Compounds > phentolamine
Page last updated: 2024-08-17

phentolamine and rx 821002

phentolamine has been researched along with rx 821002 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (60.00)18.2507
2000's3 (30.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Denis-Pouxviel, C; Devedjian, JC; Esclapez, F; Paris, H1
Harms, GS; Lohse, MJ; Steinmeyer, R; Vilardaga, JP1
Leslie, FM; Raymon, HK; Smith, TD1
Czerwiec, E; De Backer, JP; De Potter, W; De Vos, H; Vauquelin, G1
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D1
Coupar, IM; Liu, L1
Caramona, MM; Figueiredo, IV; Guimarães, S; Moura, D; Paiva, MQ1
Berlan, M; Crampes, F; Daviaud, D; Gesta, S; Hejnova, J; Saulnier-Blache, JS; Stich, V; Valet, P1
Fagerholm, V; Hein, L; Philipp, M; Scheinin, M1
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB1

Other Studies

10 other study(ies) available for phentolamine and rx 821002

ArticleYear
Further characterization of human alpha 2-adrenoceptor subtypes: [3H]RX821002 binding and definition of additional selective drugs.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Line; Dioxanes; Humans; Idazoxan; Plasmids; Radioligand Assay; Receptors, Adrenergic, alpha; Transfection

1994
Molecular basis of inverse agonism in a G protein-coupled receptor.
    Nature chemical biology, 2005, Volume: 1, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Cell Line; Fluorescence Resonance Energy Transfer; Humans; Ligands; Protein Binding; Receptors, Adrenergic, alpha-2; Receptors, G-Protein-Coupled; Signal Transduction

2005
Further pharmacological characterization of [3H]idazoxan binding sites in rat brain: evidence for predominant labeling of alpha 2-adrenergic receptors.
    Brain research, 1992, Jun-12, Volume: 582, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Buffers; Dioxanes; Epinephrine; Idazoxan; Male; Phentolamine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Drug; Tritium; Yohimbine

1992
[3H]rauwolscine behaves as an agonist for the 5-HT1A receptors in human frontal cortex membranes.
    European journal of pharmacology, 1991, May-25, Volume: 207, Issue:1

    Topics: Adrenergic alpha-Antagonists; Aged; Dioxanes; Frontal Lobe; GTP-Binding Proteins; Guanine Nucleotides; Humans; Idazoxan; In Vitro Techniques; Kinetics; Membranes; Middle Aged; Mollusk Venoms; Phentolamine; Receptors, Adrenergic, alpha; Receptors, Serotonin; Yohimbine

1991
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
    Biochemical pharmacology, 1990, Aug-01, Volume: 40, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1990
Characterisation of pre- and post-synaptic alpha-adrenoceptors in modulation of the rat ileum longitudinal and circular muscle activities.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brimonidine Tartrate; Clonidine; Electric Stimulation; Idazoxan; Ileum; In Vitro Techniques; Muscle Contraction; Oxymetazoline; Phentolamine; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Receptors, Presynaptic

1997
Prejunctional alpha2A-autoreceptors in the human gastric and ileocolic arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Arteries; Autoreceptors; Colon; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Mucosa; Humans; Idazoxan; Ileum; In Vitro Techniques; Male; Middle Aged; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha-2; Spiro Compounds; Stomach; Tritium; Yohimbine

1998
In vitro and in vivo impairment of alpha2-adrenergic receptor-dependent antilipolysis by fatty acids in human adipose tissue.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2001, Volume: 33, Issue:12

    Topics: Adipocytes; Adipose Tissue; Adrenergic Agents; Adult; Biopsy, Needle; Dietary Fats; Dose-Response Relationship, Drug; Epinephrine; Exercise; Fatty Acids; Female; Gene Expression; Glycerol; GTP-Binding Proteins; Humans; Idazoxan; Isoproterenol; Lipolysis; Middle Aged; Palmitates; Phentolamine; Receptors, Adrenergic, alpha-2

2001
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Cerebral Cortex; Idazoxan; In Vitro Techniques; Isoquinolines; Ligands; Mice; Mice, Knockout; Naphthyridines; Oxymetazoline; Phentolamine; Prazosin; Putamen; Radioligand Assay; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2004
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
    British journal of pharmacology, 2012, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei

2012