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phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide and bibp 3226

phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide has been researched along with bibp 3226 in 7 studies

Compound Research Comparison

Studies
(phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide)
Trials
(phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide)
Recent Studies (post-2010)
(phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide)
Studies
(bibp 3226)
Trials
(bibp 3226)
Recent Studies (post-2010) (bibp 3226)
276055248054
705248054

Protein Interaction Comparison

ProteinTaxonomyphenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide (IC50)bibp 3226 (IC50)
Neuropeptide Y receptor type 1Homo sapiens (human)0.0091

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (71.43)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adham, N; Artymyshyn, R; Bonini, JA; Borowsky, B; Boteju, LW; Boyle, N; Branchek, TA; Durkin, MM; Forray, C; Gerald, C; Jones, KA; Kouranova, EV; Lakhlani, PP; Ogozalek, KL; Quan, Y; Raddatz, R; Smith, KE; Tamm, JA; Vaysse, PJ; Wetzel, JM; Yao, WJ1
Chang, M; Chen, LX; Chen, Q; Fang, Q; Guo, J; Wang, R1
Chevé, G; McCurdy, CR; Mollereau, C; Vyas, N1
Chang, M; Fang, Q; Guo, J; He, F; Peng, YL; Wang, R1
Miyazaki, R; Yamada, T; Yamamoto, T1
Kakinuma, N; Kawate, T; Narita, K; Takeda, S1
Beck-Sickinger, AG; Findeisen, M; Meier, R; Meiler, J; Olsson, R; Rathmann, D; Würker, C1

Reviews

1 review(s) available for phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide and bibp 3226

ArticleYear
Structure-activity relationships of neuropeptide FF and related peptidic and non-peptidic derivatives.
    Peptides, 2006, Volume: 27, Issue:5

    Topics: Amino Acid Sequence; Animals; Arginine; CHO Cells; Cricetinae; Cricetulus; Humans; Oligopeptides; Peptide Fragments; Receptors, Neuropeptide; Structure-Activity Relationship

2006

Other Studies

6 other study(ies) available for phenylalanyl-leucyl-phenylalanyl-glutaminyl-prolyl-glutaminyl-arginyl-phenylalaninamide and bibp 3226

ArticleYear
Identification and characterization of two G protein-coupled receptors for neuropeptide FF.
    The Journal of biological chemistry, 2000, Dec-15, Volume: 275, Issue:50

    Topics: Amino Acid Sequence; Animals; Arginine; Binding Sites; Brain; Calcium; Chromosome Mapping; Cloning, Molecular; COS Cells; Cyclic AMP; DNA, Complementary; Electrophysiology; Gene Library; Humans; Kinetics; Ligands; Molecular Sequence Data; Oligopeptides; Oocytes; Phosphatidylinositols; Protein Binding; Protein Structure, Tertiary; Rats; Receptors, Cell Surface; Receptors, Neuropeptide; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution; Xenopus

2000
Neuropeptide FF receptors exert contractile activity via inhibition of nitric oxide release in the mouse distal colon.
    Peptides, 2005, Volume: 26, Issue:5

    Topics: Acetylcholine; Animals; Arginine; Biological Assay; Colon, Sigmoid; Enzyme Inhibitors; In Vitro Techniques; Mice; Muscle Contraction; Neuropeptides; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oligopeptides; Receptors, Neuropeptide

2005
In vivo inhibition of neuropeptide FF agonism by BIBP3226, an NPY Y1 receptor antagonist.
    Peptides, 2006, Volume: 27, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Arginine; Hypothermia; Male; Mice; Oligopeptides; Rats; Rats, Wistar; Receptors, Neuropeptide; Receptors, Neuropeptide Y; Tachycardia; Time Factors

2006
Intracerebroventricular administration of 26RFa produces an analgesic effect in the rat formalin test.
    Peptides, 2009, Volume: 30, Issue:9

    Topics: Analgesics, Non-Narcotic; Animals; Anti-Anxiety Agents; Arginine; Formaldehyde; Hot Temperature; Injections, Intraventricular; Male; Narcotic Antagonists; Neuropeptide Y; Neuropeptides; Oligopeptides; Pain; Pain Measurement; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, G-Protein-Coupled; Spinal Cord

2009
Multiple primary cilia modulate the fluid transcytosis in choroid plexus epithelium.
    Traffic (Copenhagen, Denmark), 2010, Volume: 11, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Arginine; Autocrine Communication; Base Sequence; Caco-2 Cells; Cattle; Cell Line, Tumor; Cerebrospinal Fluid; Choroid Plexus; Cilia; Cyclic AMP; Epithelium; Humans; Mice; Models, Biological; Molecular Sequence Data; Oligopeptides; Protein Transport; Rats; Receptors, Neuropeptide; Swine

2010
Selective mode of action of guanidine-containing non-peptides at human NPFF receptors.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Adamantane; Amino Acid Substitution; Animals; Arginine; Binding Sites; Biological Assay; Chlorocebus aethiops; COS Cells; Dipeptides; Drug Design; Guanidine; HEK293 Cells; Humans; Ligands; Microscopy, Fluorescence; Molecular Conformation; Peptidomimetics; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Structure-Activity Relationship

2012