Page last updated: 2024-08-17

phentolamine and oxymetazoline

phentolamine has been researched along with oxymetazoline in 58 studies

Research

Studies (58)

TimeframeStudies, this research(%)All Research%
pre-199039 (67.24)18.7374
1990's13 (22.41)18.2507
2000's5 (8.62)29.6817
2010's1 (1.72)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Timmermans, PB; van Zwieten, PA1
Foglar, R; Horie, K; Obika, K; Ogawa, S; Sakamoto, A; Shibata, K; Tsujimoto, G1
Bondinell, WE; Hieble, JP; Ruffolo, RR1
Harms, GS; Lohse, MJ; Steinmeyer, R; Vilardaga, JP1
Agbaba, D; Filipic, S; Nikolic, K1
Handzlik, J; Jankowska, A; Jastrzębska-Więsek, M; Kieć-Kononowicz, K; Kucwaj-Brysz, K; Kurczab, R; Nitek, W; Partyka, A; Satała, G; Siwek, A; Wesołowska, A; Żesławska, E1
Chan, CC; Kalsner, S1
Ganong, WF; Morris, BJ; Reid, IA1
Dismukes, RK; Mulder, AH1
de Boer, AA; Dismukes, K; Mulder, AH1
Synder, SH; U'Prichard, DC1
de Langen, CD; de Regt, V; Hogenboom, F; Mulder, AH1
Brown, DA; Caulfield, MP1
Miller, DD; Patil, PN; Sanders, J1
Wikberg, J1
Endoh, M; Schümann, HJ1
Ruffolo, RR1
Hoyer, D; Schoeffter, P1
Chandranath, SI; Gokhale, SD; Sharif, SI1
Hadjiconstantinou, M; Krajnc, D; Neff, NH; Rossetti, Z1
Drukarch, B; Heimans, JJ; Schepens, E; Stoof, JC1
Cervenko, FW; Loomis, CW; Milne, B; Sherman, SE1
Nobin, A; Owman, C; Törnebrandt, K1
Dickinson, KE; McKernan, RM; Miles, CM; Sever, PS1
Cools, AR1
Cools, AR; Ellenbroek, BA; Gispen, WH; Spruijt, BM1
Cervenko, F; Loomis, C; Milne, B; Sherman, S1
Coats, RA1
Montel, H; Starke, K5
Starke, K1
Altmann, KP; Starke, K1
Reinhardt, D; Wagner, J1
Endo, M; Schümann, HJ; Wagner, J1
Görlitz, BD; Montel, H; Schümann, HJ; Starke, K1
Farmer, JB; Kennedy, I; Levy, GP; Marshall, RJ1
Broekkamp, C; van Rossum, JM1
Cavero, I; Gomeni, R; Lefèvre-Borg, F; Roach, AG1
Armstrong, JM; Cavero, I; Lefèvre-Borg, F; Scatton, B1
Carpenter, CA; Saggerson, ED1
Fuder, H; Muscholl, E; Spemann, R1
Robie, NW1
Brown, DR; Malone, ED; Trent, AM; Turner, TA1
Göthert, M; Molderings, GJ1
Coupar, IM; Liu, L1
Dan, K; Hirose, H; Maruyama, H; Nakamura, K; Saruta, T; Seto, Y1
Duda, T; Sharma, RK; Venkataraman, V1
Hogenboom, F; Mulder, AH; Schoffelmeer, AN; van Royen, DE; Vanderschuren, LJ; Wardeh, G1
Arimitsu, M; Karaki, H; Koga, Y; Mitsui-Saito, M; Ozaki, H; Sato, K1
Abe, M; Hikasa, Y; Hisashi, Y; Matsuda, H; Ogasawara, S; Satoh, T1
Keef, KD; Mutafova-Yambolieva, VN1
García-Sáinz, JA; González-Espinosa, C; González-Espinosa, D; Mora-Rodríguez, DM; Romero-Avila, MT1
Fagerholm, V; Hein, L; Philipp, M; Scheinin, M1

Reviews

3 review(s) available for phentolamine and oxymetazoline

ArticleYear
alpha 2 adrenoceptors: classification, localization, mechanisms, and targets for drugs.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:12

    Topics: Adipose Tissue; Animals; Blood Platelets; Central Nervous System; Humans; Islets of Langerhans; Melanocytes; Muscle, Smooth, Vascular; Nerve Endings; Norepinephrine; Parasympathetic Nervous System; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Serotonin; Synapses

1982
Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Humans; Molecular Biology; Molecular Structure; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1995
Fundamentals of receptor theory: basics for shock research.
    Circulatory shock, 1992, Volume: 37, Issue:2

    Topics: Binding, Competitive; Drug Design; Naphazoline; Oxymetazoline; Phentolamine; Phenylephrine; Receptors, Adrenergic; Research Design; Shock, Septic; Signal Transduction; Therapeutic Equivalency

1992

Other Studies

55 other study(ies) available for phentolamine and oxymetazoline

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
KMD-3213, a novel, potent, alpha 1a-adrenoceptor-selective antagonist: characterization using recombinant human alpha 1-adrenoceptors and native tissues.
    Molecular pharmacology, 1995, Volume: 48, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Calcium; Cell Line; CHO Cells; Clonidine; Cloning, Molecular; Cricetinae; Humans; Indoles; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Sulfonamides; Tamsulosin

1995
Molecular basis of inverse agonism in a G protein-coupled receptor.
    Nature chemical biology, 2005, Volume: 1, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Cell Line; Fluorescence Resonance Energy Transfer; Humans; Ligands; Protein Binding; Receptors, Adrenergic, alpha-2; Receptors, G-Protein-Coupled; Signal Transduction

2005
QSAR study of imidazoline antihypertensive drugs.
    Bioorganic & medicinal chemistry, 2008, Aug-01, Volume: 16, Issue:15

    Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2008
Computer-aided insights into receptor-ligand interaction for novel 5-arylhydantoin derivatives as serotonin 5-HT
    European journal of medicinal chemistry, 2018, Mar-10, Volume: 147

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Computer-Aided Design; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Hydantoins; Male; Mice; Models, Molecular; Molecular Structure; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

2018
Adrenergic antagonists and the presynaptic receptor hypothesis in vascular tissue.
    The Journal of pharmacology and experimental therapeutics, 1979, Volume: 211, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Muscle, Smooth, Vascular; Oxymetazoline; Phenoxybenzamine; Phentolamine; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Yohimbine

1979
Inhibition by alpha-adrenoceptor agonists of renin release in vitro.
    European journal of pharmacology, 1979, Oct-26, Volume: 59, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Depression, Chemical; Epinephrine; In Vitro Techniques; Isoproterenol; Kidney; Male; Methoxamine; Norepinephrine; Oxymetazoline; Phentolamine; Phenylephrine; Propranolol; Rats; Renin

1979
Cyclic AMP and alpha-receptor-mediated modulation of noradrenaling release from rat brain slices.
    European journal of pharmacology, 1976, Volume: 39, Issue:2

    Topics: Animals; Brain; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Male; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Phentolamine; Phosphodiesterase Inhibitors; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synaptic Transmission; Xanthines

1976
On the mechanism of alpha-receptor mediated modulation of 3H-noradrenaline release from slices of rat brain neocortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 299, Issue:2

    Topics: Animals; Cerebral Cortex; Electric Stimulation; In Vitro Techniques; Male; Norepinephrine; Oxymetazoline; Phentolamine; Potassium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Stimulation, Chemical

1977
Differential labelling of alpha and beta-noradrenergic receptors in calf cerebellum membranes with 3H-adrenaline.
    Nature, 1977, Nov-17, Volume: 270, Issue:5634

    Topics: Animals; Binding, Competitive; Cattle; Cerebellar Cortex; Epinephrine; Kinetics; Oxymetazoline; Phentolamine; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1977
Alpha-receptor-mediated modulation of 3H-noradrenaline release from rat brain cortex synaptosomes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1978, Volume: 303, Issue:2

    Topics: Animals; Brain; Desipramine; In Vitro Techniques; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synaptosomes; Time Factors; Yohimbine

1978
Hyperpolarizing 'alpha 2'-adrenoceptors in rat sympathetic ganglia.
    British journal of pharmacology, 1979, Volume: 65, Issue:3

    Topics: Animals; Catecholamines; Clonidine; Ganglia, Autonomic; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Oxymetazoline; Phentolamine; Propranolol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Dopamine; Time Factors

1979
Alpha adrenergic and histaminergic effects of tolazoline-like imidazolines.
    The Journal of pharmacology and experimental therapeutics, 1975, Volume: 195, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Chlorpheniramine; Guinea Pigs; Heart Atria; Histamine; Imidazoles; In Vitro Techniques; Metiamide; Muscle Contraction; Myocardial Contraction; Oxymetazoline; Phentolamine; Phenylephrine; Propranolol; Rabbits; Reserpine; Tolazoline

1975
Differentiation between pre- and postjunctional alpha-receptors in guinea pig ileum and rabbit aorta.
    Acta physiologica Scandinavica, 1978, Volume: 103, Issue:3

    Topics: Animals; Aorta, Thoracic; Cimetidine; Clonidine; Dibenzylchlorethamine; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Oxymetazoline; Parasympathetic Nervous System; Phenoxybenzamine; Phentolamine; Phenylephrine; Rabbits; Receptors, Adrenergic; Tolazoline

1978
Frequency-dependence of the positive inotropic effect of methoxamine and naphazoline mediated by alpha-Adrenoceptors in the isolated rabbit papillary muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 287, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Electric Stimulation; Imidazoles; In Vitro Techniques; Methoxamine; Myocardial Contraction; Naphazoline; Oxymetazoline; Papaverine; Papillary Muscles; Phentolamine; Rabbits; Receptors, Adrenergic; Stimulation, Chemical

1975
Interaction of the alpha-adrenoceptor agonist oxymetazoline with serotonin 5-HT1A, 5-HT1B, 5-HT1C and 5-HT1D receptors.
    European journal of pharmacology, 1991, Apr-17, Volume: 196, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Brain; Cattle; Clonidine; In Vitro Techniques; Kinetics; Methiothepin; Oxymetazoline; Phentolamine; Rats; Receptors, Serotonin; Swine

1991
Pharmacological characterization of the postjunctional alpha-adrenoceptors of the rat isolated seminal vesicle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Naphazoline; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Phentolamine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Seminal Vesicles; Yohimbine

1990
Modulation of retinal aromatic L-amino acid decarboxylase via alpha 2 adrenoceptors.
    Journal of neurochemistry, 1989, Volume: 52, Issue:2

    Topics: Animals; Aromatic-L-Amino-Acid Decarboxylases; Clonidine; Cycloheximide; Darkness; Dihydroxyphenylalanine; Kinetics; Light; Male; Oxymetazoline; Phentolamine; Piperoxan; Pyridoxal Phosphate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Retina; Yohimbine

1989
Alpha 2-adrenoceptor-mediated modulation of noradrenaline release is decreased in vas deferens but not in cerebral cortex of diabetic rats.
    Journal of the neurological sciences, 1989, Volume: 91, Issue:3

    Topics: Animals; Cerebral Cortex; Diabetes Mellitus, Experimental; Electric Stimulation; In Vitro Techniques; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Streptozocin; Vas Deferens

1989
Intrathecal oxymetazoline produces analgesia via spinal alpha-adrenoceptors and potentiates spinal morphine.
    European journal of pharmacology, 1988, Apr-13, Volume: 148, Issue:3

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Drug Synergism; Imidazoles; Injections, Intravenous; Injections, Spinal; Male; Morphine; Oxymetazoline; Phentolamine; Rats; Receptors, Adrenergic, alpha; Spinal Cord

1988
Pharmacological characterization of alpha-adrenergic receptor subtypes mediating contraction in human mesenteric arteries and veins.
    Blood vessels, 1985, Volume: 22, Issue:4

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Clonidine; Drug Interactions; Female; Humans; Male; Mesenteric Arteries; Mesenteric Veins; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxymetazoline; Phentolamine; Prazosin; Vasodilation; Yohimbine

1985
Heterogeneity between soluble human and rabbit splenic alpha 2-adrenoceptors.
    Biochemical pharmacology, 1986, Oct-15, Volume: 35, Issue:20

    Topics: Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; Lectins; Oxymetazoline; Phentolamine; Prazosin; Quinolizines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Solubility; Spleen; Sulfhydryl Reagents; Yohimbine

1986
Morphine and specific changes in the sensitivity of noradrenergic receptors within the "limbic" part of the feline caudate nucleus: a behaviour study.
    Brain research bulletin, 1985, Volume: 14, Issue:3

    Topics: Animals; Cats; Caudate Nucleus; Drug Interactions; Female; Limbic System; Male; Morphine; Oxymetazoline; Phentolamine; Receptors, Adrenergic; Time Factors

1985
Dopaminergic modulation of ACTH-induced grooming.
    European journal of pharmacology, 1986, Jan-29, Volume: 120, Issue:3

    Topics: Adrenocorticotropic Hormone; Animals; Apomorphine; Catheterization; Desipramine; Ergotamine; Grooming; Haloperidol; Male; Nucleus Accumbens; Oxymetazoline; Periaqueductal Gray; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra

1986
Prolonged spinal analgesia in the rat with the alpha-adrenoceptor agonist oxymetazoline.
    European journal of pharmacology, 1987, Aug-04, Volume: 140, Issue:1

    Topics: Anesthesia, Spinal; Animals; Dose-Response Relationship, Drug; Imidazoles; Male; Oxymetazoline; Phentolamine; Rats; Rats, Inbred Strains; Reaction Time

1987
The effects of adrenoceptor agonists and antagonists on plasma potassium concentration in anaesthetized guinea-pigs, rabbits and rats.
    British journal of pharmacology, 1985, Volume: 86, Issue:4

    Topics: Anesthesia; Angiotensin II; Animals; Apamin; Blood Pressure; Epinephrine; Ethanolamines; Guinea Pigs; Isoproterenol; Male; Methoxamine; Oxymetazoline; Phentolamine; Phenylephrine; Potassium; Propranolol; Rabbits; Rats; Rats, Inbred Strains; Species Specificity; Sympatholytics; Sympathomimetics

1985
Alpha-receptor-mediated modulation of transmitter release from central noradrenergic neurones.
    Naunyn-Schmiedeberg's archives of pharmacology, 1973, Volume: 279, Issue:1

    Topics: Animals; Cerebral Cortex; Cocaine; Cresols; Feedback; Imidazoles; In Vitro Techniques; Male; Nasal Decongestants; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Phentolamine; Rats; Receptors, Adrenergic; Sensory Receptor Cells; Synaptic Transmission; Tritium

1973
Letter: Interaction between indomethacin, oxymetazoline and phentolamine on the release of (3H)noradrenaline from brain slices.
    The Journal of pharmacy and pharmacology, 1973, Volume: 25, Issue:9

    Topics: Animals; Brain; Imidazoles; In Vitro Techniques; Indomethacin; Nasal Decongestants; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Tritium

1973
Proceedings: Influence of oxymetazoline and phentolamine on noradrenaline (NA) release caused by electrical stimulation, potassium, tyramine and dimethylphenylpiperazine (DMPP).
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:Suppl

    Topics: Action Potentials; Animals; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Ganglionic Stimulants; Heart; Imidazoles; In Vitro Techniques; Myocardium; Nasal Decongestants; Neurons; Norepinephrine; Oxymetazoline; Perfusion; Phentolamine; Piperazines; Potassium; Rabbits; Sympathetic Nervous System; Tritium; Tyramine

1974
Inhibition of adrenergic neurotransmission by clonidine: an action on prejunctional -receptors.
    Neuropharmacology, 1973, Volume: 12, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Cocaine; Heart; In Vitro Techniques; Mathematics; Oxymetazoline; Phenoxybenzamine; Phentolamine; Rabbits; Receptors, Adrenergic; Sympathetic Nervous System; Synaptic Transmission

1973
Characterization of the adrenoceptors mediating the positive ino- and chronotropic effect of phenylephrine on isolated atria from guinea pigs and rabbits by means of adrenolytic drugs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Guinea Pigs; Heart; Heart Atria; Heart Rate; In Vitro Techniques; Male; Methoxamine; Naphazoline; Oxymetazoline; Perfusion; Phentolamine; Phenylephrine; Pindolol; Rabbits; Receptors, Adrenergic; Reserpine; Stimulation, Chemical

1974
Positive inotropic effects of phenylephrine in the isolated rabbit papillary muscle mediated both by alpha- and beta-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 284, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Depression, Chemical; Epinephrine; Heart; In Vitro Techniques; Isoproterenol; Methoxamine; Muscles; Naphazoline; Norepinephrine; Oxymetazoline; Papaverine; Papillary Muscles; Phentolamine; Phenylephrine; Phosphodiesterase Inhibitors; Pindolol; Rabbits; Receptors, Adrenergic; Reserpine; Stimulation, Chemical; Theophylline

1974
Local alpha-adrenoceptor mediated feed-back inhibition of catecholamine release from the adrenal medulla?
    Experientia, 1974, Oct-15, Volume: 30, Issue:10

    Topics: Adrenal Medulla; Adrenergic alpha-Antagonists; Animals; Catecholamines; Cattle; Desipramine; Feedback; Imidazoles; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Phentolamine; Potassium; Receptors, Adrenergic; Stimulation, Chemical

1974
Sympathomimetic inhibition of noradrenaline release: mediated by prostaglandins?
    Naunyn-Schmiedeberg's archives of pharmacology, 1973, Volume: 278, Issue:1

    Topics: Animals; Feedback; Heart; Indomethacin; Myocardium; Norepinephrine; Oxymetazoline; Perfusion; Phentolamine; Prostaglandins; Rabbits; Sympathetic Nervous System

1973
Pharmacology of AH 5158; a drug which blocks both - and -adrenoceptors.
    British journal of pharmacology, 1972, Volume: 45, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Cardiac Output; Catecholamines; Cocaine; Dogs; Ethanolamines; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Mesenteric Veins; Norepinephrine; Ouabain; Oxymetazoline; Phentolamine; Propranolol; Propylamines; Rats; Salicylamides; Trachea; Vas Deferens

1972
Influence of drugs with affinity for alpha-adrenoceptors on noradrenaline release by potassium, tyramine and dimethylphenylpiperazinium.
    European journal of pharmacology, 1974, Volume: 27, Issue:3

    Topics: Animals; Depression, Chemical; Dimethylphenylpiperazinium Iodide; Fluorometry; Heart; In Vitro Techniques; Myocardium; Neurons; Norepinephrine; Oxymetazoline; Perfusion; Phentolamine; Piperazines; Potassium; Rabbits; Receptors, Adrenergic; Stimulation, Chemical; Time Factors; Tritium; Tyramine

1974
Clonidine induced intrahypothalamic stimulation of eating in rats.
    Psychopharmacologia, 1972, Volume: 25, Issue:2

    Topics: Animals; Antihypertensive Agents; Behavior, Animal; Feeding Behavior; Food Deprivation; Hypothalamus; Imidazoles; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Receptors, Drug; Stereotaxic Techniques; Stimulation, Chemical

1972
Alpha-receptors regulate transmitter release from central monoamine neurones.
    Die Naturwissenschaften, 1973, Volume: 60, Issue:7

    Topics: Animals; Brain; Cocaine; Electric Stimulation; Feedback; In Vitro Techniques; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Receptors, Adrenergic; Serotonin; Tritium

1973
Pharmacological evidence favoring a similarity between alpha adrenoceptors mediating sleep in chicks and cardiac presynaptic alpha-2 receptors in rats.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Chickens; Clonidine; Guanfacine; Guanidines; Heart; Heart Rate; Male; Methoxamine; Nordefrin; Oxymetazoline; Phentolamine; Phenylacetates; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Sleep; Xylazine; Yohimbine

1982
Urethane inhibits cardiovascular responses mediated by the stimulation of alpha-2 adrenoceptors in the rat.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:2

    Topics: Adrenalectomy; Adrenergic alpha-Agonists; Animals; Clonidine; Epinephrine; Heart Rate; Kinetics; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Urethane; Vagotomy; Vagus Nerve

1982
Effect of compound D-600 (methoxyverapamil) on gluconeogenesis and on acceleration of the process by alpha-adrenergic stimuli in rat kidney tubules.
    The Biochemical journal, 1980, Aug-15, Volume: 190, Issue:2

    Topics: Angiotensin II; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Gallopamil; Gluconeogenesis; Imidazoles; In Vitro Techniques; Kidney Tubules; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Verapamil

1980
The determination of presynaptic pA2 values of yohimbine and phentolamine on the perfused rat heart under conditions of negligible autoinhibition.
    British journal of pharmacology, 1983, Volume: 79, Issue:1

    Topics: Animals; Electric Stimulation; Heart; Male; Myocardium; Oxymetazoline; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Synapses; Yohimbine

1983
Controversial evidence regarding the functional importance of presynaptic alpha receptors.
    Federation proceedings, 1984, Volume: 43, Issue:5

    Topics: Animals; Clonidine; Dogs; Electric Stimulation; Heart; Heart Rate; Kidney; Norepinephrine; Oxymetazoline; Phentolamine; Receptors, Adrenergic, alpha; Synapses; Vasoconstriction; Yohimbine

1984
Influence of adrenergic and cholinergic mediators on the equine jejunum in vitro.
    American journal of veterinary research, 1996, Volume: 57, Issue:6

    Topics: Acetylcholine; Adrenergic Agonists; Adrenergic Antagonists; Animals; Atropine; Brimonidine Tartrate; Calcium Channel Blockers; Cholinergic Agonists; Cholinergic Antagonists; Dose-Response Relationship, Drug; Horses; Isoproterenol; Jejunum; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxymetazoline; Parasympathetic Nervous System; Phentolamine; Phenylephrine; Prazosin; Quinoxalines; Sympathetic Nervous System; Tetrodotoxin; Verapamil; Yohimbine

1996
Subtype determination of presynaptic alpha 2-autoreceptors in the rabbit pulmonary artery and human saphenous vein.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Benzazepines; Cattle; Dioxanes; Electric Stimulation; Humans; Idazoxan; Imidazoles; In Vitro Techniques; Oxymetazoline; Phentolamine; Presynaptic Terminals; Pulmonary Artery; Rabbits; Rats; Receptors, Adrenergic, alpha-2; Saphenous Vein; Tritium

1995
Characterisation of pre- and post-synaptic alpha-adrenoceptors in modulation of the rat ileum longitudinal and circular muscle activities.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brimonidine Tartrate; Clonidine; Electric Stimulation; Idazoxan; Ileum; In Vitro Techniques; Muscle Contraction; Oxymetazoline; Phentolamine; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Receptors, Presynaptic

1997
Effects of alpha 2-adrenergic agonism, imidazolines, and G-protein on insulin secretion in beta cells.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:10

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Cricetinae; Glucose; GTP-Binding Proteins; Humans; Imidazoles; Indoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Kinetics; Molecular Structure; Oxymetazoline; Pancreatic Neoplasms; Pertussis Toxin; Phentolamine; Pyrroles; Quinolizines; Receptors, Adrenergic, alpha-2; Tumor Cells, Cultured; Virulence Factors, Bordetella

1997
A role for amino acid residues in the third cytoplasmic loop in defining the ligand binding characteristics of the alpha2D-adrenergic receptor.
    Molecular and cellular biochemistry, 1997, Volume: 177, Issue:1-2

    Topics: Amino Acid Sequence; Amino Acids; Animals; Cattle; Clonidine; COS Cells; Cytoplasm; Epinephrine; Humans; Ligands; Mice; Molecular Sequence Data; Mutagenesis, Site-Directed; Oxymetazoline; Phentolamine; Prazosin; Protein Binding; Rats; Receptors, Adrenergic, alpha-2; Sequence Alignment; Yohimbine

1997
Lack of alpha2-adrenoceptor autoregulation of noradrenaline release in rat nucleus accumbens slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Homeostasis; Male; Norepinephrine; Nucleus Accumbens; Oxymetazoline; Phentolamine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Yohimbine

1998
Mechanism of relaxant effect of clonidine in isolated bovine tracheal smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Cattle; Clonidine; Cyclic AMP; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxymetazoline; Phentolamine; Trachea

1998
Effects of imidazoline and non-imidazoline alpha-adrenergic agents on canine platelet aggregation.
    Pharmacology, 1999, Volume: 58, Issue:4

    Topics: Adenosine Diphosphate; Adrenergic Agents; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Collagen; Dogs; Epinephrine; Female; Imidazoles; Male; Oxymetazoline; Phentolamine; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Adrenergic, alpha; Thrombin; Yohimbine

1999
Frequency dependent alpha(2)-adrenoceptor mediated modulation of excitatory junction potentials in guinea-pig mesenteric artery.
    European journal of pharmacology, 2001, Jan-05, Volume: 411, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Electric Stimulation; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; Neuromuscular Junction; Oxymetazoline; Phentolamine; Pyridoxal Phosphate; Receptors, Adrenergic, alpha-2; Reserpine; Suramin; Yohimbine

2001
Molecular cloning and functional expression of the guinea pig alpha(1a)-adrenoceptor.
    European journal of pharmacology, 2001, Aug-31, Volume: 426, Issue:3

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cloning, Molecular; COS Cells; DNA, Complementary; Dose-Response Relationship, Drug; Epinephrine; Gene Expression; Guinea Pigs; Methoxamine; Molecular Sequence Data; Norepinephrine; Oxathiins; Oxymetazoline; Phentolamine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sulfonamides; Tamsulosin; Tritium

2001
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Cerebral Cortex; Idazoxan; In Vitro Techniques; Isoquinolines; Ligands; Mice; Mice, Knockout; Naphthyridines; Oxymetazoline; Phentolamine; Prazosin; Putamen; Radioligand Assay; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2004