Page last updated: 2024-08-17

phentolamine and mianserin

phentolamine has been researched along with mianserin in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19908 (38.10)18.7374
1990's5 (23.81)18.2507
2000's2 (9.52)29.6817
2010's5 (23.81)24.3611
2020's1 (4.76)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andrews, PR; Craik, DJ; Martin, JL1
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Andersen, K; Balle, T; Larsen, AK; Liljefors, T; Perregaard, J; Ramirez, MT; Søby, KK1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Doxey, JC; Everitt, J; Metcalf, G1
Doggrell, SA2
Roeder, T1
Bockaert, J; Lafon-Cazal, M1
Cavero, I; Gomeni, R; Lefèvre-Borg, F; Roach, AG1
Mckee, M; Nathanson, JA; Scavone, C1
Chen, X; Kombian, SB; Pittman, QJ; Zidichouski, JA1
Katayama, S; Kohno, H; Ohkubo, Y; Ohuchi, Y1
Fujiseki, Y; Inagaki, C; Kinoshita, T; Okugawa, G; Omori, K; Suzukawa, J1
Papaefthimiou, C; Theophilidis, G1
Merritt, DJ; Rigby, LM1
Kanai, A; Momohara, Y; Nagayama, T1
Barreto, YC; Belo, CAD; Borges, BT; Carlini, CR; de Almeida, CGM; Oliveira, RS; Rosa, ME; Vinadé, L; Zanatta, AP1

Other Studies

21 other study(ies) available for phentolamine and mianserin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Synthesis and structure-affinity relationship investigations of 5-heteroaryl-substituted analogues of the antipsychotic sertindole. A new class of highly selective alpha(1) adrenoceptor antagonists.
    Journal of medicinal chemistry, 2003, Jan-16, Volume: 46, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Azoles; Brain; Cell Line; Cricetinae; Humans; Imidazoles; In Vitro Techniques; Indoles; Pyridines; Pyrimidines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Receptors, Dopamine; Receptors, Serotonin; Structure-Activity Relationship; Triazoles

2003
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Mianserin--an analysis of its peripheral autonomic actions.
    European journal of pharmacology, 1978, Sep-01, Volume: 51, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Desipramine; Dibenzazepines; Electric Stimulation; Male; Mianserin; Norepinephrine; Phenoxybenzamine; Phentolamine; Rats; Tyramine; Yohimbine

1978
Mianserin potentiates responses to acetylcholine in the rat anococcygeus muscle.
    European journal of pharmacology, 1979, May-01, Volume: 55, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Dibenzazepines; Drug Synergism; Hydroxydopamines; In Vitro Techniques; Male; Mianserin; Muscle Contraction; Norepinephrine; Nortriptyline; Phentolamine; Rats

1979
A new octopamine receptor class in locust nervous tissue, the octopamine 3 (OA3) receptor.
    Life sciences, 1992, Volume: 50, Issue:1

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Animals; Binding Sites; Chlorpromazine; Female; Grasshoppers; Male; Metoclopramide; Mianserin; Neurons; Octopamine; Phentolamine; Receptors, Adrenergic; Receptors, Biogenic Amine; Regression Analysis

1992
Pharmacological characterization of octopamine-sensitive adenylate cyclase in the flight muscle of Locusta migratoria L.
    European journal of pharmacology, 1985, Dec-10, Volume: 119, Issue:1-2

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Catecholamines; Chlorphenamidine; Chlorpromazine; Flight, Animal; Grasshoppers; In Vitro Techniques; Male; Metoclopramide; Mianserin; Muscles; Octopamine; Phentolamine; Prazosin; Receptors, Adrenergic; Receptors, Biogenic Amine; Serotonin; Synephrine; Tyramine

1985
Effect of mianserin on noradrenergic transmission in the rat anococcygeus muscle.
    British journal of pharmacology, 1980, Volume: 68, Issue:2

    Topics: Animals; Dibenzazepines; Hydroxydopamines; In Vitro Techniques; Male; Mianserin; Muscle Contraction; Muscles; Neuromuscular Junction; Norepinephrine; Nortriptyline; Phentolamine; Rats; Sympathetic Nervous System; Synaptic Transmission

1980
Comparison of mianserin with desipramine, maprotiline and phentolamine on cardiac presynaptic and vascular postsynaptic alpha-adrenoceptors and noradrenaline reuptake in pithed normotensive rats.
    British journal of pharmacology, 1980, Volume: 68, Issue:2

    Topics: Animals; Anthracenes; Blood Vessels; Cardiovascular System; Clonidine; Desipramine; Dibenzazepines; Drug Interactions; Heart; Male; Maprotiline; Mianserin; Norepinephrine; Phentolamine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Spinal Cord

1980
Monoamine uptake in insect synaptosomal preparations.
    Insect biochemistry and molecular biology, 1994, Volume: 24, Issue:6

    Topics: Animals; Biological Transport; Brain; Carrier Proteins; Cell Fractionation; Cocaine; Cockroaches; Dopamine; Ganglia, Invertebrate; Mianserin; Octopamine; Optic Lobe, Nonmammalian; Phentolamine; Rats; Rats, Sprague-Dawley; Sodium; Synaptic Transmission; Synaptosomes

1994
Dopamine depresses glutamatergic synaptic transmission in the rat parabrachial nucleus in vitro.
    Neuroscience, 1999, Volume: 90, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzazepines; Dopamine; Dopamine Agonists; Dopamine Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Male; Membrane Potentials; Mianserin; Neurons; Patch-Clamp Techniques; Phentolamine; Pons; Quinpirole; Rats; Rats, Sprague-Dawley; Reaction Time; Sulpiride; Synaptic Transmission

1999
Possible neural mechanisms involved in footshock stress-induced enhancement of exploratory behavior in mice.
    Biological & pharmaceutical bulletin, 1999, Volume: 22, Issue:4

    Topics: Animals; Atropine; Central Nervous System; Diazepam; Dizocilpine Maleate; Electric Stimulation; Exploratory Behavior; Haloperidol; Male; Mianserin; Mice; Naltrexone; Phentolamine; Propranolol; Stress, Physiological

1999
Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.
    Journal of neuroendocrinology, 1999, Volume: 11, Issue:11

    Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cells, Cultured; Desipramine; Dexamethasone; Gene Expression Regulation; Haloperidol; Hippocampus; Ketanserin; Mianserin; Neurons; Paroxetine; Phentolamine; Propranolol; Radioligand Assay; Rats; Receptors, Glucocorticoid; Receptors, Mineralocorticoid; RNA, Messenger; Sulpiride; Transcription, Genetic; Tritium

1999
Octopamine--a single modulator with double action on the heart of two insect species (Apis mellifera macedonica and Bactrocera oleae): Acceleration vs. inhibition.
    Journal of insect physiology, 2011, Volume: 57, Issue:2

    Topics: Animals; Bees; Heart; Heart Rate; Mianserin; Octopamine; Phentolamine; Receptors, Biogenic Amine; Tephritidae

2011
Roles of biogenic amines in regulating bioluminescence in the Australian glowworm Arachnocampa flava.
    The Journal of experimental biology, 2011, Oct-01, Volume: 214, Issue:Pt 19

    Topics: Analysis of Variance; Animals; Biogenic Amines; Carbon Dioxide; Diptera; Image Processing, Computer-Assisted; Immunohistochemistry; Larva; Luminescent Proteins; Malpighian Tubules; Mianserin; Octopamine; Phentolamine; Queensland

2011
Aminergic control of social status in crayfish agonistic encounters.
    PloS one, 2013, Volume: 8, Issue:9

    Topics: Agonistic Behavior; Animals; Astacoidea; Behavior, Animal; Biogenic Amines; Body Size; Injections; Male; Mianserin; Octopamine; Phentolamine; Serotonin; Social Dominance

2013
The neurotoxic mechanism of Jack Bean Urease in insects involves the interplay between octopaminergic and dopaminergic pathways.
    Pesticide biochemistry and physiology, 2023, Volume: 189

    Topics: Animals; Cockroaches; Mianserin; Phentolamine; Reserpine; Urease

2023