Page last updated: 2024-08-23

phenyl acetate and repaglinide

phenyl acetate has been researched along with repaglinide in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Backman, JT; Kajosaari, LI; Neuvonen, PJ; Niemi, M1
Foti, RS; Rock, DA; VandenBrink, BM; Wahlstrom, JL; Wienkers, LC1
Goda, H; Ito, K; Komatsu, S; Kudo, T; Tanaka, R; Yokosuka, Y1
Mahajan, AN; Patel, A; Patel, D; Surti, N; Surti, Z1

Trials

1 trial(s) available for phenyl acetate and repaglinide

ArticleYear
Telithromycin, but not montelukast, increases the plasma concentrations and effects of the cytochrome P450 3A4 and 2C8 substrate repaglinide.
    Clinical pharmacology and therapeutics, 2006, Volume: 79, Issue:3

    Topics: Acetates; Adolescent; Adult; Area Under Curve; Aryl Hydrocarbon Hydroxylases; Biotransformation; Blood Glucose; Carbamates; Cross-Over Studies; Cyclopropanes; Cytochrome P-450 CYP2C8; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Drug Interactions; Female; Humans; Hypoglycemic Agents; Ketolides; Leukotriene Antagonists; Male; Piperidines; Quinolines; Sulfides

2006

Other Studies

3 other study(ies) available for phenyl acetate and repaglinide

ArticleYear
Evaluation of CYP2C8 inhibition in vitro: utility of montelukast as a selective CYP2C8 probe substrate.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:9

    Topics: Acetates; Amodiaquine; Aryl Hydrocarbon Hydroxylases; Binding Sites; Carbamates; Cyclopropanes; Cytochrome P-450 CYP2C8; Drug Interactions; Humans; Microsomes, Liver; Paclitaxel; Piperidines; Quinolines; Rosiglitazone; Sensitivity and Specificity; Substrate Specificity; Sulfides; Thiazolidinediones

2011
Estimation of the Contribution of CYP2C8 and CYP3A4 in Repaglinide Metabolism by Human Liver Microsomes Under Various Buffer Conditions.
    Journal of pharmaceutical sciences, 2017, Volume: 106, Issue:9

    Topics: Acetates; Buffers; Carbamates; Cyclopropanes; Cytochrome P-450 CYP2C8; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inducers; Cytochrome P-450 Enzyme Inhibitors; Drug Interactions; Humans; Hypoglycemic Agents; Ketoconazole; Microsomes, Liver; Piperidines; Quinolines; Sulfides

2017
Spray dried solid dispersion of repaglinide using hypromellose acetate succinate:
    Drug development and industrial pharmacy, 2020, Volume: 46, Issue:10

    Topics: Acetates; Animals; Carbamates; Chemistry, Pharmaceutical; Hypromellose Derivatives; Pharmaceutical Preparations; Piperidines; Rats; Solubility; Succinates

2020