phorbol 12,13-dibutyrate has been researched along with 1,2-dioctanoylglycerol in 41 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 16 (39.02) | 18.7374 |
1990's | 21 (51.22) | 18.2507 |
2000's | 4 (9.76) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Boscá, L; Genaro, AM; Hortelano, S | 1 |
Alexandre, A; Deana, R; Donella-Deana, A; Francesconi, M; Ruzzene, M | 1 |
Kumada, M; Takuwa, N; Takuwa, Y; Zhou, W | 1 |
Casillas, T; Delicado, EG; Miras-Portugal, MT; Sen, RP | 1 |
Doré, M; Neilsen, NR; Slauson, DO | 1 |
Bjaaland, T; Bogle, RG; Carter, TD | 1 |
Huang, CL; Ives, HE; Lowe, JH | 1 |
Jacobson, DP; O'Flaherty, JT; Redman, JF; Rossi, AG | 1 |
Godson, C; Insel, PA; Weiss, BA | 1 |
Alonso, M; Cárdenas, L; Carrera, AC; de Landázuri, MO; Sánchez-Madrid, F; Tugores, A | 1 |
Kitajima, Y; Sheu, HM; Yaoita, H | 1 |
Gillies, RJ; Hoyer, PB; Martinez, R; Sneider, JM | 1 |
Badwey, JA; Curnutte, JT; Heyworth, PG; Robinson, JM | 1 |
Lapetina, EG; Siess, W | 1 |
Inoue, Y; Rebois, RV | 1 |
Gárdos, G; Görög, G; Sarkadi, B; Tordai, A | 1 |
Conn, PM; Huckle, WR; McArdle, CA | 1 |
de Graan, PN; Eichberg, J; Gispen, WH; Schrama, LH | 1 |
Brown, G; Gordon, J; Guy, GR; Michell, RH | 1 |
Gainer, HS; Murray, AW | 1 |
Jetten, AM; Shirley, JE | 1 |
Bell, RM; Greenberg, CS; Hannun, YA | 1 |
Crouch, MF; Lapetina, EG | 1 |
Niedel, JE; Salehi, Z; Taylor, JD | 1 |
Bell, RM; Hannun, YA; Loomis, CR; Merrill, AH | 1 |
Clegg, RA; Connor, K; Ison, A; Johnson, MS; MacEwan, DJ; Mitchell, R; Simpson, J | 1 |
Hoy, K; Maccarone, P; Marley, PD; Thomson, KA | 1 |
Brooks, G; East, JA; Goss, MW; Hart, IR | 1 |
Bardes, ES; Bell, RM; Quest, AF | 1 |
Rozengurt, E; Sinnett-Smith, J; Valverde, AM; Zachary, I | 1 |
Clegg, RA; Connor, K; Johnson, MS; Lutz, EM; MacEwan, DJ; Mitchell, R; Thomson, FJ | 1 |
Clegg, RA; Connor, K; Ison, AJ; Johnson, MS; MacEwan, DJ; Mitchell, R | 1 |
Messlinger, K; Schepelmann, K; Schmidt, RF | 1 |
Ching, KN; Nicholson, WE; Orth, DN; Won, JG | 1 |
Johnson, MS; MacEwan, DJ; Mitchell, R; Thomson, FJ | 1 |
Gailly, P; Gong, MC; Somlyo, AP; Somlyo, AV | 1 |
Rösner, H; Vacun, G | 1 |
Ciereszko, RE; Dusza, L; Kaminska, B; Opalka, M | 1 |
Namiki, H; Takahashi, H | 1 |
Burger, KN; Claro, E; Egea, G; Fernández-Ulibarri, I; Jiménez, N; Lázaro-Diéguez, F; Martínez, SE; Mérida, I; Sarri, E; Vilella, M | 1 |
Blumberg, PM; Garfield, SH; Lewin, NE; Marquez, VE; Nacro, K; Nicklaus, MC; Pearce, LL; Sigano, DM; Yan, S | 1 |
41 other study(ies) available for phorbol 12,13-dibutyrate and 1,2-dioctanoylglycerol
Article | Year |
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Phorbol esters induce nitric oxide synthase activity in rat hepatocytes. Antagonism with the induction elicited by lipopolysaccharide.
Topics: Amino Acid Oxidoreductases; Animals; Arginine; Calcimycin; Carcinogens; Cells, Cultured; Cyclic GMP; Diglycerides; Enzyme Induction; Kinetics; Lipopolysaccharides; Liver; Nitric Oxide Synthase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Rats; Tetradecanoylphorbol Acetate | 1992 |
The antioxidant butylated hydroxytoluene (BHT) inhibits the dioctanoylglycerol-evoked platelet response but potentiates that elicited by ionomycin.
Topics: Adenosine Triphosphate; Alkaloids; Arachidonic Acid; Blood Platelets; Butylated Hydroxytoluene; Diglycerides; Drug Synergism; Humans; In Vitro Techniques; Ionomycin; Kinetics; Phorbol 12,13-Dibutyrate; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Platelet Aggregation; Platelet Aggregation Inhibitors; Protein Kinase C; Staurosporine | 1992 |
Activators of protein kinase C induce p34cdc2 histone H1 kinase stimulation in Swiss 3T3 fibroblasts.
Topics: 3T3 Cells; Animals; CDC2 Protein Kinase; Diglycerides; Down-Regulation; Enzyme Activation; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C | 1992 |
Control of nucleoside transport in neural cells. Effect of protein kinase C activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine; Adrenal Medulla; Animals; Biological Transport; Calcimycin; Caprylates; Cells, Cultured; Diglycerides; Dinucleoside Phosphates; Enzyme Activation; Ethers, Cyclic; Isoquinolines; Kinetics; Okadaic Acid; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Tetradecanoylphorbol Acetate; Triglycerides | 1991 |
Decreased respiratory burst activity in neonatal bovine neutrophils stimulated by protein kinase C agonists.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Animals, Newborn; Cattle; Cells, Cultured; Diglycerides; Dose-Response Relationship, Drug; Female; Isoquinolines; Neutrophils; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 1991 |
Spiking of intracellular calcium ion concentration in single cultured pig aortic endothelial cells stimulated with ATP or bradykinin.
Topics: Adenosine Triphosphate; Animals; Aorta; Bradykinin; Calcium; Cells, Cultured; Diglycerides; Endothelium, Vascular; Enzyme Activation; Phorbol 12,13-Dibutyrate; Potassium; Protein Kinase C; Swine | 1991 |
Sphingosine differentially inhibits activation of the Na+/H+ exchanger by phorbol esters and growth factors.
Topics: Animals; Animals, Newborn; Biological Transport; Carrier Proteins; Cells, Cultured; Detergents; Diglycerides; Hydrogen-Ion Concentration; Kinetics; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Platelet-Derived Growth Factor; Rats; Sodium-Hydrogen Exchangers; Sphingosine; Tetradecanoylphorbol Acetate; Thrombin | 1990 |
Translocation of protein kinase C in human polymorphonuclear neutrophils. Regulation by cytosolic Ca2(+)-independent and Ca2(+)-dependent mechanisms.
Topics: Binding, Competitive; Caenorhabditis elegans Proteins; Calcimycin; Calcium; Carrier Proteins; Cell Membrane; Cytosol; Diglycerides; Humans; Ionomycin; Kinetics; Leukotriene B4; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phorbol 12,13-Dibutyrate; Phospholipids; Protein Kinase C; Receptors, Drug; Sphingosine | 1990 |
Differential activation of protein kinase C alpha is associated with arachidonate release in Madin-Darby canine kidney cells.
Topics: Animals; Arachidonic Acids; Bradykinin; Cell Line; Diglycerides; Dogs; Enzyme Activation; Kidney; Kinetics; Phorbol 12,13-Dibutyrate; Phospholipids; Protein Kinase C; Tetradecanoylphorbol Acetate | 1990 |
Activators of protein kinase C up-regulate the cell surface expression of CD2 and CD5 T cell glycoproteins.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antibodies, Monoclonal; Antigens, Differentiation; Antigens, Differentiation, T-Lymphocyte; Calcium Channel Blockers; CD2 Antigens; CD5 Antigens; Cell Membrane; Cells, Cultured; Cycloheximide; Diglycerides; Dinoprostone; Enzyme Activation; Flow Cytometry; Humans; Isoquinolines; Membrane Glycoproteins; Phorbol 12,13-Dibutyrate; Piperazines; Protein Kinase C; Receptors, Immunologic; RNA, Messenger; Sulfonamides; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1989 |
Involvement of protein kinase C in translocation of desmoplakins from cytosol to plasma membrane during desmosome formation in human squamous cell carcinoma cells grown in low to normal calcium concentration.
Topics: Calcimycin; Calcium; Carcinoma, Squamous Cell; Cell Membrane; Cytoskeletal Proteins; Cytosol; Desmoplakins; Desmosomes; Diglycerides; Dose-Response Relationship, Drug; Humans; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Sphingosine inhibits phorbol 12-myristate 13-acetate-, but not serum-induced, activation of Na+/H+ exchange in mammalian cells.
Topics: Animals; Blood Physiological Phenomena; Carrier Proteins; Cell Line; Diglycerides; Enzyme Activation; Humans; Hydrogen-Ion Concentration; Phorbol 12,13-Dibutyrate; Protein Kinase C; Sodium-Hydrogen Exchangers; Sphingosine; Tetradecanoylphorbol Acetate | 1989 |
1,2-dioctanoyl-sn-glycerol can stimulate neutrophils by different mechanisms. Evidence for a pathway that does not involve phosphorylation of the 47-kDa protein.
Topics: Alkaloids; Animals; Diglycerides; Diterpenes; Glycerides; Guinea Pigs; Humans; Kinetics; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Proteins; Staurosporine; Superoxides; Terpenes; Tetradecanoylphorbol Acetate | 1989 |
Platelet aggregation induced by alpha 2-adrenoceptor and protein kinase C activation. A novel synergism.
Topics: Adenosine Diphosphate Ribose; Adenosine Triphosphate; Adrenergic alpha-Agonists; Blood Platelets; Brimonidine Tartrate; Calcium; Diglycerides; Drug Synergism; Enzyme Activation; Epinephrine; GTP-Binding Proteins; Humans; Immunosorbent Techniques; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phosphorylation; Platelet Aggregation; Protein Kinase C; Quinoxalines; Receptors, Adrenergic, alpha; Type C Phospholipases; Virulence Factors, Bordetella | 1989 |
Protein kinase C activity can desensitize the gonadotropin-responsive adenylate cyclase in Leydig tumor cells. But hCG-induced desensitization does not involve protein kinase C activation.
Topics: Adenylyl Cyclases; Animals; Binding Sites; Cell Line; Chorionic Gonadotropin; Diglycerides; Enzyme Activation; Inositol; Kinetics; Leydig Cell Tumor; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1989 |
Inhibition of the CD3-mediated calcium signal by protein kinase C activators in human T (Jurkat) lymphoblastoid cells.
Topics: Antigens, Differentiation, T-Lymphocyte; Calcium; Cell Line; Depression, Chemical; Diglycerides; Enzyme Activation; Glycerides; Humans; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Antigen, T-Cell; Signal Transduction; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1989 |
Differential sensitivity of agonist- and antagonist-occupied gonadotropin-releasing hormone receptors to protein kinase C activators. A marker for receptor activation.
Topics: Animals; Buserelin; Cell Membrane; Cells, Cultured; Diglycerides; Enzyme Activation; Female; Glycerides; Gonadotropin-Releasing Hormone; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Pituitary Gland; Protein Kinase C; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, LHRH; Tetradecanoylphorbol Acetate | 1988 |
Dioctanoylglycerol and phorbol diesters enhance phosphorylation of phosphoprotein B-50 in native synaptic plasma membranes.
Topics: Animals; Calcium; Diglycerides; Dose-Response Relationship, Drug; GAP-43 Protein; Glycerides; Histones; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphoproteins; Phosphorylation; Protein Kinase C; Rats; Synaptic Membranes | 1986 |
Synergism between diacylglycerols and calcium ionophore in the induction of human B cell proliferation mimics the inositol lipid polyphosphate breakdown signals induced by crosslinking surface immunoglobulin.
Topics: B-Lymphocytes; Binding, Competitive; Cell Division; Diglycerides; Drug Synergism; Enzyme Activation; Ethers; Glycerides; Humans; Ionomycin; Lymphocyte Activation; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Protein Kinase C; Protein Kinases; Receptors, Antigen, B-Cell; Staphylococcus aureus | 1985 |
The effect of cAMP on tumour promoter responses mediated by C-kinase.
Topics: Aminophylline; Animals; Bucladesine; Carcinogens; Cell Communication; Cell Line; Cyclic AMP; Diglycerides; Epidermal Growth Factor; Glycerides; Mice; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylcholines; Protein Kinase C; Tetradecanoylphorbol Acetate | 1986 |
Action of retinoic acid on the diacylglycerol-induced ornithine decarboxylase activity, reduction in EGF binding and protein kinase C activation in rat tracheal epithelial 2C5 cells.
Topics: Animals; Cell Line; Diglycerides; Enzyme Activation; Enzyme Induction; Epidermal Growth Factor; ErbB Receptors; Ornithine Decarboxylase; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Rats; Receptors, Cell Surface; Tetradecanoylphorbol Acetate; Trachea; Tretinoin | 1986 |
Sphingosine inhibition of agonist-dependent secretion and activation of human platelets implies that protein kinase C is a necessary and common event of the signal transduction pathways.
Topics: Adenosine Diphosphate; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Collagen; Diglycerides; Humans; Kinetics; Phorbol 12,13-Dibutyrate; Phorbol Esters; Platelet Activating Factor; Platelet Aggregation; Protein Kinase C; Sphingosine; Thrombin | 1987 |
Spacial isolation of protein kinase C activation in thrombin stimulated human platelets.
Topics: Blood Platelets; Blood Proteins; Calcium; Diglycerides; Enzyme Activation; Epinephrine; Fluorescent Dyes; Humans; Indoles; Kinetics; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Platelet Activating Factor; Prostaglandin Endoperoxides, Synthetic; Protein Kinase C; Thrombin | 1988 |
Dioctanoylglycerol and phorbol esters regulate transcription of c-myc in human promyelocytic leukemia cells.
Topics: Diglycerides; Enzyme Activation; Glycerides; Humans; Leukemia, Myeloid, Acute; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Proto-Oncogenes; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 1988 |
Sphingosine inhibition of protein kinase C activity and of phorbol dibutyrate binding in vitro and in human platelets.
Topics: Amines; Blood Platelets; Diglycerides; Humans; Micelles; Models, Biological; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphatidylserines; Protein Kinase C; Sphingosine; Thrombin | 1986 |
Phorbol ester and diacylglycerol activation of native protein kinase C species from various tissues.
Topics: Animals; Cattle; Cell Line; Cytosol; Diglycerides; Enzyme Activation; Isoenzymes; Mesencephalon; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Recombinant Proteins; Spleen; Tissue Distribution | 1995 |
Regulation of cyclic AMP levels by phorbol esters in bovine adrenal medullary cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adrenal Medulla; Animals; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Indoles; Pertussis Toxin; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Virulence Factors, Bordetella | 1993 |
Growth of melanocytic cells is associated with down-regulation of protein kinase C alpha, delta, and epsilon isoforms. Possible role of diacylglycerol.
Topics: Animals; Cell Division; Cells, Cultured; Diglycerides; DNA; Down-Regulation; Isoenzymes; Melanocytes; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Tetradecanoylphorbol Acetate | 1993 |
A phorbol ester binding domain of protein kinase C gamma. High affinity binding to a glutathione-S-transferase/Cys2 fusion protein.
Topics: Animals; Base Sequence; Binding Sites; Cell Line; Cloning, Molecular; Cysteine; Diglycerides; DNA Primers; Escherichia coli; Glutathione Transferase; Isoenzymes; Kinetics; Liposomes; Molecular Sequence Data; Moths; Phorbol 12,13-Dibutyrate; Phosphatidylcholines; Phosphatidylserines; Polymerase Chain Reaction; Protein Kinase C; Rats; Recombinant Fusion Proteins; Transfection | 1994 |
Bombesin stimulation of p125 focal adhesion kinase tyrosine phosphorylation. Role of protein kinase C, Ca2+ mobilization, and the actin cytoskeleton.
Topics: 3T3 Cells; Actins; Animals; Bombesin; Calcimycin; Calcium; Calcium-Transporting ATPases; Cell Adhesion Molecules; Colchicine; Cytochalasin D; Cytoskeleton; Diglycerides; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Indoles; Intracellular Signaling Peptides and Proteins; Kinetics; Maleimides; Membrane Proteins; Mice; Myristoylated Alanine-Rich C Kinase Substrate; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Proteins; Terpenes; Thapsigargin; Tyrosine | 1993 |
Evidence that protein kinase C alpha has reduced affinity towards 1,2-dioctanoyl-sn-glycerol: the effects of lipid activators on phorbol ester binding and kinase activity.
Topics: Amino Acid Sequence; Animals; Arachidonic Acids; Cerebellum; Cerebral Cortex; Cytosol; Diglycerides; Isoenzymes; Lipid Metabolism; Lung; Male; Molecular Sequence Data; Phorbol 12,13-Dibutyrate; Phosphatidylserines; Protein Kinase C; Rats; Rats, Wistar; RNA, Messenger | 1993 |
Evidence for a distinct H7-resistant form of protein kinase C in rat anterior pituitary gland.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Calcium; Diglycerides; Diterpenes; Drug Resistance; Enzyme Activation; Indoles; Isoquinolines; Lung; Male; Phorbol 12,13-Dibutyrate; Piperazines; Pituitary Gland, Anterior; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Terpenes | 1993 |
The effects of phorbol ester on slowly conducting afferents of the cat's knee joint.
Topics: Animals; Bradykinin; Bucladesine; Cats; Dibutyryl Cyclic GMP; Diglycerides; Dinoprostone; Epoprostenol; Hindlimb; Knee Joint; Neural Conduction; Neurons, Afferent; Nociceptors; Phorbol 12,13-Dibutyrate; Protein Kinase C; Signal Transduction | 1993 |
Effect of protein kinase-C depletion on inositol trisphosphate-mediated and cyclic adenosine 3',5'-monophosphate-dependent protein kinase-mediated adrenocorticotropin secretion.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenocorticotropic Hormone; Animals; Arginine Vasopressin; Cyclic AMP; Cycloheximide; Diglycerides; Inositol 1,4,5-Trisphosphate; Ionomycin; Male; Perfusion; Phorbol 12,13-Dibutyrate; Pituitary Gland, Anterior; Potassium Chloride; Protein Kinase C; Protein Kinases; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1993 |
Oestradiol-17 beta modulates the actions of pharmacologically distinct forms of protein kinase C in rat anterior pituitary cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Cytosol; Diglycerides; Enzyme Activation; Estradiol; Female; Growth Hormone; Ionomycin; Isoenzymes; Isoquinolines; Luteinizing Hormone; Ovariectomy; Phorbol 12,13-Dibutyrate; Piperazines; Pituitary Gland, Anterior; Protein Kinase C; Rats; Rats, Wistar | 1993 |
Possible role of atypical protein kinase C activated by arachidonic acid in Ca2+ sensitization of rabbit smooth muscle.
Topics: Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Arachidonic Acid; Calcium; Diglycerides; Enzyme Activation; Enzyme Inhibitors; Femoral Artery; In Vitro Techniques; Indoles; Isoenzymes; Isometric Contraction; Kinetics; Maleimides; Molecular Sequence Data; Muscle, Smooth, Vascular; Myosin Light Chains; Peptide Fragments; Phenylephrine; Phorbol 12,13-Dibutyrate; Phosphorylation; Portal Vein; Protein Kinase C; Protein Kinase C-alpha; Rabbits; Sequence Homology, Amino Acid; Substrate Specificity; Type C Phospholipases | 1997 |
1,2-dioctanoyl-s,n-glycerol-induced activation of protein kinase C results in striking, but reversible growth cone shape changes and an accumulation of f-actin and serine 41-phosphorylated GAP-43 in the axonal process.
Topics: Actins; Animals; Animals, Newborn; Axons; Brain; Chick Embryo; Culture Techniques; Diglycerides; Enzyme Activation; Enzyme Inhibitors; GAP-43 Protein; Growth Cones; Indoles; Neurons; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Rats; Serine; Spinal Cord | 1999 |
Prolactin signaling in porcine adrenocortical cells: involvement of protein kinases.
Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Androstenedione; Animals; Diglycerides; Enzyme Activators; Enzyme Inhibitors; Female; Genistein; Hydrocortisone; Ionomycin; Phorbol 12,13-Dibutyrate; Prolactin; Protein Kinase C; Protein-Tyrosine Kinases; Signal Transduction; Sphingosine; Swine; Tetradecanoylphorbol Acetate | 2002 |
Mechanism of membrane redistribution of protein kinase C by its ATP-competitive inhibitors.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Binding, Competitive; Carbazoles; Cell Membrane; Chlorocebus aethiops; COS Cells; Diglycerides; Estrenes; HeLa Cells; HL-60 Cells; Humans; Indoles; Maleimides; Membranes; Microscopy, Confocal; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Transport; Pyrrolidinones; Staurosporine | 2007 |
Diacylglycerol is required for the formation of COPI vesicles in the Golgi-to-ER transport pathway.
Topics: Animals; Biological Transport; Brefeldin A; Carrier Proteins; Cell Membrane; Chlorocebus aethiops; Coat Protein Complex I; COP-Coated Vesicles; COS Cells; Diglycerides; Endoplasmic Reticulum; Estrenes; Golgi Apparatus; GTPase-Activating Proteins; HeLa Cells; Humans; Phorbol 12,13-Dibutyrate; Propranolol; Pyrrolidinones; Rats; Receptors, Peptide; Signal Transduction | 2007 |
An optimized protein kinase C activating diacylglycerol combining high binding affinity (Ki) with reduced lipophilicity (log P).
Topics: Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Databases as Topic; Diglycerides; Enzyme Activation; Hydrogen Bonding; Kinetics; Models, Molecular; Molecular Conformation; Phorbol 12,13-Dibutyrate; Protein Conformation; Protein Kinase C; Protein Structure, Secondary; Recombinant Fusion Proteins; Structure-Activity Relationship; Transfection; Tryptophan; Tyrosine; Zinc Fingers | 2001 |