phenylalanine and quinazolines

phenylalanine has been researched along with quinazolines in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19902 (11.76)18.7374
1990's1 (5.88)18.2507
2000's7 (41.18)29.6817
2010's6 (35.29)24.3611
2020's1 (5.88)2.80

Authors

AuthorsStudies
Gröger, D; Johne, S; Waiblinger, K1
Mothes, K1
Dreslin, JA; Grizzuti, K; Gros, P; Kajiji, S1
Abraham, JA; Clowes, AW; Daum, G; Kalmes, A; Vesti, BR1
Bode, AM; Chen, N; Dong, Z; Liu, G; Ma, WY; She, QB; Wu, E1
Enrich, C; Lladó, A; Tebar, F1
Barki-Harrington, L; El-Shewy, HM; Kelly, FL; Luttrell, LM1
Armstrong, C; Durkin, AJ; Osborne, DA; Rosemurgy, AS; Yeatman, TJ; Zervos, EE1
Casas-González, P; García-Sáinz, JA1
Fu, X; Ho, WT; Ishii, T; Li, Q; Li, Z; Xing, S; Xu, M; Zhao, ZJ1
Balghi, H; Carlile, GW; de Jonge, HR; Hanrahan, JW; Kus, B; Lesimple, P; Liao, J; Liu, N; Robert, R; Rotin, D; Scholte, BJ; Thomas, DY; Wilke, M1
Bear, CE; Huan, LJ; Kim Chiaw, P; Ramjeesingh, M; Wellhauser, L1
Cantrell, DA; Feijoo, C; Finlay, D; Macintyre, AN; Okkenhaug, K; Preston, G; Sinclair, LV; Tamas, P; Waugh, CM1
Alemi, F; Bunnett, NW; Canals, M; Corvera, CU; Cottrell, GS; Godfrey, CB; Jensen, DD; Kocan, M; Korbmacher, C; Lambert, NA; Murphy, JE; Niklas, C; Poole, DP1
Cho-Clark, M; Larco, DO; Mani, SK; Semsarzadeh, NN; Vasta, F; Wu, TJ1
Al-Kali, A; Cherry, M; Ghabache, B; Khawandanah, M; Ozer, H; Selby, G; Srour, S; Zhao, ZJ1
Fukase, H; Furuie, H; Ikeda, N; Kajioka, T; Oikawa, I1

Trials

2 trial(s) available for phenylalanine and quinazolines

ArticleYear
Erlotinib is not effective in patients with JAK2V617F-positive polycythemia vera.
    Annals of hematology, 2015, Volume: 94, Issue:4

    Topics: Adult; Aged; Amino Acid Substitution; Antineoplastic Agents; Drug-Related Side Effects and Adverse Reactions; Erlotinib Hydrochloride; Female; Humans; Janus Kinase 2; Male; Middle Aged; Phenylalanine; Polycythemia Vera; Quinazolines; Treatment Outcome; Valine

2015
Food Effect on a Single High Dose of Carotegrast Methyl, an Oral Antagonist of α4-Integrin, in Healthy Male Subjects: A Randomised, Placebo-Controlled, Double-Blind Study.
    Clinical drug investigation, 2020, Volume: 40, Issue:3

    Topics: Administration, Oral; Adult; Area Under Curve; Cross-Over Studies; Double-Blind Method; Fasting; Food-Drug Interactions; Humans; Integrin alpha4; Male; Phenylalanine; Quinazolines; Quinazolinones; Young Adult

2020

Other Studies

15 other study(ies) available for phenylalanine and quinazolines

ArticleYear
[Biosynthesis of the quinazoline alkaloid arborine].
    European journal of biochemistry, 1970, Volume: 15, Issue:3

    Topics: Alkaloids; Carbon Isotopes; Methionine; Nitrogen; ortho-Aminobenzoates; Phenylalanine; Plants; Quinazolines; Radioisotopes; Tritium

1970
[Alkaloids in the metabolism of plants].
    Experientia, 1969, Mar-15, Volume: 25, Issue:3

    Topics: Alkaloids; Dopamine; Indoles; Isoquinolines; Mevalonic Acid; ortho-Aminobenzoates; Papaver; Penicillium; Phenylalanine; Pipecolic Acids; Plants, Medicinal; Pregnenolone; Quinazolines; Sparteine; Terpenes; Tryptophan; Tyrosine

1969
Structurally distinct MDR modulators show specific patterns of reversal against P-glycoproteins bearing unique mutations at serine939/941.
    Biochemistry, 1994, May-03, Volume: 33, Issue:17

    Topics: Amino Acid Sequence; Animals; Cell Survival; CHO Cells; Clone Cells; Cricetinae; Cyclosporine; Dibenzocycloheptenes; Drug Resistance; Glycoproteins; Isoquinolines; Mice; Phenylalanine; Point Mutation; Quinazolines; Quinolines; Recombinant Proteins; Serine; Transfection; Vinblastine

1994
Heparin blockade of thrombin-induced smooth muscle cell migration involves inhibition of epidermal growth factor (EGF) receptor transactivation by heparin-binding EGF-like growth factor.
    Circulation research, 2000, Jul-21, Volume: 87, Issue:2

    Topics: Animals; Anticoagulants; Aorta; Becaplermin; Cell Line; Cell Movement; Cells, Cultured; Epidermal Growth Factor; ErbB Receptors; Heparin; Heparin-binding EGF-like Growth Factor; Humans; Intercellular Signaling Peptides and Proteins; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Papio; Phenylalanine; Phosphorylation; Platelet-Derived Growth Factor; Protease Inhibitors; Proto-Oncogene Proteins c-sis; Quinazolines; Rats; Rats, Inbred F344; Signal Transduction; Thiophenes; Thrombin; Tyrphostins

2000
Transactivation of the epidermal growth factor receptor is involved in 12-O-tetradecanoylphorbol-13-acetate-induced signal transduction.
    The Journal of biological chemistry, 2001, Dec-14, Volume: 276, Issue:50

    Topics: Animals; Carcinogens; Cell Transformation, Neoplastic; Cells, Cultured; DNA; Dose-Response Relationship, Drug; Embryo, Mammalian; Enzyme Inhibitors; ErbB Receptors; Ligands; Mice; Mitogen-Activated Protein Kinases; Models, Biological; Phenylalanine; Phosphorylation; Protein Binding; Protein Structure, Tertiary; Quinazolines; Signal Transduction; Tetradecanoylphorbol Acetate; Thiophenes; Transcription Factor AP-1; Transcriptional Activation; Tyrphostins

2001
Role of calmodulin in the modulation of the MAPK signalling pathway and the transactivation of epidermal growth factor receptor mediated by PKC.
    FEBS letters, 2002, Apr-24, Volume: 517, Issue:1-3

    Topics: Animals; Calmodulin; Chlorocebus aethiops; COS Cells; Enzyme Activation; Enzyme Inhibitors; ErbB Receptors; Mitogen-Activated Protein Kinases; Phenylalanine; Protein Kinase C; Quinazolines; ras Proteins; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thiophenes; Transcriptional Activation; Tyrphostins

2002
Ectodomain shedding-dependent transactivation of epidermal growth factor receptors in response to insulin-like growth factor type I.
    Molecular endocrinology (Baltimore, Md.), 2004, Volume: 18, Issue:11

    Topics: Animals; Cell Line; Chlorocebus aethiops; Endocytosis; ErbB Receptors; Humans; Insulin-Like Growth Factor I; Metalloendopeptidases; Mice; Mitogen-Activated Protein Kinase 3; Paracrine Communication; Phenylalanine; Phosphorylation; Quinazolines; Rats; Receptors, Somatomedin; Tetradecanoylphorbol Acetate; Thiophenes; Tyrosine; Tyrphostins

2004
EGF receptor antagonism improves survival in a murine model of pancreatic adenocarcinoma.
    The Journal of surgical research, 2006, Volume: 135, Issue:1

    Topics: Adenocarcinoma; Animals; Cell Division; Cell Line, Tumor; Disease Models, Animal; ErbB Receptors; Erlotinib Hydrochloride; Gene Expression; Humans; Mice; Mice, Nude; Pancreatic Neoplasms; Phenylalanine; Protease Inhibitors; Protein Kinase Inhibitors; Quinazolines; Survival Rate; Thiophenes

2006
Role of epidermal growth factor receptor transactivation in alpha1B-adrenoceptor phosphorylation.
    European journal of pharmacology, 2006, Aug-07, Volume: 542, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Androstadienes; Animals; Antibodies; Cell Line; Cricetinae; Dose-Response Relationship, Drug; Endothelin-1; Epidermal Growth Factor; ErbB Receptors; Heparin-binding EGF-like Growth Factor; Intercellular Signaling Peptides and Proteins; Norepinephrine; Phenylalanine; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Quinazolines; Rats; Receptors, Adrenergic, alpha-1; Tetradecanoylphorbol Acetate; Thiophenes; Tyrphostins; Wortmannin

2006
Erlotinib effectively inhibits JAK2V617F activity and polycythemia vera cell growth.
    The Journal of biological chemistry, 2007, Feb-09, Volume: 282, Issue:6

    Topics: Amino Acid Substitution; Animals; Cell Line, Tumor; Cell Proliferation; Drug Delivery Systems; Enzyme Activation; Erlotinib Hydrochloride; Growth Inhibitors; Hematopoietic Stem Cells; Humans; Janus Kinase 2; Jurkat Cells; Mice; Phenylalanine; Polycythemia Vera; Protein Kinase Inhibitors; Quinazolines; Valine

2007
Correction of the Delta phe508 cystic fibrosis transmembrane conductance regulator trafficking defect by the bioavailable compound glafenine.
    Molecular pharmacology, 2010, Volume: 77, Issue:6

    Topics: Analgesics, Non-Narcotic; Animals; Biological Availability; Blotting, Western; Cell Line; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; Glafenine; Humans; Phenylalanine; Piperazines; Protein Transport; Quinazolines; Spectrometry, Fluorescence

2010
A chemical corrector modifies the channel function of F508del-CFTR.
    Molecular pharmacology, 2010, Volume: 78, Issue:3

    Topics: Animals; Cricetinae; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Mutation; Phenylalanine; Piperazines; Protein Transport; Quinazolines; Sequence Deletion

2010
Protein kinase B controls transcriptional programs that direct cytotoxic T cell fate but is dispensable for T cell metabolism.
    Immunity, 2011, Feb-25, Volume: 34, Issue:2

    Topics: 3-Phosphoinositide-Dependent Protein Kinases; Adenine; Animals; Cell Division; Cell Movement; Class I Phosphatidylinositol 3-Kinases; Cytotoxicity, Immunologic; Gene Expression Regulation; Glucose; Interferon-gamma; Interleukin-2; Mice; Mice, Inbred C57BL; Mice, Transgenic; Phenylalanine; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pore Forming Cytotoxic Proteins; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-akt; Quinazolines; Receptors, Antigen, T-Cell; Receptors, Cytokine; T-Lymphocytes, Cytotoxic; Transcription, Genetic

2011
The bile acid receptor TGR5 does not interact with β-arrestins or traffic to endosomes but transmits sustained signals from plasma membrane rafts.
    The Journal of biological chemistry, 2013, Aug-09, Volume: 288, Issue:32

    Topics: Antineoplastic Agents; Arrestins; beta-Arrestin 1; beta-Arrestin 2; beta-Arrestins; beta-Cyclodextrins; Cholagogues and Choleretics; Cyclic AMP; Deoxycholic Acid; Endocytosis; Endosomes; Enzyme Inhibitors; ErbB Receptors; G-Protein-Coupled Receptor Kinase 2; G-Protein-Coupled Receptor Kinase 5; HEK293 Cells; Humans; Membrane Microdomains; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Oleanolic Acid; Phenylalanine; Protein Transport; Quinazolines; Receptors, G-Protein-Coupled; Thiophenes; Tyrphostins

2013
GnRH-(1-5) transactivates EGFR in Ishikawa human endometrial cells via an orphan G protein-coupled receptor.
    Molecular endocrinology (Baltimore, Md.), 2014, Volume: 28, Issue:1

    Topics: Calcium Signaling; Cell Line, Tumor; Cell Movement; Endometrial Neoplasms; Epidermal Growth Factor; ErbB Receptors; Female; Gene Expression; Gonadotropin-Releasing Hormone; Humans; Matrix Metalloproteinase Inhibitors; Oligopeptides; Oncogene Proteins; Peptide Fragments; Phenylalanine; Phosphorylation; Protein Processing, Post-Translational; Pyrrolidonecarboxylic Acid; Quinazolines; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, LHRH; Thiophenes; Transcriptional Activation; Tyrphostins

2014