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phenazocine and pentazocine

phenazocine has been researched along with pentazocine in 69 studies

Research

Studies (69)

TimeframeStudies, this research(%)All Research%
pre-199030 (43.48)18.7374
1990's31 (44.93)18.2507
2000's5 (7.25)29.6817
2010's3 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creese, I; Feinberg, AP; Snyder, SH1
Hudzik, TJ; Slifer, BL1
Feuerstein, G; Gagnon, RC; Gu, JL; Lysko, PG; Yue, TL1
Angulo, JA; Ledoux, M; McEwen, BS1
Boyce, S; Cook, G; Iversen, SD; Rupniak, NM; Steventon, MJ1
Baldessarini, RJ; Booth, RG1
Gillard, J; Knight, AR; Middlemiss, DN; Wong, EH1
Brent, PJ1
Contreras, PC; Dilworth, VM; Farah, JM; Gray, NM; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL1
Dykstra, LA; Picker, MJ; Powell, K1
Contreras, PC; Dilworth, VM; Iyengar, S; Mick, SJ; Monahan, JB; Rao, TS; Wood, PL1
Connick, JH; Fox, PK; France, L; Hanlon, GM; Nicholson, CD1
Bowen, WD; DeCosta, B; Hellewell, SB; Rice, KC; Thurkauf, A; Walker, JM1
Dilworth, V; Farah, JM; Iyengar, S; Michel, J; Mick, S; Rao, TS; Wood, PL1
Bauerle, LM; DeNoble, VJ; Jones, KW1
Duffy, O; Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauche, D1
Alberici, GP; Cook, L; Steinfels, GF; Tam, SW1
Holtzman, SG1
Adler, MW; Geller, EB; Rowan, CH1
Cook, L; Steinfels, GF; Tam, SW1
Röthig, J1
Medzihradsky, F; Nandhasri, PS1
Aceto, MD; McKean, DB; Pearl, J1
Bowman, WC; Buwembo, JB1
Carr, EA; Marks, MJ; Medzihradsky, F1
Janssen, PA1
Pittman, KA; Williams, TA1
Conaghan, JP; Jacobsen, M; Rae, L; Ward-McQuaid, JN1
Fennessy, MR; Heimans, RL; Rand, MJ1
Ahmad, K; Medzihradsky, F1
Economou, G; Monson, R; Ward-McQuaid, JN1
McKean, DB; Pearl, J; Stander, H1
Rogers, KJ; Thornton, JA1
Gyand, EA; Kosterlitz, HW1
Clarke, RS; Dundee, JW; Hamilton, RC; Loan, WB; Morrison, JD1
Ben-Sreti, MM; Gonzalez, JP; Sewell, RD1
Bernardini, GL; Clark, WG; Ponder, SW1
Shannon, HE; Su, TP1
Herling, S; Woods, JH1
Adler, MW; Geller, EB; Hawk, C; Keinath, SH; Tallarida, RJ1
Moerschbaecher, JM; Thompson, DM1
Franklin, SR; Tang, AH1
Brent, PJ; Dunkley, PR; Haynes, H; Jarvie, PE; Mudge, L; Sim, AT1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC1
Matsunaga, KH; Matsuno, K; Mita, S1
Bao, WL; Sun, FY; Zhang, AZ; Zhen, FC1
Hasegawa, T; Hiramatsu, M; Itoh, J; Kameyama, T; Maurice, T; Nabeshima, T1
Kamei, H; Kameyama, T; Nabeshima, T1
Gonzalez-Alvear, GM; Werling, LL1
Allen, JT; DeHaven-Hudkins, DL; Ford-Rice, FY; Hudkins, RL1
Bergeron, R; Bouchard, P; de Montigny, C; Debonnel, G; Junien, JL; Monnet, F; Quirion, R; Roman, F1
Kobayashi, T; Matsuno, K; Mita, S1
Bowen, WD; Torrence-Campbell, C1
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA1
Bucolo, C; Cacciaguerra, S; Campana, G; Di Toro, R; Spampinato, S1
Baulieu, EE; Collin, T; Denavit-Saubié, M; Monnet, FP; Morin-Surun, MP1
Matsuno, K1
Kamei, J1
Aydar, E; Chen, Y; Jackson, MB; Lupardus, PJ; Palmer, CP; Ruoho, AE; Wilke, RA1
Furukawa, S; Hiramatsu, M; Kameyama, T; Karasawa, K; Mamiya, T; Nabeshima, T; Noda, A; Noda, Y; Yamada, K1
Furukawa, H; Ichihara, K; Kamei, H; Mamiya, T; Nabeshima, T; Nagai, T; Noda, A; Noda, Y; Sugiura, S1
HARRIS, LS; PIERSON, AK1
LASAGNA, L1
Cantero, M; Codony, X; Cozar, P; Dordal, A; Giménez, E; Guitart, X; Hernández, E; Langa, F; Lavado, A; Monroy, X; Montoliu, L; Pérez, R; Tovar, V; Zamanillo, D1
Jackson, MB; Johannessen, M; Ramachandran, S; Ramos-Serrano, A; Riemer, L; Ruoho, AE1
Isotani, K; Mori, T; Narita, M; Nomura, M; Suzuki, T; Torigoe, K; Tsukiyama, Y; Yoshizawa, K1
Akopova, I; Clark, AF; Daudt, DR; Ma, HY; Mueller, BH; Park, Y; Stankowska, DL; Yorio, T1
Ahlskog, N; Beique, JC; Bergeron, R; Biscaro, D; Hristova, E; Nassrallah, W; Ngsee, JK; Pabba, M; Snyder, M; Wong, AY1

Reviews

5 review(s) available for phenazocine and pentazocine

ArticleYear
Drug discrimination studies.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
[Analgesics. 32].
    Pharmazeutische Praxis, 1969, Volume: 5

    Topics: Alphaprodine; Analgesics; Azepines; Benzimidazoles; Bridged-Ring Compounds; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Fentanyl; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Levallorphan; Levorphanol; Lysergic Acid Diethylamide; Methadone; Morphinans; Morphine; Nalorphine; Naphthoquinones; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine

1969
[Anti-amnesic effects of sigma (sigma)-receptor agonists].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114, Issue:1

    Topics: Acetylcholine; Amnesia; Animals; Disease Models, Animal; Dopamine; Ligands; Mice; Morpholines; Pentazocine; Phenazocine; Piperazines; Receptors, sigma; Sigma-1 Receptor

1999
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases

1999
THE CLINICAL EVALUATION OF MORPHINE AND ITS SUBSTITUTES AS ANALGESICS.
    Pharmacological reviews, 1964, Volume: 16

    Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Biomedical Research; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Meperidine; Methadone; Methotrimeprazine; Morphine; Nalorphine; Narcotic Antagonists; Oxymorphone; Pentazocine; Phenazocine; Substance-Related Disorders; Toxicology

1964

Trials

3 trial(s) available for phenazocine and pentazocine

ArticleYear
Pentazocine and phenazocine. A double-blind comparison of two benzomorphan derivatives in postoperative pain.
    British journal of anaesthesia, 1966, Volume: 38, Issue:5

    Topics: Adolescent; Adult; Aged; Analgesia; Child; Clinical Trials as Topic; Female; Humans; Injections, Intramuscular; Male; Middle Aged; Pentazocine; Phenazocine; Postoperative Care

1966
Oral pentazocine and phenazocine: a comparison in postoperative pain.
    British journal of anaesthesia, 1971, Volume: 43, Issue:5

    Topics: Administration, Oral; Adolescent; Adult; Aged; Consciousness; Female; Humans; Male; Middle Aged; Nausea; Pain; Pentazocine; Phenazocine; Postoperative Complications; Time Factors; Vertigo

1971
Studies of drugs given before anaesthesia. 13. Pentazocine and other opiate antagonists.
    British journal of anaesthesia, 1967, Volume: 39, Issue:8

    Topics: Adult; Central Nervous System; Drug Antagonism; Female; Humans; Levallorphan; Meperidine; Morphine; Nalorphine; Pentazocine; Phenazocine; Preanesthetic Medication; Psychoses, Substance-Induced

1967

Other Studies

61 other study(ies) available for phenazocine and pentazocine

ArticleYear
The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists.
    Proceedings of the National Academy of Sciences of the United States of America, 1976, Volume: 73, Issue:11

    Topics: Allosteric Regulation; Dextropropoxyphene; Fentanyl; Methadone; Models, Biological; Models, Molecular; Molecular Conformation; Morphine; Nalorphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Protein Conformation; Receptors, Opioid; Structure-Activity Relationship

1976
Interaction of sigma and PCP-like drugs on operant behaviors in the rat.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: Animals; Conditioning, Operant; Dextroamphetamine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Pentazocine; Phenazocine; Phencyclidine; Psychotropic Drugs; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule

1992
Neuroprotective effects of SKF 10,047 in cultured rat cerebellar neurons and in gerbil global brain ischemia.
    Stroke, 1992, Volume: 23, Issue:3

    Topics: Animals; Body Temperature; Brain Ischemia; Cells, Cultured; Cerebellum; Cyclazocine; Dizocilpine Maleate; Gerbillinae; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Reference Values; Stereoisomerism

1992
Chronic treatment with pentazocine or SFK 10047 decrease proenkephalin mRNA levels in the rat striatum and nucleus accumbens.
    Neuroscience letters, 1991, Jan-14, Volume: 122, Issue:1

    Topics: Animals; Base Sequence; Corpus Striatum; Enkephalins; Histocytochemistry; Male; Molecular Sequence Data; Nucleic Acid Hybridization; Nucleus Accumbens; Pentazocine; Phenazocine; Protein Precursors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; RNA, Messenger

1991
Psychomotor activity and cognitive disruption attributable to NMDA, but not sigma, interactions in primates.
    Behavioural brain research, 1991, Feb-28, Volume: 42, Issue:2

    Topics: Animals; Ataxia; Cognition; Dizocilpine Maleate; Macaca mulatta; Male; Pentazocine; Phenazocine; Phencyclidine; Psychomotor Performance; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Saimiri; Space Perception

1991
(+)-6,7-benzomorphan sigma ligands stimulate dopamine synthesis in rat corpus striatum tissue.
    Brain research, 1991, Aug-23, Volume: 557, Issue:1-2

    Topics: Animals; Benzomorphans; Catecholamines; Corpus Striatum; Cyclazocine; Dopamine; In Vitro Techniques; Ligands; Male; Nerve Endings; Neural Pathways; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Stimulation, Chemical; Tyrosine 3-Monooxygenase

1991
The human sigma site, which resembles that in NCB20 cells, may correspond to a low-affinity site in guinea pig brain.
    Neuroscience letters, 1991, Oct-14, Volume: 131, Issue:2

    Topics: Animals; Brain Chemistry; Cells, Cultured; Cerebral Cortex; Cricetinae; Cricetulus; Dopamine Agents; Guanidines; Guinea Pigs; Humans; Kinetics; Male; Mice; Neuroblastoma; Pentazocine; Phenazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Tumor Cells, Cultured

1991
Similar behavioural effects of sigma agonists and PCP-like non-competitive NMDA antagonists in guinea-pigs.
    Psychopharmacology, 1991, Volume: 105, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Dizocilpine Maleate; Dopamine Agents; Dopamine Antagonists; Ergolines; Female; Guanidines; Guinea Pigs; Haloperidol; Ketamine; Male; Motor Activity; N-Methylaspartate; Pentazocine; Phenazocine; Phencyclidine; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride

1991
(+) 3-[3-hydroxyphenyl-N-(1-propyl) piperidine] selectively differentiates effects of sigma ligands on neurochemical pathways modulated by sigma receptors: evidence for subtypes, in vivo.
    Neuropharmacology, 1991, Volume: 30, Issue:8

    Topics: Adrenocorticotropic Hormone; Animals; Brain; Butaclamol; Cerebellum; Corpus Striatum; Cyclic GMP; Dopamine; Dopamine Agents; Male; Mice; Pentazocine; Phenazocine; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma

1991
Stereospecificity of mixed-action opioid agonist/antagonists in morphine-tolerant squirrel monkeys.
    NIDA research monograph, 1990, Volume: 105

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Morphine; Narcotic Antagonists; Narcotics; Pentazocine; Phenazocine; Saimiri; Stereoisomerism

1990
Sigma receptors modulate both A9 and A10 dopaminergic neurons in the rat brain: functional interaction with NMDA receptors.
    Brain research, 1990, Aug-06, Volume: 524, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Cerebral Ventricles; Dopamine; Kinetics; Male; Neurons; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma

1990
The lack of utility of the rat vas deferens as a functional bioassay for sigma ligands.
    European journal of pharmacology, 1991, Feb-07, Volume: 193, Issue:2

    Topics: Animals; Binding Sites; Biological Assay; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; Male; Muscle Contraction; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Vas Deferens

1991
Characterization of [3H] (+)-pentazocine, a highly selective sigma ligand.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Binding, Competitive; Brain; Guinea Pigs; In Vitro Techniques; Kinetics; Pentazocine; Phenazocine; Piperidines; Receptors, Opioid; Receptors, sigma

1990
Sigma receptors modulate the hypothalamic-pituitary-adrenal (HPA) axis centrally: evidence for a functional interaction with NMDA receptors, in vivo.
    Neuropharmacology, 1990, Volume: 29, Issue:3

    Topics: Adrenocorticotropic Hormone; Animals; Aspartic Acid; Cells, Cultured; Hypothalamo-Hypophyseal System; Male; N-Methylaspartate; Pentazocine; Phenazocine; Piperazines; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, sigma

1990
Differential effects of sigma and phencyclidine receptor ligands on learning.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Avoidance Learning; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Ligands; Male; Memory; Pentazocine; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Retention, Psychology

1990
Neuropeptide Y and peptide YY interact with rat brain sigma and PCP binding sites.
    European journal of pharmacology, 1989, Dec-19, Volume: 174, Issue:2-3

    Topics: Animals; Brain Chemistry; Haloperidol; In Vitro Techniques; Male; Neuropeptide Y; Pentazocine; Peptide YY; Peptides; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1989
Biochemical, behavioral, and electrophysiologic actions of the selective sigma receptor ligand (+)-pentazocine.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1988, Volume: 1, Issue:4

    Topics: Animals; Avoidance Learning; Brain; Discrimination Learning; Evoked Potentials, Visual; Male; Membranes; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Reference Values

1988
Body temperature effects of opioids in rats: intracerebroventricular administration.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:6

    Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains

1986
Discriminative stimulus properties of (+)-N-allylnormetazocine in the rat: correlations with (+)-N-allylnormetazocine and phencyclidine receptor binding.
    Psychopharmacology, 1987, Volume: 91, Issue:1

    Topics: Animals; Brain; Cyclazocine; Discrimination Learning; Ketamine; Male; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism

1987
Effects of some analgesics and antidepressants on the (Na + + K + )-adenosine triphosphatase from cortices of brain and kidney.
    Biochemical pharmacology, 1972, Aug-01, Volume: 21, Issue:15

    Topics: Adenosine Triphosphatases; Amitriptyline; Analgesics; Animals; Antidepressive Agents; Cattle; Cerebral Cortex; Chlorpromazine; Cyclazocine; Desipramine; Dose-Response Relationship, Drug; Hydralazine; Imipramine; In Vitro Techniques; Kidney; Kidney Cortex; Pentazocine; Phenazocine; Phenelzine; Potassium; Sodium; Tranylcypromine

1972
Effects of opiates and opiate antagonists on the Straub tail reaction in mice.
    British journal of pharmacology, 1969, Volume: 36, Issue:2

    Topics: Analgesics; Animals; Atropine; Bridged-Ring Compounds; Codeine; Cyclazocine; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Narcotic Antagonists; Pentazocine; Phenazocine; Stereoisomerism; Tail

1969
Effects of narcotic analgesics on contractions of the chick isolated, innervated oesophagus.
    The Journal of pharmacy and pharmacology, 1972, Volume: 24, Issue:9

    Topics: Acetylcholine; Analgesics; Animals; Chickens; Cyclazocine; Dextropropoxyphene; Electric Stimulation; Esophagus; Heroin; In Vitro Techniques; Meperidine; Methadone; Morphinans; Morphine; Muscle Contraction; Nalorphine; Pentazocine; Phenazocine; Serotonin; Tachyphylaxis; Time Factors

1972
Energy-dependent uptake of benzomorphans by leukocytes.
    Biochemical pharmacology, 1972, Jun-01, Volume: 21, Issue:11

    Topics: Animals; Cell Membrane; Chromatography, Gas; Cyclazocine; Fluorides; Glucose; Leukocytes; Male; Models, Biological; Oxygen Consumption; Pentazocine; Phenazocine; Potassium; Rats; Sodium; Structure-Activity Relationship; Time Factors

1972
Potent long-acting antagonists of the 9,9-dialkylbenzomorphan series.
    Advances in biochemical psychopharmacology, 1973, Volume: 8, Issue:0

    Topics: Alkylation; Analgesics; Animals; Butyrates; Cyclazocine; Cyclization; Isomerism; Methylation; Morphinans; Narcotic Antagonists; Pentazocine; Phenazocine; Phenols; Propionates; Rats; Structure-Activity Relationship; Time Factors

1973
Pentazocine radioimmunoassay.
    Research communications in chemical pathology and pharmacology, 1974, Volume: 7, Issue:1

    Topics: Ammonium Sulfate; Animals; Antibody Specificity; Antigen-Antibody Reactions; Azo Compounds; Carboxylic Acids; Chromatography, Gas; Cross Reactions; Cyclazocine; Levallorphan; Levorphanol; Methods; Molecular Weight; Morphine; Nalorphine; Oxidation-Reduction; Pentazocine; Phenazocine; Rabbits; Radioimmunoassay; Tritium; Urine

1974
Comparison of effect of morphine-like analgesics on transmurally stimulated guinea-pig ileum.
    British journal of pharmacology, 1969, Volume: 37, Issue:2

    Topics: Analgesics; Animals; Codeine; Cyclic N-Oxides; Drug Tolerance; Electric Stimulation; Female; Fentanyl; Guinea Pigs; Heroin; Humans; Ileum; In Vitro Techniques; Male; Meperidine; Morphinans; Morphine; Muscle Contraction; Muscle, Smooth; Nalorphine; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine; Rats; Substance-Related Disorders; Urinary Bladder

1969
The determination of benzomorphan derivatives in plasma by gas chromatography.
    Life sciences. Pt. 1: Physiology and pharmacology, 1971, Jun-15, Volume: 10, Issue:12

    Topics: Analgesics; Azocines; Cyclazocine; Humans; Methods; Narcotic Antagonists; Pentazocine; Phenazocine

1971
Effects of analgesics and other drugs on mice in phenylquinone and rotarod tests.
    The Journal of pharmacology and experimental therapeutics, 1969, Volume: 167, Issue:1

    Topics: Analgesics; Animals; Chemical Phenomena; Chemistry; Chlorpromazine; Cyclazocine; Dextroamphetamine; Levallorphan; Male; Mice; Morphine; Motor Activity; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Pilocarpine; Quinones; Salivation

1969
The interaction between monoamine oxidase inhibitors and narcotic analgesics in mice.
    British journal of pharmacology, 1969, Volume: 36, Issue:3

    Topics: Analgesics; Animals; Drug Synergism; Iproniazid; Meperidine; Mice; Monoamine Oxidase Inhibitors; Morphine; Pentazocine; Phenazocine; Tranylcypromine

1969
Agonist and antagonist actions of morphine-like drugs on the guinea-pig isolated ileum.
    British journal of pharmacology and chemotherapy, 1966, Volume: 27, Issue:3

    Topics: Analgesics; Animals; Cyclazocine; Drug Synergism; Guinea Pigs; Ileum; Levallorphan; Levorphanol; Morphine; Muscle, Smooth; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Reflex

1966
Effects of elevated calcium and calcium antagonists on 6,7-benzomorphan-induced analgesia.
    European journal of pharmacology, 1983, Jun-17, Volume: 90, Issue:4

    Topics: Analgesia; Analgesics; Analgesics, Opioid; Animals; Benzomorphans; Calcium; Calcium Channel Blockers; Cyclazocine; Egtazic Acid; Ethylketocyclazocine; Gallopamil; Male; Mice; Morphinans; Pentazocine; Phenazocine

1983
Central injection of a sigma opioid receptor agonist alters body temperature of cats.
    Brain research bulletin, 1981, Volume: 7, Issue:3

    Topics: Animals; Body Temperature Regulation; Cats; Dose-Response Relationship, Drug; Pentazocine; Phenazocine; Receptors, Opioid

1981
Effects of the combination of tripelennamine and pentazocine at the behavioral and molecular levels.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:4

    Topics: Animals; Brain; Diphenhydramine; Discrimination, Psychological; Drug Synergism; Guinea Pigs; Ileum; Learning; Male; Morphine; Pentazocine; Phenazocine; Rats; Receptors, Opioid; Synaptic Membranes; Tripelennamine

1982
Discriminative stimulus effects of etorphine in Rhesus monkeys.
    Psychopharmacology, 1981, Volume: 72, Issue:3

    Topics: Animals; Codeine; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Etorphine; Macaca mulatta; Male; Meperidine; Morphinans; Morphine; Pentazocine; Phenazocine; Sodium Chloride

1981
Subclasses of opioids based on body temperature change in rats: acute subcutaneous administration.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:2

    Topics: Animals; Body Temperature; Buprenorphine; Dose-Response Relationship, Drug; Endorphins; Injections, Subcutaneous; Male; Meperidine; Morphine; Nalbuphine; Naloxone; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains

1983
Differential effects of prototype opioid agonists on the acquisition of conditional discriminations in monkeys.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Animals; Behavior, Animal; Conditioning, Psychological; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Male; Morphine; Pentazocine; Phenazocine; Psychomotor Performance

1983
Acquisition of brightness discrimination in the rat is impaired by opiates with psychotomimetic properties.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:6

    Topics: Animals; Avoidance Learning; Cyclazocine; Discrimination Learning; Male; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Phenazocine; Photic Stimulation; Psychotropic Drugs; Rats; Rats, Inbred F344

1983
Phosphorylation of synapsin I and dynamin in rat forebrain synaptosomes: modulation by sigma (sigma) ligands.
    Neuroscience letters, 1995, May-19, Volume: 191, Issue:1-2

    Topics: Animals; Anticonvulsants; Dynamins; GTP Phosphohydrolases; Guanidines; Haloperidol; In Vitro Techniques; Microtubules; Pentazocine; Phenazocine; Phosphorylation; Prosencephalon; Rats; Receptors, sigma; Synapsins; Synaptosomes

1995
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
    Brain research, 1995, Feb-06, Volume: 671, Issue:1

    Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma

1995
Acute effects of sigma ligands on the extracellular DOPAC level in rat frontal cortex and striatum.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Corpus Striatum; Extracellular Space; Frontal Lobe; Guanidines; Kinetics; Ligands; Male; Microdialysis; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Time Factors

1995
Effects of sigma and phencyclidine receptor ligands on electric field-stimulated rabbit ear artery constriction in vitro.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1994, Volume: 15, Issue:4

    Topics: Animals; Arteries; Dizocilpine Maleate; Ear; Electric Stimulation; Female; In Vitro Techniques; Ligands; Male; Pentazocine; Phenazocine; Phencyclidine; Rabbits; Receptors, Phencyclidine; Receptors, sigma; Vasoconstriction

1994
Low dose of 1,3-di(2-tolyl)guanidine (DTG) attenuates MK-801-induced spatial working memory impairment in mice.
    Psychopharmacology, 1994, Volume: 114, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Dizocilpine Maleate; Dose-Response Relationship, Drug; Guanidines; Male; Memory; Mice; Mice, Inbred Strains; Motor Activity; Pentazocine; Phenazocine; Pyrimidines; Receptors, sigma; Space Perception

1994
SKF-10,047 reverses stress-induced motor suppression: interaction with dopaminergic system.
    European journal of pharmacology, 1994, Jul-21, Volume: 260, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anticonvulsants; Apomorphine; Dopamine; Electroshock; Guanidines; Male; Methamphetamine; Mice; Mice, Inbred Strains; Motor Activity; Oxidopamine; Pentazocine; Phenazocine; Pimozide; Pyrimidines; Receptors, sigma; Stress, Psychological

1994
Regulation of [3H]dopamine release from rat striatal slices by sigma receptor ligands.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:1

    Topics: Animals; Atropine; Corpus Striatum; Dopamine; Flavonoids; In Vitro Techniques; N-Methylaspartate; Naloxone; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma

1994
Allosteric modulation of ligand binding to [3H](+)pentazocine-defined sigma recognition sites by phenytoin.
    Life sciences, 1993, Volume: 53, Issue:1

    Topics: Allosteric Regulation; Animals; Binding Sites; Cyclopentanes; Dextromethorphan; Dextrorphan; Guinea Pigs; Ligands; Male; Pentazocine; Phenazocine; Phenytoin; Piperidines; Radioligand Assay; Receptors, sigma; Tritium

1993
In vivo modulation of sigma receptor sites by calcitonin gene-related peptide in the mouse and rat hippocampal formation: radioligand binding and electrophysiological studies.
    The European journal of neuroscience, 1995, Sep-01, Volume: 7, Issue:9

    Topics: Animals; Antipsychotic Agents; Calcitonin Gene-Related Peptide; Dopamine Antagonists; Electrophysiology; Haloperidol; Hippocampus; In Vitro Techniques; Iontophoresis; Male; Membranes; Mice; Narcotics; Neuropeptide Y; Pentazocine; Phenazocine; Pyramidal Cells; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma

1995
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:1

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens

1996
Differential solubilization of rat liver sigma 1 and sigma 2 receptors: retention of sigma 2 sites in particulate fractions.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Animals; Binding, Competitive; Cell Fractionation; Cell Membrane; Cholic Acids; Detergents; Guanidines; Haloperidol; In Vitro Techniques; Liver; Male; Pentazocine; Phenazocine; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Solubility; Subcellular Fractions

1996
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
    Journal of neuroimmunology, 1997, Volume: 72, Issue:1

    Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium

1997
Sigma1 recognition sites in rabbit iris-ciliary body: topical sigma1-site agonists lower intraocular pressure.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: Animals; Anisoles; Antipsychotic Agents; Binding, Competitive; Cell Membrane; Ciliary Body; Functional Laterality; Guanidines; Intraocular Pressure; Iris; Kinetics; Lens, Crystalline; Male; Pentazocine; Phenazocine; Propylamines; Rabbits; Receptors, sigma; Retina; Tritium

1999
Intracellular sigma1 receptor modulates phospholipase C and protein kinase C activities in the brainstem.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, Jul-06, Volume: 96, Issue:14

    Topics: Action Potentials; Animals; Antipsychotic Agents; Brain Stem; Cell Membrane; Cytoplasm; GTP-Binding Proteins; Guinea Pigs; Haloperidol; In Vitro Techniques; Isoenzymes; Ligands; Male; Pentazocine; Pertussis Toxin; Phenazocine; Protein Kinase C; Protein Kinase C beta; Receptors, sigma; Respiratory Mechanics; Reverse Transcriptase Polymerase Chain Reaction; Type C Phospholipases; Virulence Factors, Bordetella

1999
Membrane-delimited coupling between sigma receptors and K+ channels in rat neurohypophysial terminals requires neither G-protein nor ATP.
    The Journal of physiology, 2000, Aug-01, Volume: 526 Pt 3

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Antipsychotic Agents; Cells, Cultured; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine Triphosphate; In Vitro Techniques; Ligands; Oocytes; Patch-Clamp Techniques; Pentazocine; Phenazocine; Phosphorylation; Pituitary Gland, Posterior; Potassium; Potassium Channels; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptic Membranes; Xenopus laevis

2000
Effects of sigma receptor agonists on the impairment of spontaneous alternation behavior and decrease of cyclic GMP level induced by nitric oxide synthase inhibitors in mice.
    Neuropharmacology, 2000, Volume: 39, Issue:12

    Topics: Analgesics, Opioid; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Behavior, Animal; Brain Chemistry; Cyclic GMP; Enzyme Inhibitors; Guanidines; Indazoles; Male; Methylene Blue; Mice; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Pentazocine; Phenazocine; Pyrimidines; Receptors, sigma

2000
Phencyclidine impairs latent learning in mice: interaction between glutamatergic systems and sigma(1) receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 24, Issue:4

    Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Behavior, Animal; Cycloserine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Exploratory Behavior; Glutamic Acid; Learning; Male; Mice; Mice, Inbred Strains; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Piperazines; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism

2001
SOME NARCOTIC ANTAGONISTS IN THE BENZOMORPHAN SERIES.
    The Journal of pharmacology and experimental therapeutics, 1964, Volume: 143

    Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Antipyretics; Azocines; Benzomorphans; Cats; Cyclazocine; Haplorhini; Heterocyclic Compounds; Meperidine; Mice; Morphine; Nalorphine; Narcotic Antagonists; Pentazocine; Pharmacology; Phenazocine; Rats; Research; Toxicology

1964
Generation and phenotypic analysis of sigma receptor type I (sigma 1) knockout mice.
    The European journal of neuroscience, 2003, Volume: 18, Issue:8

    Topics: Animals; Animals, Newborn; Antidepressive Agents; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Blotting, Northern; Blotting, Southern; Blotting, Western; Body Weight; Cells, Cultured; Embryo, Mammalian; Endorphins; Heterozygote; Hyperkinesis; In Situ Hybridization; Mice; Mice, Knockout; Narcotic Antagonists; Oligonucleotides, Antisense; Pentazocine; Peptide Fragments; Phenazocine; Phenotype; Radioligand Assay; Receptors, sigma; Sigma-1 Receptor; Time Factors

2003
Voltage-gated sodium channel modulation by sigma-receptors in cardiac myocytes and heterologous systems.
    American journal of physiology. Cell physiology, 2009, Volume: 296, Issue:5

    Topics: Adenosine Triphosphate; Animals; Antipsychotic Agents; Cell Line; Chlorocebus aethiops; COS Cells; Guanosine Triphosphate; Haloperidol; Humans; Kidney; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Proteins; Myocytes, Cardiac; Narcotics; NAV1.5 Voltage-Gated Sodium Channel; Patch-Clamp Techniques; Pentazocine; Phenazocine; Receptors, sigma; RNA, Small Interfering; Sodium; Sodium Channels

2009
Sigma-1 receptor function is critical for both the discriminative stimulus and aversive effects of the kappa-opioid receptor agonist U-50488H.
    Addiction biology, 2012, Volume: 17, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anisoles; Avoidance Learning; Conditioning, Psychological; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Propylamines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor

2012
Sigma-1 receptor stimulation attenuates calcium influx through activated L-type Voltage Gated Calcium Channels in purified retinal ganglion cells.
    Experimental eye research, 2013, Volume: 107

    Topics: Animals; Animals, Newborn; Blotting, Western; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Ethylenediamines; Fluorescent Antibody Technique, Indirect; Fura-2; Microscopy, Fluorescence; Pentazocine; Phenazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Retinal Ganglion Cells; Sigma-1 Receptor; Verapamil

2013
NMDA receptors are upregulated and trafficked to the plasma membrane after sigma-1 receptor activation in the rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Aug-20, Volume: 34, Issue:34

    Topics: Animals; Cell Membrane; Disks Large Homolog 4 Protein; Ethylenediamines; Hippocampus; Intracellular Signaling Peptides and Proteins; Male; Membrane Proteins; Mice; Mice, Knockout; Morpholines; Pentazocine; Phenazocine; Piperazines; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Subcellular Fractions; Time Factors; Up-Regulation

2014