Page last updated: 2024-08-21

phenazocine and phencyclidine

phenazocine has been researched along with phencyclidine in 129 studies

Research

Studies (129)

TimeframeStudies, this research(%)All Research%
pre-199090 (69.77)18.7374
1990's34 (26.36)18.2507
2000's4 (3.10)29.6817
2010's1 (0.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Grynne, BH; Holmen, AT; Maurset, A1
Abraham, P; Bai, X; Brine, GA; Carroll, FI; Martin, BR; Mascarella, SW; May, EL; Parham, K; Sauss, C; Zhang, X1
Lemaire, S; Rogers, C1
Hudzik, TJ; Slifer, BL1
Boyce, S; Cook, G; Iversen, SD; Rupniak, NM; Steventon, MJ1
deCosta, BR; Hardwick, WC; McMillan, DE; Rice, KC1
Katki, AG; Munson, PJ; Rodbard, D; Schwarz, S; Zhou, GZ1
Carter, AJ; Müller, RE1
Pèzzola, A; Popoli, P; Sagratella, S; Scotti de Carolis, A1
Brent, PJ1
Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauché, D1
Burke, M; Earley, B; Gouret, CJ; Junien, JL; Leonard, BE1
Feuerstein, G; Lysko, PG1
Connick, JH; Fox, PK; France, L; Hanlon, GM; Nicholson, CD1
Su, TP; Wu, XZ1
Bejanian, M; George, R; Pechnick, RN1
Bauerle, LM; DeNoble, VJ; Jones, KW1
Bueno, L; Fioramonti, J; Gue, M; Junien, JL; Pascaud, X1
Beinfeld, MC; Brog, JS1
Katki, AG; Rodbard, D; Schwarz, S; Zhou, GZ1
DeLander, GE; Wahl, JJ1
Oswald, RE; Papke, RL1
France, CP; Snyder, AM; Woods, JH1
Alerhand, S; Itzhak, Y1
Cheng, BK; Contreras, PC; Gray, NM; Lair, CM; Mick, SJ1
Wann, KT; Wardley-Smith, B1
Iversen, SD; Oles, RJ; Preston, C; Singh, L; Tricklebank, MD1
Gussio, RP; Marquis, KL; Moreton, JE; Paquette, NC1
Allikmets, LKh; Kharro, IaE; Lang, AE; Vasar, EE1
Duffy, O; Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauche, D1
Jackson, A; Sanger, DJ3
McMillan, DE; Wessinger, WD1
Iversen, SD; Oles, RJ; Singh, L; Tricklebank, MD; Wong, EH1
Catt, KJ; Dufau, ML; Stojilković, SS1
Knight, AR; Wong, EH; Woodruff, GN1
Beart, PM; Manallack, DT1
Itzhak, Y; Khouri, M1
Kushner, L; Zukin, RS; Zukin, SR1
Contreras, PC; DiMaggio, DA; O'Donohue, TL1
Alberici, GP; Cook, L; Steinfels, GF; Tam, SW1
Holtzman, SG2
Downes, CP; Lewis, PE; Stone, MA1
French, ED1
Chang, KJ; Ferris, RM; Russell, A; Tang, FL1
Chung, JM; Kim, J; Shin, HK; Willcockson, WS; Willis, WD1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Braunwalder, AF; Lehmann, J; Loo, PS; Sills, MA; Williams, M1
Itzhak, Y2
Furukawa, H; Hiramatsu, M; Kameyama, T; Nabeshima, T1
Gundlach, AL; Largent, BL; Snyder, SH4
Goldman, ME; Jacobson, AE; Paul, SM; Rice, KC1
Greenberg, BD; Segal, DS1
Jacobson, AE; Koek, W; Lessor, RA; Rice, KC; Woods, JH1
Ieni, JR; Nichtenhauser, R; Sircar, R; Zukin, SR1
Su, TP; Weissman, AD; Yeh, SY1
Sircar, R; Zukin, SR3
Contreras, PC; DiMaggio, DA; O'Donohue, TL; Quirion, R1
Contreras, PC; O'Donohue, TL; Quirion, R2
Hiramatsu, M; Kameyama, T; Nabeshima, T2
Dykstra, LA; Slifer, BL2
Cook, L; Steinfels, GF; Tam, SW2
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR1
Coan, EJ; Collingridge, GL1
Iwamoto, ET1
Carroll, ME1
Bartschat, DK; Blaustein, MP1
Dykstra, LA; Picker, M1
Iversen, LL; Kemp, JA; Knight, AR; Priestley, T; Wong, EH; Woodruff, GN1
McCann, DJ; Rabin, RA; Winter, JC1
Kozlowski, MR1
Mattia, A; Moreton, JE1
Risner, ME; Shannon, HE; Vaupel, DB1
McLaughlin, JT; Oswald, RE; Pennow, NN1
Bigelow, J; Michel, L; Oswald, RE1
McCann, DJ; Winter, JC1
Leccese, AP; Marquis, KL; Mattia, A; Moreton, JE1
Clark, RD; Katz, JL; Spealman, RD1
Bergman, J; Hassoun, J; Schuster, CR1
Bunney, BS; Freeman, AS1
Hillman, GR; Johnson, KM1
Cone, EJ; Goldberg, SR; Gorodetzky, CW; Herling, S; Risner, ME; Shannon, HE; Vaupel, DB1
French, ED; Vantini, G1
Balster, RL; Brady, KT; Slifer, BL; Zukin, SR1
Balster, RL; Brady, KT; May, EL1
Hammer, RP; Herkenham, M; Pert, CB; Quirion, R1
Morton, EC; Vaupel, DB1
Pert, CB; Quirion, R1
Vaupel, DB1
Tam, SW1
Greenfield, LJ; Guyenet, PG; Hackett, JT; Stringer, JL1
Stafford, I; Tomie, A; Wagner, GC1
Holtzman, SG; White, JM2
Johnson, KM; Leventer, SM1
Contreras, CM; Ervin, FR; Guzman-Flores, C; Mexicano, G; Palmour, R1
Shannon, HE2
Bao, WL; Sun, FY; Zhang, AZ; Zhen, FC1
Pechnick, RN; Poland, RE1
Ajima, A; Araki, H; Imagawa, Y; Muramatsu, M; Nakazato, A; Ogawa, S; Okuyama, S; Tanaka, M; Yamaguchi, K; Yoshida, M1
Chaki, S; Imagawa, Y; Muramatsu, M; Okuyama, S; Otomo, S; Tanaka, M1
De Souza, EB; Wolfe, SA1
Shi, GG; Xu, SF1
Masaki, H; Mishina, M; Mori, H; Shimoji, K; Yamakura, T1
della Puppa, A; Kimes, AS; London, ED1
Kamei, H; Kameyama, T; Nabeshima, T1
Amano, M; Matsuno, K; Nabeshima, T; Yamada, K1
Jin, J; Watanabe, S; Yamamoto, T1
Kobayashi, T; Matsuno, K; Mita, S1
Ahmed, MS; Enna, SJ; Mather, A1
Horikomi, K; Iizuka, K; Mita, N; Miwa, T; Nagase, H; Sakai, K; Sonehara, K; Takagi, K; Takahashi, S1
Furukawa, H; Ichihara, K; Kamei, H; Mamiya, T; Nabeshima, T; Nagai, T; Noda, A; Noda, Y; Sugiura, S1
Horikomi, K; Karasawa, J; Sagi, N; Sora, I; Yamamoto, H; Yamamoto, T1
Sun, W; Wessinger, WD1
Tanabe, M1
Isotani, K; Mori, T; Narita, M; Nomura, M; Suzuki, T; Torigoe, K; Tsukiyama, Y; Yoshizawa, K1

Reviews

3 review(s) available for phenazocine and phencyclidine

ArticleYear
Drug discrimination studies.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Sigma and phencyclidine receptors in the brain-endocrine-immune axis.
    NIDA research monograph, 1993, Volume: 133

    Topics: Animals; Autoradiography; Brain Chemistry; Endocrine Glands; Humans; Hypophysectomy; Lymphocytes; Phenazocine; Phencyclidine; Receptors, Phencyclidine; Receptors, sigma

1993
[Neuropharmacological effects of sigma receptor ligands: anxiolytic, anti-amnesic and neuroprotective effects].
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1996, Volume: 16, Issue:3

    Topics: Animals; Antipsychotic Agents; Anxiety; Brain Ischemia; Cinnamates; Cyclopropanes; Humans; Learning Disabilities; Memory Disorders; Phenazocine; Phencyclidine; Receptors, sigma

1996

Other Studies

126 other study(ies) available for phenazocine and phencyclidine

ArticleYear
Evidence for distinct phencyclidine and SKF10047 receptors following detergent treatment of rat brain membranes.
    Pharmacology & toxicology, 1992, Volume: 70, Issue:1

    Topics: Animals; Brain Chemistry; Cell Membrane; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Synaptosomes; Tritium

1992
Enantiomeric N-substituted N-normetazocines: a comparative study of affinities at sigma, PCP, and mu opioid receptors.
    Journal of medicinal chemistry, 1992, Jul-24, Volume: 35, Issue:15

    Topics: Animals; Brain; Guinea Pigs; Male; Narcotics; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism; Substrate Specificity

1992
Characterization of [3H]desmethylimipramine binding in bovine adrenal medulla: interactions with sigma- and (or) phencyclidine-receptor ligands.
    Canadian journal of physiology and pharmacology, 1992, Volume: 70, Issue:11

    Topics: Adrenal Medulla; Animals; Binding Sites; Cattle; Desipramine; Dextromethorphan; Dizocilpine Maleate; Phenazocine; Phencyclidine; Piperidines; Potassium Chloride; Receptors, Opioid, delta; Receptors, Phencyclidine; Tranquilizing Agents

1992
Interaction of sigma and PCP-like drugs on operant behaviors in the rat.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: Animals; Conditioning, Operant; Dextroamphetamine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Pentazocine; Phenazocine; Phencyclidine; Psychotropic Drugs; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule

1992
Psychomotor activity and cognitive disruption attributable to NMDA, but not sigma, interactions in primates.
    Behavioural brain research, 1991, Feb-28, Volume: 42, Issue:2

    Topics: Animals; Ataxia; Cognition; Dizocilpine Maleate; Macaca mulatta; Male; Pentazocine; Phenazocine; Phencyclidine; Psychomotor Performance; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Saimiri; Space Perception

1991
Effects of drugs that bind to PCP and sigma receptors on punished responding.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Animals; Buspirone; Dizocilpine Maleate; Haloperidol; Learning; Male; Pentobarbital; Phenazocine; Phencyclidine; Punishment; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1991
Quantitative characterization of multiple binding sites for phencyclidine and N-allylnormetazocine in membranes from rat and guinea pig brain.
    Neuropharmacology, 1991, Volume: 30, Issue:7

    Topics: Animals; Binding Sites; Brain; Cell Membrane; Guinea Pigs; Male; Phenazocine; Phencyclidine; Psychotropic Drugs; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1991
Activation of excitatory amino acid receptors cannot alone account for anoxia-induced impairment of protein synthesis in rat hippocampal slices.
    Journal of neurochemistry, 1991, Volume: 57, Issue:3

    Topics: Animals; Aspartic Acid; Carbon Radioisotopes; Dizocilpine Maleate; Glutamates; Glutamic Acid; Hippocampus; Hypoxia; Kainic Acid; Lysine; Male; N-Methylaspartate; Nerve Tissue Proteins; Phenazocine; Phencyclidine; Quisqualic Acid; Rats; Receptors, Amino Acid; Receptors, Cell Surface; Receptors, N-Methyl-D-Aspartate

1991
Behavioural and electoencephalographic interactions between haloperidol and PCP/sigma ligands in the rat.
    Psychopharmacology, 1991, Volume: 105, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Catalepsy; Electroencephalography; Haloperidol; Isoquinolines; Kinetics; Male; Phenazocine; Phencyclidine; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Spiperone

1991
Similar behavioural effects of sigma agonists and PCP-like non-competitive NMDA antagonists in guinea-pigs.
    Psychopharmacology, 1991, Volume: 105, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Dizocilpine Maleate; Dopamine Agents; Dopamine Antagonists; Ergolines; Female; Guanidines; Guinea Pigs; Haloperidol; Ketamine; Male; Motor Activity; N-Methylaspartate; Pentazocine; Phenazocine; Phencyclidine; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride

1991
JO 1784, a potent and selective ligand for rat and mouse brain sigma-sites.
    The Journal of pharmacy and pharmacology, 1990, Volume: 42, Issue:6

    Topics: Animals; Brain Chemistry; Cinnamates; Cyclopropanes; In Vitro Techniques; Male; Mice; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta

1990
A comparison of the psychopharmacological profiles of phencyclidine, ketamine and (+) SKF 10,047 in the trimethyltin rat model.
    Neuropharmacology, 1990, Volume: 29, Issue:8

    Topics: Animals; Avoidance Learning; Behavior, Animal; Brain Chemistry; Ketamine; Learning; Male; Nervous System Diseases; Neurotransmitter Agents; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine; Swimming; Trimethyltin Compounds

1990
Excitatory amino acid neurotoxicity at the N-methyl-D-aspartate receptor in cultured neurons: protection by SKF 10,047.
    Neuroscience letters, 1990, Dec-11, Volume: 120, Issue:2

    Topics: Animals; Cell Survival; Cells, Cultured; Cerebellum; Dopamine Agents; Glutamates; Glutamic Acid; Neurons; Neurotoxins; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine

1990
The lack of utility of the rat vas deferens as a functional bioassay for sigma ligands.
    European journal of pharmacology, 1991, Feb-07, Volume: 193, Issue:2

    Topics: Animals; Binding Sites; Biological Assay; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; Male; Muscle Contraction; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Vas Deferens

1991
Guinea pig vas deferens contains sigma but not phencyclidine receptors.
    Neuroscience letters, 1990, Jan-22, Volume: 108, Issue:3

    Topics: Animals; Binding, Competitive; Guinea Pigs; Male; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Vas Deferens

1990
Effects of acute and chronic administration of (+)-SKF 10,047 on body temperature in the rat: cross-sensitization with phencyclidine.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Animals; Body Temperature; Body Weight; Dose-Response Relationship, Drug; Drug Interactions; Injections, Subcutaneous; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism

1990
Differential effects of sigma and phencyclidine receptor ligands on learning.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Avoidance Learning; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Ligands; Male; Memory; Pentazocine; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Retention, Psychology

1990
Selective stimulation of colonic motor response to a meal by sigma ligands in dogs.
    Gastroenterology, 1990, Volume: 99, Issue:3

    Topics: Animals; Cinnamates; Colon; Cyclopropanes; Dogs; Drug Antagonism; Eating; Gastrointestinal Motility; Guanidines; Injections, Intravenous; Injections, Intraventricular; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism

1990
Inhibition of carbachol-induced inositol phosphate accumulation by phencyclidine, phencyclidine-like ligands and sigma agonists involves blockade of the muscarinic cholinergic receptor: a novel dioxadrol-preferring interaction.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:3

    Topics: Animals; Brain; Carbachol; Culture Techniques; Dibenzocycloheptenes; Dioxolanes; Dizocilpine Maleate; Inositol Phosphates; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Sigma Factor; Transcription Factors

1990
Differential modulation by cations of sigma and phencyclidine binding sites in rat brain.
    Journal of receptor research, 1990, Volume: 10, Issue:1-2

    Topics: Animals; Binding Sites; Brain; Cations; Dose-Response Relationship, Drug; Haloperidol; Ligands; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Sigma Factor; Tritium

1990
In vivo characterization of phencyclidine/sigma agonist-mediated inhibition of nociception.
    European journal of pharmacology, 1989, Jan-10, Volume: 159, Issue:2

    Topics: Animals; Anticonvulsants; Aspartic Acid; Behavior, Animal; Binding, Competitive; Dibenzocycloheptenes; Dizocilpine Maleate; Male; Mice; N-Methylaspartate; Nociceptors; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, Opioid, delta; Substance P

1989
Mechanisms of noncompetitive inhibition of acetylcholine-induced single-channel currents.
    The Journal of general physiology, 1989, Volume: 93, Issue:5

    Topics: Acetylcholine; Biomechanical Phenomena; Cell Line; Electric Conductivity; Electrophysiology; Ion Channels; Phenazocine; Phencyclidine; Tetracaine; Time Factors

1989
Analgesic effects of phencyclidine-like drugs in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Alfentanil; Analgesia; Analgesics; Anesthetics; Animals; Anticonvulsants; Dextrorphan; Dibenzocycloheptenes; Discrimination, Psychological; Dizocilpine Maleate; Dose-Response Relationship, Drug; Fentanyl; Ketamine; Macaca mulatta; Phenazocine; Phencyclidine; Pyrrolidines

1989
Differential regulation of sigma and PCP receptors after chronic administration of haloperidol and phencyclidine in mice.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1989, Volume: 3, Issue:7

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Hallucinogens; Haloperidol; Male; Mice; Mice, Inbred Strains; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Time Factors

1989
Phencyclidine-like effects of tetrahydroisoquinolines and related compounds.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:6

    Topics: Animals; Ataxia; Behavior, Animal; Chemical Phenomena; Chemistry; Isoquinolines; Male; Molecular Structure; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereotyped Behavior; Structure-Activity Relationship; Tetrahydroisoquinolines

1989
The effects of non-competitive NMDA receptor antagonists on rats exposed to hyperbaric pressure.
    European journal of pharmacology, 1989, Jun-08, Volume: 165, Issue:1

    Topics: Animals; Binding, Competitive; Dibenzocycloheptenes; Dizocilpine Maleate; Hyperbaric Oxygenation; Ketamine; Male; Myoclonus; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Seizures; Tremor

1989
The behavioural effects of MK-801: a comparison with antagonists acting non-competitively and competitively at the NMDA receptor.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Animals; Anticonvulsants; Aspartic Acid; Behavior, Animal; Binding, Competitive; Dibenzocycloheptenes; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Male; Motor Activity; N-Methylaspartate; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Seizures

1989
Comparative electroencephalographic and behavioral effects of phencyclidine, (+)-SKF-10,047 and MK-801 in rats.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:3

    Topics: Animals; Anticonvulsants; Dibenzocycloheptenes; Dizocilpine Maleate; Electroencephalography; Female; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, sigma; Stereotyped Behavior

1989
[Adaptive changes in sigma and phencyclidine receptors during the long-term use of haloperidol and raclopride in rats].
    Biulleten' eksperimental'noi biologii i meditsiny, 1989, Volume: 108, Issue:9

    Topics: Adaptation, Physiological; Animals; Apomorphine; Behavior, Animal; Drug Interactions; Haloperidol; Ketamine; Phenazocine; Phencyclidine; Raclopride; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Salicylamides; Time Factors; Tritium

1989
Neuropeptide Y and peptide YY interact with rat brain sigma and PCP binding sites.
    European journal of pharmacology, 1989, Dec-19, Volume: 174, Issue:2-3

    Topics: Animals; Brain Chemistry; Haloperidol; In Vitro Techniques; Male; Neuropeptide Y; Pentazocine; Peptide YY; Peptides; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1989
Conditioned taste aversions induced by phencyclidine and other antagonists of N-methyl-D-aspartate.
    Neuropharmacology, 1989, Volume: 28, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Avoidance Learning; Conditioning, Operant; Male; N-Methylaspartate; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Taste

1989
Effects of phencyclidine and other N-methyl-D-aspartate antagonists on the schedule-controlled behavior of rats.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Animals; Aspartic Acid; Conditioning, Psychological; Dibenzocycloheptenes; Dizocilpine Maleate; Male; N-Methylaspartate; Phenazocine; Phencyclidine; Piperazines; Piperidines; Punishment; Rats; Rats, Inbred Strains; Reinforcement Schedule; Stereoisomerism

1989
Interaction of the discriminative stimulus effects of phencyclidine with those of (+)-N-allylnormetazocine, pentobarbital and d-amphetamine.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:3

    Topics: Amphetamines; Animals; Columbidae; Discrimination Learning; Drug Interactions; Pentobarbital; Phenazocine; Phencyclidine; Substance-Related Disorders

1989
A role for receptors of N-methyl-D-aspartic acid in the discriminative stimulus properties of phencyclidine.
    European journal of pharmacology, 1987, Sep-23, Volume: 141, Issue:3

    Topics: Animals; Discrimination, Psychological; Generalization, Stimulus; Haloperidol; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1987
Receptors and secretory actions of sigma/phencyclidine agonists in anterior pituitary cells.
    Endocrinology, 1987, Volume: 121, Issue:6

    Topics: Animals; Cell Membrane; Cells, Cultured; Etorphine; Female; Kinetics; Luteinizing Hormone; Phenazocine; Phencyclidine; Pituitary Gland, Anterior; Potassium; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Thermodynamics

1987
[3H]MK-801 labels a site on the N-methyl-D-aspartate receptor channel complex in rat brain membranes.
    Journal of neurochemistry, 1988, Volume: 50, Issue:1

    Topics: Animals; Anticonvulsants; Brain; Cations, Divalent; Cell Membrane; Cerebral Cortex; Dibenzocycloheptenes; Dizocilpine Maleate; Kinetics; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Tissue Distribution; Tritium

1988
Quantitative conformational analyses predict distinct receptor sites for PCP-like and sigma drugs.
    European journal of pharmacology, 1987, Dec-01, Volume: 144, Issue:2

    Topics: Animals; Binding Sites; Brain; Computer Graphics; Dibenzocycloheptenes; Dizocilpine Maleate; In Vitro Techniques; Isoquinolines; Male; Molecular Conformation; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1987
Regulation of the binding of sigma- and phencyclidine (PCP)-receptor ligands in rat brain membranes by guanine nucleotides and ions.
    Neuroscience letters, 1988, Feb-15, Volume: 85, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cations; Guanine Nucleotides; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine; Subcellular Fractions

1988
Characterization of opioid, sigma, and phencyclidine receptors in the neuroblastoma-brain hybrid cell line NCB-20.
    Molecular pharmacology, 1988, Volume: 34, Issue:5

    Topics: Animals; Brain Chemistry; Cell Line; Cricetinae; Hybrid Cells; Kinetics; Mice; Neuroblastoma; Phenazocine; Phencyclidine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1988
An endogenous ligand for the sigma opioid binding site.
    Synapse (New York, N.Y.), 1987, Volume: 1, Issue:1

    Topics: Animals; Brain; Endorphins; Kinetics; Ligands; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Swine

1987
Biochemical, behavioral, and electrophysiologic actions of the selective sigma receptor ligand (+)-pentazocine.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1988, Volume: 1, Issue:4

    Topics: Animals; Avoidance Learning; Brain; Discrimination Learning; Evoked Potentials, Visual; Male; Membranes; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Reference Values

1988
A comparison of the binding of sigma opioids and phencyclidine, and the interaction with antipsychotic drugs in rat brain membranes.
    British journal of pharmacology, 1986, Volume: 88, Issue:1

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Brain; Corpus Striatum; Endorphins; Haloperidol; In Vitro Techniques; Male; Membranes; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, delta

1986
Effects of N-allylnormetazocine (SKF 10,047), phencyclidine, and other psychomotor stimulants in the rat following 6-hydroxydopamine lesion of the ventral tegmental area.
    Neuropharmacology, 1986, Volume: 25, Issue:4

    Topics: Amphetamine; Animals; Apomorphine; Caffeine; Central Nervous System Stimulants; Dopamine; Hydroxydopamines; Male; Motor Activity; Oxidopamine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Scopolamine; Tegmentum Mesencephali

1986
Evidence that the potential antipsychotic agent rimcazole (BW 234U) is a specific, competitive antagonist of sigma sites in brain.
    Life sciences, 1986, Jun-23, Volume: 38, Issue:25

    Topics: Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Brain; Carbazoles; Clozapine; Guinea Pigs; Kinetics; Male; Methylphenidate; Mice; Phenazocine; Phencyclidine; Phenoxybenzamine; Propranolol; Receptors, Opioid; Receptors, sigma; Sulpiride

1986
Actions of opioids on primate spinothalamic tract neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:9

    Topics: Animals; Dynorphins; Enkephalin, Methionine; Macaca fascicularis; Morphine; Naloxone; Narcotics; Neurons; Phenazocine; Phencyclidine; Spinal Cord; Thalamus

1986
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:3

    Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid

1987
Interaction of L-glutamate and magnesium with phencyclidine recognition sites in rat brain: evidence for multiple affinity states of the phencyclidine/N-methyl-D-aspartate receptor complex.
    Molecular pharmacology, 1987, Volume: 32, Issue:6

    Topics: Animals; Brain; Glutamates; Glutamic Acid; In Vitro Techniques; Kinetics; Magnesium; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine

1987
Pharmacological specificity of some psychotomimetic and antipsychotic agents for the sigma and PCP binding sites.
    Life sciences, 1988, Volume: 42, Issue:7

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Haloperidol; In Vitro Techniques; Male; Phenazocine; Phencyclidine; Piperidines; Psychotropic Drugs; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1988
Different effects of ethylketocyclazocine on phencyclidine- and N-allylnormetazocine-induced stereotyped behaviors in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:4

    Topics: Analgesics, Opioid; Animals; Cyclazocine; Ethylketocyclazocine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereotyped Behavior

1987
Is the discriminative stimulus produced by phencyclidine due to an interaction with N-methyl-D-aspartate receptors?
    Psychopharmacology, 1988, Volume: 96, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Anticonvulsants; Chlordiazepoxide; Dibenzocycloheptenes; Discrimination, Psychological; Dizocilpine Maleate; Drug Interactions; Generalization, Stimulus; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1988
Phencyclidine and sigma opiate receptors in brain: biochemical and autoradiographical differentiation.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Autoradiography; Brain; Humans; In Vitro Techniques; Membranes; Phenazocine; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine

1985
Differentiation of [3H]phencyclidine and (+)-[3H]SKF-10,047 binding sites in rat cerebral cortex.
    FEBS letters, 1985, Oct-14, Volume: 190, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism

1985
Evidence for multiple opiate receptor involvement in different phencyclidine-induced unconditioned behaviors in rats.
    Psychopharmacology, 1986, Volume: 88, Issue:1

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Eating; Habituation, Psychophysiologic; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereotyped Behavior

1986
Metaphit, a proposed phencyclidine receptor acylator: phencyclidine-like behavioral effects and evidence of absence of antagonist activity in pigeons and in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Acylation; Animals; Ataxia; Catalepsy; Columbidae; Discrimination Learning; Drug Synergism; Ketamine; Macaca mulatta; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Species Specificity; Stereotyped Behavior

1986
Characterization and autoradiographic visualization of (+)-[3H]SKF10,047 binding in rat and mouse brain: further evidence for phencyclidine/"sigma opiate" receptor commonality.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Autoradiography; Brain Chemistry; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Species Specificity; Tritium

1986
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays.
    Life sciences, 1986, Jun-16, Volume: 38, Issue:24

    Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma

1986
Characterization of phencyclidine and sigma receptor-binding sites in brain.
    NIDA research monograph, 1986, Volume: 64

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Kinetics; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tritium

1986
Further evidence of phencyclidine/sigma opioid receptor commonality.
    NIDA research monograph, 1986, Volume: 64

    Topics: Animals; Autoradiography; Brain; Kinetics; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tissue Distribution; Tritium

1986
Isolation and identification of an endogenous ligand for the phencyclidine receptor.
    NIDA research monograph, 1986, Volume: 64

    Topics: Animals; Binding, Competitive; Brain; Brain Chemistry; Endopeptidases; Nerve Tissue Proteins; Neuropeptides; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Swine; Tissue Distribution

1986
Agonistic and antagonistic effects of PCP-derivatives and sigma opioids in PCP behavioral and receptor assays.
    NIDA research monograph, 1986, Volume: 64

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclazocine; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereotyped Behavior; Structure-Activity Relationship; Tritium

1986
Sigma receptors on NCB-20 hybrid neurotumor cells labeled with (+)[3H]SKF 10,047 and (+)[3H]3-PPP.
    European journal of pharmacology, 1986, May-13, Volume: 124, Issue:1-2

    Topics: Animals; Brain; Cells, Cultured; Cricetinae; Cricetulus; Hybrid Cells; Kinetics; Neuroblastoma; Phenazocine; Phencyclidine; Piperidines; Receptors, Opioid; Receptors, Opioid, delta; Stereoisomerism

1986
Autoradiographic distribution of phencyclidine receptors in the rat brain using [3H]1-(1-(2-thienyl)cyclohexyl)piperidine ([3H]TCP).
    Neuroscience letters, 1986, Jun-18, Volume: 67, Issue:2

    Topics: Animals; Autoradiography; Brain; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine

1986
Pharmacological and autoradiographic discrimination of sigma and phencyclidine receptor binding sites in brain with (+)-[3H]SKF 10,047, (+)-[3H]-3-[3-hydroxyphenyl]-N-(1-propyl)piperidine and [3H]-1-[1-(2-thienyl)cyclohexyl]piperidine.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; In Vitro Techniques; Kinetics; Male; Phenazocine; Phencyclidine; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism

1986
Phencyclidine-induced stereotyped behaviors after injection of morphine and N-allylnormetazocine (SKF 10,047) in rats.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:6

    Topics: Animals; Male; Morphine; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereotyped Behavior

1986
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
    Journal of pharmacobio-dynamics, 1986, Volume: 9, Issue:5

    Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid

1986
Discriminative stimulus effects of N-allylnormetazocine in rats trained to discriminate a kappa from a sigma agonist.
    Life sciences, 1987, Jan-26, Volume: 40, Issue:4

    Topics: Animals; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, sigma; Stereoisomerism

1987
Discriminative stimulus properties of (+)-N-allylnormetazocine in the rat: correlations with (+)-N-allylnormetazocine and phencyclidine receptor binding.
    Psychopharmacology, 1987, Volume: 91, Issue:1

    Topics: Animals; Brain; Cyclazocine; Discrimination Learning; Ketamine; Male; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism

1987
The effects of N-allylnormetazocine on electric shock titration in squirrel monkeys.
    Alcohol and drug research, 1987, Volume: 7, Issue:4

    Topics: Animals; Avoidance Learning; Electroshock; Male; Morphine; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma; Reinforcement Schedule; Saimiri; Stereoisomerism

1987
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
    Life sciences, 1987, Jun-01, Volume: 40, Issue:22

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism

1987
[3H]PCP-3-OH and (+)[3H]SKF 10047 binding sites in rat brain membranes: evidence of multiplicity.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Haloperidol; In Vitro Techniques; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine

1987
Effects of phencyclidine, SKF 10,047 and related psychotomimetic agents on N-methyl-D-aspartate receptor mediated synaptic responses in rat hippocampal slices.
    British journal of pharmacology, 1987, Volume: 91, Issue:3

    Topics: Analgesics; Animals; Dioxolanes; Hallucinogens; Hippocampus; In Vitro Techniques; Ketamine; Kinetics; Magnesium; Neuromuscular Depolarizing Agents; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Synapses; Synaptic Transmission

1987
Comparison of the pharmacologic effects of N-allylnormetazocine and phencyclidine: sensitization, cross-sensitization, and opioid antagonist activity.
    Psychopharmacology, 1986, Volume: 89, Issue:2

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Male; Morphine Dependence; Motor Activity; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereoisomerism

1986
Oral self-administration of N-allylnormetazocine (SKF-10,047) stereoisomers in rhesus monkeys: substitution during phencyclidine self-administration and withdrawal.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:2

    Topics: Administration, Oral; Animals; Macaca mulatta; Male; Phenazocine; Phencyclidine; Self Administration; Stereoisomerism; Substance Withdrawal Syndrome

1988
Psychotomimetic sigma-ligands, dexoxadrol and phencyclidine block the same presynaptic potassium channel in rat brain.
    The Journal of physiology, 1988, Volume: 403

    Topics: Animals; Brain; Cyclazocine; Dioxolanes; Dioxoles; Dose-Response Relationship, Drug; Hallucinogens; In Vitro Techniques; Naloxone; Phenazocine; Phencyclidine; Piperidines; Potassium Channels; Rats; Synaptosomes

1988
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors

1987
The anticonvulsant MK-801 is a potent N-methyl-D-aspartate antagonist.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:18

    Topics: Animals; Anticonvulsants; Aspartic Acid; Binding Sites; Brain; Dibenzocycloheptenes; Dizocilpine Maleate; In Vitro Techniques; Ketamine; Male; N-Methylaspartate; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains

1986
Use of the radial maze in studies of phencyclidine and other drugs of abuse.
    Physiology & behavior, 1987, Volume: 40, Issue:6

    Topics: Animals; Brain; Learning; Lysergic Acid Diethylamide; Memory; Organ Specificity; Phenazocine; Phencyclidine; Scopolamine; Substance-Related Disorders; Verapamil

1987
Effects of sigma agonist compounds on local cerebral glucose utilization: relationship to psychotomimetic properties.
    Brain research, 1986, Jun-18, Volume: 376, Issue:1

    Topics: Animals; Brain; Dioxolanes; Dioxoles; Glucose; Hallucinogens; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains

1986
Electroencephalographic (EEG), EEG power spectra, and behavioral correlates in rats given phencyclidine.
    Neuropharmacology, 1986, Volume: 25, Issue:7

    Topics: Animals; Arousal; Behavior, Animal; Cerebral Cortex; Electroencephalography; Female; Ketamine; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereotyped Behavior

1986
Pharmacologic and reinforcing properties of phencyclidine and the enantiomers of N-allylnormetazocine in the dog.
    Drug and alcohol dependence, 1986, Volume: 18, Issue:2

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Decerebrate State; Dogs; Female; Morphine; Naltrexone; Phenazocine; Phencyclidine; Reinforcement Schedule; Self Administration; Stereoisomerism

1986
(+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine [(+)-3-PPP] but not (-)-3-PPP produces (+)-N-allylnormetazocine-like (SKF 10,047) discriminative stimuli.
    Life sciences, 1986, Dec-29, Volume: 39, Issue:26

    Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Isomerism; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred F344

1986
Demonstration and affinity labeling of a stereoselective binding site for a benzomorphan opiate on acetylcholine receptor-rich membranes from Torpedo electroplaque.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:3

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Electric Organ; Electrophoresis, Polyacrylamide Gel; Kinetics; Phenazocine; Phencyclidine; Photochemistry; Receptors, Cholinergic; Torpedo

1985
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
    Molecular pharmacology, 1986, Volume: 29, Issue:2

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine

1986
Effects of phencyclidine, N-allyl-N-normetazocine (SKF-10,047), and verapamil on performance in a radial maze.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:2

    Topics: Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Male; Memory; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Time Factors; Verapamil

1986
The convulsant and anticonvulsant effects of phencyclidine (PCP) and PCP analogues in the rat.
    Behavioural brain research, 1986, Volume: 19, Issue:2

    Topics: Animals; Anticonvulsants; Chemical Phenomena; Chemistry; Convulsants; Dose-Response Relationship, Drug; Female; Ketamine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1986
Stereoselective behavioral effects of N-allylnormetazocine in pigeons and squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:2

    Topics: Animals; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Morphine; Naloxone; Phenazocine; Phencyclidine; Reinforcement Schedule; Saimiri; Stereoisomerism

1985
Behavioral effects of selected opiates and phencyclidine in the nondependent and cyclazocine-dependent rhesus monkey.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Food; Macaca mulatta; Male; Naloxone; Phenazocine; Phencyclidine; Stereoisomerism; Substance-Related Disorders

1985
The effects of phencyclidine and N-allylnormetazocine on midbrain dopamine neuronal activity.
    European journal of pharmacology, 1984, Sep-17, Volume: 104, Issue:3-4

    Topics: Animals; Haloperidol; Iontophoresis; Male; Mesencephalon; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism

1984
Comparisons between phencyclidine, its monohydroxylated metabolites, and the stereoisomers of N-allyl-N-normetazocine (SKF 10047) as inhibitors of the muscarinic receptor and acetylcholinesterase.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:7

    Topics: Acetylcholinesterase; Animals; Behavior, Animal; Cholinesterase Inhibitors; In Vitro Techniques; Male; Membranes; Parasympatholytics; Phenazocine; Phencyclidine; Quinuclidinyl Benzilate; Rats; Stereoisomerism

1982
Progress report from the NIDA Addiction Research Center (preclinical laboratory), Lexington, Kentucky.
    NIDA research monograph, 1983, Volume: 43

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Cocaine; Dogs; Guinea Pigs; Humans; Kinetics; Male; Nicotine; Opioid-Related Disorders; Oxymorphone; Phenazocine; Phencyclidine; Rats; Self Administration; Stereoisomerism

1983
Phencyclidine-induced locomotor activity in the rat is blocked by 6-hydroxydopamine lesion of the nucleus accumbens: comparisons to other psychomotor stimulants.
    Psychopharmacology, 1984, Volume: 82, Issue:1-2

    Topics: Animals; Caffeine; Central Nervous System Stimulants; Dextroamphetamine; Hydroxydopamines; Motor Activity; Nucleus Accumbens; Oxidopamine; Phenazocine; Phencyclidine; Rats; Receptors, Dopamine; Scopolamine; Septal Nuclei

1984
Behavioral and biochemical stereoselectivity of sigma opiate/PCP receptors.
    Brain research, 1984, Feb-27, Volume: 294, Issue:1

    Topics: Animals; Behavior, Animal; Brain; Cyclazocine; Hydromorphone; In Vitro Techniques; Ketamine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism

1984
Stereoisomers of N-allylnormetazocine: phencyclidine-like behavioral effects in squirrel monkeys and rats.
    Science (New York, N.Y.), 1982, Jan-08, Volume: 215, Issue:4529

    Topics: Animals; Behavior, Animal; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Saimiri; Stereoisomerism; Structure-Activity Relationship

1982
Autoradiographic localization of the phencyclidine/sigma "opiate" receptor in rat brain.
    NIDA research monograph, 1982, Volume: 41

    Topics: Animals; Autoradiography; Brain; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tritium

1982
Anorexia and hyperphagia produced by five pharmacologic classes of hallucinogens.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:3

    Topics: Amphetamine; Animals; Anorexia; Atropine; Dextroamphetamine; Dogs; Dronabinol; Feeding and Eating Disorders; Feeding Behavior; Female; Hallucinogens; Humans; Lysergic Acid Diethylamide; Male; Phenazocine; Phencyclidine

1982
Modulation of phencyclidine receptor sensitivity.
    NIDA research monograph, 1983, Volume: 43

    Topics: Amantadine; Animals; In Vitro Techniques; Olfactory Bulb; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Stereoisomerism

1983
Naltrexone fails to antagonize the sigma effects of PCP and SKF 10,047 in the dog.
    European journal of pharmacology, 1983, Sep-02, Volume: 92, Issue:3-4

    Topics: Animals; Body Temperature; Dogs; Female; Heart Rate; Morphine; Naloxone; Naltrexone; Paraplegia; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Reflex

1983
Naloxone-inaccessible sigma receptor in rat central nervous system.
    Proceedings of the National Academy of Sciences of the United States of America, 1983, Volume: 80, Issue:21

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalins; Ethylketocyclazocine; Kinetics; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Spinal Cord; Tissue Distribution

1983
Blockade of long-term potentiation by phencyclidine and sigma opiates in the hippocampus in vivo and in vitro.
    Brain research, 1983, Nov-28, Volume: 280, Issue:1

    Topics: Animals; Cyclazocine; Drug Synergism; Hippocampus; Male; Membrane Potentials; Morphine; Naloxone; Narcotics; Phenazocine; Phencyclidine; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synapses; Synaptic Transmission

1983
Effects of SKF-10047 in the phencyclidine-dependent rat: evidence for common receptor mechanisms.
    Drug and alcohol dependence, 1983, Volume: 12, Issue:2

    Topics: Animals; Drug Tolerance; Female; Humans; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Substance Withdrawal Syndrome

1983
Ontogeny of sigma opiate/phencyclidine-binding sites in rat brain.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Aging; Animals; Brain; Female; Fetus; Gestational Age; Phenazocine; Phencyclidine; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1983
Characterization of specific sigma opiate/phencyclidine (PCP)-binding sites in the human brain.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Brain; Humans; Kinetics; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tissue Distribution

1983
Further characterization of the three-choice morphine, cyclazocine and saline discrimination paradigm: opioids with agonist and antagonist properties.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:1

    Topics: Animals; Cyclazocine; Discrimination Learning; Discrimination, Psychological; Ethylketocyclazocine; Male; Morphine; Narcotic Antagonists; Narcotics; Phenazocine; Phencyclidine; Rats; Sodium Chloride; Stereoisomerism

1983
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
    Life sciences, 1984, Feb-20, Volume: 34, Issue:8

    Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains

1984
Three-choice drug discrimination: phencyclidine-like stimulus effects of opioids.
    Psychopharmacology, 1983, Volume: 80, Issue:1

    Topics: Animals; Choice Behavior; Cyclazocine; Dextroamphetamine; Discrimination, Psychological; Male; Naltrexone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Secobarbital

1983
Spike and wave complexes produced by four hallucinogenic compounds in the cat.
    Physiology & behavior, 1984, Volume: 33, Issue:6

    Topics: Animals; Behavior, Animal; Cats; Electroencephalography; Hallucinogens; Ketamine; Limbic System; Phenazocine; Phencyclidine; Quipazine

1984
Phencyclidine-like discriminative stimulus properties of opioids in the squirrel monkey.
    Psychopharmacology, 1982, Volume: 77, Issue:4

    Topics: Animals; Cyclazocine; Discrimination Learning; Female; Male; Naltrexone; Narcotics; Phenazocine; Phencyclidine; Saimiri; Time Factors

1982
Pharmacological evaluation of N-allynormetazocine (SKF 10,047) on the basis of its discriminative stimulus properties in the rat.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:1

    Topics: Animals; Benzomorphans; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Male; Naloxone; Phenazocine; Phencyclidine; Propranolol; Rats; Rats, Inbred F344; Stereoisomerism

1983
Phencyclidine-like discriminative stimuli of (+)- and (-)-N-allylnormetazocine in rats.
    European journal of pharmacology, 1982, Oct-22, Volume: 84, Issue:3-4

    Topics: Animals; Discrimination Learning; Discrimination, Psychological; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Reinforcement Schedule; Stereoisomerism

1982
Effects of sigma and phencyclidine receptor ligands on electric field-stimulated rabbit ear artery constriction in vitro.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1994, Volume: 15, Issue:4

    Topics: Animals; Arteries; Dizocilpine Maleate; Ear; Electric Stimulation; Female; In Vitro Techniques; Ligands; Male; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Receptors, Phencyclidine; Receptors, sigma; Vasoconstriction

1994
Neuroendocrine responses produced by enantiomeric pairs of drugs that interact with phencyclidine and sigma receptors.
    European journal of pharmacology, 1994, Sep-22, Volume: 263, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Analgesics; Animals; Corticosterone; Dioxolanes; Drug Interactions; Hypothalamo-Hypophyseal System; Injections, Subcutaneous; Male; Phenazocine; Phencyclidine; Piperidines; Pituitary-Adrenal System; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stereoisomerism; Sympathomimetics

1994
NE-100, a novel sigma receptor ligand: in vivo tests.
    Life sciences, 1993, Volume: 53, Issue:18

    Topics: Animals; Anisoles; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Catalepsy; Dopamine Agents; Drug Interactions; Locomotion; Male; Phenazocine; Phencyclidine; Propylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Rats, Wistar; Receptors, sigma; Stereotyped Behavior

1993
FH-510, a potent and selective ligand for rat brain sigma recognition sites.
    European journal of pharmacology, 1993, Jul-06, Volume: 238, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain; Carbazoles; Dopamine; Haloperidol; Male; Mice; Phenazocine; Phencyclidine; Propylamines; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma; Stereotyped Behavior

1993
Effect of phencyclidine on contraction of porcine coronary vessel strips.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1993, Volume: 14, Issue:3

    Topics: Animals; Biological Assay; Coronary Vessels; Dextromethorphan; Dizocilpine Maleate; Haloperidol; In Vitro Techniques; Muscle, Smooth, Vascular; Myocardial Contraction; Phenazocine; Phencyclidine; Receptors, Phencyclidine; Receptors, sigma; Swine

1993
Different sensitivities of NMDA receptor channel subtypes to non-competitive antagonists.
    Neuroreport, 1993, Volume: 4, Issue:6

    Topics: Amino Acid Sequence; Animals; Dizocilpine Maleate; Ketamine; Magnesium; Molecular Sequence Data; Mutagenesis; Oocytes; Phenazocine; Phencyclidine; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Xenopus

1993
Dose-dependent effects of D-N-allylnormetazocine on regional cerebral metabolic rates for glucose.
    Brain research, 1993, Feb-12, Volume: 603, Issue:1

    Topics: Animals; Blood Glucose; Blood Pressure; Brain Chemistry; Brain Mapping; Deoxyglucose; Dose-Response Relationship, Drug; Glucose; Heart Rate; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Phencyclidine; Receptors, sigma

1993
(+)-SKF-10,047 and dextromethorphan ameliorate conditioned fear stress through the activation of phenytoin-regulated sigma 1 sites.
    European journal of pharmacology, 1996, Mar-28, Volume: 299, Issue:1-3

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Behavior, Animal; Dextromethorphan; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Male; Mice; Motor Activity; Phenazocine; Phencyclidine; Phenytoin; Pyrimidines; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Stress, Physiological

1996
The involvement of sigma receptors in the choice reaction performance deficits induced by phencyclidine.
    European journal of pharmacology, 1997, Jan-29, Volume: 319, Issue:2-3

    Topics: Animals; Anisoles; Antipsychotic Agents; Excitatory Amino Acid Agonists; Ligands; Male; Phenazocine; Phencyclidine; Piperidines; Propylamines; Psychomotor Performance; Rats; Rats, Wistar; Reaction Time; Receptors, sigma

1997
Sigma1 receptor subtype does not interact with stereotyped behaviors in rats.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 61, Issue:4

    Topics: Animals; Antipsychotic Agents; Male; Nootropic Agents; Phenazocine; Phencyclidine; Piperazines; Rats; Rats, Wistar; Receptors, sigma; Stereotyped Behavior

1998
Binding of [3H]desglycinyl remacemide to rat brain membranes: association with the benzomorphan attachment site of the N-methyl-D-aspartic acid receptor channel.
    Brain research, 1999, May-08, Volume: 827, Issue:1-2

    Topics: Animals; Antipsychotic Agents; Benzomorphans; Binding Sites; Brain Chemistry; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Haloperidol; Male; Membrane Proteins; Neurons; Phenazocine; Phencyclidine; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Subcellular Fractions; Tritium

1999
Pharmacological profile of MS-377, a novel antipsychotic agent with selective affinity for sigma receptors.
    Psychopharmacology, 1999, Volume: 145, Issue:3

    Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Dopamine Agonists; Free Radical Scavengers; Guinea Pigs; Haloperidol; Head Movements; Male; Mice; Phenazocine; Phencyclidine; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, sigma; Risperidone; Serotonin; Serotonin Antagonists; Stereotyped Behavior; Sulpiride; Tartrates

1999
Phencyclidine impairs latent learning in mice: interaction between glutamatergic systems and sigma(1) receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 24, Issue:4

    Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Behavior, Animal; Cycloserine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Exploratory Behavior; Glutamic Acid; Learning; Male; Mice; Mice, Inbred Strains; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Piperazines; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism

2001
MS-377, a selective sigma receptor ligand, indirectly blocks the action of PCP in the N-methyl-D-aspartate receptor ion-channel complex in primary cultured rat neuronal cells.
    Life sciences, 2002, Feb-22, Volume: 70, Issue:14

    Topics: Animals; Antipsychotic Agents; Calcium; Cells, Cultured; Dizocilpine Maleate; Female; Ion Channels; Neurons; Phenazocine; Phencyclidine; Piperazines; Pregnancy; Pyrrolidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Tartrates; Tritium

2002
Characterization of the non-competitive antagonist binding site of the NMDA receptor in dark Agouti rats.
    Life sciences, 2004, Aug-06, Volume: 75, Issue:12

    Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dioxolanes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Female; Ketamine; N-Methylaspartate; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Mutant Strains; Receptors, N-Methyl-D-Aspartate; Scintillation Counting; Tritium

2004
Inhibition of hyperpolarization-activated cation currents by phencyclidine and some sigma ligands in rat hippocampal CA1 pyramidal neurons in vitro.
    Neuropharmacology, 2007, Volume: 53, Issue:3

    Topics: Animals; Animals, Newborn; Cesium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Ion Channels; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Phenazocine; Phencyclidine; Pyramidal Cells; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma

2007
Sigma-1 receptor function is critical for both the discriminative stimulus and aversive effects of the kappa-opioid receptor agonist U-50488H.
    Addiction biology, 2012, Volume: 17, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anisoles; Avoidance Learning; Conditioning, Psychological; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Propylamines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor

2012