phorbol 12,13-dibutyrate has been researched along with phorbols in 149 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 134 (89.93) | 18.7374 |
1990's | 14 (9.40) | 18.2507 |
2000's | 1 (0.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Byrne, JH; Critz, SD | 1 |
Raufman, JP | 1 |
Arienti, D; Bendinelli, P; Bernelli-Zazzera, A; Piccoletti, R | 1 |
Gross, JL; Horuk, R | 1 |
Sacktor, TC; Schwartz, JH | 1 |
Alterman, RL; Kornblith, PL; Maleci, A; Moskal, JR; Sundstrom, D | 1 |
Brown, BL; Dobson, PR; Quilliam, LA | 1 |
Bauer, KD; Dunn, MM; Kamp, DW; Knap, A | 1 |
Hirata, Y | 1 |
Chuang, DM; Dillon-Carter, O | 1 |
Zatz, M | 1 |
Bauer, KD; Dunn, MM; Kamp, DW; Rubin, DB | 1 |
de Graan, PN; Eichberg, J; Gispen, WH; Schrama, LH | 1 |
Drummond, AH; MacIntyre, DE; McNicol, A | 1 |
Besterman, JM; Cragoe, EJ; Cuatrecasas, P; LeVine, H; May, WS | 1 |
Iwashima, A; Kitagawa, K; Nishino, H | 1 |
Bell, RM; Czech, MP; Davis, RJ; Ganong, BR | 1 |
Lapetina, EG; Watson, SP | 1 |
Civan, MM; Mauro, T; O'Brien, TG; Rubenstein, D | 1 |
Benveniste, R; Ilekis, J | 1 |
Patel, J; Rebois, RV | 1 |
Lapetina, EG; Negro-Vilar, A | 1 |
Madshus, IH; Olsnes, S; Sandvig, K | 1 |
Strnad, CF; Wong, K | 1 |
Gainer, HS; Murray, AW | 1 |
el-Fakahany, EE; Lai, WS | 2 |
Cavender, D; Haskard, D; Ziff, M | 1 |
Bell, RM; Ebeling, JG; Ganong, BR; Kuhn, LJ; Niedel, JE; Vandenbark, GR | 1 |
Blumberg, PM; Leach, KL | 1 |
Häring, HU; Kirsch, D; Obermaier, B | 1 |
Brown, EJ; Frank, MM; Gaither, TA; O'Shea, JJ; Takahashi, T | 1 |
Rodriguez-Pena, A; Rozengurt, E | 2 |
Anderson, D; Dewdney, RS; Soper, CJ | 1 |
de Laat, SW; Mummery, CL; Snoek, GT; van den Brink, CE; van der Saag, PT | 1 |
Bayard, F; Darbon, JM; Valette, A | 1 |
Murphy, RL; Smith, ME | 1 |
Chobanian, MC; Hammerman, MR | 1 |
Blumberg, PM; Sharkey, NA | 2 |
Fearon, CW; Tashjian, AH; Wolfson, G | 1 |
Baylin, SB; Berger, CL; de Bustros, A; Leong, SS; Nelkin, BD; Roos, BA | 1 |
Argov, S; Cuatrecasas, P; Hebdon, M; Koren, HS | 1 |
Aguelon-Pegouries, AM; Enomoto, T; Furstenberger, G; Marks, F; Martel, N; Yamasaki, H | 1 |
Gescher, A; Reed, DJ | 1 |
Bressler, JP; Kornblith, PL; Weingarten, D | 1 |
Chang, EB; Rao, MC; Wang, NS | 1 |
Arcoleo, JP; Brothman, AR; Liskamp, RM; Miller, OJ; Weinstein, IB | 1 |
Finlay, TH; Kadner, SS; Katz, J; Levitz, M | 1 |
Klein, E; Masucci, MG; Ramos, OF | 1 |
Chen, BD; Wilkins, KL | 1 |
Lefkowitz, RJ; Nambi, P; Sibley, DR | 1 |
Pettit, GR; Smith, JB; Smith, L | 1 |
Adams, DO; Hamilton, TA; Rigsbee, JE; Scott, WA | 1 |
Blumberg, PM; Jeng, AY; Lichti, U; Strickland, JE | 1 |
Enomoto, T; Kanno, Y; Martel, N; Yamasaki, H | 1 |
Arcoleo, J; Backer, J; Gattoni-Celli, S; Hsiao, WL; Jeffrey, A; Kirschmeier, P; Okin, E; Weinstein, IB | 1 |
Blumberg, PM; Chritton, S; Lew, KK | 1 |
Ono, T; Tanaka, K | 1 |
Enomoto, T; Kanno, Y; Martel, N; Shiba, Y; Yamasaki, H | 1 |
Carstensen, A; Klein, E; Masucci, MG; Pear, W; Torsteinsdottir, S | 1 |
Aub, DL; Leslie, BA; McKinney, JS; Putney, JW | 1 |
Blumberg, PM; Jaken, S; Jeng, AY; König, B; Leach, KL; Sharkey, NA | 1 |
Dicker, P; Rozengurt, E | 1 |
Salomon, DS | 1 |
Greenebaum, E; Horowitz, AD; Nicolaides, M; Weinstein, IB; Woodward, K | 1 |
Logani, MK; Slaga, TJ; Solanki, V | 1 |
Dulbecco, R; Okada, S; Sonnenberg, A | 1 |
Castagna, M; Horowitz, AD; Sala, M; Schachter, D; Tran, PL; Vassent, G; Weinstein, LB | 1 |
Jaken, S; Phillips, MA | 1 |
Fürstenberger, G; Marks, F; Sachs, L; Simantov, R | 1 |
Eisinger, M; Greenebaum, E; Nicolaides, M; Vogel, RH; Weinstein, IB | 1 |
Colburn, NH; Dalal, B; Gindhart, TD; Hegamyer, GA | 1 |
Blumberg, PM; Delclos, KB; Jaken, S | 1 |
Collins, M; McKay, I; Rozengurt, E; Taylor-Papadimitriou, J | 1 |
Chen, BD; Hsu, S; Lin, HS | 1 |
Ishii, DN; Spinelli, W | 1 |
Cabot, MC | 1 |
Blumberg, PM; James, ML; Leach, KL | 1 |
Blumberg, PM; Delclos, KB; Dunn, JA; Jaken, S; Leach, KL; Yeh, E | 1 |
Blumberg, PM; Dunn, JA | 1 |
Misukonis, MA; Weinberg, JB | 1 |
Eisen, HJ; Hankinson, O; Kärenlampi, SO; Nebert, DW | 1 |
Kikkawa, U; Miyake, R; Nishizuka, Y; Takai, Y; Tanaka, Y | 1 |
Blumberg, PM; Feldman, H; Jaken, S; Tashjian, AH | 1 |
Rodriguez-Pena, M; Rozengurt, E; Smith, KA | 1 |
Gearhart, JD; Gould, RJ; Murphy, KM; Oster-Granite, ML; Snyder, SH | 1 |
Goodwin, BJ; Misukonis, MA; Weinberg, JB | 1 |
Fox, CF; Iwashita, S | 1 |
Kuhn, LJ; Niedel, JE; Vandenbark, GR | 1 |
Blumberg, PM; Jaken, S; Jeng, AY; König, B; Leach, KL; Sharkey, NA; Yeh, E | 1 |
Pastan, I; Werth, DK | 1 |
Cuatrecasas, P; Jacobs, S; May, WS | 1 |
Besterman, JM; Cuatrecasas, P | 1 |
Estensen, RD; Mascioli, DW | 1 |
Block, A; Hromchak, R; Sakagami, H | 1 |
Isakson, PC; Simpson, L | 1 |
Biberfeld, P; Klein, E; Klein, G; Patarroyo, M | 1 |
Peterfreund, RA; Vale, WW | 1 |
Franson, RC; Kramer, CM; Rubin, RP | 1 |
O'Brien, T; Perussia, B; Shade, M; Trinchieri, G | 1 |
Jones, MJ; Murray, AW | 1 |
Cohen, LE; Koeffler, HP; Lehrer, RI | 1 |
Chida, K; Kuroki, T | 1 |
Anderson, NL; Callaham, MF; Gemmell, MA; Huberman, E; Murao, S | 1 |
Burczak, JD; Fairley, JL; Moskal, JR; Sweeley, CC; Trosko, JE | 1 |
Gordon, J; Jondal, M; Klein, E; Patarroyo, M | 1 |
Burns, CP; Rozengurt, E | 1 |
Elliott, MS; Katze, JR; Trewyn, RW | 1 |
Gahmberg, CG; Patarroyo, M | 1 |
Schorderet-Slatkine, S; Urner, F | 1 |
Janowsky, A; Labarca, R; Patel, J; Paul, SM | 1 |
Clarke, PR; Varani, J | 1 |
Honikman-Leban, E; Moulé, Y | 1 |
Dawson, G; Golomb, HM; Lockney, MW | 1 |
Blumberg, PM; Jaken, S; Shupnik, MA; Tashjian, AH | 1 |
Cassel, DL; Cooper, RA; Hoxie, JA | 1 |
Bejarano, MT; Klein, E; Masucci, MG; Ramos, OF | 1 |
Cooper, RA; Gerson, SL | 1 |
Blumberg, PM; Jaken, S; Tashjian, AH | 1 |
Collins, M; Rozengurt, E | 1 |
Hoffman, DR; Huberman, E | 1 |
Blumberg, PM; Castagna, M; Jaken, S; Nagle, DS | 1 |
Callaham, M; Huberman, E; Slaga, TJ; Solanki, V | 1 |
Slaga, TJ; Solanki, V | 1 |
Blumberg, PM; Castagna, M; Dunphy, WG; Kochenburger, RJ | 1 |
Cogan, U; Fisher, PB; Horowitz, AD; Schachter, D; Weinstein, IB | 1 |
Shoyab, M; Todaro, GJ; Warren, TC | 3 |
Blumberg, PM; Butler-Gralla, E; Herschman, HR | 1 |
Shoyab, M; Todaro, GJ | 1 |
Callaham, M; Huberman, E; Slaga, T; Solanki, V; Weeks, C | 1 |
Guy, GR; Murray, AW | 1 |
Goodwin, BJ; Weinberg, JB | 1 |
Drevon, C; Martel, N; Yamasaki, H | 1 |
Biberfeld, P; Klein, E; Klein, G; Patarroyo, M; Yogeeswaran, G | 1 |
Farrar, JJ; Hilfiker, ML; Salomon, DS; Sando, JJ | 1 |
Blumberg, PM; Delclos, KB; Dunphy, WG; Jaken, S | 1 |
Black, SC; Chi, L; Fagbemi, SO; Friedrichs, GS; Lucchesi, BR | 1 |
Ichikawa, K; Ito, M; Itoh, H; Konishi, T; Nakano, T; Okubo, S; Shimomura, A | 1 |
Ashby, CR; Edwards, E; Wang, RY | 1 |
Hirsh, JK; Redman, RS; Searl, TJ; Silinsky, EM | 1 |
Hirono, M; Suzuki, N; Takagi, H; Yoshioka, T | 1 |
Colbert, CM; Johnston, D | 1 |
Bhagavan, S; Etcheberrigaray, R; Ibarreta, D; Kozikowski, AP; Ma, D | 1 |
Conn, PJ; Macek, TA; Schaffhauser, H | 1 |
Cubillos, S; Guerra, A; Lima, L | 1 |
4 review(s) available for phorbol 12,13-dibutyrate and phorbols
Article | Year |
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Molecular mechanisms of tumor promotion and multistage carcinogenesis.
Topics: Adenosine Triphosphate; Animals; Base Sequence; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Transformation, Neoplastic; ErbB Receptors; Humans; Lyngbya Toxins; Molecular Conformation; Neoplasms; Oncogenes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1983 |
Phorbol ester receptors-insights into the initial events in the mechanism of action of the phorbol esters.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Membrane; Cytosol; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Protein Kinases; Receptors, Drug; Receptors, Immunologic; Solubility; Structure-Activity Relationship; Ultraviolet Rays | 1983 |
Phorbol ester receptors and the in vitro effects of tumor promoters.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Mice; Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin Neoplasms; Structure-Activity Relationship | 1983 |
Specific binding of phorbol ester tumor promoters to mouse tissues and cultured cells.
Topics: Animals; Biological Evolution; Brain; Caenorhabditis elegans Proteins; Calcium; Carcinogens; Carrier Proteins; Cell Membrane; Cells, Cultured; Humans; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Skin; Spleen; Structure-Activity Relationship; Temperature; Tetradecanoylphorbol Acetate; Thermodynamics | 1982 |
145 other study(ies) available for phorbol 12,13-dibutyrate and phorbols
Article | Year |
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Modulation of IK,Ca by phorbol ester-mediated activation of PKC in pleural sensory neurons of Aplysia.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Aplysia; Calcium; Dose-Response Relationship, Drug; Enzyme Activation; Ganglia; In Vitro Techniques; Isoquinolines; Kinetics; Membrane Potentials; Neurons, Afferent; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Piperazines; Potassium Channels; Protein Kinase C; Protein Kinase Inhibitors; Second Messenger Systems; Tetradecanoylphorbol Acetate; Tetraethylammonium; Tetraethylammonium Compounds | 1992 |
Actions of phorbol esters on levels of cAMP in cholera toxin-treated chief cells from guinea pig stomach.
Topics: Animals; Calcimycin; Calmodulin; Carbachol; Cholera Toxin; Gastric Mucosa; Guinea Pigs; Imidazoles; In Vitro Techniques; Kinetics; Male; Phorbol 12,13-Dibutyrate; Phorbols; Signal Transduction; Sincalide; Tetradecanoylphorbol Acetate | 1992 |
State and activity of protein kinase C in postischemic reperfused liver.
Topics: Animals; Cell Fractionation; Cell Membrane; Cytosol; Diglycerides; Immunoblotting; Lipids; Liver; Male; Phorbol 12,13-Dibutyrate; Phorbols; Phosphatidylcholines; Phosphatidylethanolamines; Phospholipids; Protein Kinase C; Rats; Rats, Inbred Strains; Reperfusion Injury; Tritium | 1992 |
Protein kinase C-linked inactivation of the interleukin-1 receptor in a human transformed B-cell line.
Topics: B-Lymphocytes; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Cell Membrane; Enzyme Activation; Humans; Interleukin-1; Kinetics; Lymphoma; Phorbol 12,13-Dibutyrate; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Receptors, Interleukin-1; Recombinant Proteins; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1990 |
Sensitizing stimuli cause translocation of protein kinase C in Aplysia sensory neurons.
Topics: Animals; Aplysia; Caenorhabditis elegans Proteins; Carrier Proteins; Cyclic AMP; Ganglia; Histones; In Vitro Techniques; Magnesium; Neurons, Afferent; Phorbol 12,13-Dibutyrate; Phorbols; Phosphorylation; Protein Kinase C; Receptors, Drug; Serotonin; Subcellular Fractions; Thionucleotides | 1990 |
Effect of phorbol esters on the susceptibility of a glioma cell line to lymphokine-activated killer cell activity.
Topics: Cell Division; Glioma; Humans; Killer Cells, Lymphokine-Activated; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Tetradecanoylphorbol Acetate; Thymidine; Tumor Cells, Cultured | 1990 |
Modulation of cyclic AMP accumulation in GH3 cells by a phorbol ester and thyroliberin.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Animals; Bacterial Toxins; Cell Line; Cholera Toxin; Cyclic AMP; GTP-Binding Proteins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pituitary Gland; Pituitary Neoplasms; Rats; Thyrotropin-Releasing Hormone; Time Factors; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1985 |
Contrasting effects of inflammatory stimuli on neutrophil and monocyte adherence to endothelial cells.
Topics: Animals; Cattle; Cells, Cultured; Diglycerides; Dose-Response Relationship, Drug; Endothelium, Vascular; Hydrogen Peroxide; Immune Adherence Reaction; Ionomycin; Monocytes; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbols; Protein Kinase C; Second Messenger Systems; Superoxides | 1989 |
Heterologous down-regulation of vascular atrial natriuretic peptide receptors by phorbol esters.
Topics: Animals; Dose-Response Relationship, Drug; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Atrial Natriuretic Factor; Receptors, Cell Surface; Temperature; Tetradecanoylphorbol Acetate; Time Factors | 1988 |
Characterization of bradykinin-induced phosphoinositide turnover in neurohybrid NCB-20 cells.
Topics: Animals; Bradykinin; Cell Line; Diphenhydramine; GTP-Binding Proteins; Kinetics; Lithium; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylinositols; Triprolidine; Type C Phospholipases | 1988 |
Phorbol esters mimic alpha-Adrenergic potentiation of serotonin N-acetyltransferase induction in the rat pineal.
Topics: Acetyltransferases; Adrenergic alpha-Agonists; Animals; Arylamine N-Acetyltransferase; Enzyme Induction; Isoproterenol; Male; Phenylephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pineal Gland; Rats; Rats, Inbred Strains | 1985 |
Tumor-promoting phorbol esters inhibit monocyte adherence to endothelial cells.
Topics: Animals; Aorta; Carcinogens; Cell Adhesion; Cells, Cultured; Endothelium, Vascular; Male; Monocytes; Phorbol 12,13-Dibutyrate; Phorbols; Tetradecanoylphorbol Acetate | 1989 |
Dioctanoylglycerol and phorbol diesters enhance phosphorylation of phosphoprotein B-50 in native synaptic plasma membranes.
Topics: Animals; Calcium; Diglycerides; Dose-Response Relationship, Drug; GAP-43 Protein; Glycerides; Histones; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphoproteins; Phosphorylation; Protein Kinase C; Rats; Synaptic Membranes | 1986 |
Tumour-promoting phorbol esters inhibit agonist-induced phosphatidate formation and Ca2+ flux in human platelets.
Topics: Blood Platelets; Calcium; Carcinogens; Enzyme Activation; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylinositols; Platelet Activating Factor; Protein Kinase C; Protein Kinases; Tetradecanoylphorbol Acetate; Thrombin; Vasopressins | 1985 |
Amiloride inhibits phorbol ester-stimulated Na+/H+ exchange and protein kinase C. An amiloride analog selectively inhibits Na+/H+ exchange.
Topics: Amiloride; Carrier Proteins; Cell Adhesion; Cell Differentiation; Cell Line; Humans; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Pyrazines; Receptors, Cell Surface; Receptors, Transferrin; Sodium-Hydrogen Exchangers | 1985 |
Ca2+-dependent stimulation of 3-O-methylglucose transport in mouse fibroblast Swiss 3T3 cells induced by phorbol-12,13-dibutyrate.
Topics: 3-O-Methylglucose; Animals; Biological Transport, Active; Calcimycin; Calcium; Cell Transformation, Viral; Egtazic Acid; Fibroblasts; Methylglucosides; Methylglycosides; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Simian virus 40; Time Factors | 1985 |
Structural requirements for diacylglycerols to mimic tumor-promoting phobol diester action on the epidermal growth factor receptor.
Topics: Animals; Carcinogens; Cell Line; Diglycerides; ErbB Receptors; Glycerides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1985 |
1,2-Diacylglycerol and phorbol ester inhibit agonist-induced formation of inositol phosphates in human platelets: possible implications for negative feedback regulation of inositol phospholipid hydrolysis.
Topics: Blood Platelets; Diglycerides; Feedback; Glycerides; Humans; Hydrolysis; In Vitro Techniques; Inositol Phosphates; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Phosphatidylinositols; Sugar Phosphates; Thrombin | 1985 |
Effects of tumor promoters on sodium ion transport across frog skin.
Topics: Amiloride; Animals; Biological Transport, Active; Carcinogens; Cyclic AMP; Indomethacin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rana pipiens; Skin; Sodium; Tetradecanoylphorbol Acetate | 1985 |
Effects of epidermal growth factor, phorbol myristate acetate, and arachidonic acid on choriogonadotropin secretion by cultured human choriocarcinoma cells.
Topics: Arachidonic Acid; Arachidonic Acids; Caenorhabditis elegans Proteins; Carrier Proteins; Catechols; Cells, Cultured; Choriocarcinoma; Chorionic Gonadotropin; Dose-Response Relationship, Drug; Epidermal Growth Factor; ErbB Receptors; Female; Humans; Indomethacin; Masoprocol; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pregnancy; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Uterine Neoplasms | 1985 |
Phorbol ester causes desensitization of gonadotropin-responsive adenylate cyclase in a murine Leydig tumor cell line.
Topics: Adenylyl Cyclases; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Chorionic Gonadotropin; Diglycerides; Dose-Response Relationship, Drug; Kinetics; Leydig Cell Tumor; Male; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Receptors, Immunologic; Receptors, LH; Testicular Neoplasms; Tetradecanoylphorbol Acetate | 1985 |
1,2-Didecanoylglycerol and phorbol 12,13-dibutyrate enhance anterior pituitary hormone secretion in vitro.
Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; Diglycerides; Dose-Response Relationship, Drug; Endorphins; Enzyme Activation; Follicle Stimulating Hormone; Glycerides; Growth Hormone; Luteinizing Hormone; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pituitary Gland, Anterior; Prolactin; Protein Kinase C; Protein Kinases; Rats; Thyrotropin; Time Factors | 1985 |
Tumor-promoting phorbol esters and vanadate alter the sensitivity of HeLa S3 cells to poliovirus type 1.
Topics: Cell Membrane; HeLa Cells; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Poliovirus; Tetradecanoylphorbol Acetate; Vanadates; Vanadium | 1985 |
Effect of the calcium ionophore A23187 on superoxide generation in phorbol ester stimulated human neutrophils.
Topics: Calcimycin; Calcium; Humans; In Vitro Techniques; Kinetics; L-Lactate Dehydrogenase; Lysosomes; Neutrophils; Oxygen Consumption; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Superoxides; Tetradecanoylphorbol Acetate | 1985 |
The effect of cAMP on tumour promoter responses mediated by C-kinase.
Topics: Aminophylline; Animals; Bucladesine; Carcinogens; Cell Communication; Cell Line; Cyclic AMP; Diglycerides; Epidermal Growth Factor; Glycerides; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylcholines; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Phorbol ester-induced inhibition of cyclic GMP formation mediated by muscarinic receptors in murine neuroblastoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Carbachol; Cell Line; Cyclic GMP; Dose-Response Relationship, Drug; Histamine; Isoquinolines; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Piperazines; Receptors, Muscarinic; Tetradecanoylphorbol Acetate | 1987 |
Phorbol ester-stimulated T lymphocytes show enhanced adhesion to human endothelial cell monolayers.
Topics: Cell Adhesion; Cells, Cultured; Endothelium; Fibroblasts; Gelatin; Humans; Interferon-gamma; Interleukin-1; Lipopolysaccharides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; T-Lymphocytes; Tetradecanoylphorbol Acetate; Umbilical Veins | 1986 |
Diacylglycerols mimic phorbol diester induction of leukemic cell differentiation.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Differentiation; Cell Line; Diglycerides; Enzyme Activation; Glycerides; Humans; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Drug; Receptors, Immunologic | 1985 |
Modulation of protein kinase C activity and [3H]phorbol 12,13-dibutyrate binding by various tumor promoters in mouse brain cytosol.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Brain; Carcinogens; Cytosol; Fatty Acids; Female; In Vitro Techniques; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases | 1985 |
Phorbolesters enhance basal D-glucose transport but inhibit insulin stimulation of D-glucose transport and insulin binding in isolated rat adipocytes.
Topics: Adipose Tissue; Animals; Biological Transport, Active; Glucose; Insulin; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Protein-Tyrosine Kinases; Rats; Rats, Inbred Strains; Receptor, Insulin; Tetradecanoylphorbol Acetate | 1985 |
Tumor-promoting phorbol esters induce rapid internalization of the C3b receptor via a cytoskeleton-dependent mechanism.
Topics: Antibodies, Monoclonal; Binding, Competitive; Cytochalasin B; Cytoskeleton; Fibronectins; Humans; Immunoglobulin Fab Fragments; Neutrophils; Phagocytosis; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Receptors, Complement; Receptors, Complement 3b; Temperature; Tetradecanoylphorbol Acetate | 1985 |
Serum, like phorbol esters, rapidly activates protein kinase C in intact quiescent fibroblasts.
Topics: Animals; Culture Media; Enzyme Activation; Fibroblasts; Interphase; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphorylation; Platelet-Derived Growth Factor; Protein Kinase C; Protein Kinases | 1985 |
Characterization of lymphocyte stimulation by phorbol related compounds.
Topics: Adolescent; Adult; Animals; Humans; Irritants; Lymphocyte Activation; Male; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phytohemagglutinins; Skin Tests; Tetradecanoylphorbol Acetate | 1988 |
Regulation of [3H]phorbol-12,13-dibutyrate binding sites in mouse neuroblastoma cells: simultaneous down-regulation by phorbol esters and desensitization of their inhibition of muscarinic receptor function.
Topics: Animals; Binding Sites; Carbachol; Clone Cells; Enzyme Activation; Kinetics; Mice; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Muscarinic | 1988 |
Protein kinase C and phorbol ester receptor expression related to growth and differentiation of nullipotent and pluripotent embryonal carcinoma cells.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Differentiation; Cell Division; Cell Line; DNA Replication; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Teratoma; Tetradecanoylphorbol Acetate; Thymidine | 1986 |
Phorbol esters inhibit the proliferation of MCF-7 cells. Possible implication of protein kinase C.
Topics: Breast Neoplasms; Cell Division; Cell Line; Dose-Response Relationship, Drug; Female; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Effects of diacylglycerol and phorbol ester on acetylcholine release and action at the neuromuscular junction in mice.
Topics: Animals; Benzylamines; Calcium; Diaphragm; Diglycerides; Electric Stimulation; Glycerides; In Vitro Techniques; Magnesium; Membrane Potentials; Mice; Motor Endplate; Neuromuscular Junction; Pargyline; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phrenic Nerve; Stereoisomerism; Tubocurarine | 1987 |
Phorbol esters inhibit ammoniagenesis and gluconeogenesis in proximal tubular segments.
Topics: Ammonia; Animals; Dimethyl Sulfoxide; Dogs; Gluconeogenesis; Glutamine; Kidney Tubules, Proximal; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1987 |
Comparison of the activity of phorbol 12-myristate 13-acetate and the diglyceride glycerol 1-myristate 2-acetate.
Topics: Animals; Cell Line; Diglycerides; Epidermal Growth Factor; Fibroblasts; Glycerides; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Radioimmunoassay for phorbol esters using rabbit antisera against phorbol succinate.
Topics: Animals; Carcinogens; Cross Reactions; Immune Sera; Kinetics; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rabbits; Radioimmunoassay; Rats; Rats, Inbred Strains; Succinates; Tritium | 1985 |
Highly lipophilic phorbol esters as inhibitors of specific [3H]phorbol 12,13-dibutyrate binding.
Topics: Animals; Binding, Competitive; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cytosol; Detergents; Female; Kinetics; Mice; Octoxynol; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylserines; Polyethylene Glycols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Solubility; Structure-Activity Relationship | 1985 |
Phorbol esters increase calcitonin gene transcription and decrease c-myc mRNA levels in cultured human medullary thyroid carcinoma.
Topics: Calcitonin; Carcinogens; Cell Line; DNA; Genes; Humans; Kinetics; Oncogenes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; RNA, Messenger; Tetradecanoylphorbol Acetate; Thyroid Neoplasms; Transcription, Genetic | 1985 |
Phorbol ester-induced lymphocyte adherence: selective action on NK cells.
Topics: Antibody-Dependent Cell Cytotoxicity; Cell Adhesion; Cell Line; Cell Separation; Cytotoxicity, Immunologic; Humans; Interferon Type I; Killer Cells, Natural; Kinetics; Leukemia, Erythroblastic, Acute; Lymphocyte Activation; Phenotype; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols | 1985 |
Comparative effects of a complete tumor promoter, TPA, and a second-stage tumor promoter, RPA, on intercellular communication, cell differentiation and cell transformation.
Topics: Animals; Cell Communication; Cell Differentiation; Cell Transformation, Neoplastic; Cells, Cultured; Mice; Mice, Inbred BALB C; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1985 |
Characterization of the growth inhibition induced by tumor-promoting phorbol esters and of their receptor binding in A549 human lung carcinoma cells.
Topics: Caenorhabditis elegans Proteins; Carcinoma; Carrier Proteins; Cell Division; Cells, Cultured; Humans; Lung Neoplasms; Male; Middle Aged; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Tritium; Type C Phospholipases | 1985 |
Glucocorticoid-mediated increases in glycerol phosphate dehydrogenase activity is inhibited by the phorbol ester tumor promoters.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Dexamethasone; Enzyme Induction; Glioma; Glycerolphosphate Dehydrogenase; Oligodendroglia; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Theophylline | 1985 |
Phorbol ester stimulation of active anion secretion in intestine.
Topics: Animals; Anions; Carcinogens; Chickens; Epithelial Cells; Epithelium; Ileum; Intestinal Mucosa; Kinetics; Membrane Potentials; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rabbits | 1985 |
Cellular uptake and localization of fluorescent derivatives of phorbol ester tumor promoters.
Topics: Animals; Binding, Competitive; Cattle; Cell Line; Chick Embryo; Cytoplasm; Dansyl Compounds; Enzyme Activation; Fluorescent Dyes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1985 |
The 65-kDa phorbol-diester hydrolase in mouse plasma is esterase 1 and is immunologically distinct from the 56-kDa phorbol-diester hydrolase in mouse liver.
Topics: Animals; Antibody Specificity; Carboxylesterase; Carboxylic Ester Hydrolases; Chromatography, High Pressure Liquid; Cross Reactions; Estradiol; Kinetics; Liver; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1985 |
Modulation of human blood lymphocyte cytotoxicity by the phorbol ester tumor promoter P(Bu)2: increase of target binding, impairment of effector recycling, and activation of lytic potential which is independent of IL-2.
Topics: Animals; Antibodies, Monoclonal; Burkitt Lymphoma; Cell Count; Cell Line; Cytotoxicity, Immunologic; Humans; Interferon Type I; Interleukin-2; Killer Cells, Natural; Kinetics; Leukemia, Myeloid; Lymphocyte Activation; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; T-Lymphocytes, Cytotoxic | 1985 |
Role of phorbol ester receptors in the 12-0-tetradecanoyl-phorbol-13-acetate (TPA)-induced down-regulation of colony-stimulating factor (CSF-1) binding to murine peritoneal exudate macrophages.
Topics: Animals; Ascitic Fluid; Caenorhabditis elegans Proteins; Carrier Proteins; Colony-Stimulating Factors; Macrophages; Mice; Mice, Inbred C3H; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Temperature; Tetradecanoylphorbol Acetate; Time Factors | 1985 |
Sensitization of frog erythrocyte adenylate cyclase system by tumor-promoting phorbol diesters.
Topics: Adenylyl Cyclases; Animals; Carcinogens; Erythrocyte Membrane; Erythrocytes; Fluorides; Isoproterenol; Kinetics; Manganese; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rana pipiens; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1985 |
Bryostatins: potent, new mitogens that mimic phorbol ester tumor promoters.
Topics: Animals; Bryostatins; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cells, Cultured; Insulin; Lactones; Macrolides; Mice; Mitogens; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Thymidine | 1985 |
gamma-Interferon enhances the secretion of arachidonic acid metabolites from murine peritoneal macrophages stimulated with phorbol diesters.
Topics: Adjuvants, Immunologic; Animals; Arachidonic Acid; Arachidonic Acids; Interferon-gamma; Macrophage Activation; Macrophages; Mice; Mice, Inbred C57BL; Peritoneal Cavity; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins; SRS-A; Tetradecanoylphorbol Acetate; Thromboxane B2 | 1985 |
Similar effects of phospholipase C and phorbol ester tumor promoters on primary mouse epidermal cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Caenorhabditis elegans Proteins; Carrier Proteins; Cells, Cultured; Diglycerides; Enzyme Induction; Epidermal Growth Factor; Epidermis; Mice; Mice, Inbred BALB C; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Tritium; Type C Phospholipases | 1985 |
Inhibition of cell communication between Balb/c 3T3 cells by tumor promoters and protection by cAMP.
Topics: Animals; Bucladesine; Caenorhabditis elegans Proteins; Caffeine; Carcinogens; Carrier Proteins; Cell Communication; Cells, Cultured; Cricetinae; Cricetulus; Cyclic AMP; Fluorescent Dyes; Isoquinolines; Lung; Mice; Mice, Inbred BALB C; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate | 1984 |
Biological responsiveness to the phorbol esters and specific binding of [3H]phorbol 12,13-dibutyrate in the nematode Caenorhabditis elegans, a manipulable genetic system.
Topics: Animals; Caenorhabditis; Carcinogens; Movement; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Tritium | 1982 |
Characterization of specific binding of 3H-phorbol dibutyrate to Friend leukemia cells.
Topics: Animals; Antipsychotic Agents; Binding Sites; Caenorhabditis elegans Proteins; Calmodulin; Carrier Proteins; Cell Line; Depression, Chemical; Friend murine leukemia virus; Kinetics; Leukemia, Experimental; Mice; Neuraminidase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipases; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug | 1983 |
Tumour promoter-mediated reversible inhibition of cell-cell communication (electrical coupling). Relationship with phorbol ester binding and de novo macromolecule synthesis.
Topics: Binding Sites; Cell Communication; Cell Line; Cycloheximide; Dactinomycin; Diterpenes; Electrophysiology; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Biosynthesis; RNA; Terpenes; Tetradecanoylphorbol Acetate | 1983 |
Disappearance of Ca2+-sensitive, phospholipid-dependent protein kinase activity in phorbol ester-treated 3T3 cells.
Topics: Animals; Calcium; Cell Line; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Protein Kinase Inhibitors; Time Factors | 1984 |
Phorbol esters inhibit the functional activation of cytotoxic precursors in mixed lymphocyte cultures.
Topics: Antigens, Surface; Cytotoxicity, Immunologic; Humans; Immunosuppressive Agents; Interferon Type I; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Mitogens; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Stem Cells; T-Lymphocytes, Cytotoxic; T-Lymphocytes, Regulatory | 1984 |
Phorbol ester-induced protein secretion in rat parotid gland. Relationship to the role of inositol lipid breakdown and protein kinase C activation in stimulus-secretion coupling.
Topics: Animals; Calcium; Carcinogens; Egtazic Acid; Ethers; In Vitro Techniques; Inositol; Ionomycin; Kinetics; Male; Methacholine Chloride; Methacholine Compounds; Parotid Gland; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Proteins; Rats; Tritium | 1984 |
Phorbol ester stimulation of Na influx and Na-K pump activity in Swiss 3T3 cells.
Topics: Animals; Biological Transport, Active; Carcinogens; Cells, Cultured; Kinetics; Mice; Mice, Inbred Strains; Monensin; Ouabain; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rubidium; Sodium; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate | 1981 |
Inhibition of epidermal growth factor binding to mouse embryonal carcinoma cells by phorbol esters mediated by specific phorbol ester receptors.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Epidermal Growth Factor; ErbB Receptors; Kinetics; Mice; Neoplasms, Experimental; Peptides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Teratoma; Tetradecanoylphorbol Acetate | 1981 |
Inhibition of phorbol ester-receptor binding by a factor from human serum.
Topics: Animals; Arachidonic Acids; Blood; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Cell Membrane; Choline; Embryo, Mammalian; Epidermal Growth Factor; ErbB Receptors; Female; Humans; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Pregnancy; Protein Kinase C; Rats; Receptors, Cell Surface; Receptors, Drug; Sex Characteristics | 1982 |
Effect of tunicamycin on receptors for tumor promoters.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Epidermal Growth Factor; Glucosamine; Glycoproteins; Mannose; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin; Tunicamycin | 1982 |
Tumor promoter binding to rat mammary cell cultures: role of receptors in the inhibition of dome formation.
Topics: Animals; Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Female; Mammary Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Cell Surface; Receptors, Drug; Temperature; Tetradecanoylphorbol Acetate; Time Factors | 1983 |
Differential effect of tumor promoters on phorbol-ester-receptor binding and membrane fluorescence anisotropy in C3H 10T 1/2 cells.
Topics: Alkaloids; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Membrane; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Fibroblasts; Fluorescence Polarization; Kinetics; Lyngbya Toxins; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Species Specificity; Temperature | 1983 |
Specific desensitization to tumor-promoting phorbol esters in mouse pituitary cells. Evidence that desensitization is a two-step process.
Topics: Adrenocorticotropic Hormone; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pituitary Neoplasms; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
Control of endogenous cell regulators by the second-stage tumor promoter phorbol-12-retinoate 13-acetate.
Topics: Animals; Binding, Competitive; Cell Differentiation; Cells, Cultured; Cyclic AMP; Glycoproteins; Growth Inhibitors; Interleukin-6; Leukemia Inhibitory Factor; Leukemia, Myeloid; Lymphokines; Mice; Muramidase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins E; Tetradecanoylphorbol Acetate | 1983 |
Binding of phorbol dibutyrate and epidermal growth factor to cultured human epidermal cells.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Epidermal Growth Factor; ErbB Receptors; Humans; Melanoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin Neoplasms; Tetradecanoylphorbol Acetate | 1983 |
The role of phorbol ester receptor binding in responses to promoters by mouse and human cells.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Differentiation; Cell Line; Clone Cells; Drug Resistance; Humans; Leukemia, Myeloid, Acute; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin; Tetradecanoylphorbol Acetate | 1983 |
Tissue and species specificity for phorbol ester receptors.
Topics: Animals; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cattle; Chickens; Cricetinae; Erythrocytes; Female; Humans; Mice; Organ Specificity; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Species Specificity | 1983 |
An inhibitory effect of tumour promoters on human epithelial cell growth can be dissociated from an effect on junctional communication.
Topics: Breast Neoplasms; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Communication; Cell Division; Cell Line; Cell Transformation, Viral; Epidermal Cells; Epidermis; Humans; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
Tumor-promoting phorbol esters inhibit the binding of colony-stimulating factor (CSF-1) to murine peritoneal exudate macrophages.
Topics: Animals; Ascitic Fluid; Colony-Stimulating Factors; Dose-Response Relationship, Drug; Kinetics; Macrophages; Mice; Mice, Inbred C3H; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Receptors, Cell Surface; Receptors, Colony-Stimulating Factor; Temperature; Tetradecanoylphorbol Acetate | 1983 |
Tumor promoter receptors regulating neurite formation in cultured human neuroblastoma cells.
Topics: Axons; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Humans; Kinetics; Neuroblastoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug | 1983 |
Effect of cellular phospholipid modification on phorbol diester binding.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tritium | 1983 |
Characterization of a specific phorbol ester aporeceptor in mouse brain cytosol.
Topics: Animals; Apoproteins; Binding, Competitive; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cytosol; Female; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug | 1983 |
Specific binding of [20-3H]12-deoxyphorbol 13-isobutyrate to phorbol ester receptor subclasses in mouse skin particulate preparations.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Female; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Skin; Structure-Activity Relationship | 1983 |
Phorbol diester-induced H2O2 production by peritoneal macrophages. Different H2O2 production by macrophages from normal and BCG-infected mice despite comparable phorbol diester receptors.
Topics: Animals; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cells, Cultured; Female; Hydrogen Peroxide; Kinetics; Macrophages; Mice; Mice, Inbred Strains; Mycobacterium bovis; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1983 |
Effects of cytochrome P1-450 inducers on the cell-surface receptors for epidermal growth factor, phorbol 12,13-dibutyrate, or insulin of cultured mouse hepatoma cells.
Topics: Animals; Benz(a)Anthracenes; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Cytochrome P-450 Enzyme System; Enzyme Induction; ErbB Receptors; Liver Neoplasms, Experimental; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Polychlorinated Dibenzodioxins; Protein Kinase C; Receptor, Insulin; Receptors, Cell Surface; Receptors, Drug | 1983 |
Protein kinase C as a possible receptor protein of tumor-promoting phorbol esters.
Topics: Animals; Binding, Competitive; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Protein Kinases; Rats; Receptors, Cell Surface; Receptors, Drug | 1983 |
Association of phorbol ester receptor down modulation with a cryptic receptor state.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Line; Cell Nucleus; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pituitary Neoplasms; Protein Kinase C; Rats; Receptors, Cell Surface; Receptors, Drug; Thyrotropin-Releasing Hormone | 1983 |
Phorbol esters, phospholipase C, and growth factors rapidly stimulate the phosphorylation of a Mr 80,000 protein in intact quiescent 3T3 cells.
Topics: Animals; Carcinogens; Cells, Cultured; Clostridium perfringens; Kinetics; Mice; Molecular Weight; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipases; Phosphoproteins; Phosphorus Radioisotopes; Phosphorylation; Platelet-Derived Growth Factor; Proteins; Type C Phospholipases | 1983 |
Phorbol ester receptors: autoradiographic identification in the developing rat.
Topics: Animals; Autoradiography; Brain; Brain Chemistry; Caenorhabditis elegans Proteins; Carrier Proteins; Cell Communication; Cell Division; Central Nervous System; Eye; Fetus; Intestines; Lens, Crystalline; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Drug | 1983 |
Human leukemia cell lines with comparable receptor binding characteristics but different phenotypic responses to phorbol diesters.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Adhesion; Cell Aggregation; Cell Line; Humans; Kinetics; Leukemia; Phenotype; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug | 1984 |
Epidermal growth factor and potent phorbol tumor promoters induce epidermal growth factor receptor phosphorylation in a similar but distinctively different manner in human epidermoid carcinoma A431 cells.
Topics: Carcinogens; Carcinoma, Squamous Cell; Cell Line; Epidermal Growth Factor; ErbB Receptors; Humans; Kinetics; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphorylation; Receptors, Cell Surface; Tetradecanoylphorbol Acetate | 1984 |
Possible mechanism of phorbol diester-induced maturation of human promyelocytic leukemia cells.
Topics: Caenorhabditis elegans Proteins; Carrier Proteins; Cell Differentiation; Cell Line; Enzyme Activation; Humans; Leukemia, Myeloid; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Receptors, Drug; Tetradecanoylphorbol Acetate | 1984 |
Mechanism of action of the phorbol ester tumor promoters: specific receptors for lipophilic ligands.
Topics: Animals; Brain Chemistry; Caenorhabditis elegans Proteins; Calcium; Carrier Proteins; Diglycerides; Humans; Neoplasms; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Protein Kinases; Receptors, Cell Surface; Receptors, Drug; Tritium | 1984 |
Vinculin phosphorylation in response to calcium and phorbol esters in intact cells.
Topics: Animals; Bucladesine; Calcium; Cells, Cultured; Chick Embryo; Dibutyryl Cyclic GMP; Fibroblasts; Kinetics; Mice; Muscle Proteins; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphopeptides; Phosphorylation; Tetradecanoylphorbol Acetate; Trypsin; Vinculin | 1984 |
Association of phorbol ester-induced hyperphosphorylation and reversible regulation of transferrin membrane receptors in HL60 cells.
Topics: Carcinogens; Cell Line; Cell Membrane; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphorylation; Receptors, Cell Surface; Receptors, Transferrin; Transferrin | 1984 |
Phorbol esters rapidly stimulate amiloride-sensitive Na+/H+ exchange in a human leukemic cell line.
Topics: Amiloride; Carrier Proteins; Cell Line; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pyrazines; Sodium-Hydrogen Exchangers; Tetradecanoylphorbol Acetate | 1984 |
Analysis of human promyelocytic leukemia cell (HL60) variants insensitive to phorbol ester tumor promoters.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Line; Genetic Variation; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug; Superoxide Dismutase; Tetradecanoylphorbol Acetate | 1984 |
Prevention of phorbol ester receptor down modulation in human myeloblastic leukemia ML-1 cells by differentiation-stimulating serum components.
Topics: Animals; Binding, Competitive; Blood; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cattle; Cell Differentiation; Cell Line; Culture Media; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Cell Surface; Receptors, Drug | 1984 |
Phorbol esters inhibit murine B cell differentiation to immunoglobulin secretion but not proliferation.
Topics: Animals; Antibody-Producing Cells; B-Lymphocytes; Cell Differentiation; Dose-Response Relationship, Immunologic; Female; Immunoglobulin G; Immunoglobulin M; Immunosuppressive Agents; Kinetics; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Structure-Activity Relationship; Tetradecanoylphorbol Acetate | 1984 |
Phorbol 12,13-dibutyrate (P(Bu)2)-treated human blood mononuclear cells bind to each other.
Topics: Animals; Cell Aggregation; Cell Communication; Cycloheximide; Deoxyglucose; Edetic Acid; Energy Metabolism; Humans; Leukocytes; Lymphocyte Activation; Lymphocytes; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols | 1983 |
Phorbol diesters stimulate somatostatin secretion from cultured brain cells.
Topics: Alkaloids; Animals; Cell Line; Cerebral Cortex; Female; gamma-Aminobutyric Acid; Hypothalamus; Lyngbya Toxins; Peptides; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pregnancy; Rats; Tetradecanoylphorbol Acetate; Verapamil | 1983 |
Regulation of phosphatidylinositol turnover, calcium metabolism and enzyme secretion by phorbol dibutyrate in neutrophils.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcium; Dose-Response Relationship, Drug; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphates; Phosphatidylinositols; Phospholipases; Phospholipases A; Phospholipases A2; Rabbits; Time Factors | 1984 |
Phorbol esters enhance spontaneous cytotoxicity of human lymphocytes, abrogate Fc receptor expression, and inhibit antibody-dependent lymphocyte-mediated cytotoxicity.
Topics: Animals; Antibody-Dependent Cell Cytotoxicity; Antigens, Surface; Cell Line; Cytotoxicity, Immunologic; Humans; Interferon-gamma; Killer Cells, Natural; Lymphocyte Activation; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Receptors, Fc | 1984 |
Decreased [20-3H]phorbol-12,13-dibutyrate binding to phospholipase C pretreated epidermal cells.
Topics: Animals; Binding Sites; Carcinogens; Cell Line; Dose-Response Relationship, Drug; Epidermis; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipases; Time Factors; Type C Phospholipases | 1983 |
Specific binding of [3H]phorbol dibutyrate to phorbol diester-responsive and -resistant clones of a human myeloid leukemia (KG-1) line 1.
Topics: Cell Differentiation; Cell Line; Clone Cells; Humans; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols | 1983 |
Presence of specific binding sites for phorbol ester tumor promoters in human epidermal and dermal cells in culture but lack of down regulation in epidermal cells.
Topics: Binding Sites; Binding, Competitive; Cells, Cultured; Diterpenes; Epidermis; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Terpenes; Tetradecanoylphorbol Acetate | 1983 |
Control of macrophage cell differentiation in human promyelocytic HL-60 leukemia cells by 1,25-dihydroxyvitamin D3 and phorbol-12-myristate-13-acetate.
Topics: Antibodies, Monoclonal; Calcitriol; Cell Differentiation; Cell Line; Dimethyl Sulfoxide; Humans; Leukemia, Myeloid, Acute; Macrophages; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1983 |
Phorbol ester-associated changes in ganglioside metabolism.
Topics: Animals; Carcinogens; Cell Division; Cell Line; Contact Inhibition; Cricetinae; Gangliosides; Palmitic Acid; Palmitic Acids; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Sialic Acids; Sialyltransferases; Tetradecanoylphorbol Acetate | 1983 |
Characterization of the phorbol 12,13-dibutyrate (P(Bu)2) induced binding between human lymphocytes.
Topics: Amino Acids; Cell Adhesion; Cell Aggregation; Humans; Lymphocytes; Membrane Proteins; Neuraminidase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protease Inhibitors; Trypsin | 1983 |
Serum, platelet-derived growth factor, vasopressin and phorbol esters increase intracellular pH in Swiss 3T3 cells.
Topics: Animals; Body Fluids; Carcinogens; Cells, Cultured; Culture Media; Humans; Hydrogen-Ion Concentration; Intracellular Fluid; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Platelet-Derived Growth Factor; Vasopressins | 1983 |
Relationship between a tumor promoter-induced decrease in queuine modification of transfer RNA in normal human cells and the expression of an altered cell phenotype.
Topics: Carcinogens; Cells, Cultured; Fibroblasts; Guanine; Humans; Infant, Newborn; Kinetics; Male; Phenotype; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; RNA, Transfer; Skin; Tritium | 1984 |
Phorbol 12,13-dibutyrate enhances lateral redistribution of membrane glycoproteins in human blood lymphocytes.
Topics: Glycoproteins; Humans; Immunologic Capping; Lymphocytes; Membrane Proteins; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protease Inhibitors; Tetradecanoylphorbol Acetate | 1984 |
Inhibition of denuded mouse oocyte meiotic maturation by tumor-promoting phorbol esters and its reversal by retinoids.
Topics: Animals; Colforsin; Diterpenes; Drug Interactions; Female; Meiosis; Mice; Oocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Retinoids; Tetradecanoylphorbol Acetate | 1984 |
Phorbol esters inhibit agonist-induced [3H] inositol-1-phosphate accumulation in rat hippocampal slices.
Topics: Animals; Caenorhabditis elegans Proteins; Carbachol; Carcinogens; Carrier Proteins; Hippocampus; Inositol; Inositol Phosphates; Male; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rats; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate | 1984 |
Phorbol ester binding to chemotactically responding and nonresponding Walker 256 carcinosarcoma cells.
Topics: Animals; Binding, Competitive; Caenorhabditis elegans Proteins; Carcinogens; Carcinoma 256, Walker; Carrier Proteins; Chemotaxis; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Receptors, Immunologic | 1984 |
Biological activity of a fluorescent 12-O-tetradecanoyl-phorbol-13-acetate derivative.
Topics: Animals; Cricetinae; Cricetulus; Dansyl Compounds; Fluorescence; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1984 |
Phorbol ester tumor promoters specifically stimulate choline phospholipid metabolism in human leukemic cells.
Topics: Acetates; Acetic Acid; Caenorhabditis elegans Proteins; Carbon Radioisotopes; Carcinogens; Carrier Proteins; Cells, Cultured; Choline; Humans; Leukemia, Hairy Cell; Microscopy, Electron, Scanning; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylcholines; Protein Kinase C; Receptors, Drug; Receptors, Immunologic; Tetradecanoylphorbol Acetate; Tritium | 1984 |
Relationship between mezerein-mediated biological responses and phorbol ester receptor occupancy.
Topics: Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Dinoprostone; Diterpenes; Epidermal Growth Factor; Humans; Kinetics; Osteosarcoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins E; Protein Kinase C; Receptors, Drug; Terpenes; Tetradecanoylphorbol Acetate | 1983 |
Phorbol ester modulation of T-cell antigens in the Jurkat lymphoblastic leukemia cell line.
Topics: Antigens, Surface; Cell Division; Cell Line; Humans; Leukemia, Lymphoid; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rosette Formation; T-Lymphocytes | 1983 |
The tumor promoter phorbol-12,13-dibutyrate [P(Bu)2] stimulates cytotoxic activity of human blood lymphocytes.
Topics: Cell Adhesion; Cytotoxicity, Immunologic; Humans; In Vitro Techniques; Killer Cells, Natural; Lymphocyte Activation; Lymphocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; T-Lymphocytes, Cytotoxic; Tetradecanoylphorbol Acetate; Time Factors | 1983 |
Release of granulocyte-specific colony-stimulating activity by human bone marrow exposed to phorbol esters.
Topics: Alprostadil; Bone Marrow; Bone Marrow Cells; Colony-Forming Units Assay; Colony-Stimulating Factors; Granulocytes; Hematopoiesis; Hematopoietic Stem Cells; Humans; Monocytes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Prostaglandins E; Time Factors | 1984 |
Characterization of phorbol ester receptors and their down-modulation in GH4C1 rat pituitary cells.
Topics: Animals; Binding Sites; Caenorhabditis elegans Proteins; Carrier Proteins; Dose-Response Relationship, Drug; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pituitary Gland; Protein Kinase C; Rats; Receptors, Drug; Thyrotropin-Releasing Hormone; Time Factors | 1981 |
Stimulation of DNA synthesis in murine fibroblasts by the tumour promoter teleocidin: relationship to phorbol esters and vasopressin.
Topics: Alkaloids; Animals; Carcinogens; Cells, Cultured; DNA; Drug Synergism; Fibroblasts; Growth Substances; Lyngbya Toxins; Mice; Mice, Inbred BALB C; Mitogens; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Vasopressins | 1982 |
The control of phospholipid methylation by phorbol diesters in differentiating human myeloid HL-60 leukemia cells.
Topics: Alkaloids; Cell Differentiation; Cell Line; Humans; Leukemia, Myeloid, Acute; Lyngbya Toxins; Methylation; Methyltransferases; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylethanolamine N-Methyltransferase; Phospholipids; Tetradecanoylphorbol Acetate | 1982 |
Variation with embryonic development and regional localization of specific [3H]phorbol 12,13-dibutyrate binding to brain.
Topics: Animals; Brain; Brain Mapping; Caenorhabditis elegans Proteins; Carrier Proteins; Cattle; Chick Embryo; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Propranolol; Protein Kinase C; Receptors, Drug | 1981 |
Down regulation of specific binding of [20-3H]phorbol 12,13-dibutyrate and phorbol ester-induced differentiation of human promyelocytic leukemia cells.
Topics: Binding Sites; Binding, Competitive; Carcinogens; Cell Differentiation; Cell Line; Humans; Kinetics; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate | 1981 |
Specific binding of phorbol ester tumor promoters to intact primary epidermal cells from Sencar mice.
Topics: Animals; Animals, Newborn; Binding, Competitive; Caenorhabditis elegans Proteins; Carrier Proteins; Epidermis; Fluocinolone Acetonide; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Tretinoin | 1981 |
Kinetics and subcellular localization of specific [3H]phorbol 12, 13-dibutyrate binding by mouse brain.
Topics: Animals; Binding Sites; Brain; Calcium; Cell Fractionation; Centrifugation, Density Gradient; Hydrogen-Ion Concentration; Intracellular Membranes; Kinetics; Mice; Mitochondria; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Temperature | 1981 |
TPA-resistance in Friend erythroleukemia cells: role of membrane lipid fluidity.
Topics: Animals; Carcinogens; Cell Line; Clone Cells; Diphenylhexatriene; Drug Resistance; Kinetics; Leukemia, Experimental; Membrane Fluidity; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Spectrometry, Fluorescence; Tetradecanoylphorbol Acetate | 1981 |
Isolation and characterization of an ester hydrolase active on phorbol diesters from murine liver.
Topics: Animals; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Membrane; Cytosol; Esterases; Kinetics; Liver; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Substrate Specificity | 1981 |
Analysis of phorbol ester receptors in phorbol ester unresponsive 3T3 cell variants.
Topics: Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Cells, Cultured; Genetic Variation; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1981 |
Partial purification and characterization of a binding protein for biologically active phorbol and ingenol esters from murine sera.
Topics: Animals; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Cell Membrane; Diterpenes; Humans; Kinetics; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Species Specificity | 1982 |
Tissue and species distribution and developmental variation of specific receptors for biologically active phorbol and ingenol esters.
Topics: Aging; Animals; Brain; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Diterpenes; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Rabbits; Receptors, Drug; Species Specificity; Spleen; Tissue Distribution | 1981 |
Phorbol-12,13-diester 12-ester hydrolase may prevent tumour promotion by phorbol diesters in skin.
Topics: Animals; Carboxylic Ester Hydrolases; Cats; Child, Preschool; Cricetinae; Dogs; Female; Guinea Pigs; Humans; Kinetics; Macaca mulatta; Mice; Neoplasms, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Rabbits; Rats; Skin Neoplasms; Species Specificity; Swine | 1982 |
Cell differentiation, alterations in polyamine levels, and specific binding of phorbol diesters in cultured human cells.
Topics: Binding Sites; Carcinogens; Cell Differentiation; Cell Line; Cell Membrane; Humans; Leukemia, Myeloid, Acute; Melanoma; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Polyamines; Tetradecanoylphorbol Acetate | 1982 |
Modulation of HeLa cell phospholipid metabolism and ornithine decarboxylase activity by tumour promoters: regulation of response to phorbol-12,13-dibutyrate by receptor occupancy time.
Topics: Caenorhabditis elegans Proteins; Carboxy-Lyases; Carrier Proteins; Enzyme Induction; HeLa Cells; Humans; Kinetics; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phospholipids; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1982 |
Receptor-mediated modulation of human monocyte, neutrophil, lymphocyte, and platelet function by phorbol diesters.
Topics: Blood Cells; Blood Platelets; Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Humans; Hydrogen Peroxide; Leukocytes; Lymphocytes; Monocytes; Neutrophils; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Serotonin; Thymidine | 1982 |
Specific binding of phorbol esters to Friend erythroleukemia cells--general properties, down regulation and relationship to cell differentiation.
Topics: Animals; Binding Sites; Cell Differentiation; Diterpenes; Friend murine leukemia virus; Leukemia, Erythroblastic, Acute; Leukemia, Experimental; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Tetradecanoylphorbol Acetate; Tritium | 1982 |
Morphological changes, cell aggregation and cell membrane alterations caused by phorbol 12,13-dibutyrate in human blood lymphocytes.
Topics: Carcinogens; Cell Aggregation; Cell Membrane; Glycosphingolipids; Humans; Lymphocytes; Membrane Proteins; Microscopy, Electron, Scanning; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols | 1982 |
Specific receptors for phorbol esters in lymphoid cell populations: role in enhanced production of T-cell growth factor.
Topics: Caenorhabditis elegans Proteins; Carcinogens; Carrier Proteins; Humans; Interleukin-2; Kinetics; Lymphokines; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Receptors, Drug; Structure-Activity Relationship; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1981 |
Phorbol ester-induced ventricular fibrillation in the Langendorff-perfused rabbit heart: antagonism by staurosporine and glibenclamide.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Diglycerides; Glyburide; Guanidines; Isoquinolines; Perfusion; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Pinacidil; Piperazines; Protein Kinase C; Rabbits; Staurosporine; Ventricular Fibrillation | 1993 |
Inhibition of myosin light chain phosphatase during Ca(2+)-independent vasocontraction.
Topics: Animals; Aorta, Thoracic; Calcium; Colforsin; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbols; Phosphates; Phosphoprotein Phosphatases; Phosphorus Radioisotopes; Rats; Rats, Wistar; Vasoconstriction; Vasodilator Agents | 1993 |
Further characterization of 5-HT- and 5-HT3 receptor agonists'-stimulated phosphoinositol phosphates accumulation.
Topics: Animals; GTP-Binding Proteins; Inositol Phosphates; Male; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbols; Phosphatidylinositols; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1993 |
Opposing effects of phorbol esters on transmitter release and calcium currents at frog motor nerve endings.
Topics: Acetylcholine; Animals; Calcium Channel Blockers; Calcium Channels; Electrophysiology; Enzyme Activation; Motor Endplate; Motor Neurons; Nerve Endings; Neurotransmitter Agents; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Potassium Channel Blockers; Protein Kinase C; Rana pipiens | 1997 |
Facilitation of Ca2+ action potential frequency by a small G protein Rab3A in rat pituitary GH3 cells.
Topics: Action Potentials; Animals; Calcium; Enzyme Inhibitors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Patch-Clamp Techniques; Peptide Fragments; Peptides; Phorbol 12,13-Dibutyrate; Phorbols; Pituitary Gland; Protein Kinase C; rab3 GTP-Binding Proteins; rab5 GTP-Binding Proteins; ras Proteins; Rats; Thionucleotides; Thyrotropin-Releasing Hormone; Tumor Cells, Cultured | 1997 |
Protein kinase C activation decreases activity-dependent attenuation of dendritic Na+ current in hippocampal CA1 pyramidal neurons.
Topics: Action Potentials; Animals; Dendrites; Electric Stimulation; Enzyme Activation; Hippocampus; In Vitro Techniques; Male; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Protein Kinase C; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Sodium Channels | 1998 |
Restoration of TEA-induced calcium responses in fibroblasts from Alzheimer's disease patients by a PKC activator.
Topics: Alzheimer Disease; Calcium; Carcinogens; Cells, Cultured; Dimethyl Sulfoxide; Enzyme Activation; Excipients; Fibroblasts; Humans; Immunoblotting; Lactams; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Phorbols; Potassium Channels; Protein Kinase C; Tetraethylammonium | 1998 |
Activation of PKC disrupts presynaptic inhibition by group II and group III metabotropic glutamate receptors and uncouples the receptor from GTP-binding proteins.
Topics: Adenosine; Animals; Dihydropyridines; Enzyme Activation; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Phorbol 12,13-Dibutyrate; Phorbols; Propionates; Protein Kinase C; Receptor, Adenosine A3; Receptors, Metabotropic Glutamate; Receptors, Purinergic P1; Synaptic Transmission | 1999 |
Regulation of high affinity taurine transport in goldfish and rat retinal cells.
Topics: Animals; Biological Transport; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Goldfish; Okadaic Acid; Phorbol 12,13-Dibutyrate; Phorbols; Phosphoprotein Phosphatases; Protein Kinase C; Rats; Retina; Taurine | 2000 |