phenazocine has been researched along with phencyclidine in 129 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 90 (69.77) | 18.7374 |
1990's | 34 (26.36) | 18.2507 |
2000's | 4 (3.10) | 29.6817 |
2010's | 1 (0.78) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Grynne, BH; Holmen, AT; Maurset, A | 1 |
Abraham, P; Bai, X; Brine, GA; Carroll, FI; Martin, BR; Mascarella, SW; May, EL; Parham, K; Sauss, C; Zhang, X | 1 |
Lemaire, S; Rogers, C | 1 |
Hudzik, TJ; Slifer, BL | 1 |
Boyce, S; Cook, G; Iversen, SD; Rupniak, NM; Steventon, MJ | 1 |
deCosta, BR; Hardwick, WC; McMillan, DE; Rice, KC | 1 |
Katki, AG; Munson, PJ; Rodbard, D; Schwarz, S; Zhou, GZ | 1 |
Carter, AJ; Müller, RE | 1 |
Pèzzola, A; Popoli, P; Sagratella, S; Scotti de Carolis, A | 1 |
Brent, PJ | 1 |
Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauché, D | 1 |
Burke, M; Earley, B; Gouret, CJ; Junien, JL; Leonard, BE | 1 |
Feuerstein, G; Lysko, PG | 1 |
Connick, JH; Fox, PK; France, L; Hanlon, GM; Nicholson, CD | 1 |
Su, TP; Wu, XZ | 1 |
Bejanian, M; George, R; Pechnick, RN | 1 |
Bauerle, LM; DeNoble, VJ; Jones, KW | 1 |
Bueno, L; Fioramonti, J; Gue, M; Junien, JL; Pascaud, X | 1 |
Beinfeld, MC; Brog, JS | 1 |
Katki, AG; Rodbard, D; Schwarz, S; Zhou, GZ | 1 |
DeLander, GE; Wahl, JJ | 1 |
Oswald, RE; Papke, RL | 1 |
France, CP; Snyder, AM; Woods, JH | 1 |
Alerhand, S; Itzhak, Y | 1 |
Cheng, BK; Contreras, PC; Gray, NM; Lair, CM; Mick, SJ | 1 |
Wann, KT; Wardley-Smith, B | 1 |
Iversen, SD; Oles, RJ; Preston, C; Singh, L; Tricklebank, MD | 1 |
Gussio, RP; Marquis, KL; Moreton, JE; Paquette, NC | 1 |
Allikmets, LKh; Kharro, IaE; Lang, AE; Vasar, EE | 1 |
Duffy, O; Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauche, D | 1 |
Jackson, A; Sanger, DJ | 3 |
McMillan, DE; Wessinger, WD | 1 |
Iversen, SD; Oles, RJ; Singh, L; Tricklebank, MD; Wong, EH | 1 |
Catt, KJ; Dufau, ML; Stojilković, SS | 1 |
Knight, AR; Wong, EH; Woodruff, GN | 1 |
Beart, PM; Manallack, DT | 1 |
Itzhak, Y; Khouri, M | 1 |
Kushner, L; Zukin, RS; Zukin, SR | 1 |
Contreras, PC; DiMaggio, DA; O'Donohue, TL | 1 |
Alberici, GP; Cook, L; Steinfels, GF; Tam, SW | 1 |
Holtzman, SG | 2 |
Downes, CP; Lewis, PE; Stone, MA | 1 |
French, ED | 1 |
Chang, KJ; Ferris, RM; Russell, A; Tang, FL | 1 |
Chung, JM; Kim, J; Shin, HK; Willcockson, WS; Willis, WD | 1 |
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K | 1 |
Braunwalder, AF; Lehmann, J; Loo, PS; Sills, MA; Williams, M | 1 |
Itzhak, Y | 2 |
Furukawa, H; Hiramatsu, M; Kameyama, T; Nabeshima, T | 1 |
Gundlach, AL; Largent, BL; Snyder, SH | 4 |
Goldman, ME; Jacobson, AE; Paul, SM; Rice, KC | 1 |
Greenberg, BD; Segal, DS | 1 |
Jacobson, AE; Koek, W; Lessor, RA; Rice, KC; Woods, JH | 1 |
Ieni, JR; Nichtenhauser, R; Sircar, R; Zukin, SR | 1 |
Su, TP; Weissman, AD; Yeh, SY | 1 |
Sircar, R; Zukin, SR | 3 |
Contreras, PC; DiMaggio, DA; O'Donohue, TL; Quirion, R | 1 |
Contreras, PC; O'Donohue, TL; Quirion, R | 2 |
Hiramatsu, M; Kameyama, T; Nabeshima, T | 2 |
Dykstra, LA; Slifer, BL | 2 |
Cook, L; Steinfels, GF; Tam, SW | 2 |
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR | 1 |
Coan, EJ; Collingridge, GL | 1 |
Iwamoto, ET | 1 |
Carroll, ME | 1 |
Bartschat, DK; Blaustein, MP | 1 |
Dykstra, LA; Picker, M | 1 |
Iversen, LL; Kemp, JA; Knight, AR; Priestley, T; Wong, EH; Woodruff, GN | 1 |
McCann, DJ; Rabin, RA; Winter, JC | 1 |
Kozlowski, MR | 1 |
Mattia, A; Moreton, JE | 1 |
Risner, ME; Shannon, HE; Vaupel, DB | 1 |
McLaughlin, JT; Oswald, RE; Pennow, NN | 1 |
Bigelow, J; Michel, L; Oswald, RE | 1 |
McCann, DJ; Winter, JC | 1 |
Leccese, AP; Marquis, KL; Mattia, A; Moreton, JE | 1 |
Clark, RD; Katz, JL; Spealman, RD | 1 |
Bergman, J; Hassoun, J; Schuster, CR | 1 |
Bunney, BS; Freeman, AS | 1 |
Hillman, GR; Johnson, KM | 1 |
Cone, EJ; Goldberg, SR; Gorodetzky, CW; Herling, S; Risner, ME; Shannon, HE; Vaupel, DB | 1 |
French, ED; Vantini, G | 1 |
Balster, RL; Brady, KT; Slifer, BL; Zukin, SR | 1 |
Balster, RL; Brady, KT; May, EL | 1 |
Hammer, RP; Herkenham, M; Pert, CB; Quirion, R | 1 |
Morton, EC; Vaupel, DB | 1 |
Pert, CB; Quirion, R | 1 |
Vaupel, DB | 1 |
Tam, SW | 1 |
Greenfield, LJ; Guyenet, PG; Hackett, JT; Stringer, JL | 1 |
Stafford, I; Tomie, A; Wagner, GC | 1 |
Holtzman, SG; White, JM | 2 |
Johnson, KM; Leventer, SM | 1 |
Contreras, CM; Ervin, FR; Guzman-Flores, C; Mexicano, G; Palmour, R | 1 |
Shannon, HE | 2 |
Bao, WL; Sun, FY; Zhang, AZ; Zhen, FC | 1 |
Pechnick, RN; Poland, RE | 1 |
Ajima, A; Araki, H; Imagawa, Y; Muramatsu, M; Nakazato, A; Ogawa, S; Okuyama, S; Tanaka, M; Yamaguchi, K; Yoshida, M | 1 |
Chaki, S; Imagawa, Y; Muramatsu, M; Okuyama, S; Otomo, S; Tanaka, M | 1 |
De Souza, EB; Wolfe, SA | 1 |
Shi, GG; Xu, SF | 1 |
Masaki, H; Mishina, M; Mori, H; Shimoji, K; Yamakura, T | 1 |
della Puppa, A; Kimes, AS; London, ED | 1 |
Kamei, H; Kameyama, T; Nabeshima, T | 1 |
Amano, M; Matsuno, K; Nabeshima, T; Yamada, K | 1 |
Jin, J; Watanabe, S; Yamamoto, T | 1 |
Kobayashi, T; Matsuno, K; Mita, S | 1 |
Ahmed, MS; Enna, SJ; Mather, A | 1 |
Horikomi, K; Iizuka, K; Mita, N; Miwa, T; Nagase, H; Sakai, K; Sonehara, K; Takagi, K; Takahashi, S | 1 |
Furukawa, H; Ichihara, K; Kamei, H; Mamiya, T; Nabeshima, T; Nagai, T; Noda, A; Noda, Y; Sugiura, S | 1 |
Horikomi, K; Karasawa, J; Sagi, N; Sora, I; Yamamoto, H; Yamamoto, T | 1 |
Sun, W; Wessinger, WD | 1 |
Tanabe, M | 1 |
Isotani, K; Mori, T; Narita, M; Nomura, M; Suzuki, T; Torigoe, K; Tsukiyama, Y; Yoshizawa, K | 1 |
3 review(s) available for phenazocine and phencyclidine
Article | Year |
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Drug discrimination studies.
Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Sigma and phencyclidine receptors in the brain-endocrine-immune axis.
Topics: Animals; Autoradiography; Brain Chemistry; Endocrine Glands; Humans; Hypophysectomy; Lymphocytes; Phenazocine; Phencyclidine; Receptors, Phencyclidine; Receptors, sigma | 1993 |
[Neuropharmacological effects of sigma receptor ligands: anxiolytic, anti-amnesic and neuroprotective effects].
Topics: Animals; Antipsychotic Agents; Anxiety; Brain Ischemia; Cinnamates; Cyclopropanes; Humans; Learning Disabilities; Memory Disorders; Phenazocine; Phencyclidine; Receptors, sigma | 1996 |
126 other study(ies) available for phenazocine and phencyclidine
Article | Year |
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Evidence for distinct phencyclidine and SKF10047 receptors following detergent treatment of rat brain membranes.
Topics: Animals; Brain Chemistry; Cell Membrane; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Synaptosomes; Tritium | 1992 |
Enantiomeric N-substituted N-normetazocines: a comparative study of affinities at sigma, PCP, and mu opioid receptors.
Topics: Animals; Brain; Guinea Pigs; Male; Narcotics; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism; Substrate Specificity | 1992 |
Characterization of [3H]desmethylimipramine binding in bovine adrenal medulla: interactions with sigma- and (or) phencyclidine-receptor ligands.
Topics: Adrenal Medulla; Animals; Binding Sites; Cattle; Desipramine; Dextromethorphan; Dizocilpine Maleate; Phenazocine; Phencyclidine; Piperidines; Potassium Chloride; Receptors, Opioid, delta; Receptors, Phencyclidine; Tranquilizing Agents | 1992 |
Interaction of sigma and PCP-like drugs on operant behaviors in the rat.
Topics: Animals; Conditioning, Operant; Dextroamphetamine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Pentazocine; Phenazocine; Phencyclidine; Psychotropic Drugs; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule | 1992 |
Psychomotor activity and cognitive disruption attributable to NMDA, but not sigma, interactions in primates.
Topics: Animals; Ataxia; Cognition; Dizocilpine Maleate; Macaca mulatta; Male; Pentazocine; Phenazocine; Phencyclidine; Psychomotor Performance; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Saimiri; Space Perception | 1991 |
Effects of drugs that bind to PCP and sigma receptors on punished responding.
Topics: Animals; Buspirone; Dizocilpine Maleate; Haloperidol; Learning; Male; Pentobarbital; Phenazocine; Phencyclidine; Punishment; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1991 |
Quantitative characterization of multiple binding sites for phencyclidine and N-allylnormetazocine in membranes from rat and guinea pig brain.
Topics: Animals; Binding Sites; Brain; Cell Membrane; Guinea Pigs; Male; Phenazocine; Phencyclidine; Psychotropic Drugs; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma | 1991 |
Activation of excitatory amino acid receptors cannot alone account for anoxia-induced impairment of protein synthesis in rat hippocampal slices.
Topics: Animals; Aspartic Acid; Carbon Radioisotopes; Dizocilpine Maleate; Glutamates; Glutamic Acid; Hippocampus; Hypoxia; Kainic Acid; Lysine; Male; N-Methylaspartate; Nerve Tissue Proteins; Phenazocine; Phencyclidine; Quisqualic Acid; Rats; Receptors, Amino Acid; Receptors, Cell Surface; Receptors, N-Methyl-D-Aspartate | 1991 |
Behavioural and electoencephalographic interactions between haloperidol and PCP/sigma ligands in the rat.
Topics: 2-Amino-5-phosphonovalerate; Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Catalepsy; Electroencephalography; Haloperidol; Isoquinolines; Kinetics; Male; Phenazocine; Phencyclidine; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Spiperone | 1991 |
Similar behavioural effects of sigma agonists and PCP-like non-competitive NMDA antagonists in guinea-pigs.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Dizocilpine Maleate; Dopamine Agents; Dopamine Antagonists; Ergolines; Female; Guanidines; Guinea Pigs; Haloperidol; Ketamine; Male; Motor Activity; N-Methylaspartate; Pentazocine; Phenazocine; Phencyclidine; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride | 1991 |
JO 1784, a potent and selective ligand for rat and mouse brain sigma-sites.
Topics: Animals; Brain Chemistry; Cinnamates; Cyclopropanes; In Vitro Techniques; Male; Mice; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta | 1990 |
A comparison of the psychopharmacological profiles of phencyclidine, ketamine and (+) SKF 10,047 in the trimethyltin rat model.
Topics: Animals; Avoidance Learning; Behavior, Animal; Brain Chemistry; Ketamine; Learning; Male; Nervous System Diseases; Neurotransmitter Agents; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine; Swimming; Trimethyltin Compounds | 1990 |
Excitatory amino acid neurotoxicity at the N-methyl-D-aspartate receptor in cultured neurons: protection by SKF 10,047.
Topics: Animals; Cell Survival; Cells, Cultured; Cerebellum; Dopamine Agents; Glutamates; Glutamic Acid; Neurons; Neurotoxins; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1990 |
The lack of utility of the rat vas deferens as a functional bioassay for sigma ligands.
Topics: Animals; Binding Sites; Biological Assay; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; Male; Muscle Contraction; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Vas Deferens | 1991 |
Guinea pig vas deferens contains sigma but not phencyclidine receptors.
Topics: Animals; Binding, Competitive; Guinea Pigs; Male; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Vas Deferens | 1990 |
Effects of acute and chronic administration of (+)-SKF 10,047 on body temperature in the rat: cross-sensitization with phencyclidine.
Topics: Animals; Body Temperature; Body Weight; Dose-Response Relationship, Drug; Drug Interactions; Injections, Subcutaneous; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1990 |
Differential effects of sigma and phencyclidine receptor ligands on learning.
Topics: Animals; Avoidance Learning; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Ligands; Male; Memory; Pentazocine; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Retention, Psychology | 1990 |
Selective stimulation of colonic motor response to a meal by sigma ligands in dogs.
Topics: Animals; Cinnamates; Colon; Cyclopropanes; Dogs; Drug Antagonism; Eating; Gastrointestinal Motility; Guanidines; Injections, Intravenous; Injections, Intraventricular; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1990 |
Inhibition of carbachol-induced inositol phosphate accumulation by phencyclidine, phencyclidine-like ligands and sigma agonists involves blockade of the muscarinic cholinergic receptor: a novel dioxadrol-preferring interaction.
Topics: Animals; Brain; Carbachol; Culture Techniques; Dibenzocycloheptenes; Dioxolanes; Dizocilpine Maleate; Inositol Phosphates; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Sigma Factor; Transcription Factors | 1990 |
Differential modulation by cations of sigma and phencyclidine binding sites in rat brain.
Topics: Animals; Binding Sites; Brain; Cations; Dose-Response Relationship, Drug; Haloperidol; Ligands; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Sigma Factor; Tritium | 1990 |
In vivo characterization of phencyclidine/sigma agonist-mediated inhibition of nociception.
Topics: Animals; Anticonvulsants; Aspartic Acid; Behavior, Animal; Binding, Competitive; Dibenzocycloheptenes; Dizocilpine Maleate; Male; Mice; N-Methylaspartate; Nociceptors; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, Opioid, delta; Substance P | 1989 |
Mechanisms of noncompetitive inhibition of acetylcholine-induced single-channel currents.
Topics: Acetylcholine; Biomechanical Phenomena; Cell Line; Electric Conductivity; Electrophysiology; Ion Channels; Phenazocine; Phencyclidine; Tetracaine; Time Factors | 1989 |
Analgesic effects of phencyclidine-like drugs in rhesus monkeys.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Alfentanil; Analgesia; Analgesics; Anesthetics; Animals; Anticonvulsants; Dextrorphan; Dibenzocycloheptenes; Discrimination, Psychological; Dizocilpine Maleate; Dose-Response Relationship, Drug; Fentanyl; Ketamine; Macaca mulatta; Phenazocine; Phencyclidine; Pyrrolidines | 1989 |
Differential regulation of sigma and PCP receptors after chronic administration of haloperidol and phencyclidine in mice.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Hallucinogens; Haloperidol; Male; Mice; Mice, Inbred Strains; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Time Factors | 1989 |
Phencyclidine-like effects of tetrahydroisoquinolines and related compounds.
Topics: Animals; Ataxia; Behavior, Animal; Chemical Phenomena; Chemistry; Isoquinolines; Male; Molecular Structure; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereotyped Behavior; Structure-Activity Relationship; Tetrahydroisoquinolines | 1989 |
The effects of non-competitive NMDA receptor antagonists on rats exposed to hyperbaric pressure.
Topics: Animals; Binding, Competitive; Dibenzocycloheptenes; Dizocilpine Maleate; Hyperbaric Oxygenation; Ketamine; Male; Myoclonus; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Seizures; Tremor | 1989 |
The behavioural effects of MK-801: a comparison with antagonists acting non-competitively and competitively at the NMDA receptor.
Topics: Animals; Anticonvulsants; Aspartic Acid; Behavior, Animal; Binding, Competitive; Dibenzocycloheptenes; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Male; Motor Activity; N-Methylaspartate; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Seizures | 1989 |
Comparative electroencephalographic and behavioral effects of phencyclidine, (+)-SKF-10,047 and MK-801 in rats.
Topics: Animals; Anticonvulsants; Dibenzocycloheptenes; Dizocilpine Maleate; Electroencephalography; Female; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, sigma; Stereotyped Behavior | 1989 |
[Adaptive changes in sigma and phencyclidine receptors during the long-term use of haloperidol and raclopride in rats].
Topics: Adaptation, Physiological; Animals; Apomorphine; Behavior, Animal; Drug Interactions; Haloperidol; Ketamine; Phenazocine; Phencyclidine; Raclopride; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Salicylamides; Time Factors; Tritium | 1989 |
Neuropeptide Y and peptide YY interact with rat brain sigma and PCP binding sites.
Topics: Animals; Brain Chemistry; Haloperidol; In Vitro Techniques; Male; Neuropeptide Y; Pentazocine; Peptide YY; Peptides; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1989 |
Conditioned taste aversions induced by phencyclidine and other antagonists of N-methyl-D-aspartate.
Topics: Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Avoidance Learning; Conditioning, Operant; Male; N-Methylaspartate; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Taste | 1989 |
Effects of phencyclidine and other N-methyl-D-aspartate antagonists on the schedule-controlled behavior of rats.
Topics: Animals; Aspartic Acid; Conditioning, Psychological; Dibenzocycloheptenes; Dizocilpine Maleate; Male; N-Methylaspartate; Phenazocine; Phencyclidine; Piperazines; Piperidines; Punishment; Rats; Rats, Inbred Strains; Reinforcement Schedule; Stereoisomerism | 1989 |
Interaction of the discriminative stimulus effects of phencyclidine with those of (+)-N-allylnormetazocine, pentobarbital and d-amphetamine.
Topics: Amphetamines; Animals; Columbidae; Discrimination Learning; Drug Interactions; Pentobarbital; Phenazocine; Phencyclidine; Substance-Related Disorders | 1989 |
A role for receptors of N-methyl-D-aspartic acid in the discriminative stimulus properties of phencyclidine.
Topics: Animals; Discrimination, Psychological; Generalization, Stimulus; Haloperidol; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter | 1987 |
Receptors and secretory actions of sigma/phencyclidine agonists in anterior pituitary cells.
Topics: Animals; Cell Membrane; Cells, Cultured; Etorphine; Female; Kinetics; Luteinizing Hormone; Phenazocine; Phencyclidine; Pituitary Gland, Anterior; Potassium; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Thermodynamics | 1987 |
[3H]MK-801 labels a site on the N-methyl-D-aspartate receptor channel complex in rat brain membranes.
Topics: Animals; Anticonvulsants; Brain; Cations, Divalent; Cell Membrane; Cerebral Cortex; Dibenzocycloheptenes; Dizocilpine Maleate; Kinetics; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Tissue Distribution; Tritium | 1988 |
Quantitative conformational analyses predict distinct receptor sites for PCP-like and sigma drugs.
Topics: Animals; Binding Sites; Brain; Computer Graphics; Dibenzocycloheptenes; Dizocilpine Maleate; In Vitro Techniques; Isoquinolines; Male; Molecular Conformation; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1987 |
Regulation of the binding of sigma- and phencyclidine (PCP)-receptor ligands in rat brain membranes by guanine nucleotides and ions.
Topics: Animals; Binding, Competitive; Brain; Cations; Guanine Nucleotides; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine; Subcellular Fractions | 1988 |
Characterization of opioid, sigma, and phencyclidine receptors in the neuroblastoma-brain hybrid cell line NCB-20.
Topics: Animals; Brain Chemistry; Cell Line; Cricetinae; Hybrid Cells; Kinetics; Mice; Neuroblastoma; Phenazocine; Phencyclidine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1988 |
An endogenous ligand for the sigma opioid binding site.
Topics: Animals; Brain; Endorphins; Kinetics; Ligands; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Swine | 1987 |
Biochemical, behavioral, and electrophysiologic actions of the selective sigma receptor ligand (+)-pentazocine.
Topics: Animals; Avoidance Learning; Brain; Discrimination Learning; Evoked Potentials, Visual; Male; Membranes; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Reference Values | 1988 |
A comparison of the binding of sigma opioids and phencyclidine, and the interaction with antipsychotic drugs in rat brain membranes.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Brain; Corpus Striatum; Endorphins; Haloperidol; In Vitro Techniques; Male; Membranes; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, delta | 1986 |
Effects of N-allylnormetazocine (SKF 10,047), phencyclidine, and other psychomotor stimulants in the rat following 6-hydroxydopamine lesion of the ventral tegmental area.
Topics: Amphetamine; Animals; Apomorphine; Caffeine; Central Nervous System Stimulants; Dopamine; Hydroxydopamines; Male; Motor Activity; Oxidopamine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Scopolamine; Tegmentum Mesencephali | 1986 |
Evidence that the potential antipsychotic agent rimcazole (BW 234U) is a specific, competitive antagonist of sigma sites in brain.
Topics: Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Brain; Carbazoles; Clozapine; Guinea Pigs; Kinetics; Male; Methylphenidate; Mice; Phenazocine; Phencyclidine; Phenoxybenzamine; Propranolol; Receptors, Opioid; Receptors, sigma; Sulpiride | 1986 |
Actions of opioids on primate spinothalamic tract neurons.
Topics: Animals; Dynorphins; Enkephalin, Methionine; Macaca fascicularis; Morphine; Naloxone; Narcotics; Neurons; Phenazocine; Phencyclidine; Spinal Cord; Thalamus | 1986 |
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid | 1987 |
Interaction of L-glutamate and magnesium with phencyclidine recognition sites in rat brain: evidence for multiple affinity states of the phencyclidine/N-methyl-D-aspartate receptor complex.
Topics: Animals; Brain; Glutamates; Glutamic Acid; In Vitro Techniques; Kinetics; Magnesium; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1987 |
Pharmacological specificity of some psychotomimetic and antipsychotic agents for the sigma and PCP binding sites.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Haloperidol; In Vitro Techniques; Male; Phenazocine; Phencyclidine; Piperidines; Psychotropic Drugs; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1988 |
Different effects of ethylketocyclazocine on phencyclidine- and N-allylnormetazocine-induced stereotyped behaviors in rats.
Topics: Analgesics, Opioid; Animals; Cyclazocine; Ethylketocyclazocine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereotyped Behavior | 1987 |
Is the discriminative stimulus produced by phencyclidine due to an interaction with N-methyl-D-aspartate receptors?
Topics: Adrenergic beta-Antagonists; Animals; Anticonvulsants; Chlordiazepoxide; Dibenzocycloheptenes; Discrimination, Psychological; Dizocilpine Maleate; Drug Interactions; Generalization, Stimulus; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter | 1988 |
Phencyclidine and sigma opiate receptors in brain: biochemical and autoradiographical differentiation.
Topics: Autoradiography; Brain; Humans; In Vitro Techniques; Membranes; Phenazocine; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine | 1985 |
Differentiation of [3H]phencyclidine and (+)-[3H]SKF-10,047 binding sites in rat cerebral cortex.
Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism | 1985 |
Evidence for multiple opiate receptor involvement in different phencyclidine-induced unconditioned behaviors in rats.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Eating; Habituation, Psychophysiologic; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereotyped Behavior | 1986 |
Metaphit, a proposed phencyclidine receptor acylator: phencyclidine-like behavioral effects and evidence of absence of antagonist activity in pigeons and in rhesus monkeys.
Topics: Acylation; Animals; Ataxia; Catalepsy; Columbidae; Discrimination Learning; Drug Synergism; Ketamine; Macaca mulatta; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Species Specificity; Stereotyped Behavior | 1986 |
Characterization and autoradiographic visualization of (+)-[3H]SKF10,047 binding in rat and mouse brain: further evidence for phencyclidine/"sigma opiate" receptor commonality.
Topics: Animals; Autoradiography; Brain Chemistry; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Species Specificity; Tritium | 1986 |
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays.
Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma | 1986 |
Characterization of phencyclidine and sigma receptor-binding sites in brain.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Kinetics; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tritium | 1986 |
Further evidence of phencyclidine/sigma opioid receptor commonality.
Topics: Animals; Autoradiography; Brain; Kinetics; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tissue Distribution; Tritium | 1986 |
Isolation and identification of an endogenous ligand for the phencyclidine receptor.
Topics: Animals; Binding, Competitive; Brain; Brain Chemistry; Endopeptidases; Nerve Tissue Proteins; Neuropeptides; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Swine; Tissue Distribution | 1986 |
Agonistic and antagonistic effects of PCP-derivatives and sigma opioids in PCP behavioral and receptor assays.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclazocine; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereotyped Behavior; Structure-Activity Relationship; Tritium | 1986 |
Sigma receptors on NCB-20 hybrid neurotumor cells labeled with (+)[3H]SKF 10,047 and (+)[3H]3-PPP.
Topics: Animals; Brain; Cells, Cultured; Cricetinae; Cricetulus; Hybrid Cells; Kinetics; Neuroblastoma; Phenazocine; Phencyclidine; Piperidines; Receptors, Opioid; Receptors, Opioid, delta; Stereoisomerism | 1986 |
Autoradiographic distribution of phencyclidine receptors in the rat brain using [3H]1-(1-(2-thienyl)cyclohexyl)piperidine ([3H]TCP).
Topics: Animals; Autoradiography; Brain; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1986 |
Pharmacological and autoradiographic discrimination of sigma and phencyclidine receptor binding sites in brain with (+)-[3H]SKF 10,047, (+)-[3H]-3-[3-hydroxyphenyl]-N-(1-propyl)piperidine and [3H]-1-[1-(2-thienyl)cyclohexyl]piperidine.
Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; In Vitro Techniques; Kinetics; Male; Phenazocine; Phencyclidine; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism | 1986 |
Phencyclidine-induced stereotyped behaviors after injection of morphine and N-allylnormetazocine (SKF 10,047) in rats.
Topics: Animals; Male; Morphine; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereotyped Behavior | 1986 |
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid | 1986 |
Discriminative stimulus effects of N-allylnormetazocine in rats trained to discriminate a kappa from a sigma agonist.
Topics: Animals; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, sigma; Stereoisomerism | 1987 |
Discriminative stimulus properties of (+)-N-allylnormetazocine in the rat: correlations with (+)-N-allylnormetazocine and phencyclidine receptor binding.
Topics: Animals; Brain; Cyclazocine; Discrimination Learning; Ketamine; Male; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism | 1987 |
The effects of N-allylnormetazocine on electric shock titration in squirrel monkeys.
Topics: Animals; Avoidance Learning; Electroshock; Male; Morphine; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma; Reinforcement Schedule; Saimiri; Stereoisomerism | 1987 |
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1987 |
[3H]PCP-3-OH and (+)[3H]SKF 10047 binding sites in rat brain membranes: evidence of multiplicity.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Haloperidol; In Vitro Techniques; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1987 |
Effects of phencyclidine, SKF 10,047 and related psychotomimetic agents on N-methyl-D-aspartate receptor mediated synaptic responses in rat hippocampal slices.
Topics: Analgesics; Animals; Dioxolanes; Hallucinogens; Hippocampus; In Vitro Techniques; Ketamine; Kinetics; Magnesium; Neuromuscular Depolarizing Agents; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Synapses; Synaptic Transmission | 1987 |
Comparison of the pharmacologic effects of N-allylnormetazocine and phencyclidine: sensitization, cross-sensitization, and opioid antagonist activity.
Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Male; Morphine Dependence; Motor Activity; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereoisomerism | 1986 |
Oral self-administration of N-allylnormetazocine (SKF-10,047) stereoisomers in rhesus monkeys: substitution during phencyclidine self-administration and withdrawal.
Topics: Administration, Oral; Animals; Macaca mulatta; Male; Phenazocine; Phencyclidine; Self Administration; Stereoisomerism; Substance Withdrawal Syndrome | 1988 |
Psychotomimetic sigma-ligands, dexoxadrol and phencyclidine block the same presynaptic potassium channel in rat brain.
Topics: Animals; Brain; Cyclazocine; Dioxolanes; Dioxoles; Dose-Response Relationship, Drug; Hallucinogens; In Vitro Techniques; Naloxone; Phenazocine; Phencyclidine; Piperidines; Potassium Channels; Rats; Synaptosomes | 1988 |
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors | 1987 |
The anticonvulsant MK-801 is a potent N-methyl-D-aspartate antagonist.
Topics: Animals; Anticonvulsants; Aspartic Acid; Binding Sites; Brain; Dibenzocycloheptenes; Dizocilpine Maleate; In Vitro Techniques; Ketamine; Male; N-Methylaspartate; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains | 1986 |
Use of the radial maze in studies of phencyclidine and other drugs of abuse.
Topics: Animals; Brain; Learning; Lysergic Acid Diethylamide; Memory; Organ Specificity; Phenazocine; Phencyclidine; Scopolamine; Substance-Related Disorders; Verapamil | 1987 |
Effects of sigma agonist compounds on local cerebral glucose utilization: relationship to psychotomimetic properties.
Topics: Animals; Brain; Dioxolanes; Dioxoles; Glucose; Hallucinogens; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains | 1986 |
Electroencephalographic (EEG), EEG power spectra, and behavioral correlates in rats given phencyclidine.
Topics: Animals; Arousal; Behavior, Animal; Cerebral Cortex; Electroencephalography; Female; Ketamine; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereotyped Behavior | 1986 |
Pharmacologic and reinforcing properties of phencyclidine and the enantiomers of N-allylnormetazocine in the dog.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Decerebrate State; Dogs; Female; Morphine; Naltrexone; Phenazocine; Phencyclidine; Reinforcement Schedule; Self Administration; Stereoisomerism | 1986 |
(+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine [(+)-3-PPP] but not (-)-3-PPP produces (+)-N-allylnormetazocine-like (SKF 10,047) discriminative stimuli.
Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Isomerism; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred F344 | 1986 |
Demonstration and affinity labeling of a stereoselective binding site for a benzomorphan opiate on acetylcholine receptor-rich membranes from Torpedo electroplaque.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Electric Organ; Electrophoresis, Polyacrylamide Gel; Kinetics; Phenazocine; Phencyclidine; Photochemistry; Receptors, Cholinergic; Torpedo | 1985 |
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine | 1986 |
Effects of phencyclidine, N-allyl-N-normetazocine (SKF-10,047), and verapamil on performance in a radial maze.
Topics: Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Male; Memory; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Time Factors; Verapamil | 1986 |
The convulsant and anticonvulsant effects of phencyclidine (PCP) and PCP analogues in the rat.
Topics: Animals; Anticonvulsants; Chemical Phenomena; Chemistry; Convulsants; Dose-Response Relationship, Drug; Female; Ketamine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Structure-Activity Relationship | 1986 |
Stereoselective behavioral effects of N-allylnormetazocine in pigeons and squirrel monkeys.
Topics: Animals; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Morphine; Naloxone; Phenazocine; Phencyclidine; Reinforcement Schedule; Saimiri; Stereoisomerism | 1985 |
Behavioral effects of selected opiates and phencyclidine in the nondependent and cyclazocine-dependent rhesus monkey.
Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Food; Macaca mulatta; Male; Naloxone; Phenazocine; Phencyclidine; Stereoisomerism; Substance-Related Disorders | 1985 |
The effects of phencyclidine and N-allylnormetazocine on midbrain dopamine neuronal activity.
Topics: Animals; Haloperidol; Iontophoresis; Male; Mesencephalon; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism | 1984 |
Comparisons between phencyclidine, its monohydroxylated metabolites, and the stereoisomers of N-allyl-N-normetazocine (SKF 10047) as inhibitors of the muscarinic receptor and acetylcholinesterase.
Topics: Acetylcholinesterase; Animals; Behavior, Animal; Cholinesterase Inhibitors; In Vitro Techniques; Male; Membranes; Parasympatholytics; Phenazocine; Phencyclidine; Quinuclidinyl Benzilate; Rats; Stereoisomerism | 1982 |
Progress report from the NIDA Addiction Research Center (preclinical laboratory), Lexington, Kentucky.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Cocaine; Dogs; Guinea Pigs; Humans; Kinetics; Male; Nicotine; Opioid-Related Disorders; Oxymorphone; Phenazocine; Phencyclidine; Rats; Self Administration; Stereoisomerism | 1983 |
Phencyclidine-induced locomotor activity in the rat is blocked by 6-hydroxydopamine lesion of the nucleus accumbens: comparisons to other psychomotor stimulants.
Topics: Animals; Caffeine; Central Nervous System Stimulants; Dextroamphetamine; Hydroxydopamines; Motor Activity; Nucleus Accumbens; Oxidopamine; Phenazocine; Phencyclidine; Rats; Receptors, Dopamine; Scopolamine; Septal Nuclei | 1984 |
Behavioral and biochemical stereoselectivity of sigma opiate/PCP receptors.
Topics: Animals; Behavior, Animal; Brain; Cyclazocine; Hydromorphone; In Vitro Techniques; Ketamine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism | 1984 |
Stereoisomers of N-allylnormetazocine: phencyclidine-like behavioral effects in squirrel monkeys and rats.
Topics: Animals; Behavior, Animal; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Saimiri; Stereoisomerism; Structure-Activity Relationship | 1982 |
Autoradiographic localization of the phencyclidine/sigma "opiate" receptor in rat brain.
Topics: Animals; Autoradiography; Brain; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tritium | 1982 |
Anorexia and hyperphagia produced by five pharmacologic classes of hallucinogens.
Topics: Amphetamine; Animals; Anorexia; Atropine; Dextroamphetamine; Dogs; Dronabinol; Feeding and Eating Disorders; Feeding Behavior; Female; Hallucinogens; Humans; Lysergic Acid Diethylamide; Male; Phenazocine; Phencyclidine | 1982 |
Modulation of phencyclidine receptor sensitivity.
Topics: Amantadine; Animals; In Vitro Techniques; Olfactory Bulb; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Stereoisomerism | 1983 |
Naltrexone fails to antagonize the sigma effects of PCP and SKF 10,047 in the dog.
Topics: Animals; Body Temperature; Dogs; Female; Heart Rate; Morphine; Naloxone; Naltrexone; Paraplegia; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Reflex | 1983 |
Naloxone-inaccessible sigma receptor in rat central nervous system.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalins; Ethylketocyclazocine; Kinetics; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Spinal Cord; Tissue Distribution | 1983 |
Blockade of long-term potentiation by phencyclidine and sigma opiates in the hippocampus in vivo and in vitro.
Topics: Animals; Cyclazocine; Drug Synergism; Hippocampus; Male; Membrane Potentials; Morphine; Naloxone; Narcotics; Phenazocine; Phencyclidine; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synapses; Synaptic Transmission | 1983 |
Effects of SKF-10047 in the phencyclidine-dependent rat: evidence for common receptor mechanisms.
Topics: Animals; Drug Tolerance; Female; Humans; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Substance Withdrawal Syndrome | 1983 |
Ontogeny of sigma opiate/phencyclidine-binding sites in rat brain.
Topics: Aging; Animals; Brain; Female; Fetus; Gestational Age; Phenazocine; Phencyclidine; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1983 |
Characterization of specific sigma opiate/phencyclidine (PCP)-binding sites in the human brain.
Topics: Brain; Humans; Kinetics; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tissue Distribution | 1983 |
Further characterization of the three-choice morphine, cyclazocine and saline discrimination paradigm: opioids with agonist and antagonist properties.
Topics: Animals; Cyclazocine; Discrimination Learning; Discrimination, Psychological; Ethylketocyclazocine; Male; Morphine; Narcotic Antagonists; Narcotics; Phenazocine; Phencyclidine; Rats; Sodium Chloride; Stereoisomerism | 1983 |
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains | 1984 |
Three-choice drug discrimination: phencyclidine-like stimulus effects of opioids.
Topics: Animals; Choice Behavior; Cyclazocine; Dextroamphetamine; Discrimination, Psychological; Male; Naltrexone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Secobarbital | 1983 |
Spike and wave complexes produced by four hallucinogenic compounds in the cat.
Topics: Animals; Behavior, Animal; Cats; Electroencephalography; Hallucinogens; Ketamine; Limbic System; Phenazocine; Phencyclidine; Quipazine | 1984 |
Phencyclidine-like discriminative stimulus properties of opioids in the squirrel monkey.
Topics: Animals; Cyclazocine; Discrimination Learning; Female; Male; Naltrexone; Narcotics; Phenazocine; Phencyclidine; Saimiri; Time Factors | 1982 |
Pharmacological evaluation of N-allynormetazocine (SKF 10,047) on the basis of its discriminative stimulus properties in the rat.
Topics: Animals; Benzomorphans; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Male; Naloxone; Phenazocine; Phencyclidine; Propranolol; Rats; Rats, Inbred F344; Stereoisomerism | 1983 |
Phencyclidine-like discriminative stimuli of (+)- and (-)-N-allylnormetazocine in rats.
Topics: Animals; Discrimination Learning; Discrimination, Psychological; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Reinforcement Schedule; Stereoisomerism | 1982 |
Effects of sigma and phencyclidine receptor ligands on electric field-stimulated rabbit ear artery constriction in vitro.
Topics: Animals; Arteries; Dizocilpine Maleate; Ear; Electric Stimulation; Female; In Vitro Techniques; Ligands; Male; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Receptors, Phencyclidine; Receptors, sigma; Vasoconstriction | 1994 |
Neuroendocrine responses produced by enantiomeric pairs of drugs that interact with phencyclidine and sigma receptors.
Topics: Adrenocorticotropic Hormone; Analgesics; Animals; Corticosterone; Dioxolanes; Drug Interactions; Hypothalamo-Hypophyseal System; Injections, Subcutaneous; Male; Phenazocine; Phencyclidine; Piperidines; Pituitary-Adrenal System; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stereoisomerism; Sympathomimetics | 1994 |
NE-100, a novel sigma receptor ligand: in vivo tests.
Topics: Animals; Anisoles; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Catalepsy; Dopamine Agents; Drug Interactions; Locomotion; Male; Phenazocine; Phencyclidine; Propylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Rats, Wistar; Receptors, sigma; Stereotyped Behavior | 1993 |
FH-510, a potent and selective ligand for rat brain sigma recognition sites.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain; Carbazoles; Dopamine; Haloperidol; Male; Mice; Phenazocine; Phencyclidine; Propylamines; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma; Stereotyped Behavior | 1993 |
Effect of phencyclidine on contraction of porcine coronary vessel strips.
Topics: Animals; Biological Assay; Coronary Vessels; Dextromethorphan; Dizocilpine Maleate; Haloperidol; In Vitro Techniques; Muscle, Smooth, Vascular; Myocardial Contraction; Phenazocine; Phencyclidine; Receptors, Phencyclidine; Receptors, sigma; Swine | 1993 |
Different sensitivities of NMDA receptor channel subtypes to non-competitive antagonists.
Topics: Amino Acid Sequence; Animals; Dizocilpine Maleate; Ketamine; Magnesium; Molecular Sequence Data; Mutagenesis; Oocytes; Phenazocine; Phencyclidine; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Xenopus | 1993 |
Dose-dependent effects of D-N-allylnormetazocine on regional cerebral metabolic rates for glucose.
Topics: Animals; Blood Glucose; Blood Pressure; Brain Chemistry; Brain Mapping; Deoxyglucose; Dose-Response Relationship, Drug; Glucose; Heart Rate; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Phencyclidine; Receptors, sigma | 1993 |
(+)-SKF-10,047 and dextromethorphan ameliorate conditioned fear stress through the activation of phenytoin-regulated sigma 1 sites.
Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Behavior, Animal; Dextromethorphan; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Male; Mice; Motor Activity; Phenazocine; Phencyclidine; Phenytoin; Pyrimidines; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Stress, Physiological | 1996 |
The involvement of sigma receptors in the choice reaction performance deficits induced by phencyclidine.
Topics: Animals; Anisoles; Antipsychotic Agents; Excitatory Amino Acid Agonists; Ligands; Male; Phenazocine; Phencyclidine; Piperidines; Propylamines; Psychomotor Performance; Rats; Rats, Wistar; Reaction Time; Receptors, sigma | 1997 |
Sigma1 receptor subtype does not interact with stereotyped behaviors in rats.
Topics: Animals; Antipsychotic Agents; Male; Nootropic Agents; Phenazocine; Phencyclidine; Piperazines; Rats; Rats, Wistar; Receptors, sigma; Stereotyped Behavior | 1998 |
Binding of [3H]desglycinyl remacemide to rat brain membranes: association with the benzomorphan attachment site of the N-methyl-D-aspartic acid receptor channel.
Topics: Animals; Antipsychotic Agents; Benzomorphans; Binding Sites; Brain Chemistry; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Haloperidol; Male; Membrane Proteins; Neurons; Phenazocine; Phencyclidine; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Subcellular Fractions; Tritium | 1999 |
Pharmacological profile of MS-377, a novel antipsychotic agent with selective affinity for sigma receptors.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Dopamine Agonists; Free Radical Scavengers; Guinea Pigs; Haloperidol; Head Movements; Male; Mice; Phenazocine; Phencyclidine; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, sigma; Risperidone; Serotonin; Serotonin Antagonists; Stereotyped Behavior; Sulpiride; Tartrates | 1999 |
Phencyclidine impairs latent learning in mice: interaction between glutamatergic systems and sigma(1) receptors.
Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Behavior, Animal; Cycloserine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Exploratory Behavior; Glutamic Acid; Learning; Male; Mice; Mice, Inbred Strains; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Piperazines; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism | 2001 |
MS-377, a selective sigma receptor ligand, indirectly blocks the action of PCP in the N-methyl-D-aspartate receptor ion-channel complex in primary cultured rat neuronal cells.
Topics: Animals; Antipsychotic Agents; Calcium; Cells, Cultured; Dizocilpine Maleate; Female; Ion Channels; Neurons; Phenazocine; Phencyclidine; Piperazines; Pregnancy; Pyrrolidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Tartrates; Tritium | 2002 |
Characterization of the non-competitive antagonist binding site of the NMDA receptor in dark Agouti rats.
Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dioxolanes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Female; Ketamine; N-Methylaspartate; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Mutant Strains; Receptors, N-Methyl-D-Aspartate; Scintillation Counting; Tritium | 2004 |
Inhibition of hyperpolarization-activated cation currents by phencyclidine and some sigma ligands in rat hippocampal CA1 pyramidal neurons in vitro.
Topics: Animals; Animals, Newborn; Cesium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Ion Channels; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Phenazocine; Phencyclidine; Pyramidal Cells; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma | 2007 |
Sigma-1 receptor function is critical for both the discriminative stimulus and aversive effects of the kappa-opioid receptor agonist U-50488H.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anisoles; Avoidance Learning; Conditioning, Psychological; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Propylamines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor | 2012 |