Acetate | 1986 |
Effects of tumor promoters on LLC-PK1 renal epithelial tight junctions and transepithelial fluxes.
Topics: Carcinogens; Cell Line; Diffusion; Epithelium; Intercellular Junctions; Kidney; Membrane Potentials; Phorbol 12,13-Dibutyrate; Phorbol Esters; Sodium Chloride; Tetradecanoylphorbol Acetate | 1986 |
Factors influencing chelator-stable, detergent-extractable, phorbol diester-induced membrane association of protein kinase C. Differences between Ca2+-induced and phorbol ester-stabilized membrane bindings of protein kinase C.
Topics: Animals; Calcium; Calcium Chloride; Cell Line; Cell Membrane; Cells, Cultured; Detergents; Diglycerides; Glycerides; Organoids; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phospholipases; Protein Binding; Protein Kinase C; Tetradecanoylphorbol Acetate; Trypsin | 1986 |
Three activators of protein kinase C, bryostatins, dioleins, and phorbol esters, show differing specificities of action on GH4 pituitary cells.
Topics: Animals; Binding Sites; Binding, Competitive; Bryostatins; Cell Line; Diglycerides; Enzyme Activation; Eukaryota; Glycerides; Kinetics; Lactones; Macrolides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Possible involvement of protein kinase C in platelet-derived growth factor-stimulated DNA synthesis in vascular smooth muscle cells.
Topics: Animals; Cell Division; Cells, Cultured; DNA; Enzyme Activation; Humans; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Platelet-Derived Growth Factor; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate | 1987 |
Down regulation of protein kinase C in neuronal cells: effects on neurotransmitter release.
Topics: Animals; Cells, Cultured; Ethers; Ionomycin; Neurons; Nitrendipine; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Sympathetic Nervous System; Tetradecanoylphorbol Acetate | 1987 |
Catalytic and receptor-binding properties of the calcium-sensitive phospholipid-dependent protein kinase (protein kinase C) in swine luteal cytosol.
Topics: Animals; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Corpus Luteum; Cytosol; Diglycerides; Enzyme Activation; Female; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Polymyxin B; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Swine; Tetradecanoylphorbol Acetate | 1987 |
Phorbol esters inhibit ammoniagenesis and gluconeogenesis in proximal tubular segments.
Topics: Ammonia; Animals; Dimethyl Sulfoxide; Dogs; Gluconeogenesis; Glutamine; Kidney Tubules, Proximal; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1987 |
Substitution of phosphatidylserine by lipid A in the activation of purified rabbit brain protein kinase C.
Topics: Animals; Brain; Enzyme Activation; Lipid A; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate | 1987 |
Distinct functions of down-regulation-sensitive and -resistant types of protein kinase C in rabbit aortic smooth muscle cells.
Topics: Animals; Aorta, Thoracic; Calcium; Cytoplasm; DNA; Drug Resistance; Male; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate | 1987 |
Divergent effects of co-carcinogenic phorbol esters and a synthetic diacylglycerol on human neutrophil chemokinesis and granular enzyme secretion.
Topics: Calcium; Chemotaxis, Leukocyte; Cocarcinogenesis; Cytoplasmic Granules; Diglycerides; Glycerides; Humans; Muramidase; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 1987 |
TPA induces subcellular translocation and subsequent down-regulation of both phorbol ester binding and protein kinase C activities in MCF-7 cells.
Topics: Animals; Binding Sites; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Subcellular Fractions; Tetradecanoylphorbol Acetate; Time Factors | 1987 |
Differences between human and goose erythrocytes in response to phorbol esters and expression of phorbol ester receptors.
Topics: 4-Chloro-7-nitrobenzofurazan; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Erythrocytes; Geese; Glucosamine; Humans; Oxadiazoles; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Species Specificity; Temperature; Tetradecanoylphorbol Acetate | 1987 |
Phorbol myristate acetate inhibits growth in S49 cells: isolation of resistant variants.
Topics: Animals; Cell Division; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Lymphoma; Mice; Molecular Weight; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1987 |
4 beta-PDBu contracts parenchymal strip and synergizes with raised cytosolic calcium.
Topics: Animals; Calcium; Cytosol; Dimethyl Sulfoxide; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate | 1987 |
Purification and characterization of calcium/phospholipid-dependent kinase from adult human epidermis.
Topics: Adult; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Cell Membrane; Cytosol; Diglycerides; Epidermis; Humans; Membrane Proteins; Molecular Weight; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1987 |
1,2-Diacylglycerols but not phorbol esters stimulate sphingomyelin hydrolysis in GH3 pituitary cells.
Topics: Animals; Ceramides; Choline; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Glycerides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Neoplasms; Rats; Sphingomyelin Phosphodiesterase; Sphingomyelins; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured | 1987 |
Phorbol-ester-induced alterations of free calcium ion transients in single rat hepatocytes.
Topics: Aequorin; Animals; Arginine Vasopressin; Biological Transport; Calcium; In Vitro Techniques; Liver; Male; Phenylephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1987 |
Comparison of the activity of phorbol 12-myristate 13-acetate and the diglyceride glycerol 1-myristate 2-acetate.
Topics: Animals; Cell Line; Diglycerides; Epidermal Growth Factor; Fibroblasts; Glycerides; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Antagonistic effects of phorbol esters on lymphocyte activation. Evidence that protein kinase C provides an early signal associated with lytic function.
Topics: Animals; Cell Line; Kinetics; Lymphocyte Activation; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; T-Lymphocytes, Cytotoxic; Tetradecanoylphorbol Acetate | 1986 |
Altered protein kinase C in a mast cell variant defective in exocytosis.
Topics: Animals; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Cell Line; Exocytosis; Genetic Variation; Interleukin-3; Mast Cells; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Serotonin; Tetradecanoylphorbol Acetate | 1987 |
Inhibition of DNA synthesis by phorbol esters through protein kinase C in cultured rabbit aortic smooth muscle cells.
Topics: Animals; Aorta, Thoracic; Cells, Cultured; DNA Replication; Epidermal Growth Factor; Male; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Platelet-Derived Growth Factor; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate | 1987 |
Perturbation of cultured human vascular endothelial cells by phorbol ester or thrombin alters the cellular von Willebrand factor distribution.
Topics: Cells, Cultured; Endothelium, Vascular; Extracellular Matrix; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; RNA, Messenger; Subcellular Fractions; Tetradecanoylphorbol Acetate; Thrombin; von Willebrand Factor | 1987 |
Synergistic interaction between interleukin 4 and anti-Bp50 (CDw40) revealed in a novel B cell restimulation assay.
Topics: Antibodies, Monoclonal; Antigens, Differentiation; B-Lymphocytes; DNA; Ethers; Humans; Interleukin-4; Interleukins; Ionomycin; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate | 1987 |
Protein kinase C-mediated feed back inhibition of the Ca2+ response at the EGF receptor.
Topics: Calcium; Carcinoma, Squamous Cell; Enzyme Activation; Epidermal Growth Factor; ErbB Receptors; Feedback; Inositol Phosphates; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1987 |
Phorbol ester-stimulated phosphorylation of basolateral membranes from canine kidney.
Topics: Adenosine Triphosphate; alpha-Glucosidases; Amino Acids; Animals; Dogs; In Vitro Techniques; Kidney; Membranes; Microvilli; Osmolar Concentration; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phospholipids; Phosphorylation; Stimulation, Chemical; Tetradecanoylphorbol Acetate; Tritium | 1986 |
Quantitation of protein kinase C by immunoblot--expression in different cell lines and response to phorbol esters.
Topics: Animals; Antigen-Antibody Complex; Cattle; Cell Line; Glioma; Humans; Immunologic Techniques; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rabbits; Rats; Tetradecanoylphorbol Acetate | 1987 |
Phorbol esters increase calcitonin gene transcription and decrease c-myc mRNA levels in cultured human medullary thyroid carcinoma.
Topics: Calcitonin; Carcinogens; Cell Line; DNA; Genes; Humans; Kinetics; Oncogenes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; RNA, Messenger; Tetradecanoylphorbol Acetate; Thyroid Neoplasms; Transcription, Genetic | 1985 |
Comparative effects of a complete tumor promoter, TPA, and a second-stage tumor promoter, RPA, on intercellular communication, cell differentiation and cell transformation.
Topics: Animals; Cell Communication; Cell Differentiation; Cell Transformation, Neoplastic; Cells, Cultured; Mice; Mice, Inbred BALB C; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1985 |
Characterization of the growth inhibition induced by tumor-promoting phorbol esters and of their receptor binding in A549 human lung carcinoma cells.
Topics: Caenorhabditis elegans Proteins; Carcinoma; Carrier Proteins; Cell Division; Cells, Cultured; Humans; Lung Neoplasms; Male; Middle Aged; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Tritium; Type C Phospholipases | 1985 |
Glucocorticoid-mediated increases in glycerol phosphate dehydrogenase activity is inhibited by the phorbol ester tumor promoters.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Dexamethasone; Enzyme Induction; Glioma; Glycerolphosphate Dehydrogenase; Oligodendroglia; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Theophylline | 1985 |
Induction and desensitization of plasminogen activator gene expression by tumor promoters.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcitonin; Carcinogens; Cell Line; Cycloheximide; Dexamethasone; Diterpenes; Dose-Response Relationship, Drug; Enzyme Induction; Gene Expression Regulation; Kidney; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; RNA, Messenger; Swine; Terpenes; Tetradecanoylphorbol Acetate; Transcription, Genetic; Urokinase-Type Plasminogen Activator | 1985 |
Cellular uptake and localization of fluorescent derivatives of phorbol ester tumor promoters.
Topics: Animals; Binding, Competitive; Cattle; Cell Line; Chick Embryo; Cytoplasm; Dansyl Compounds; Enzyme Activation; Fluorescent Dyes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1985 |
Effects of 6-thioguanine on communication competence and factors affecting reversibility of phorbol ester inhibition in V79 cells measured by the metabolic cooperation assay and by dye coupling.
Topics: Animals; Cell Communication; Cells, Cultured; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Hypoxanthine Phosphoribosyltransferase; Isoquinolines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate; Thioguanine | 1985 |
The 65-kDa phorbol-diester hydrolase in mouse plasma is esterase 1 and is immunologically distinct from the 56-kDa phorbol-diester hydrolase in mouse liver.
Topics: Animals; Antibody Specificity; Carboxylesterase; Carboxylic Ester Hydrolases; Chromatography, High Pressure Liquid; Cross Reactions; Estradiol; Kinetics; Liver; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1985 |
Role of phorbol ester receptors in the 12-0-tetradecanoyl-phorbol-13-acetate (TPA)-induced down-regulation of colony-stimulating factor (CSF-1) binding to murine peritoneal exudate macrophages.
Topics: Animals; Ascitic Fluid; Caenorhabditis elegans Proteins; Carrier Proteins; Colony-Stimulating Factors; Macrophages; Mice; Mice, Inbred C3H; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Temperature; Tetradecanoylphorbol Acetate; Time Factors | 1985 |
Sensitization of frog erythrocyte adenylate cyclase system by tumor-promoting phorbol diesters.
Topics: Adenylyl Cyclases; Animals; Carcinogens; Erythrocyte Membrane; Erythrocytes; Fluorides; Isoproterenol; Kinetics; Manganese; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rana pipiens; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1985 |
Bryostatins: potent, new mitogens that mimic phorbol ester tumor promoters.
Topics: Animals; Bryostatins; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cells, Cultured; Insulin; Lactones; Macrolides; Mice; Mitogens; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Thymidine | 1985 |
Effects of phorbol myristate acetate, phorbol dibutyrate, ethanol, dimethylsulfoxide, phenol, and seven metabolites of phenol on metabolic cooperation between Chinese hamster V79 lung fibroblasts.
Topics: Animals; Carcinogens; Cell Communication; Cells, Cultured; Cricetinae; Cricetulus; Dimethyl Sulfoxide; Ethanol; Fibroblasts; Lung; Phenol; Phenols; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1985 |
Reversibility of phorbol diester-induced macrophage spreading.
Topics: Animals; Female; Macrophages; Mice; Mice, Inbred ICR; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1985 |
gamma-Interferon enhances the secretion of arachidonic acid metabolites from murine peritoneal macrophages stimulated with phorbol diesters.
Topics: Adjuvants, Immunologic; Animals; Arachidonic Acid; Arachidonic Acids; Interferon-gamma; Macrophage Activation; Macrophages; Mice; Mice, Inbred C57BL; Peritoneal Cavity; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins; SRS-A; Tetradecanoylphorbol Acetate; Thromboxane B2 | 1985 |
Similar effects of phospholipase C and phorbol ester tumor promoters on primary mouse epidermal cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Caenorhabditis elegans Proteins; Carrier Proteins; Cells, Cultured; Diglycerides; Enzyme Induction; Epidermal Growth Factor; Epidermis; Mice; Mice, Inbred BALB C; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Tritium; Type C Phospholipases | 1985 |
Inhibition of cell communication between Balb/c 3T3 cells by tumor promoters and protection by cAMP.
Topics: Animals; Bucladesine; Caenorhabditis elegans Proteins; Caffeine; Carcinogens; Carrier Proteins; Cell Communication; Cells, Cultured; Cricetinae; Cricetulus; Cyclic AMP; Fluorescent Dyes; Isoquinolines; Lung; Mice; Mice, Inbred BALB C; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate | 1984 |
Biological responsiveness to the phorbol esters and specific binding of [3H]phorbol 12,13-dibutyrate in the nematode Caenorhabditis elegans, a manipulable genetic system.
Topics: Animals; Caenorhabditis; Carcinogens; Movement; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Tritium | 1982 |
Tumour promoter-mediated reversible inhibition of cell-cell communication (electrical coupling). Relationship with phorbol ester binding and de novo macromolecule synthesis.
Topics: Binding Sites; Cell Communication; Cell Line; Cycloheximide; Dactinomycin; Diterpenes; Electrophysiology; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Biosynthesis; RNA; Terpenes; Tetradecanoylphorbol Acetate | 1983 |
Activation of protein kinase C by non-phorbol tumor promoter, mezerein.
Topics: Animals; Brain; Carcinogens; Diterpenes; Enzyme Activation; Humans; In Vitro Techniques; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phospholipids; Protein Binding; Protein Kinase C; Protein Kinases; Rats; Structure-Activity Relationship; Terpenes; Tetradecanoylphorbol Acetate | 1984 |
Phorbol ester stimulation of Na influx and Na-K pump activity in Swiss 3T3 cells.
Topics: Animals; Biological Transport, Active; Carcinogens; Cells, Cultured; Kinetics; Mice; Mice, Inbred Strains; Monensin; Ouabain; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rubidium; Sodium; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate | 1981 |
Inhibition of epidermal growth factor binding to mouse embryonal carcinoma cells by phorbol esters mediated by specific phorbol ester receptors.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Epidermal Growth Factor; ErbB Receptors; Kinetics; Mice; Neoplasms, Experimental; Peptides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Teratoma; Tetradecanoylphorbol Acetate | 1981 |
Tumor promoter binding to rat mammary cell cultures: role of receptors in the inhibition of dome formation.
Topics: Animals; Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Female; Mammary Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Cell Surface; Receptors, Drug; Temperature; Tetradecanoylphorbol Acetate; Time Factors | 1983 |
Specific desensitization to tumor-promoting phorbol esters in mouse pituitary cells. Evidence that desensitization is a two-step process.
Topics: Adrenocorticotropic Hormone; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pituitary Neoplasms; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
Control of endogenous cell regulators by the second-stage tumor promoter phorbol-12-retinoate 13-acetate.
Topics: Animals; Binding, Competitive; Cell Differentiation; Cells, Cultured; Cyclic AMP; Glycoproteins; Growth Inhibitors; Interleukin-6; Leukemia Inhibitory Factor; Leukemia, Myeloid; Lymphokines; Mice; Muramidase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins E; Tetradecanoylphorbol Acetate | 1983 |
Binding of phorbol dibutyrate and epidermal growth factor to cultured human epidermal cells.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Epidermal Growth Factor; ErbB Receptors; Humans; Melanoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin Neoplasms; Tetradecanoylphorbol Acetate | 1983 |
Characterization of a high-affinity receptor for phorbol esters in rat alveolar macrophages.
Topics: Animals; Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Kinetics; Macrophages; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Pulmonary Alveoli; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
The role of phorbol ester receptor binding in responses to promoters by mouse and human cells.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Differentiation; Cell Line; Clone Cells; Drug Resistance; Humans; Leukemia, Myeloid, Acute; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin; Tetradecanoylphorbol Acetate | 1983 |
An inhibitory effect of tumour promoters on human epithelial cell growth can be dissociated from an effect on junctional communication.
Topics: Breast Neoplasms; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Communication; Cell Division; Cell Line; Cell Transformation, Viral; Epidermal Cells; Epidermis; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
Tumor-promoting phorbol esters inhibit the binding of colony-stimulating factor (CSF-1) to murine peritoneal exudate macrophages.
Topics: Animals; Ascitic Fluid; Colony-Stimulating Factors; Dose-Response Relationship, Drug; Kinetics; Macrophages; Mice; Mice, Inbred C3H; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Receptors, Cell Surface; Receptors, Colony-Stimulating Factor; Temperature; Tetradecanoylphorbol Acetate | 1983 |
Antagonist of phorbol ester receptor-mediated chemotaxis in mouse peritoneal macrophages.
Topics: Animals; Ascitic Fluid; Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Chemotaxis; Female; Macrophages; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate; Time Factors | 1983 |
Phorbol diester-induced H2O2 production by peritoneal macrophages. Different H2O2 production by macrophages from normal and BCG-infected mice despite comparable phorbol diester receptors.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cells, Cultured; Female; Hydrogen Peroxide; Kinetics; Macrophages; Mice; Mice, Inbred Strains; Mycobacterium bovis; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
Epidermal growth factor and potent phorbol tumor promoters induce epidermal growth factor receptor phosphorylation in a similar but distinctively different manner in human epidermoid carcinoma A431 cells.
Topics: Carcinogens; Carcinoma, Squamous Cell; Cell Line; Epidermal Growth Factor; ErbB Receptors; Humans; Kinetics; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphorylation; Receptors, Cell Surface; Tetradecanoylphorbol Acetate | 1984 |
Possible mechanism of phorbol diester-induced maturation of human promyelocytic leukemia cells.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Differentiation; Cell Line; Enzyme Activation; Humans; Leukemia, Myeloid; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1984 |
Vinculin phosphorylation in response to calcium and phorbol esters in intact cells.
Topics: Animals; Bucladesine; Calcium; Cells, Cultured; Chick Embryo; Dibutyryl Cyclic GMP; Fibroblasts; Kinetics; Mice; Muscle Proteins; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphopeptides; Phosphorylation; Tetradecanoylphorbol Acetate; Trypsin; Vinculin | 1984 |
Communication between receptors for different ligands on a single cell: ligation of fibronectin receptors induces a reversible alteration in the function of complement receptors on cultured human monocytes.
Topics: Cell Communication; Fibronectins; Humans; Macrophage-1 Antigen; Monocytes; Phagocytosis; Phorbol 12,13-Dibutyrate; Phorbol Esters; Receptors, Cell Surface; Receptors, Complement; Receptors, Fibronectin; Serum Albumin; Tetradecanoylphorbol Acetate | 1984 |
Phorbol esters rapidly stimulate amiloride-sensitive Na+/H+ exchange in a human leukemic cell line.
Topics: Amiloride; Carrier Proteins; Cell Line; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pyrazines; Sodium-Hydrogen Exchangers; Tetradecanoylphorbol Acetate | 1984 |
Analysis of human promyelocytic leukemia cell (HL60) variants insensitive to phorbol ester tumor promoters.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Genetic Variation; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Superoxide Dismutase; Tetradecanoylphorbol Acetate | 1984 |
Phorbol esters inhibit murine B cell differentiation to immunoglobulin secretion but not proliferation.
Topics: Animals; Antibody-Producing Cells; B-Lymphocytes; Cell Differentiation; Dose-Response Relationship, Immunologic; Female; Immunoglobulin G; Immunoglobulin M; Immunosuppressive Agents; Kinetics; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1984 |
Phorbol diesters stimulate somatostatin secretion from cultured brain cells.
Topics: Alkaloids; Animals; Cell Line; Cerebral Cortex; Female; gamma-Aminobutyric Acid; Hypothalamus; Lyngbya Toxins; Peptides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pregnancy; Rats; Tetradecanoylphorbol Acetate; Verapamil | 1983 |
Teleocidin-induced phenotypic changes in thymic ALL cell line, HPB-ALL.
Topics: Adolescent; Alkaloids; Binding, Competitive; Carcinogens; Cell Differentiation; Cell Line; DNA; Humans; Leukemia, Lymphoid; Lyngbya Toxins; Male; Phenotype; Phorbol 12,13-Dibutyrate; Phorbol Esters; Rosette Formation; Tetradecanoylphorbol Acetate | 1983 |
Presence of specific binding sites for phorbol ester tumor promoters in human epidermal and dermal cells in culture but lack of down regulation in epidermal cells.
Topics: Binding Sites; Binding, Competitive; Cells, Cultured; Diterpenes; Epidermis; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Terpenes; Tetradecanoylphorbol Acetate | 1983 |
Control of macrophage cell differentiation in human promyelocytic HL-60 leukemia cells by 1,25-dihydroxyvitamin D3 and phorbol-12-myristate-13-acetate.
Topics: Antibodies, Monoclonal; Calcitriol; Cell Differentiation; Cell Line; Dimethyl Sulfoxide; Humans; Leukemia, Myeloid, Acute; Macrophages; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1983 |
Phorbol ester-associated changes in ganglioside metabolism.
Topics: Animals; Carcinogens; Cell Division; Cell Line; Contact Inhibition; Cricetinae; Gangliosides; Palmitic Acid; Palmitic Acids; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Sialic Acids; Sialyltransferases; Tetradecanoylphorbol Acetate | 1983 |
Phorbol 12,13-dibutyrate enhances lateral redistribution of membrane glycoproteins in human blood lymphocytes.
Topics: Glycoproteins; Humans; Immunologic Capping; Lymphocytes; Membrane Proteins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protease Inhibitors; Tetradecanoylphorbol Acetate | 1984 |
Inhibition of denuded mouse oocyte meiotic maturation by tumor-promoting phorbol esters and its reversal by retinoids.
Topics: Animals; Colforsin; Diterpenes; Drug Interactions; Female; Meiosis; Mice; Oocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Retinoids; Tetradecanoylphorbol Acetate | 1984 |
Phorbol esters inhibit agonist-induced [3H] inositol-1-phosphate accumulation in rat hippocampal slices.
Topics: Animals; Caenorhabditis elegans Proteins; Carbachol; Carcinogens; Carrier Proteins; Hippocampus; Inositol; Inositol Phosphates; Male; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate | 1984 |
Biological activity of a fluorescent 12-O-tetradecanoyl-phorbol-13-acetate derivative.
Topics: Animals; Cricetinae; Cricetulus; Dansyl Compounds; Fluorescence; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1984 |
Phorbol ester tumor promoters specifically stimulate choline phospholipid metabolism in human leukemic cells.
Topics: Acetates; Acetic Acid; Caenorhabditis elegans Proteins; Carbon Radioisotopes; Carcinogens; Carrier Proteins; Cells, Cultured; Choline; Humans; Leukemia, Hairy Cell; Microscopy, Electron, Scanning; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylcholines; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Tritium | 1984 |
Relationship between mezerein-mediated biological responses and phorbol ester receptor occupancy.
Topics: Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Dinoprostone; Diterpenes; Epidermal Growth Factor; Humans; Kinetics; Osteosarcoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins E; Protein Kinase C; Receptors, Drug; Terpenes; Tetradecanoylphorbol Acetate | 1983 |
The tumor promoter phorbol-12,13-dibutyrate [P(Bu)2] stimulates cytotoxic activity of human blood lymphocytes.
Topics: Cell Adhesion; Cytotoxicity, Immunologic; Humans; In Vitro Techniques; Killer Cells, Natural; Lymphocyte Activation; Lymphocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; T-Lymphocytes, Cytotoxic; Tetradecanoylphorbol Acetate; Time Factors | 1983 |
The control of phospholipid methylation by phorbol diesters in differentiating human myeloid HL-60 leukemia cells.
Topics: Alkaloids; Cell Differentiation; Cell Line; Humans; Leukemia, Myeloid, Acute; Lyngbya Toxins; Methylation; Methyltransferases; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylethanolamine N-Methyltransferase; Phospholipids; Tetradecanoylphorbol Acetate | 1982 |
Down regulation of specific binding of [20-3H]phorbol 12,13-dibutyrate and phorbol ester-induced differentiation of human promyelocytic leukemia cells.
Topics: Binding Sites; Binding, Competitive; Carcinogens; Cell Differentiation; Cell Line; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1981 |
TPA-resistance in Friend erythroleukemia cells: role of membrane lipid fluidity.
Topics: Animals; Carcinogens; Cell Line; Clone Cells; Diphenylhexatriene; Drug Resistance; Kinetics; Leukemia, Experimental; Membrane Fluidity; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Spectrometry, Fluorescence; Tetradecanoylphorbol Acetate | 1981 |
Analysis of phorbol ester receptors in phorbol ester unresponsive 3T3 cell variants.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cells, Cultured; Genetic Variation; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1981 |
Cell differentiation, alterations in polyamine levels, and specific binding of phorbol diesters in cultured human cells.
Topics: Binding Sites; Carcinogens; Cell Differentiation; Cell Line; Cell Membrane; Humans; Leukemia, Myeloid, Acute; Melanoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Polyamines; Tetradecanoylphorbol Acetate | 1982 |
Modulation of HeLa cell phospholipid metabolism and ornithine decarboxylase activity by tumour promoters: regulation of response to phorbol-12,13-dibutyrate by receptor occupancy time.
Topics: Caenorhabditis elegans Proteins; Carboxy-Lyases; Carrier Proteins; Enzyme Induction; HeLa Cells; Humans; Kinetics; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1982 |
Specific binding of phorbol esters to Friend erythroleukemia cells--general properties, down regulation and relationship to cell differentiation.
Topics: Animals; Binding Sites; Cell Differentiation; Diterpenes; Friend murine leukemia virus; Leukemia, Erythroblastic, Acute; Leukemia, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate; Tritium | 1982 |
Specific receptors for phorbol esters in lymphoid cell populations: role in enhanced production of T-cell growth factor.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Humans; Interleukin-2; Kinetics; Lymphokines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Structure-Activity Relationship; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1981 |
Endotoxin-induced tissue factor in human monocytes is dependent upon protein kinase C activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Endotoxins; Enzyme Activation; Gene Expression Regulation; Humans; Isoquinolines; Monocytes; Naphthalenes; Naphthol AS D Esterase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Polycyclic Compounds; Protein Kinase C; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Thromboplastin | 1993 |
Direct stimulation of Vav guanine nucleotide exchange activity for Ras by phorbol esters and diglycerides.
Topics: Alkaloids; Amino Acid Sequence; Animals; Base Sequence; Benzoquinones; Cell Cycle Proteins; Cell Line; Ceramides; Chlorocebus aethiops; Diglycerides; DNA Primers; GTP-Binding Proteins; Guanosine Diphosphate; Humans; Kinetics; Lactams, Macrocyclic; Molecular Sequence Data; Muromonab-CD3; Mutagenesis, Site-Directed; Naphthalenes; Phorbol 12,13-Dibutyrate; Point Mutation; Polycyclic Compounds; Protein Kinase C; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-vav; Proto-Oncogene Proteins p21(ras); Quinones; Receptor Protein-Tyrosine Kinases; Rifabutin; Staurosporine; T-Lymphocytes; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 1994 |
Possible role of protein kinase C-epsilon isoenzyme in inhibition of interleukin 1 beta induction of nitric oxide synthase in rat renal mesangial cells.
Topics: Amino Acid Oxidoreductases; Animals; Blotting, Northern; Cells, Cultured; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Induction; Glomerular Mesangium; Interleukin-1; Isoenzymes; NADH Dehydrogenase; Naphthalenes; Nitric Oxide Synthase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Polycyclic Compounds; Protein Kinase C; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate | 1994 |
Loss of adenosine-induced negative inotropic effect in hyperexcited rabbit hearts: relationship to PKC.
Topics: Acetylcholine; Adenosine; Angiotensin II; Animals; Behavior, Animal; Biphenyl Compounds; Blood Pressure; Depression, Chemical; Enzyme Activation; Heart Rate; Imidazoles; In Vitro Techniques; Losartan; Male; Myocardial Contraction; Naphthalenes; Norepinephrine; Perfusion; Phentolamine; Phorbol 12,13-Dibutyrate; Polycyclic Compounds; Propranolol; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Tetrazoles | 1995 |
The protein kinase C isoforms leading to MAP-kinase activation in CHO cells.
Topics: Amino Acid Sequence; Animals; Binding Sites; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; CHO Cells; Chromatography; Chromatography, Gel; Chromatography, Ion Exchange; Cricetinae; Cytosol; Durapatite; Enzyme Activation; Immunoblotting; Isoenzymes; Kinetics; Molecular Sequence Data; Phorbol 12,13-Dibutyrate; Phosphotyrosine; Protein Kinase C; Tetradecanoylphorbol Acetate; Tyrosine | 1995 |
Phorbol esters elicit Ca(2+)-dependent delayed contractions in diabetic rat aorta.
Topics: Alkaloids; Animals; Aorta; Body Weight; Calcium; Diabetes Mellitus, Experimental; Male; Muscle Contraction; Muscle, Smooth, Vascular; Organ Size; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate | 1995 |
Dissociation between changes in cytoplasmic free Ca2+ concentration and insulin secretion as evidenced from measurements in mouse single pancreatic islets.
Topics: Animals; Biological Transport; Calcium; Cell Compartmentation; Colforsin; Cytoplasm; Enzyme Inhibitors; Ethers, Cyclic; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Isoenzymes; Membranes; Mice; Mice, Obese; Okadaic Acid; Phorbol 12,13-Dibutyrate; Potassium; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Radioimmunoassay; Tetradecanoylphorbol Acetate | 1995 |
Determinants of PKC-dependent modulation of a family of neuronal calcium channels.
Topics: Animals; Calcium; Calcium Channels; Egtazic Acid; Electric Conductivity; Female; GTP-Binding Proteins; Indicators and Reagents; Kinetics; Macromolecular Substances; Neurons; Oocytes; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Metabotropic Glutamate; Second Messenger Systems; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella; Xenopus laevis | 1995 |
Mechanism of interaction of protein kinase C with phorbol esters. Reversibility and nature of membrane association.
Topics: Calcium; Diglycerides; Kinetics; Liposomes; Membrane Fluidity; Osmolar Concentration; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylcholines; Protein Binding; Protein Kinase C; Spectrometry, Fluorescence; Tetradecanoylphorbol Acetate; Tryptophan | 1995 |
Depression of the spontaneous activity by phorbol esters in young embryonic chick cardiomyocytes.
Topics: Action Potentials; Animals; Calcium Channels; Cardiac Pacing, Artificial; Chick Embryo; Computer Simulation; Heart Conduction System; Heart Ventricles; Myocardium; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Potassium Channels; Protein Kinase C; Temperature; Tetradecanoylphorbol Acetate | 1995 |
Influence of protein kinase C activation on basophils from patients with atopic dermatitis in comparison with nonatopic controls.
Topics: Adolescent; Adult; Aged; Basophils; Bombesin; Dermatitis, Atopic; Diglycerides; Diterpenes; Eczema; Enzyme Activation; Female; Histamine; Histamine Release; Humans; Immunoglobulin E; Male; Middle Aged; Phorbol 12,13-Dibutyrate; Protein Kinase C; Signal Transduction; Terpenes; Tetradecanoylphorbol Acetate | 1993 |
Differential effects of putative protein kinase C inhibitors on contraction of rat aortic smooth muscle.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Aorta; Dose-Response Relationship, Drug; Isoquinolines; Male; Muscle, Smooth, Vascular; Naphthalenes; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Polycyclic Compounds; Potassium Chloride; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors; Vasoconstriction | 1993 |
Calcium dependent positive inotropic effects of low phorbol ester concentrations in isolated rat hearts.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Chloride; Dose-Response Relationship, Drug; Drug Interactions; Energy Metabolism; Male; Myocardial Contraction; Myocardium; Phorbol 12,13-Dibutyrate; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Time Factors | 1993 |
Regulation of parathyroid hormone messenger RNA levels by protein kinase A and C in bovine parathyroid cells.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Alkaloids; Analysis of Variance; Animals; Calcium; Cattle; Cells, Cultured; Cholera Toxin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Gene Expression Regulation, Enzymologic; Nucleic Acid Hybridization; Parathyroid Glands; Parathyroid Hormone; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Protein Kinase C; RNA, Messenger; RNA, Ribosomal, 18S; Staurosporine; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1995 |
Up- and down-modulation of a cloned Aplysia K+ channel (AKv1.1a) by the activators of protein kinase C.
Topics: Amino Acid Sequence; Animals; Aplysia; Base Sequence; Cloning, Molecular; Diglycerides; DNA, Complementary; Down-Regulation; Enzyme Activation; Kinetics; Molecular Sequence Data; Phorbol 12,13-Dibutyrate; Phosphorylation; Potassium Channels; Protein Kinase C; Shaker Superfamily of Potassium Channels; Tetradecanoylphorbol Acetate; Up-Regulation; Xenopus | 1995 |
Multiple intracellular signallings are involved in thyrotropin-releasing hormone (TRH)-induced c-fos and jun B mRNA levels in clonal prolactin cells.
Topics: Adenylyl Cyclases; Animals; Calcium; Clone Cells; Colforsin; Cyclic AMP; Gene Expression Regulation, Neoplastic; Genes, fos; Genes, jun; Ionomycin; Neoplasm Proteins; Nuclear Proteins; Phorbol 12,13-Dibutyrate; Pituitary Gland, Anterior; Pituitary Neoplasms; Prolactin; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Rats; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Tumor Cells, Cultured | 1995 |
Activation of protein kinase C by phorbol esters disrupts the tegument of Schistosoma mansoni.
Topics: Animals; Biomphalaria; Enzyme Activation; Female; Humans; Male; Mice; Microscopy, Electron; Microscopy, Electron, Scanning; Phorbol 12,13-Dibutyrate; Protein Kinase C; Schistosoma mansoni; Tetradecanoylphorbol Acetate | 1994 |
Mutual antagonistic interactions between the thyrotropin (adenosine 3',5'-monophosphate) and protein kinase C/epidermal growth factor (tyrosine kinase) pathways in cell proliferation and differentiation of cultured human thyroid follicles.
Topics: Alkaloids; Cell Differentiation; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Epidermal Growth Factor; Humans; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein-Tyrosine Kinases; Second Messenger Systems; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin | 1995 |
Differentiation- and protein kinase C-dependent regulation of alanine transport via system B.
Topics: Alanine; beta-Alanine; Biological Transport; Cell Differentiation; Cell Line; Cellular Senescence; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Protein Kinase C; Sodium; Tetradecanoylphorbol Acetate | 1995 |
Mechanism of transferrin receptor down-regulation in K562 cells in response to protein kinase C activation.
Topics: Bryostatins; Cell Compartmentation; Down-Regulation; Endocytosis; Enzyme Activation; Humans; Lactones; Macrolides; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Transferrin; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1995 |
Induction of c-fos in pituitary cells by thyrotrophin-releasing hormone and phorbol 12-myristate 13-acetate depends upon Ca2+ influx.
Topics: Alkaloids; Animals; Calcium; Cell Line; Culture Media, Serum-Free; Cytoplasm; Down-Regulation; Edetic Acid; Egtazic Acid; Epidermal Growth Factor; Gene Expression Regulation; Genes, fos; Phorbol 12,13-Dibutyrate; Pituitary Gland; Protein Kinase C; RNA, Messenger; Staurosporine; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Transcription, Genetic | 1994 |
Heterologous sensitization of adenylate cyclase activity by serotonin in the rat cerebral cortex.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Colforsin; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Phorbol 12,13-Dibutyrate; Propanolamines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Somatostatin; Tetradecanoylphorbol Acetate; Vasoactive Intestinal Peptide | 1993 |
Phorbol esters impair endothelium-dependent and independent relaxation in rat aortic rings.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Calcimycin; Endothelium, Vascular; Enzyme Activation; Female; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroprusside; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1994 |
Translocation of protein kinase Cs in Aplysia neurons: evidence for complex regulation.
Topics: Animals; Aplysia; Ganglia, Invertebrate; Immunoblotting; In Vitro Techniques; Isoenzymes; Kinetics; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Processing, Post-Translational; Synaptosomes; Tetradecanoylphorbol Acetate | 1994 |
Phorbol ester-, but not ligand-mediated activation of protein kinase C increases angiotensin binding to rat intestinal epithelial (RIE-1) cells.
Topics: Angiotensin II; Animals; Cell Line; Enzyme Activation; Epithelial Cells; Intestinal Mucosa; Ionomycin; Ligands; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Receptors, Angiotensin; Tetradecanoylphorbol Acetate; Up-Regulation | 1994 |
Tobacco smoke tumor promoters, catechol and hydroquinone, induce oxidative regulation of protein kinase C and influence invasion and metastasis of lung carcinoma cells.
Topics: Animals; Carcinogens; Catechols; Cell Membrane; Chelating Agents; Cytosol; Hydroquinones; Lung Neoplasms; Mice; Mice, Inbred C57BL; Neoplasm Invasiveness; Neoplasm Metastasis; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred Lew; Smoke; Smoking; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1994 |
Elevation of intracellular Ca2+ concentration by protein kinase C stimulation in isolated single rabbit sino-atrial node cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Electrophysiology; Fura-2; In Vitro Techniques; Isoproterenol; Isoquinolines; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rabbits; Sinoatrial Node; Stimulation, Chemical; Tetradecanoylphorbol Acetate | 1994 |
Protein kinase C and adaptation to ethanol.
Topics: Acclimatization; Animals; Calcium; Calcium Channels; Cell Differentiation; Ethanol; Isoenzymes; Nerve Growth Factors; Neurites; Neurons; PC12 Cells; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; RNA, Messenger; Signal Transduction; Sphingosine; Tetradecanoylphorbol Acetate | 1994 |
Overexpressed protein kinase C-delta and -epsilon subtypes in NIH 3T3 cells exhibit differential subcellular localization and differential regulation of sodium-dependent phosphate uptake.
Topics: 3T3 Cells; Animals; Biological Transport; Blotting, Western; Cell Division; Electrophoresis, Polyacrylamide Gel; Enzyme Induction; Gene Expression; Isoenzymes; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phosphates; Protein Binding; Protein Kinase C; Sodium; Subcellular Fractions; Tetradecanoylphorbol Acetate; Transfection; Zinc | 1994 |
Involvement of protein kinase C activation in regulation of acetylcholine release from rat hippocampal slices by minaprine.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Acetylcholine; Alkaloids; Animals; Enzyme Activation; Hippocampus; In Vitro Techniques; Isoquinolines; Male; Phorbol 12,13-Dibutyrate; Piperazines; Potassium; Protein Kinase C; Pyridazines; Rats; Rats, Wistar; Serotonin; Staurosporine; Synaptosomes; Tetradecanoylphorbol Acetate | 1994 |
Schistosoma mansoni: myogenic characteristics of phorbol ester-induced muscle contraction.
Topics: Acetylcholine; Animals; Cadmium; Calcimycin; Calcium; Calcium Channels; Carbachol; Cell Membrane Permeability; Dose-Response Relationship, Drug; Electromyography; Hydrogen-Ion Concentration; Male; Membrane Potentials; Microelectrodes; Muscle Contraction; Nicardipine; Phorbol 12,13-Dibutyrate; Praziquantel; Protein Kinase C; Schistosoma mansoni; Serotonin; Sodium; Tetradecanoylphorbol Acetate | 1994 |
Interplay between differentiation and cell cycle arrest at G1 in phorbol diester-treated human myelocytic leukemia cells.
Topics: Cell Differentiation; G1 Phase; Humans; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1993 |
Growth of melanocytic cells is associated with down-regulation of protein kinase C alpha, delta, and epsilon isoforms. Possible role of diacylglycerol.
Topics: Animals; Cell Division; Cells, Cultured; Diglycerides; DNA; Down-Regulation; Isoenzymes; Melanocytes; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1993 |
1,25-Dihydroxyvitamin D3 and macrophage colony-stimulating factor-1 synergistically phosphorylate talin.
Topics: Alkaloids; Animals; Calcitriol; Cell Line; Drug Synergism; Genistein; Isoflavones; L Cells; Macrophage Colony-Stimulating Factor; Macrophages; Mice; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Phosphoserine; Protein Kinase C; Protein-Tyrosine Kinases; Receptor, Macrophage Colony-Stimulating Factor; Staurosporine; Talin; Tetradecanoylphorbol Acetate | 1993 |
Phorbol ester sequentially downregulates cAMP-regulated basolateral and apical Cl- transport pathways in T84 cells.
Topics: Biological Transport; Carrier Proteins; Cell Line; Cell Membrane; Chlorides; Colforsin; Colon; Cyclic AMP; Electrophysiology; Humans; Phorbol 12,13-Dibutyrate; Potassium; Protein Kinase C; Sodium-Potassium-Chloride Symporters; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate; Time Factors | 1993 |
Effects of tannic acid on 12-O-tetradecanoylphorbol-13-acetate-induced protein kinase C activation in NIH 3T3 cells.
Topics: 3T3 Cells; Animals; DNA; Drug Interactions; Enzyme Activation; Hydrolyzable Tannins; Mice; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate | 1993 |
Phorbol 12-myristate 13-acetate stimulates proliferation and ductal morphogenesis and inhibits functional differentiation of normal rat mammary epithelial cells in primary culture.
Topics: Animals; Caseins; Cell Differentiation; Cell Division; Cells, Cultured; Epithelial Cells; Epithelium; Female; Mammary Glands, Animal; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Reference Values; Tetradecanoylphorbol Acetate | 1994 |
Effects of phorbol esters on contraction and protein kinase C activation in rabbit aorta.
Topics: Animals; Aorta, Thoracic; Enzyme Activation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate | 1994 |
Diradylglycerols stimulate phospholipase A2 and subsequent exocytosis in ram spermatozoa. Evidence that the effect is not mediated via protein kinase C.
Topics: Acrosome; Animals; Arachidonic Acid; Calcimycin; Calcium; Diglycerides; Enzyme Activation; Exocytosis; Glycerides; Male; Phorbol 12,13-Dibutyrate; Phospholipases A; Phospholipases A2; Protein Kinase C; Sheep; Spermatozoa; Tetradecanoylphorbol Acetate | 1994 |
Toxicity of phorbol esters for human epithelial cells expressing a mutant ras oncogene.
Topics: Antineoplastic Agents; Bryostatins; Cell Division; Cell Line; DNA; Epithelial Cells; Epithelium; Gene Expression Regulation; Genes, ras; Humans; Lactones; Macrolides; Models, Biological; Mutation; Phorbol 12,13-Dibutyrate; Phorbol Esters; Proto-Oncogene Proteins p21(ras); Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Thyroid Gland; Zinc | 1993 |
Phorbol esters and norepinephrine destabilize alpha 1B-adrenergic receptor mRNA in vascular smooth muscle cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aorta; Bradykinin; Cells, Cultured; Diglycerides; Down-Regulation; Ethers, Cyclic; Inositol Phosphates; Isoquinolines; Kinetics; Models, Biological; Muscle, Smooth, Vascular; Norepinephrine; Okadaic Acid; Phorbol 12,13-Dibutyrate; Phosphoprotein Phosphatases; Piperazines; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha-1; RNA, Messenger; Tetradecanoylphorbol Acetate | 1994 |
Protein kinase C-mediated inhibition of vascular smooth muscle cell proliferation: the isoforms that may mediate G1/S inhibition.
Topics: Animals; Cell Cycle; Cells, Cultured; In Vitro Techniques; Isoenzymes; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Protein Kinase C; S Phase; Swine; Tetradecanoylphorbol Acetate | 1993 |
Protein kinase C modulates glutamate receptor inhibition of Ca2+ channels and synaptic transmission.
Topics: Animals; Calcium Channels; Cyclopentanes; Dimethyl Sulfoxide; Enzyme Activation; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kinetics; Membrane Potentials; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Pyramidal Tracts; Rats; Receptors, Glutamate; Synapses; Synaptic Transmission; Tetradecanoylphorbol Acetate | 1993 |
Phorbol esters inhibit insulin-induced receptor down-regulation in cultured human lymphocytes: association with diminished insulin receptor autophosphorylation.
Topics: Cell Line; Down-Regulation; Enzyme Activation; Humans; Insulin; Lymphocytes; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Receptor, Insulin; Sphingosine; Tetradecanoylphorbol Acetate | 1993 |
Type-specific stimulation of adenylylcyclase by protein kinase C.
Topics: Adenylyl Cyclases; Alkaloids; Cells, Cultured; Cyclic AMP; DNA; Enzyme Activation; Humans; Isoenzymes; Phorbol 12,13-Dibutyrate; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1993 |
alpha-Adrenergic augmentation of myogenic response in rat arterioles: role of protein kinase C.
Topics: Animals; Arterioles; In Vitro Techniques; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate; Vasoconstriction | 1993 |
Mechanisms by which glucose can control insulin release independently from its action on adenosine triphosphate-sensitive K+ channels in mouse B cells.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Diazoxide; Diterpenes; Glucose; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Keto Acids; Kinetics; Male; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Potassium; Potassium Channels; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate | 1993 |
Phorbol ester-stimulated exocytosis in lacrimal gland: PKC might not be the sole effector.
Topics: Alkaloids; Animals; Benzophenanthridines; Bucladesine; Diglycerides; Exocytosis; In Vitro Techniques; Lacrimal Apparatus; Male; Phenanthridines; Phorbol 12,13-Dibutyrate; Protein Kinase C; Proteins; Rats; Rats, Sprague-Dawley; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate; Trifluoperazine | 1993 |
Genistein induces apoptosis in immature human thymocytes by inhibiting topoisomerase-II.
Topics: Apoptosis; Benzoquinones; Cells, Cultured; Chromatin; DNA Damage; Etoposide; Genistein; Humans; Immunophenotyping; Infant; Isoflavones; Kinetics; Lactams, Macrocyclic; Methylprednisolone; Novobiocin; Phorbol 12,13-Dibutyrate; Protein-Tyrosine Kinases; Quinones; Rifabutin; T-Lymphocytes; Tetradecanoylphorbol Acetate; Thymus Gland; Time Factors; Topoisomerase II Inhibitors | 1993 |
Modulation of beta-amyloid precursor protein secretion in differentiated and nondifferentiated cells.
Topics: Amyloid beta-Protein Precursor; Animals; Bucladesine; Calcimycin; Carcinogens; Cell Differentiation; Cell Line; Culture Media; PC12 Cells; Phorbol 12,13-Dibutyrate; Phorbol Esters; Tetradecanoylphorbol Acetate | 1993 |
Effect of protein kinase-C depletion on inositol trisphosphate-mediated and cyclic adenosine 3',5'-monophosphate-dependent protein kinase-mediated adrenocorticotropin secretion.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenocorticotropic Hormone; Animals; Arginine Vasopressin; Cyclic AMP; Cycloheximide; Diglycerides; Inositol 1,4,5-Trisphosphate; Ionomycin; Male; Perfusion; Phorbol 12,13-Dibutyrate; Pituitary Gland, Anterior; Potassium Chloride; Protein Kinase C; Protein Kinases; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1993 |
Further characterization of 5-HT- and 5-HT3 receptor agonists'-stimulated phosphoinositol phosphates accumulation.
Topics: Animals; GTP-Binding Proteins; Inositol Phosphates; Male; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbols; Phosphatidylinositols; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1993 |
Possible involvement of protein kinase C in gonadotropin-induced ovulation in the rat ovary.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bucladesine; Cells, Cultured; Female; Gonadotropins, Equine; Granulosa Cells; Isoquinolines; Luteinizing Hormone; Ovary; Ovulation; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Tissue Plasminogen Activator | 1993 |
Phorbol myristate acetate induction of chemotactic migration of human polymorphonuclear neutrophils.
Topics: Chemotaxis, Leukocyte; Humans; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate | 1993 |
Evidence for an altered protein kinase C (PKC) signaling pathway in psoriasis.
Topics: Alkaloids; Cells, Cultured; Fluorometry; Humans; Isoelectric Focusing; Keratinocytes; Phorbol 12,13-Dibutyrate; Protein Kinase C; Psoriasis; Reference Values; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate | 1993 |
Role for protein kinase C in the mediation of increased fibronectin accumulation by mesangial cells grown in high-glucose medium.
Topics: Animals; Cell Line; Dose-Response Relationship, Drug; Female; Fibronectins; Glomerular Mesangium; Glucose; Intracellular Signaling Peptides and Proteins; Kinetics; Membrane Proteins; Molecular Weight; Myristoylated Alanine-Rich C Kinase Substrate; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Protein Kinase C; Proteins; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1993 |
Two phorbol ester receptor affinities in partially transformed human urothelial cells and decrease of receptor binding in desensitized cells.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line, Transformed; Cell Transformation, Neoplastic; Dose-Response Relationship, Drug; Humans; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate; Urinary Bladder; Urinary Bladder Neoplasms | 1993 |
Stimulation of calcium uptake in Saccharomyces cerevisiae by bovine protein kinase C alpha.
Topics: Amino Acid Sequence; Animals; Base Sequence; Calcium; Cattle; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Oligopeptides; Phorbol 12,13-Dibutyrate; Plasmids; Protein Binding; Protein Kinase C; Recombinant Proteins; Saccharomyces cerevisiae; Substrate Specificity; Tetradecanoylphorbol Acetate | 1993 |
Role of protein kinase C in bradykinin-induced prostaglandin formation in osteoblasts.
Topics: Alkaloids; Animals; Bradykinin; Calcimycin; Cell Membrane; Cells, Cultured; Dinoprostone; Enzyme Activation; Hydrocortisone; Indomethacin; Mice; Osteoblasts; Phorbol 12,13-Dibutyrate; Prostaglandins; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate | 1993 |
Cobra venom cardiotoxin (cytotoxin) isoforms and neurotoxin: comparative potency of protein kinase C inhibition and cancer cell cytotoxicity and modes of enzyme inhibition.
Topics: Amino Acid Sequence; Animals; Brain; Cell Differentiation; Cell Survival; Cytotoxins; Elapid Venoms; Humans; Kinetics; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Promyelocytic, Acute; Molecular Sequence Data; Neurotoxins; Phorbol 12,13-Dibutyrate; Protein Kinase C; Sequence Homology, Amino Acid; Structure-Activity Relationship; Swine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1993 |
Characterization of [3H]staurosporine binding in protein kinase C-II purified from rat brain.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenine Nucleotides; Alkaloids; Animals; Brain; Calcium; Carbazoles; Guanine Nucleotides; Indole Alkaloids; Isoquinolines; Phorbol 12,13-Dibutyrate; Phosphatidylserines; Piperazines; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate; Zinc | 1993 |
Ethanol and protein kinase C in rat brain.
Topics: Animals; Autoradiography; Brain; Ethanol; Hippocampus; Male; Nerve Tissue Proteins; Phorbol 12,13-Dibutyrate; Phosphatidylserines; Phosphorylation; Protein Kinase C; Rats; Rats, Wistar; Synaptosomes; Tetradecanoylphorbol Acetate | 1993 |
Inhibition of protein kinase C suppresses megakaryocytic differentiation and stimulates erythroid differentiation in HEL cells.
Topics: Aphidicolin; Biomarkers; Blood Proteins; Cell Cycle; Cell Differentiation; Enzyme Inhibitors; Erythroid Precursor Cells; Gene Expression Regulation, Leukemic; Globins; Glycophorins; Hematopoietic Stem Cells; Hemin; Humans; Indoles; Leukemia, Erythroblastic, Acute; Maleimides; Megakaryocytes; Neoplasm Proteins; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Processing, Post-Translational; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1996 |
LY290181, an inhibitor of diabetes-induced vascular dysfunction, blocks protein kinase C-stimulated transcriptional activation through inhibition of transcription factor binding to a phorbol response element.
Topics: Animals; Base Sequence; Capillaries; Cattle; Cells, Cultured; Chloramphenicol O-Acetyltransferase; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Endothelium, Vascular; Enzyme Inhibitors; Fibroblasts; Humans; Male; Molecular Sequence Data; Naphthalenes; Oligodeoxyribonucleotides; Phorbol 12,13-Dibutyrate; Promoter Regions, Genetic; Protein Kinase C; Pyrans; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Retinal Vessels; Skin; Tetradecanoylphorbol Acetate; Transcription Factors; Transcriptional Activation; Urokinase-Type Plasminogen Activator | 1996 |
The role of protein kinase C in carbachol-induced and of cAMP-dependent protein kinase in isoproterenol-induced secretion in primary cultured guinea pig parotid acinar cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; alpha-Amylases; Animals; Calcium; Carbachol; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Inhibitors; Exocytosis; Guinea Pigs; Immunoblotting; Isoproterenol; Isoquinolines; Male; Parotid Gland; Phorbol 12,13-Dibutyrate; Piperazines; Protein Binding; Protein Kinase C; Sulfonamides; Tetradecanoylphorbol Acetate | 1996 |
Tamoxifen modulates protein kinase C via oxidative stress in estrogen receptor-negative breast cancer cells.
Topics: Animals; Antioxidants; Breast Neoplasms; Cattle; Cell Division; Cell Membrane; Enzyme Inhibitors; Estrogen Antagonists; Female; Humans; In Vitro Techniques; Oxidative Stress; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rabbits; Receptors, Estrogen; Second Messenger Systems; Tamoxifen; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Vitamin E | 1996 |
Mechanism of bile salt-induced mucin secretion by cultured dog gallbladder epithelial cells.
Topics: Acetylglucosamine; Animals; Bile Acids and Salts; Calcimycin; Cells, Cultured; Cyclic AMP; Dinoprostone; Dogs; Edetic Acid; Enzyme Activation; Epithelium; Gallbladder; Ionomycin; Kinetics; Mucins; Phorbol 12,13-Dibutyrate; Protein Kinase C; Second Messenger Systems; Taurochenodeoxycholic Acid; Taurocholic Acid; Tetradecanoylphorbol Acetate; Tritium | 1996 |
The role of the 90-kDa heat shock protein in cell cycle control and differentiation of the monoblastoid cell line U937.
Topics: Antigens, CD; Cell Adhesion; Cell Adhesion Molecules; Cell Cycle; Cell Differentiation; Cell Division; Cell Line; DNA, Antisense; Gene Expression; Heat-Shock Proteins; Heat-Shock Response; HSP90 Heat-Shock Proteins; Humans; Mitogens; Monocytes; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate; Transfection | 1996 |
Separate upstream and convergent downstream pathways of G-protein- and phorbol ester-mediated Ca2+ sensitization of myosin light chain phosphorylation in smooth muscle.
Topics: Animals; Calcium; Carbachol; Cell Membrane; Cytosol; Femoral Artery; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Ileum; In Vitro Techniques; Isoenzymes; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Myosin Light Chains; Phorbol 12,13-Dibutyrate; Phosphorylation; Portal Vein; Protein Kinase C; Rabbits; Staphylococcus aureus; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1996 |
Phorbol esters but not the cholinergic agonists oxotremorine-M and carbachol increase release of the amyloid precursor protein in cultured rat cortical neurons.
Topics: Amyloid beta-Protein Precursor; Animals; Atropine; Carbachol; Cells, Cultured; Cerebral Cortex; Embryo, Mammalian; Muscarinic Agonists; Neurons; Oxotremorine; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Signal Transduction; Tetradecanoylphorbol Acetate | 1996 |
The structural requirements for phorbol esters to enhance noradrenaline and dopamine release from rat brain cortex.
Topics: Animals; Cerebral Cortex; Dopamine; In Vitro Techniques; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Tritium | 1996 |
Calcitonin-induced changes in the cytoskeleton are mediated by a signal pathway associated with protein kinase A in osteoclasts.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Animals; Animals, Newborn; Bucladesine; Calcitonin; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytoskeleton; Dentin; Enzyme Activation; Hematopoietic Stem Cells; Male; Mice; Mice, Inbred Strains; Osteoblasts; Phorbol 12,13-Dibutyrate; Protein Kinase C; Signal Transduction; Skull; Tetradecanoylphorbol Acetate; Thionucleotides | 1996 |
Phorbol-12,13-dibutyrate and pinacidil cardioplegia. Novel forms of myoprotection.
Topics: Animals; Diastole; Female; Guanidines; Heart; Heart Arrest, Induced; Hemodynamics; Male; Myocardial Contraction; Phorbol 12,13-Dibutyrate; Pinacidil; Potassium Channels; Protein Kinase C; Sheep; Tetradecanoylphorbol Acetate | 1996 |
Protein kinase C activation and phosphate uptake are altered in intact mucolipidosis type-4 skin fibroblasts.
Topics: Blotting, Western; Fibroblasts; Humans; Mucolipidoses; Phorbol 12,13-Dibutyrate; Phosphates; Protein Kinase C; Skin; Tetradecanoylphorbol Acetate | 1996 |
Involvement of mitogen-activated protein kinase and translocation of cytosolic phospholipase A2 to the nuclear envelope in acetylcholine-induced prostacyclin synthesis in rabbit coronary endothelial cells.
Topics: 6-Ketoprostaglandin F1 alpha; Acetylcholine; Amino Acid Sequence; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Membrane; Cells, Cultured; Coronary Vessels; Cytosol; Endothelium, Vascular; Enzyme Activation; Epoprostenol; Molecular Sequence Data; Naphthalenes; Nitriles; Nitrophenols; Nuclear Envelope; Okadaic Acid; Phorbol 12,13-Dibutyrate; Phospholipases A; Phospholipases A2; Phosphorylation; Rabbits; Tetradecanoylphorbol Acetate; Tyrphostins | 1996 |
Protein kinase C modulates flow-initiated contraction.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Male; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rabbits; Regional Blood Flow; Staurosporine; Tetradecanoylphorbol Acetate; Vasoconstriction | 1996 |
Activation of protein kinase C-alpha and translocation of the myristoylated alanine-rich C-kinase substrate correlate with phorbol ester-enhanced noradrenaline release from SH-SY5Y human neuroblastoma cells.
Topics: Alanine; Enzyme Activation; Humans; Intracellular Signaling Peptides and Proteins; Isoenzymes; Membrane Proteins; Myristoylated Alanine-Rich C Kinase Substrate; Neuroblastoma; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Phosphotransferases; Protein Kinase C; Proteins; Subcellular Fractions; Substrate Specificity; Tetradecanoylphorbol Acetate; Tissue Distribution; Translocation, Genetic; Tumor Cells, Cultured | 1997 |
The catalytic domain of protein kinase C-delta in reciprocal delta and epsilon chimeras mediates phorbol ester-induced macrophage differentiation of mouse promyelocytes.
Topics: Animals; Antigens, Differentiation; Cell Adhesion; Cell Differentiation; Cell Line; Hematopoiesis; Isoenzymes; Macrophage Activation; Macrophage-1 Antigen; Macrophages; Mice; Phagocytosis; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate | 1997 |
Metabotropic glutamate receptor activation modulates kainate and serotonin calcium response in astrocytes.
Topics: Amino Acids, Dicarboxylic; Aminobutyrates; Animals; Astrocytes; Biological Transport; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Cerebral Cortex; Cycloleucine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Glutamic Acid; Kainic Acid; Nimodipine; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Protein Kinase C; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Receptors, Metabotropic Glutamate; Second Messenger Systems; Serotonin; Suprachiasmatic Nucleus; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1997 |
Antiproliferative effect of Pygeum africanum extract on rat prostatic fibroblasts.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carcinogens; Cell Division; DNA; Dose-Response Relationship, Drug; Epidermal Growth Factor; Fatty Alcohols; Fibroblast Growth Factor 10; Fibroblast Growth Factor 2; Fibroblast Growth Factor 7; Fibroblast Growth Factors; Fibroblasts; Growth Substances; Insulin-Like Growth Factor I; Male; Phorbol 12,13-Dibutyrate; Plant Extracts; Prostate; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1997 |
Blockade of protein kinase C is involved in the inhibition by cycloheterophyllin of neutrophil superoxide anion generation.
Topics: Animals; Arachidonic Acid; Carcinogens; Cyclic AMP-Dependent Protein Kinases; Cytosol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Inositol 1,4,5-Trisphosphate; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Neutrophil Activation; Neutrophils; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate | 1997 |
Turning of nerve growth cones induced by the activation of protein kinase C.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Calcium Channels; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Isoenzymes; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Purinergic Antagonists; Spinal Cord; Tetradecanoylphorbol Acetate; Xenopus | 1997 |
Bryostatin 1 induces biphasic activation of protein kinase D in intact cells.
Topics: 3T3 Cells; Animals; Bryostatins; Dose-Response Relationship, Drug; Enzyme Activation; Kinetics; Lactones; Macrolides; Mice; Mitogens; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Tetradecanoylphorbol Acetate | 1997 |
Effects of phorbol ester on carbachol-induced contraction in bovine ciliary muscle: possible involvement of protein kinase C.
Topics: Animals; Carbachol; Cattle; Ciliary Body; Drug Interactions; Histones; In Vitro Techniques; Muscarinic Agonists; Muscle Contraction; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Receptors, Muscarinic; Stimulation, Chemical; Tetradecanoylphorbol Acetate | 1997 |
Inhibition by protein kinase C of the 86Rb+ efflux and vasorelaxation induced by P1075, a K(ATP) channel opener, in rat isolated aorta.
Topics: Adenosine Triphosphate; Animals; Aorta; Enzyme Activation; Enzyme Inhibitors; Guanidines; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Potassium Channels; Protein Binding; Protein Kinase C; Pyridines; Rats; Rats, Sprague-Dawley; Rubidium Radioisotopes; Tetradecanoylphorbol Acetate | 1997 |
Potentiation of ara-C-induced apoptosis by the protein kinase C activator bryostatin 1 in human leukemia cells (HL-60) involves a process dependent upon c-Myc.
Topics: Antineoplastic Agents; Apoptosis; Bryostatins; Cell Cycle; Cytarabine; Diterpenes; DNA Fragmentation; Drug Synergism; Enzyme Activation; HL-60 Cells; Humans; Kinetics; Lactones; Macrolides; Oligonucleotides, Antisense; Phorbol 12,13-Dibutyrate; Protein Kinase C; Proto-Oncogene Proteins c-myc; Terpenes; Tetradecanoylphorbol Acetate; Thionucleotides | 1997 |
Evidence for the involvement of protein kinase C inhibition by norathyriol in the reduction of phorbol ester-induced neutrophil superoxide anion generation and aggregation.
Topics: Animals; Cell Aggregation; Cyclic AMP-Dependent Protein Kinases; Neutrophils; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Respiratory Burst; Superoxides; Tetradecanoylphorbol Acetate; Trypsin; Xanthenes | 1997 |
Selenocompounds induce a redox modulation of protein kinase C in the cell, compartmentally independent from cytosolic glutathione: its role in inhibition of tumor promotion.
Topics: Animals; Anticarcinogenic Agents; Carcinogens; Cell Line; Cell Transformation, Neoplastic; Chromatography, DEAE-Cellulose; Cystine; Cytosol; Glutathione; Glutathione Disulfide; Isoenzymes; Kinetics; Mice; Organoselenium Compounds; Oxidation-Reduction; Phorbol 12,13-Dibutyrate; Protein Kinase C; Sodium Selenite; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1997 |
Acetylcholine agonists stimulate mitogen-activated protein kinase in oligodendrocyte progenitors by muscarinic receptors.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Animals, Newborn; Atropine; Brain; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cells, Cultured; Cholinergic Agents; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Indoles; Maleimides; Mitogen-Activated Protein Kinase 1; Oligodendroglia; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Signal Transduction; Stem Cells; Tetradecanoylphorbol Acetate | 1997 |
Protein kinase C inhibition enhances platelet-activating factor-induced eicosanoid production in human eosinophils.
Topics: Arachidonic Acid; Calcium; Catalase; Eicosanoids; Enzyme Inhibitors; Eosinophils; Female; Humans; Indoles; Leukotriene C4; Male; Maleimides; Naphthalenes; Phorbol 12,13-Dibutyrate; Platelet Activating Factor; Protein Kinase C; Respiratory Burst; Superoxides; Tetradecanoylphorbol Acetate; Thromboxane B2 | 1998 |
Regulation of aquaporin-4 water channels by phorbol ester-dependent protein phosphorylation.
Topics: Animals; Aquaporin 4; Aquaporins; Biological Transport; Enzyme Activation; Ion Channels; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Protein Kinase C; Rats; Recombinant Proteins; Tetradecanoylphorbol Acetate; Water | 1998 |
Inhibition of cromolyn-induced phosphorylation of a 78-kDa protein by phorbol esters in rat peritoneal mast cells.
Topics: Animals; Cells, Cultured; Cromolyn Sodium; Histamine Release; Immunoglobulin E; Male; Mast Cells; Peritoneal Cavity; Phorbol 12,13-Dibutyrate; Phosphorylation; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1998 |
Dietary lipid varying in corn and coconut oil influences protein kinase C in phorbol ester-treated mouse skin.
Topics: Animals; Biological Transport; Cell Membrane; Coconut Oil; Corn Oil; Dietary Fats; Female; Isoenzymes; Mice; Phorbol 12,13-Dibutyrate; Plant Oils; Protein Kinase C; Signal Transduction; Skin; Skin Neoplasms; Tetradecanoylphorbol Acetate | 1998 |
Different effects of phorbol ester derivates on human immunodeficiency virus 1 replication in lymphocytic and monocytic human cells.
Topics: HIV-1; Humans; Jurkat Cells; Lymphocytes; Monocytes; Phorbol 12,13-Dibutyrate; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Virus Replication | 1997 |
Endogenous activation of apoptosis in bursal lymphocytes: inhibition by phorbol esters and protein synthesis inhibitors.
Topics: Animals; Apoptosis; B-Lymphocytes; Bursa of Fabricius; Cell Differentiation; Cells, Cultured; Chickens; DNA Fragmentation; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Protein Synthesis Inhibitors; Signal Transduction; Tetradecanoylphorbol Acetate | 1998 |
Taurine might be acting as a trophic factor in the retina by modulating phosphorylation of cellular proteins.
Topics: Animals; Antineoplastic Agents, Hormonal; Benzylamines; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carcinogens; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Eye Proteins; Goldfish; Growth Substances; Indoles; Lactams; Marine Toxins; Okadaic Acid; Optic Nerve; Oxazoles; Phorbol 12,13-Dibutyrate; Phosphoric Monoester Hydrolases; Phosphorylation; Protein Kinase C; Retina; Sulfonamides; Tamoxifen; Taurine; Tetradecanoylphorbol Acetate | 1998 |
Assessment of the mechanism by which prolactin stimulates progesterone production by early corpora lutea of pigs.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Carcinogens; Cells, Cultured; Corpus Luteum; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Female; Ionomycin; Ionophores; Lipoproteins, LDL; Luteal Phase; Phorbol 12,13-Dibutyrate; Progesterone; Prolactin; Protein Kinase C; Staurosporine; Stimulation, Chemical; Swine; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1998 |
Mucin secretion by the human colon cell line LS174T is regulated by bile salts.
Topics: Adenocarcinoma; Animals; Bile Acids and Salts; Colon; Colonic Neoplasms; Dogs; Enzyme Activation; Epithelium; Humans; Mucins; Phorbol 12,13-Dibutyrate; Protein Kinase C; Solutions; Structure-Activity Relationship; Taurochenodeoxycholic Acid; Tetradecanoylphorbol Acetate; Tritium; Tumor Cells, Cultured | 1999 |
Thrombopoietin potentiates the protein-kinase-C-mediated activation of mitogen-activated protein kinase/ERK kinases and extracellular signal-regulated kinases in human platelets.
Topics: Adult; Blood Platelets; Calcium-Calmodulin-Dependent Protein Kinases; Cytoskeleton; Detergents; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Humans; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phorbol 12,13-Dibutyrate; Platelet Aggregation; Protein Kinase C; Proto-Oncogene Proteins c-raf; Solubility; Tetradecanoylphorbol Acetate; Thrombin; Thrombopoietin; Time Factors | 1998 |
Biphasic effect of protein kinase C on rat renal cortical Na+, K+-ATPase.
Topics: Amiloride; Amphotericin B; Animals; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Ibuprofen; Kidney Cortex; Male; Oxazines; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate | 1998 |
Adhesion of human monocytic THP-1 cells to endothelial cell adhesion molecules or extracellular matrix proteins via beta1 integrins regulates heparin binding epidermal growth factor-like growth factor (HB-EGF) expression.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cell Adhesion; Cell Adhesion Molecules; Cell Line; Colforsin; COS Cells; E-Selectin; Endothelium, Vascular; Epidermal Growth Factor; Extracellular Matrix Proteins; Gene Expression Regulation; Heparin; Heparin-binding EGF-like Growth Factor; Humans; Integrin beta1; Intercellular Adhesion Molecule-1; Intercellular Signaling Peptides and Proteins; Monocytes; Phorbol 12,13-Dibutyrate; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection; Vascular Cell Adhesion Molecule-1 | 1999 |
Redox modulation of intracellular free calcium concentration in thyroid FRTL-5 cells: evidence for an enhanced extrusion of calcium.
Topics: Animals; Barium; Calcium; Calcium-Transporting ATPases; Cell Line; Enzyme Activation; Hydrogen-Ion Concentration; Imidazoles; Membrane Potentials; Mercaptoethanol; Oxidation-Reduction; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Binding; Protein Kinase C; Rats; Staurosporine; tert-Butylhydroperoxide; Tetradecanoylphorbol Acetate; Thapsigargin; Thimerosal; Thyroid Gland; Vanadates | 1999 |
Regulation of L-type Ca2+ channels in rabbit portal vein by G protein alphas and betagamma subunits.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium Channels; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; GTP-Binding Proteins; In Vitro Techniques; Indoles; Male; Maleimides; Models, Biological; Muscle, Smooth, Vascular; Naphthalenes; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Portal Vein; Protein Conformation; Protein Kinase C; Pyrroles; Rabbits; Signal Transduction; Tetradecanoylphorbol Acetate; Thionucleotides | 1999 |
Regulation of calcium-dependent [3H]noradrenaline release from rat cerebrocortical synaptosomes by protein kinase C and modulation of the actin cytoskeleton.
Topics: Actins; Animals; Calcium; Cerebral Cortex; Cytoskeleton; Deoxyribonuclease I; Enzyme Inhibitors; Female; Male; Norepinephrine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar; Synaptosomes; Tetradecanoylphorbol Acetate; Tritium | 1999 |
Protein kinase C-alpha produces reciprocal effects on the phorbol ester stimulated tyrosine phosphorylation of a 50 kDa kinase in Jurkat cells.
Topics: Adenosine; Affinity Labels; Cell Extracts; Enzyme Activation; Enzyme Inhibitors; Humans; Isoenzymes; Jurkat Cells; Kinetics; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Protein Kinase C-alpha; Substrate Specificity; Tetradecanoylphorbol Acetate; Tyrosine | 1999 |
Phorbol ester modulation of active ion transport across the rabbit conjunctival epithelium.
Topics: Animals; Biological Transport, Active; Bumetanide; Chlorine; Conjunctiva; Culture Techniques; Enzyme Inhibitors; Female; Ion Transport; Male; Ouabain; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rabbits; Staurosporine; Tetradecanoylphorbol Acetate | 1999 |
Inositol hexaphosphate reduces 12-O-tetradecanoylphorbol-13-acetate-induced ornithine decarboxylase independent of protein kinase C isoform expression in keratinocytes.
Topics: Animals; Blotting, Western; Cell Division; Cell Line; Dose-Response Relationship, Drug; Enzyme Induction; Epidermis; Female; Humans; Isoenzymes; Keratinocytes; Mice; Mice, Inbred SENCAR; Ornithine Decarboxylase; Ornithine Decarboxylase Inhibitors; Phorbol 12,13-Dibutyrate; Phytic Acid; Protein Kinase C; Proto-Oncogene Proteins c-myc; RNA, Messenger; Tetradecanoylphorbol Acetate | 1999 |
Requirement for protein kinase C in reactive oxygen species-induced apoptosis of vascular smooth muscle cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apoptosis; Cells, Cultured; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Flow Cytometry; Hydrogen Peroxide; Immunohistochemistry; In Situ Nick-End Labeling; Muscle, Smooth, Vascular; Naphthalenes; Necrosis; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Reactive Oxygen Species; Staurosporine; Tetradecanoylphorbol Acetate | 1999 |
Protein kinase C-delta is a target of B-cell antigen receptor signaling.
Topics: Animals; B-Lymphocytes; Biological Transport; Enzyme Activation; Estrenes; Humans; Ionomycin; Isoenzymes; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Phorbol 12,13-Dibutyrate; Phosphatidylinositol Diacylglycerol-Lyase; Phosphorylation; Protein Kinase C; Protein Kinase C-delta; Protein Processing, Post-Translational; Pyrrolidinones; Receptors, Antigen, B-Cell; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Type C Phospholipases | 1999 |
The involvement of protein kinase C in the regulation of choline cotransport in Limulus.
Topics: Animals; Arachidonic Acids; Biological Transport; Brain; Carcinogens; Carrier Proteins; Choline; Cholinergic Agents; Enzyme Inhibitors; Hemicholinium 3; Horseshoe Crabs; Nervous System; Organ Culture Techniques; Phorbol 12,13-Dibutyrate; Phospholipases A; Phospholipases A2; Potassium Chloride; Protein Kinase C; Quinacrine; Staurosporine; Tetradecanoylphorbol Acetate; Tritium | 1999 |
Protein kinase C and the opposite regulation of sodium channel alpha- and beta1-subunit mRNA levels in adrenal chromaffin cells.
Topics: Adrenal Medulla; Animals; Cattle; Cell Nucleus; Cells, Cultured; Chromaffin Cells; Cycloheximide; Down-Regulation; Enzyme Activation; Gene Expression Regulation; Kinetics; Macromolecular Substances; Phorbol 12,13-Dibutyrate; Protein Kinase C; RNA, Messenger; Sodium Channels; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1999 |
Structural determinants of phorbol ester binding in synaptosomes: pharmacokinetics and pharmacodynamics.
Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Kinetics; Male; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Binding; Protein Kinase C; Rats; Rats, Sprague-Dawley; Synaptic Membranes; Synaptosomes; Tetradecanoylphorbol Acetate; Time Factors; Tritium | 1999 |
TPA-enhanced motility and invasion in a highly metastatic variant (L-10) of human rectal adenocarcinoma cell line RCM-1: selective role of PKC-alpha and its inhibition by a combination of PDBu-induced PKC downregulation and antisense oligonucleotides trea
Topics: Adenocarcinoma; Base Sequence; Carbazoles; Down-Regulation; Humans; Indoles; Isoenzymes; Naphthalenes; Neoplasm Invasiveness; Neoplasm Metastasis; Oligonucleotides, Antisense; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Protein Kinase C-alpha; Rectal Neoplasms; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1999 |
The lipophilicity of phorbol esters as a critical factor in determining the pattern of translocation of protein kinase C delta fused to green fluorescent protein.
Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Green Fluorescent Proteins; Isoenzymes; Lipid Metabolism; Luminescent Proteins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Protein Kinase C-delta; Recombinant Fusion Proteins; Spectrometry, Fluorescence; Tetradecanoylphorbol Acetate | 2000 |
Phosphorylation regulates spontaneous and evoked transmitter release at a giant terminal in the rat auditory brainstem.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 2-Amino-5-phosphonovalerate; Animals; Cochlear Nucleus; Enzyme Inhibitors; Evoked Potentials; Excitatory Postsynaptic Potentials; In Vitro Techniques; Indoles; Maleimides; Phorbol 12,13-Dibutyrate; Phosphorylation; Presynaptic Terminals; Protein Kinase C; Rats; Rats, Wistar; Synaptic Transmission; Tetradecanoylphorbol Acetate | 2000 |
Phorbol ester-regulated cleavage of normal prion protein in HEK293 human cells and murine neurons.
Topics: Amino Acid Sequence; Animals; Blotting, Western; Bucladesine; Carcinogens; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Humans; Kinetics; Methanol; Mice; Molecular Sequence Data; Neurons; Phorbol 12,13-Dibutyrate; Phorbol Esters; Precipitin Tests; Prions; Protein Isoforms; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors; Transfection; Up-Regulation | 2000 |
Properties of the inward-rectifying Cl- channel in rat choroid plexus: regulation by intracellular messengers and inhibition by divalent cations.
Topics: Adenosine Triphosphate; Animals; Cadmium; Cations, Divalent; Chloride Channels; Choroid Plexus; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Electric Conductivity; Electrodes; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Naphthalenes; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Sprague-Dawley; Solutions; Tetradecanoylphorbol Acetate; Zinc | 2000 |
Regulation of conjunctival goblet cell secretion by Ca(2+)and protein kinase C.
Topics: Animals; Blotting, Western; Calcium; Chelating Agents; Conjunctiva; Glycoproteins; Goblet Cells; Ionomycin; Ionophores; Male; Microscopy, Fluorescence; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 2000 |
Parathyroid hormone-related protein down-regulates bone sialoprotein gene expression in cementoblasts: role of the protein kinase A pathway.
Topics: 1-Methyl-3-isobutylxanthine; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Dactinomycin; Dental Cementum; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Integrin-Binding Sialoprotein; Kinetics; Parathyroid Hormone-Related Protein; Phorbol 12,13-Dibutyrate; Proteins; RNA, Messenger; Second Messenger Systems; Sialoglycoproteins; Tetradecanoylphorbol Acetate; Thionucleotides | 2000 |
Activation of dopamine D(1)-like receptor causes phosphorylation of alpha(1)-subunit of Na(+),K(+)-ATPase in rat renal proximal tubules.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cell Line; Dopamine Agonists; Enzyme Inhibitors; In Vitro Techniques; Kidney Tubules, Proximal; Male; Mutation; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Sodium-Potassium-Exchanging ATPase; Staurosporine; Tetradecanoylphorbol Acetate | 2001 |
Regulation of adenohypophyseal pyroglutamyl aminopeptidase II activity by thyrotropin-releasing hormone and phorbol esters.
Topics: Aminopeptidases; Animals; Cells, Cultured; Cyclic AMP; Female; Homeostasis; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland, Anterior; Protein Kinase C; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Sex Characteristics; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Triiodothyronine | 2000 |
Constitutive alpha-secretase cleavage of the beta-amyloid precursor protein in the furin-deficient LoVo cell line: involvement of the pro-hormone convertase 7 and the disintegrin metalloprotease ADAM10.
Topics: Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Aspartic Acid Endopeptidases; Cell Line; Endopeptidases; Furin; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Proprotein Convertases; Protein Kinase C; Recombinant Proteins; Subtilisins; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 2001 |
G-protein-coupled receptor stimulation of the p42/p44 mitogen-activated protein kinase pathway is attenuated by lipid phosphate phosphatases 1, 1a, and 2 in human embryonic kidney 293 cells.
Topics: Cell Line; Cell Membrane; GTP-Binding Proteins; Humans; Isoenzymes; Kidney; Kinetics; Lysophospholipids; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phorbol 12,13-Dibutyrate; Phosphatidate Phosphatase; Phosphatidic Acids; Phospholipase D; Receptors, Cell Surface; Recombinant Proteins; Sphingosine; Substrate Specificity; Tetradecanoylphorbol Acetate; Transfection; Virulence Factors, Bordetella | 2001 |
Phorbol esters promote postsynaptic accumulation of Vesl-1S/Homer-1a protein.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alternative Splicing; Animals; Anisomycin; Carcinogens; Carrier Proteins; Cells, Cultured; Excitatory Amino Acid Antagonists; Hippocampus; Homer Scaffolding Proteins; Microscopy, Immunoelectron; Neurons; Neuropeptides; Phorbol 12,13-Dibutyrate; Potassium; Protein Synthesis Inhibitors; Rats; Rats, Wistar; Synaptic Membranes; Tetradecanoylphorbol Acetate; Tetrodotoxin | 2001 |
Deterioration of the protein kinase C-K(ATP) channel pathway in regulation of coronary flow in hypercholesterolaemic rabbits.
Topics: Adenosine Triphosphate; Animals; Coronary Circulation; Enzyme Inhibitors; Heart Ventricles; Hypercholesterolemia; In Vitro Techniques; Male; Phorbol 12,13-Dibutyrate; Potassium Channels; Protein Kinase C; Rabbits; Staurosporine; Tetradecanoylphorbol Acetate | 2001 |
Diacylglycerol (DAG)-lactones, a new class of protein kinase C (PKC) agonists, induce apoptosis in LNCaP prostate cancer cells by selective activation of PKCalpha.
Topics: Apoptosis; Diglycerides; Enzyme Inhibitors; Humans; Isoenzymes; Lactones; Male; Phorbol 12,13-Dibutyrate; Prostatic Neoplasms; Protein Kinase C; Proto-Oncogene Proteins c-bcl-2; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2002 |
Activity of protein kinase C modulates the apoptosis induced by polychlorinated biphenyls in human leukemic HL-60 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Apoptosis; Chlorodiphenyl (54% Chlorine); Diglycerides; DNA Fragmentation; Electrophoresis, Agar Gel; Enzyme Inhibitors; HL-60 Cells; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate | 2002 |
Modulation of the human protein kinase C alpha gene promoter by activator protein-2.
Topics: 5' Untranslated Regions; Base Sequence; Cloning, Molecular; DNA-Binding Proteins; Enzyme Activation; Gene Expression Regulation, Neoplastic; Glioblastoma; Humans; Isoenzymes; Molecular Sequence Data; Phorbol 12,13-Dibutyrate; Promoter Regions, Genetic; Protein Kinase C; Protein Kinase C-alpha; Second Messenger Systems; Sp1 Transcription Factor; Tetradecanoylphorbol Acetate; Transcription Factor AP-2; Transcription Factors; Transcription Initiation Site; Transfection; Tumor Cells, Cultured | 2002 |
Prolactin signaling in porcine adrenocortical cells: involvement of protein kinases.
Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Androstenedione; Animals; Diglycerides; Enzyme Activators; Enzyme Inhibitors; Female; Genistein; Hydrocortisone; Ionomycin; Phorbol 12,13-Dibutyrate; Prolactin; Protein Kinase C; Protein-Tyrosine Kinases; Signal Transduction; Sphingosine; Swine; Tetradecanoylphorbol Acetate | 2002 |
Protein kinase C-mediated Ca2+ entry in HEK 293 cells transiently expressing human TRPV4.
Topics: Calcium; Cation Transport Proteins; Cell Line; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Gene Expression; Humans; Hypotonic Solutions; Indoles; Ion Channels; Maleimides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; TRPV Cation Channels | 2003 |
Mechanisms of arginine-vasopressin-induced Ca2+ oscillations in beta-cells (HIT-T15): a role for oscillating protein kinase C.
Topics: Animals; Arginine Vasopressin; Biological Transport; Calcium; Calcium Channels; Cell Line; Enzyme Activation; Enzyme Inhibitors; Inositol 1,4,5-Trisphosphate; Islets of Langerhans; Isoenzymes; Oscillometry; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 2004 |
Activation of arylalkylamine N-acetyltransferase by phorbol esters in bovine pinealocytes suggests a novel regulatory pathway in melatonin synthesis.
Topics: Animals; Arylalkylamine N-Acetyltransferase; Calcium Signaling; Cattle; Cyclic AMP; Enzyme Activation; Female; Male; Melatonin; Organ Culture Techniques; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pineal Gland; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate | 2004 |
Bidirectional regulation of renal cortical Na+,K+-ATPase by protein kinase C.
Topics: Amiloride; Animals; Arachidonic Acids; Brefeldin A; Cytochrome P-450 Enzyme System; Endocytosis; Enzyme Activation; Enzyme Inhibitors; Kidney Cortex; Kinetics; Male; Models, Biological; Nocodazole; Okadaic Acid; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositol 3-Kinases; Protein Kinase C; Rats; Rats, Wistar; Sodium; Sodium-Potassium-Exchanging ATPase; Staurosporine; Tetradecanoylphorbol Acetate | 2004 |
Role of phorbol ester localization in determining protein kinase C or RasGRP3 translocation: real-time analysis using fluorescent ligands and proteins.
Topics: Animals; Biological Transport; CHO Cells; Cricetinae; Fluorescent Dyes; Guanine Nucleotide Exchange Factors; Humans; Kinetics; Ligands; Microscopy, Confocal; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Transport; ras Guanine Nucleotide Exchange Factors; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate | 2005 |
Individual C1 domains of PKD3 in phorbol ester-induced plasma membrane translocation of PKD3 in intact cells.
Topics: Animals; Catalysis; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Enzyme Activation; Enzyme Inhibitors; Mutation; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Structure, Tertiary; Protein Transport; Radioligand Assay; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate | 2005 |
Enhancement of cisplatin sensitivity of cisplatin-resistant human cervical carcinoma cells by bryostatin 1.
Topics: Antineoplastic Agents; Apoptosis; Blotting, Western; Bryostatins; Caspase 3; Caspases; Cell Survival; Cisplatin; Dose-Response Relationship, Drug; Down-Regulation; Drug Resistance, Neoplasm; Drug Synergism; Enzyme Activation; Female; HeLa Cells; Humans; Indoles; Lactams; Macrolides; Phorbol 12,13-Dibutyrate; Poly(ADP-ribose) Polymerases; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; RNA Interference; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Transfection; Uterine Cervical Neoplasms | 2005 |
Functional characterization of a human organic anion transporter hOAT4 in placental BeWo cells.
Topics: Cell Line; Dehydroepiandrosterone Sulfate; Enzyme Activation; Estradiol; Estrone; Humans; Kinetics; Organic Anion Transporters, Sodium-Independent; Phorbol 12,13-Dibutyrate; Placenta; Protein Kinase C; Tetradecanoylphorbol Acetate; Transfection | 2006 |
Directional sensing of a phorbol ester gradient requires CD44 and is regulated by CD44 phosphorylation.
Topics: Amino Acid Sequence; Cell Line, Tumor; Chemotaxis; Cyclic AMP-Dependent Protein Kinases; Humans; Hyaluronan Receptors; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Serine; Signal Transduction; Tetradecanoylphorbol Acetate | 2006 |
Cytotoxic action of phorbol esters on human pancreatic cancer cells.
Topics: Animals; Apoptosis; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Indoles; Inhibitory Concentration 50; Intracellular Signaling Peptides and Proteins; Maleimides; Membrane Proteins; Mice; Myristoylated Alanine-Rich C Kinase Substrate; Pancreatic Neoplasms; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Xenograft Model Antitumor Assays | 2007 |
Differential roles of PKCalpha and PKCepsilon in controlling the gene expression of Nox4 in human endothelial cells.
Topics: Cells, Cultured; Down-Regulation; Endothelial Cells; Gene Expression Regulation; Humans; NADPH Oxidase 4; NADPH Oxidases; Phorbol 12,13-Dibutyrate; Protein Kinase C-alpha; Protein Kinase C-epsilon; RNA, Small Interfering; Superoxides; Tetradecanoylphorbol Acetate; Umbilical Veins; Up-Regulation | 2008 |
Two PKC consensus sites on human acid-sensing ion channel 1b differentially regulate its function.
Topics: Acid Sensing Ion Channels; Amino Acid Sequence; Animals; Benzophenanthridines; Consensus Sequence; Enzyme Activation; Enzyme Activators; Humans; Ion Channel Gating; Kinetics; Membrane Potentials; Molecular Sequence Data; Mutation; Nerve Tissue Proteins; Oocytes; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Conformation; Protein Kinase C; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Sodium Channels; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Xenopus laevis | 2009 |
Does PKC activation increase the homologous desensitization of μ opioid receptors?
Topics: Analgesics, Opioid; Animals; Brain; Enkephalin, Methionine; HEK293 Cells; Humans; Male; Mice, Transgenic; Morphine; Muscarine; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Transport; Rats, Sprague-Dawley; Receptors, Opioid, mu; Tetradecanoylphorbol Acetate | 2015 |
Vasorelaxing Effect of Resveratrol on Bovine Retinal Arteries.
Topics: Animals; Antioxidants; Cattle; Dose-Response Relationship, Drug; Endothelium, Vascular; Isometric Contraction; Muscle, Smooth, Vascular; Myography; Nitric Oxide; Phorbol 12,13-Dibutyrate; Potassium Channels; Protein Kinase C; Resveratrol; Retinal Artery; Stilbenes; Tetradecanoylphorbol Acetate; Vasodilation; Vasodilator Agents | 2016 |