phenazocine has been researched along with pentazocine in 69 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 30 (43.48) | 18.7374 |
1990's | 31 (44.93) | 18.2507 |
2000's | 5 (7.25) | 29.6817 |
2010's | 3 (4.35) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creese, I; Feinberg, AP; Snyder, SH | 1 |
Hudzik, TJ; Slifer, BL | 1 |
Feuerstein, G; Gagnon, RC; Gu, JL; Lysko, PG; Yue, TL | 1 |
Angulo, JA; Ledoux, M; McEwen, BS | 1 |
Boyce, S; Cook, G; Iversen, SD; Rupniak, NM; Steventon, MJ | 1 |
Baldessarini, RJ; Booth, RG | 1 |
Gillard, J; Knight, AR; Middlemiss, DN; Wong, EH | 1 |
Brent, PJ | 1 |
Contreras, PC; Dilworth, VM; Farah, JM; Gray, NM; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL | 1 |
Dykstra, LA; Picker, MJ; Powell, K | 1 |
Contreras, PC; Dilworth, VM; Iyengar, S; Mick, SJ; Monahan, JB; Rao, TS; Wood, PL | 1 |
Connick, JH; Fox, PK; France, L; Hanlon, GM; Nicholson, CD | 1 |
Bowen, WD; DeCosta, B; Hellewell, SB; Rice, KC; Thurkauf, A; Walker, JM | 1 |
Dilworth, V; Farah, JM; Iyengar, S; Michel, J; Mick, S; Rao, TS; Wood, PL | 1 |
Bauerle, LM; DeNoble, VJ; Jones, KW | 1 |
Duffy, O; Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauche, D | 1 |
Alberici, GP; Cook, L; Steinfels, GF; Tam, SW | 1 |
Holtzman, SG | 1 |
Adler, MW; Geller, EB; Rowan, CH | 1 |
Cook, L; Steinfels, GF; Tam, SW | 1 |
Röthig, J | 1 |
Medzihradsky, F; Nandhasri, PS | 1 |
Aceto, MD; McKean, DB; Pearl, J | 1 |
Bowman, WC; Buwembo, JB | 1 |
Carr, EA; Marks, MJ; Medzihradsky, F | 1 |
Janssen, PA | 1 |
Pittman, KA; Williams, TA | 1 |
Conaghan, JP; Jacobsen, M; Rae, L; Ward-McQuaid, JN | 1 |
Fennessy, MR; Heimans, RL; Rand, MJ | 1 |
Ahmad, K; Medzihradsky, F | 1 |
Economou, G; Monson, R; Ward-McQuaid, JN | 1 |
McKean, DB; Pearl, J; Stander, H | 1 |
Rogers, KJ; Thornton, JA | 1 |
Gyand, EA; Kosterlitz, HW | 1 |
Clarke, RS; Dundee, JW; Hamilton, RC; Loan, WB; Morrison, JD | 1 |
Ben-Sreti, MM; Gonzalez, JP; Sewell, RD | 1 |
Bernardini, GL; Clark, WG; Ponder, SW | 1 |
Shannon, HE; Su, TP | 1 |
Herling, S; Woods, JH | 1 |
Adler, MW; Geller, EB; Hawk, C; Keinath, SH; Tallarida, RJ | 1 |
Moerschbaecher, JM; Thompson, DM | 1 |
Franklin, SR; Tang, AH | 1 |
Brent, PJ; Dunkley, PR; Haynes, H; Jarvie, PE; Mudge, L; Sim, AT | 1 |
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA | 1 |
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC | 1 |
Matsunaga, KH; Matsuno, K; Mita, S | 1 |
Bao, WL; Sun, FY; Zhang, AZ; Zhen, FC | 1 |
Hasegawa, T; Hiramatsu, M; Itoh, J; Kameyama, T; Maurice, T; Nabeshima, T | 1 |
Kamei, H; Kameyama, T; Nabeshima, T | 1 |
Gonzalez-Alvear, GM; Werling, LL | 1 |
Allen, JT; DeHaven-Hudkins, DL; Ford-Rice, FY; Hudkins, RL | 1 |
Bergeron, R; Bouchard, P; de Montigny, C; Debonnel, G; Junien, JL; Monnet, F; Quirion, R; Roman, F | 1 |
Kobayashi, T; Matsuno, K; Mita, S | 1 |
Bowen, WD; Torrence-Campbell, C | 1 |
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA | 1 |
Bucolo, C; Cacciaguerra, S; Campana, G; Di Toro, R; Spampinato, S | 1 |
Baulieu, EE; Collin, T; Denavit-Saubié, M; Monnet, FP; Morin-Surun, MP | 1 |
Matsuno, K | 1 |
Kamei, J | 1 |
Aydar, E; Chen, Y; Jackson, MB; Lupardus, PJ; Palmer, CP; Ruoho, AE; Wilke, RA | 1 |
Furukawa, S; Hiramatsu, M; Kameyama, T; Karasawa, K; Mamiya, T; Nabeshima, T; Noda, A; Noda, Y; Yamada, K | 1 |
Furukawa, H; Ichihara, K; Kamei, H; Mamiya, T; Nabeshima, T; Nagai, T; Noda, A; Noda, Y; Sugiura, S | 1 |
HARRIS, LS; PIERSON, AK | 1 |
LASAGNA, L | 1 |
Cantero, M; Codony, X; Cozar, P; Dordal, A; Giménez, E; Guitart, X; Hernández, E; Langa, F; Lavado, A; Monroy, X; Montoliu, L; Pérez, R; Tovar, V; Zamanillo, D | 1 |
Jackson, MB; Johannessen, M; Ramachandran, S; Ramos-Serrano, A; Riemer, L; Ruoho, AE | 1 |
Isotani, K; Mori, T; Narita, M; Nomura, M; Suzuki, T; Torigoe, K; Tsukiyama, Y; Yoshizawa, K | 1 |
Akopova, I; Clark, AF; Daudt, DR; Ma, HY; Mueller, BH; Park, Y; Stankowska, DL; Yorio, T | 1 |
Ahlskog, N; Beique, JC; Bergeron, R; Biscaro, D; Hristova, E; Nassrallah, W; Ngsee, JK; Pabba, M; Snyder, M; Wong, AY | 1 |
5 review(s) available for phenazocine and pentazocine
Article | Year |
---|---|
Drug discrimination studies.
Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
[Analgesics. 32].
Topics: Alphaprodine; Analgesics; Azepines; Benzimidazoles; Bridged-Ring Compounds; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Fentanyl; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Levallorphan; Levorphanol; Lysergic Acid Diethylamide; Methadone; Morphinans; Morphine; Nalorphine; Naphthoquinones; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine | 1969 |
[Anti-amnesic effects of sigma (sigma)-receptor agonists].
Topics: Acetylcholine; Amnesia; Animals; Disease Models, Animal; Dopamine; Ligands; Mice; Morpholines; Pentazocine; Phenazocine; Piperazines; Receptors, sigma; Sigma-1 Receptor | 1999 |
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases | 1999 |
THE CLINICAL EVALUATION OF MORPHINE AND ITS SUBSTITUTES AS ANALGESICS.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Biomedical Research; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Meperidine; Methadone; Methotrimeprazine; Morphine; Nalorphine; Narcotic Antagonists; Oxymorphone; Pentazocine; Phenazocine; Substance-Related Disorders; Toxicology | 1964 |
3 trial(s) available for phenazocine and pentazocine
Article | Year |
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Pentazocine and phenazocine. A double-blind comparison of two benzomorphan derivatives in postoperative pain.
Topics: Adolescent; Adult; Aged; Analgesia; Child; Clinical Trials as Topic; Female; Humans; Injections, Intramuscular; Male; Middle Aged; Pentazocine; Phenazocine; Postoperative Care | 1966 |
Oral pentazocine and phenazocine: a comparison in postoperative pain.
Topics: Administration, Oral; Adolescent; Adult; Aged; Consciousness; Female; Humans; Male; Middle Aged; Nausea; Pain; Pentazocine; Phenazocine; Postoperative Complications; Time Factors; Vertigo | 1971 |
Studies of drugs given before anaesthesia. 13. Pentazocine and other opiate antagonists.
Topics: Adult; Central Nervous System; Drug Antagonism; Female; Humans; Levallorphan; Meperidine; Morphine; Nalorphine; Pentazocine; Phenazocine; Preanesthetic Medication; Psychoses, Substance-Induced | 1967 |
61 other study(ies) available for phenazocine and pentazocine
Article | Year |
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The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists.
Topics: Allosteric Regulation; Dextropropoxyphene; Fentanyl; Methadone; Models, Biological; Models, Molecular; Molecular Conformation; Morphine; Nalorphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Protein Conformation; Receptors, Opioid; Structure-Activity Relationship | 1976 |
Interaction of sigma and PCP-like drugs on operant behaviors in the rat.
Topics: Animals; Conditioning, Operant; Dextroamphetamine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Pentazocine; Phenazocine; Phencyclidine; Psychotropic Drugs; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule | 1992 |
Neuroprotective effects of SKF 10,047 in cultured rat cerebellar neurons and in gerbil global brain ischemia.
Topics: Animals; Body Temperature; Brain Ischemia; Cells, Cultured; Cerebellum; Cyclazocine; Dizocilpine Maleate; Gerbillinae; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Reference Values; Stereoisomerism | 1992 |
Chronic treatment with pentazocine or SFK 10047 decrease proenkephalin mRNA levels in the rat striatum and nucleus accumbens.
Topics: Animals; Base Sequence; Corpus Striatum; Enkephalins; Histocytochemistry; Male; Molecular Sequence Data; Nucleic Acid Hybridization; Nucleus Accumbens; Pentazocine; Phenazocine; Protein Precursors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; RNA, Messenger | 1991 |
Psychomotor activity and cognitive disruption attributable to NMDA, but not sigma, interactions in primates.
Topics: Animals; Ataxia; Cognition; Dizocilpine Maleate; Macaca mulatta; Male; Pentazocine; Phenazocine; Phencyclidine; Psychomotor Performance; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Saimiri; Space Perception | 1991 |
(+)-6,7-benzomorphan sigma ligands stimulate dopamine synthesis in rat corpus striatum tissue.
Topics: Animals; Benzomorphans; Catecholamines; Corpus Striatum; Cyclazocine; Dopamine; In Vitro Techniques; Ligands; Male; Nerve Endings; Neural Pathways; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Stimulation, Chemical; Tyrosine 3-Monooxygenase | 1991 |
The human sigma site, which resembles that in NCB20 cells, may correspond to a low-affinity site in guinea pig brain.
Topics: Animals; Brain Chemistry; Cells, Cultured; Cerebral Cortex; Cricetinae; Cricetulus; Dopamine Agents; Guanidines; Guinea Pigs; Humans; Kinetics; Male; Mice; Neuroblastoma; Pentazocine; Phenazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Tumor Cells, Cultured | 1991 |
Similar behavioural effects of sigma agonists and PCP-like non-competitive NMDA antagonists in guinea-pigs.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Dizocilpine Maleate; Dopamine Agents; Dopamine Antagonists; Ergolines; Female; Guanidines; Guinea Pigs; Haloperidol; Ketamine; Male; Motor Activity; N-Methylaspartate; Pentazocine; Phenazocine; Phencyclidine; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride | 1991 |
(+) 3-[3-hydroxyphenyl-N-(1-propyl) piperidine] selectively differentiates effects of sigma ligands on neurochemical pathways modulated by sigma receptors: evidence for subtypes, in vivo.
Topics: Adrenocorticotropic Hormone; Animals; Brain; Butaclamol; Cerebellum; Corpus Striatum; Cyclic GMP; Dopamine; Dopamine Agents; Male; Mice; Pentazocine; Phenazocine; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma | 1991 |
Stereospecificity of mixed-action opioid agonist/antagonists in morphine-tolerant squirrel monkeys.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Morphine; Narcotic Antagonists; Narcotics; Pentazocine; Phenazocine; Saimiri; Stereoisomerism | 1990 |
Sigma receptors modulate both A9 and A10 dopaminergic neurons in the rat brain: functional interaction with NMDA receptors.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Cerebral Ventricles; Dopamine; Kinetics; Male; Neurons; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma | 1990 |
The lack of utility of the rat vas deferens as a functional bioassay for sigma ligands.
Topics: Animals; Binding Sites; Biological Assay; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; Male; Muscle Contraction; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Vas Deferens | 1991 |
Characterization of [3H] (+)-pentazocine, a highly selective sigma ligand.
Topics: Animals; Binding, Competitive; Brain; Guinea Pigs; In Vitro Techniques; Kinetics; Pentazocine; Phenazocine; Piperidines; Receptors, Opioid; Receptors, sigma | 1990 |
Sigma receptors modulate the hypothalamic-pituitary-adrenal (HPA) axis centrally: evidence for a functional interaction with NMDA receptors, in vivo.
Topics: Adrenocorticotropic Hormone; Animals; Aspartic Acid; Cells, Cultured; Hypothalamo-Hypophyseal System; Male; N-Methylaspartate; Pentazocine; Phenazocine; Piperazines; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, sigma | 1990 |
Differential effects of sigma and phencyclidine receptor ligands on learning.
Topics: Animals; Avoidance Learning; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Ligands; Male; Memory; Pentazocine; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Retention, Psychology | 1990 |
Neuropeptide Y and peptide YY interact with rat brain sigma and PCP binding sites.
Topics: Animals; Brain Chemistry; Haloperidol; In Vitro Techniques; Male; Neuropeptide Y; Pentazocine; Peptide YY; Peptides; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1989 |
Biochemical, behavioral, and electrophysiologic actions of the selective sigma receptor ligand (+)-pentazocine.
Topics: Animals; Avoidance Learning; Brain; Discrimination Learning; Evoked Potentials, Visual; Male; Membranes; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Reference Values | 1988 |
Body temperature effects of opioids in rats: intracerebroventricular administration.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1986 |
Discriminative stimulus properties of (+)-N-allylnormetazocine in the rat: correlations with (+)-N-allylnormetazocine and phencyclidine receptor binding.
Topics: Animals; Brain; Cyclazocine; Discrimination Learning; Ketamine; Male; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism | 1987 |
Effects of some analgesics and antidepressants on the (Na + + K + )-adenosine triphosphatase from cortices of brain and kidney.
Topics: Adenosine Triphosphatases; Amitriptyline; Analgesics; Animals; Antidepressive Agents; Cattle; Cerebral Cortex; Chlorpromazine; Cyclazocine; Desipramine; Dose-Response Relationship, Drug; Hydralazine; Imipramine; In Vitro Techniques; Kidney; Kidney Cortex; Pentazocine; Phenazocine; Phenelzine; Potassium; Sodium; Tranylcypromine | 1972 |
Effects of opiates and opiate antagonists on the Straub tail reaction in mice.
Topics: Analgesics; Animals; Atropine; Bridged-Ring Compounds; Codeine; Cyclazocine; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Narcotic Antagonists; Pentazocine; Phenazocine; Stereoisomerism; Tail | 1969 |
Effects of narcotic analgesics on contractions of the chick isolated, innervated oesophagus.
Topics: Acetylcholine; Analgesics; Animals; Chickens; Cyclazocine; Dextropropoxyphene; Electric Stimulation; Esophagus; Heroin; In Vitro Techniques; Meperidine; Methadone; Morphinans; Morphine; Muscle Contraction; Nalorphine; Pentazocine; Phenazocine; Serotonin; Tachyphylaxis; Time Factors | 1972 |
Energy-dependent uptake of benzomorphans by leukocytes.
Topics: Animals; Cell Membrane; Chromatography, Gas; Cyclazocine; Fluorides; Glucose; Leukocytes; Male; Models, Biological; Oxygen Consumption; Pentazocine; Phenazocine; Potassium; Rats; Sodium; Structure-Activity Relationship; Time Factors | 1972 |
Potent long-acting antagonists of the 9,9-dialkylbenzomorphan series.
Topics: Alkylation; Analgesics; Animals; Butyrates; Cyclazocine; Cyclization; Isomerism; Methylation; Morphinans; Narcotic Antagonists; Pentazocine; Phenazocine; Phenols; Propionates; Rats; Structure-Activity Relationship; Time Factors | 1973 |
Pentazocine radioimmunoassay.
Topics: Ammonium Sulfate; Animals; Antibody Specificity; Antigen-Antibody Reactions; Azo Compounds; Carboxylic Acids; Chromatography, Gas; Cross Reactions; Cyclazocine; Levallorphan; Levorphanol; Methods; Molecular Weight; Morphine; Nalorphine; Oxidation-Reduction; Pentazocine; Phenazocine; Rabbits; Radioimmunoassay; Tritium; Urine | 1974 |
Comparison of effect of morphine-like analgesics on transmurally stimulated guinea-pig ileum.
Topics: Analgesics; Animals; Codeine; Cyclic N-Oxides; Drug Tolerance; Electric Stimulation; Female; Fentanyl; Guinea Pigs; Heroin; Humans; Ileum; In Vitro Techniques; Male; Meperidine; Morphinans; Morphine; Muscle Contraction; Muscle, Smooth; Nalorphine; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine; Rats; Substance-Related Disorders; Urinary Bladder | 1969 |
The determination of benzomorphan derivatives in plasma by gas chromatography.
Topics: Analgesics; Azocines; Cyclazocine; Humans; Methods; Narcotic Antagonists; Pentazocine; Phenazocine | 1971 |
Effects of analgesics and other drugs on mice in phenylquinone and rotarod tests.
Topics: Analgesics; Animals; Chemical Phenomena; Chemistry; Chlorpromazine; Cyclazocine; Dextroamphetamine; Levallorphan; Male; Mice; Morphine; Motor Activity; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Pilocarpine; Quinones; Salivation | 1969 |
The interaction between monoamine oxidase inhibitors and narcotic analgesics in mice.
Topics: Analgesics; Animals; Drug Synergism; Iproniazid; Meperidine; Mice; Monoamine Oxidase Inhibitors; Morphine; Pentazocine; Phenazocine; Tranylcypromine | 1969 |
Agonist and antagonist actions of morphine-like drugs on the guinea-pig isolated ileum.
Topics: Analgesics; Animals; Cyclazocine; Drug Synergism; Guinea Pigs; Ileum; Levallorphan; Levorphanol; Morphine; Muscle, Smooth; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Reflex | 1966 |
Effects of elevated calcium and calcium antagonists on 6,7-benzomorphan-induced analgesia.
Topics: Analgesia; Analgesics; Analgesics, Opioid; Animals; Benzomorphans; Calcium; Calcium Channel Blockers; Cyclazocine; Egtazic Acid; Ethylketocyclazocine; Gallopamil; Male; Mice; Morphinans; Pentazocine; Phenazocine | 1983 |
Central injection of a sigma opioid receptor agonist alters body temperature of cats.
Topics: Animals; Body Temperature Regulation; Cats; Dose-Response Relationship, Drug; Pentazocine; Phenazocine; Receptors, Opioid | 1981 |
Effects of the combination of tripelennamine and pentazocine at the behavioral and molecular levels.
Topics: Animals; Brain; Diphenhydramine; Discrimination, Psychological; Drug Synergism; Guinea Pigs; Ileum; Learning; Male; Morphine; Pentazocine; Phenazocine; Rats; Receptors, Opioid; Synaptic Membranes; Tripelennamine | 1982 |
Discriminative stimulus effects of etorphine in Rhesus monkeys.
Topics: Animals; Codeine; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Etorphine; Macaca mulatta; Male; Meperidine; Morphinans; Morphine; Pentazocine; Phenazocine; Sodium Chloride | 1981 |
Subclasses of opioids based on body temperature change in rats: acute subcutaneous administration.
Topics: Animals; Body Temperature; Buprenorphine; Dose-Response Relationship, Drug; Endorphins; Injections, Subcutaneous; Male; Meperidine; Morphine; Nalbuphine; Naloxone; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1983 |
Differential effects of prototype opioid agonists on the acquisition of conditional discriminations in monkeys.
Topics: Animals; Behavior, Animal; Conditioning, Psychological; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Male; Morphine; Pentazocine; Phenazocine; Psychomotor Performance | 1983 |
Acquisition of brightness discrimination in the rat is impaired by opiates with psychotomimetic properties.
Topics: Animals; Avoidance Learning; Cyclazocine; Discrimination Learning; Male; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Phenazocine; Photic Stimulation; Psychotropic Drugs; Rats; Rats, Inbred F344 | 1983 |
Phosphorylation of synapsin I and dynamin in rat forebrain synaptosomes: modulation by sigma (sigma) ligands.
Topics: Animals; Anticonvulsants; Dynamins; GTP Phosphohydrolases; Guanidines; Haloperidol; In Vitro Techniques; Microtubules; Pentazocine; Phenazocine; Phosphorylation; Prosencephalon; Rats; Receptors, sigma; Synapsins; Synaptosomes | 1995 |
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc | 1994 |
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma | 1995 |
Acute effects of sigma ligands on the extracellular DOPAC level in rat frontal cortex and striatum.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Corpus Striatum; Extracellular Space; Frontal Lobe; Guanidines; Kinetics; Ligands; Male; Microdialysis; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Time Factors | 1995 |
Effects of sigma and phencyclidine receptor ligands on electric field-stimulated rabbit ear artery constriction in vitro.
Topics: Animals; Arteries; Dizocilpine Maleate; Ear; Electric Stimulation; Female; In Vitro Techniques; Ligands; Male; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Receptors, Phencyclidine; Receptors, sigma; Vasoconstriction | 1994 |
Low dose of 1,3-di(2-tolyl)guanidine (DTG) attenuates MK-801-induced spatial working memory impairment in mice.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Dizocilpine Maleate; Dose-Response Relationship, Drug; Guanidines; Male; Memory; Mice; Mice, Inbred Strains; Motor Activity; Pentazocine; Phenazocine; Pyrimidines; Receptors, sigma; Space Perception | 1994 |
SKF-10,047 reverses stress-induced motor suppression: interaction with dopaminergic system.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anticonvulsants; Apomorphine; Dopamine; Electroshock; Guanidines; Male; Methamphetamine; Mice; Mice, Inbred Strains; Motor Activity; Oxidopamine; Pentazocine; Phenazocine; Pimozide; Pyrimidines; Receptors, sigma; Stress, Psychological | 1994 |
Regulation of [3H]dopamine release from rat striatal slices by sigma receptor ligands.
Topics: Animals; Atropine; Corpus Striatum; Dopamine; Flavonoids; In Vitro Techniques; N-Methylaspartate; Naloxone; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma | 1994 |
Allosteric modulation of ligand binding to [3H](+)pentazocine-defined sigma recognition sites by phenytoin.
Topics: Allosteric Regulation; Animals; Binding Sites; Cyclopentanes; Dextromethorphan; Dextrorphan; Guinea Pigs; Ligands; Male; Pentazocine; Phenazocine; Phenytoin; Piperidines; Radioligand Assay; Receptors, sigma; Tritium | 1993 |
In vivo modulation of sigma receptor sites by calcitonin gene-related peptide in the mouse and rat hippocampal formation: radioligand binding and electrophysiological studies.
Topics: Animals; Antipsychotic Agents; Calcitonin Gene-Related Peptide; Dopamine Antagonists; Electrophysiology; Haloperidol; Hippocampus; In Vitro Techniques; Iontophoresis; Male; Membranes; Mice; Narcotics; Neuropeptide Y; Pentazocine; Phenazocine; Pyramidal Cells; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma | 1995 |
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens | 1996 |
Differential solubilization of rat liver sigma 1 and sigma 2 receptors: retention of sigma 2 sites in particulate fractions.
Topics: Animals; Binding, Competitive; Cell Fractionation; Cell Membrane; Cholic Acids; Detergents; Guanidines; Haloperidol; In Vitro Techniques; Liver; Male; Pentazocine; Phenazocine; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Solubility; Subcellular Fractions | 1996 |
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium | 1997 |
Sigma1 recognition sites in rabbit iris-ciliary body: topical sigma1-site agonists lower intraocular pressure.
Topics: Animals; Anisoles; Antipsychotic Agents; Binding, Competitive; Cell Membrane; Ciliary Body; Functional Laterality; Guanidines; Intraocular Pressure; Iris; Kinetics; Lens, Crystalline; Male; Pentazocine; Phenazocine; Propylamines; Rabbits; Receptors, sigma; Retina; Tritium | 1999 |
Intracellular sigma1 receptor modulates phospholipase C and protein kinase C activities in the brainstem.
Topics: Action Potentials; Animals; Antipsychotic Agents; Brain Stem; Cell Membrane; Cytoplasm; GTP-Binding Proteins; Guinea Pigs; Haloperidol; In Vitro Techniques; Isoenzymes; Ligands; Male; Pentazocine; Pertussis Toxin; Phenazocine; Protein Kinase C; Protein Kinase C beta; Receptors, sigma; Respiratory Mechanics; Reverse Transcriptase Polymerase Chain Reaction; Type C Phospholipases; Virulence Factors, Bordetella | 1999 |
Membrane-delimited coupling between sigma receptors and K+ channels in rat neurohypophysial terminals requires neither G-protein nor ATP.
Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Antipsychotic Agents; Cells, Cultured; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine Triphosphate; In Vitro Techniques; Ligands; Oocytes; Patch-Clamp Techniques; Pentazocine; Phenazocine; Phosphorylation; Pituitary Gland, Posterior; Potassium; Potassium Channels; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptic Membranes; Xenopus laevis | 2000 |
Effects of sigma receptor agonists on the impairment of spontaneous alternation behavior and decrease of cyclic GMP level induced by nitric oxide synthase inhibitors in mice.
Topics: Analgesics, Opioid; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Behavior, Animal; Brain Chemistry; Cyclic GMP; Enzyme Inhibitors; Guanidines; Indazoles; Male; Methylene Blue; Mice; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Pentazocine; Phenazocine; Pyrimidines; Receptors, sigma | 2000 |
Phencyclidine impairs latent learning in mice: interaction between glutamatergic systems and sigma(1) receptors.
Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Behavior, Animal; Cycloserine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Exploratory Behavior; Glutamic Acid; Learning; Male; Mice; Mice, Inbred Strains; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Piperazines; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism | 2001 |
SOME NARCOTIC ANTAGONISTS IN THE BENZOMORPHAN SERIES.
Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Antipyretics; Azocines; Benzomorphans; Cats; Cyclazocine; Haplorhini; Heterocyclic Compounds; Meperidine; Mice; Morphine; Nalorphine; Narcotic Antagonists; Pentazocine; Pharmacology; Phenazocine; Rats; Research; Toxicology | 1964 |
Generation and phenotypic analysis of sigma receptor type I (sigma 1) knockout mice.
Topics: Animals; Animals, Newborn; Antidepressive Agents; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Blotting, Northern; Blotting, Southern; Blotting, Western; Body Weight; Cells, Cultured; Embryo, Mammalian; Endorphins; Heterozygote; Hyperkinesis; In Situ Hybridization; Mice; Mice, Knockout; Narcotic Antagonists; Oligonucleotides, Antisense; Pentazocine; Peptide Fragments; Phenazocine; Phenotype; Radioligand Assay; Receptors, sigma; Sigma-1 Receptor; Time Factors | 2003 |
Voltage-gated sodium channel modulation by sigma-receptors in cardiac myocytes and heterologous systems.
Topics: Adenosine Triphosphate; Animals; Antipsychotic Agents; Cell Line; Chlorocebus aethiops; COS Cells; Guanosine Triphosphate; Haloperidol; Humans; Kidney; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Proteins; Myocytes, Cardiac; Narcotics; NAV1.5 Voltage-Gated Sodium Channel; Patch-Clamp Techniques; Pentazocine; Phenazocine; Receptors, sigma; RNA, Small Interfering; Sodium; Sodium Channels | 2009 |
Sigma-1 receptor function is critical for both the discriminative stimulus and aversive effects of the kappa-opioid receptor agonist U-50488H.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anisoles; Avoidance Learning; Conditioning, Psychological; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Propylamines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor | 2012 |
Sigma-1 receptor stimulation attenuates calcium influx through activated L-type Voltage Gated Calcium Channels in purified retinal ganglion cells.
Topics: Animals; Animals, Newborn; Blotting, Western; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Ethylenediamines; Fluorescent Antibody Technique, Indirect; Fura-2; Microscopy, Fluorescence; Pentazocine; Phenazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Retinal Ganglion Cells; Sigma-1 Receptor; Verapamil | 2013 |
NMDA receptors are upregulated and trafficked to the plasma membrane after sigma-1 receptor activation in the rat hippocampus.
Topics: Animals; Cell Membrane; Disks Large Homolog 4 Protein; Ethylenediamines; Hippocampus; Intracellular Signaling Peptides and Proteins; Male; Membrane Proteins; Mice; Mice, Knockout; Morpholines; Pentazocine; Phenazocine; Piperazines; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Subcellular Fractions; Time Factors; Up-Regulation | 2014 |