Page last updated: 2024-08-21

phenazocine and rimcazole

phenazocine has been researched along with rimcazole in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19905 (29.41)18.7374
1990's10 (58.82)18.2507
2000's2 (11.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burke, M; Earley, B; Gouret, CJ; Junien, JL; Leonard, BE1
Balestra, B; Candura, SM; Coccini, T; Costa, LG; Iapadre, N; Manzo, L; Tonini, M1
Henderson, G; Jarvis, GE; Kennedy, C1
Iwamoto, ET1
Beart, PM; Manallack, DT; O'Shea, RD1
Chang, KJ; Ferris, RM; Russell, A; Tang, FL1
Ford-Rice, FY; London, ED; Schell, SE; Su, TP1
Ceci, A; French, ED; Smith, M1
Cuomo, V; d'Istria, M; Maj, M; Monteleone, P; Serino, I; Steardo, L1
Bastianetto, S; Perrault, G; Sanger, DJ1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
Matsunaga, KH; Matsuno, K; Mita, S1
Glennon, RA; Herndon, JL; Young, R1
Kobayashi, T; Matsuno, K; Mita, S1
Kamei, J1
Bridges, S; Miller, C; Thompson, TL1
Dikranian, K; Farber, NB; Heinkel, C; Jiang, XP; Kim, SH1

Reviews

1 review(s) available for phenazocine and rimcazole

ArticleYear
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases

1999

Other Studies

16 other study(ies) available for phenazocine and rimcazole

ArticleYear
Evidence for an anti-amnesic effect of JO 1784 in the rat: a potent and selective ligand for the sigma receptor.
    Brain research, 1991, Apr-19, Volume: 546, Issue:2

    Topics: Amnesia; Animals; Antipsychotic Agents; Avoidance Learning; Behavior, Animal; Carbazoles; Cinnamates; Cyclopropanes; Dopamine Agents; Dose-Response Relationship, Drug; Guanidines; Ligands; Male; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Scopolamine

1991
Two subtypes of enteric non-opioid sigma receptors in guinea-pig cholinergic motor neurons.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Carbazoles; Dextromethorphan; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Motor Neurons; Myenteric Plexus; Parasympathetic Nervous System; Phenazocine; Pyrimidines; Receptors, Opioid; Receptors, sigma

1991
The sigma [corrected] ligand rimcazole antagonises (+)SKF 10,047, but not (+)3-PPP, in the mouse isolated vas deferens.
    European journal of pharmacology, 1990, Jun-08, Volume: 181, Issue:3

    Topics: Animals; Antipsychotic Agents; Carbazoles; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Muscle, Smooth; Phenazocine; Piperidines; Stereoisomerism; Vas Deferens

1990
Evidence for a model of activation of central sigma systems.
    Life sciences, 1989, Volume: 44, Issue:21

    Topics: Animals; Benzazepines; Benzomorphans; Butaclamol; Carbazoles; Dopamine Antagonists; Haloperidol; Kinetics; Male; Models, Biological; Motor Activity; Naltrexone; Narcotic Antagonists; Phenazocine; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Sulpiride

1989
Regulation of sigma-receptors: high- and low-affinity agonist states, GTP shifts, and up-regulation by rimcazole and 1,3-Di(2-tolyl)guanidine.
    Journal of neurochemistry, 1989, Volume: 53, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Binding, Competitive; Brain; Carbazoles; Cyclazocine; Dopamine; Dopamine Agents; GTP-Binding Proteins; Guanidines; Guanosine Triphosphate; Magnesium; Male; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1989
Evidence that the potential antipsychotic agent rimcazole (BW 234U) is a specific, competitive antagonist of sigma sites in brain.
    Life sciences, 1986, Jun-23, Volume: 38, Issue:25

    Topics: Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Brain; Carbazoles; Clozapine; Guinea Pigs; Kinetics; Male; Methylphenidate; Mice; Phenazocine; Phencyclidine; Phenoxybenzamine; Propranolol; Receptors, Opioid; Receptors, sigma; Sulpiride

1986
Correlation of inhibitory potencies of putative antagonists for sigma receptors in brain and spleen.
    European journal of pharmacology, 1988, Apr-13, Volume: 148, Issue:3

    Topics: Animals; Antipsychotic Agents; Brain Chemistry; Carbazoles; Guinea Pigs; Haloperidol; In Vitro Techniques; Isoquinolines; Male; Phenazocine; Piperazines; Pyrimidines; Receptors, Opioid; Receptors, sigma; Spleen; Tritium

1988
Activation of the A10 mesolimbic system by the sigma-receptor agonist (+)SKF 10,047 can be blocked by rimcazole, a novel putative antipsychotic.
    European journal of pharmacology, 1988, Sep-01, Volume: 154, Issue:1

    Topics: Animals; Antipsychotic Agents; Carbazoles; Dose-Response Relationship, Drug; Limbic System; Male; Motor Activity; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Receptors, sigma

1988
(+)-N-allylnormetazocine enhances N-acetyltransferase activity and melatonin synthesis: preliminary evidence for a functional role of sigma receptors in the rat pineal gland.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Antipsychotic Agents; Arylamine N-Acetyltransferase; Carbazoles; Male; Melatonin; Phenazocine; Pineal Gland; Rats; Rats, Sprague-Dawley; Receptors, sigma

1995
Pharmacological evidence for the involvement of sigma sites in DTG-induced contralateral circling in rats.
    Neuropharmacology, 1995, Volume: 34, Issue:1

    Topics: Animals; Anticonvulsants; Behavior, Animal; Carbazoles; Dose-Response Relationship, Drug; Guanidines; Haloperidol; Injections, Spinal; Male; Motor Activity; Phenazocine; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, sigma; Salicylamides

1995
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
Acute effects of sigma ligands on the extracellular DOPAC level in rat frontal cortex and striatum.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Corpus Striatum; Extracellular Space; Frontal Lobe; Guanidines; Kinetics; Ligands; Male; Microdialysis; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Time Factors

1995
Antagonism of a (+)N-allylnormetazocine stimulus by (-)PPAP and several structurally related analogs.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amines; Animals; Antipsychotic Agents; Buspirone; Carbazoles; Generalization, Stimulus; Male; Phenazocine; Phenols; Piperazines; Propylamines; Rats; Rats, Sprague-Dawley; Receptors, Phencyclidine; Receptors, sigma; Serotonin Receptor Agonists

1993
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:1

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens

1996
Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands.
    Neuroscience letters, 2001, Oct-26, Volume: 312, Issue:3

    Topics: Animals; Antipsychotic Agents; Carbazoles; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Haloperidol; Ligands; Neurons; Nomifensine; Nucleus Accumbens; Phenazocine; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, sigma; Spiperone; Sulpiride; Synaptosomes; Tritium

2001
Receptor mechanisms and circuitry underlying NMDA antagonist neurotoxicity.
    Molecular psychiatry, 2002, Volume: 7, Issue:1

    Topics: Adrenergic alpha-Agonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Carbachol; Carbazoles; Cerebral Cortex; Clonidine; Dizocilpine Maleate; Drug Interactions; Excitatory Amino Acid Antagonists; Female; Kainic Acid; Models, Neurological; Muscarinic Antagonists; Nerve Tissue Proteins; Neurons; Neuroprotective Agents; Phenazocine; Prosencephalon; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Receptors, Muscarinic; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Scopolamine

2002