phenazocine has been researched along with naloxone in 72 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 63 (87.50) | 18.7374 |
1990's | 7 (9.72) | 18.2507 |
2000's | 1 (1.39) | 29.6817 |
2010's | 1 (1.39) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creese, I; Feinberg, AP; Snyder, SH | 1 |
Chiba, S; Nishida, N; Yasuhara, Y | 1 |
Defaux, JP; Junien, JL; Pascaud, X; Rozé, C | 1 |
Goldberg, SR; Schindler, CW; White, MF | 1 |
Kobylyansky, AG | 1 |
Kamei, H; Kameyama, T; Nabeshima, T | 1 |
Holtzman, SG | 1 |
Cowan, A; Jacoby, HI; Vaught, JL | 1 |
Chung, JM; Kim, J; Shin, HK; Willcockson, WS; Willis, WD | 1 |
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K | 1 |
Cohen, S; Ouyang, A; Vos, P | 1 |
Adler, MW; Geller, EB; Rowan, CH | 1 |
George, R; Pechnick, R; Poland, RE | 1 |
Adler, MW; Geller, EB; Kirby, A; Messner, S; Robin, M | 1 |
Calligaro, D; el-Fakahany, EE; Hong, O; Khazan, N; Young, GA | 1 |
Eisenberg, RM | 1 |
Baba, Y; Ban, M; Fujimura, H; Hori, M; Imai, E; Iwata, N; Morita, T; Niwa, M; Nozaki, M; Suzuki, Y | 1 |
Starr, MS | 1 |
Greenberg, BD; Segal, DS | 1 |
DeRossett, SE; Holtzman, SG | 1 |
Ieni, JR; Nichtenhauser, R; Sircar, R; Zukin, SR | 1 |
Su, TP; Weissman, AD; Yeh, SY | 1 |
Contreras, PC; O'Donohue, TL; Quirion, R | 1 |
Hiramatsu, M; Kameyama, T; Nabeshima, T | 1 |
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR | 1 |
Giles, TD; Given, MB; Lowe, RF; Sander, GE | 1 |
Bartschat, DK; Blaustein, MP | 1 |
Dzhumbaev, SU; Egamov, IuS; Polonskiĭ, VM; Vinogradov, VA | 1 |
Dykstra, LA; Picker, M | 1 |
Dykstra, LA; Heise, JW; Picker, M | 1 |
Harris, LS; May, EL | 1 |
Costa, T; Dunn, LL; Hubbell, CL; Hunter, GA; Reid, LD | 1 |
Clark, RD; Katz, JL; Spealman, RD | 1 |
Bergman, J; Hassoun, J; Schuster, CR | 1 |
Pierson, AK | 1 |
Pert, CB; Snyder, SH | 1 |
Cowan, A; Gmerek, DE | 2 |
Miller, RJ | 1 |
Tung, AS; Yaksh, TL | 1 |
Leander, JD | 1 |
Enger, M; Grynne, BH; Holmen, AT; Maurset, AR | 1 |
Billington, CJ; Gerritsen, GC; Levine, AS; Morley, JE | 1 |
Rackham, A; Wood, PL | 1 |
Balster, RL; Brady, KT; May, EL | 1 |
Harris, RA; Snell, D | 1 |
Nishimura, S; Pasternak, GW; Wolozin, BL | 1 |
Nishimura, S; Pasternak, GW | 1 |
Bearden, LJ; Snead, OC | 1 |
Kandasamy, SB; Williams, BA | 1 |
Cicero, TJ; Meyer, ER; Owens, DP; Schmoeker, PF | 1 |
Johnson, N; Pasternak, GW | 1 |
Aceto, MD; May, EL | 1 |
Vaupel, DB | 1 |
Martin, WR; Wu, KM | 1 |
Tam, SW | 1 |
Gosnell, BA; Levine, AS; Morley, JE | 1 |
Greenfield, LJ; Guyenet, PG; Hackett, JT; Stringer, JL | 1 |
Code, RA; Tang, AH | 1 |
Michne, WF; Pierson, AK; Ward, SJ | 1 |
Johnson, KM; Leventer, SM | 1 |
Commissaris, RL; Henck, JW; Mokler, DJ; Rech, RH | 1 |
Colpaert, FC; Janssen, PA | 1 |
Shannon, HE | 2 |
Adler, MW; Geller, EB; Hawk, C; Keinath, SH; Tallarida, RJ | 1 |
Gonzalez-Alvear, GM; Werling, LL | 1 |
Brent, PJ; Chahl, LA | 1 |
Su, TP; Tsao, LI | 1 |
Lashkari, SB; Shafiee, A; Tabatabai, SA; Zarrindast, MR | 1 |
Botros, M; Carlsson, A; Fransson, R; Gordh, T; Hallberg, M; Nyberg, F; Sandström, A; Zhou, Q | 1 |
Hall, FS; Kitanaka, J; Kitanaka, N; Nishiyama, N; Takemura, M; Tanaka, K; Uhl, GR | 1 |
3 review(s) available for phenazocine and naloxone
Article | Year |
---|---|
Drug discrimination studies.
Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Assays for narcotic antagonist activity in rodents.
Topics: Analgesics; Animals; Depression, Chemical; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Heroin; Hot Temperature; Lens, Crystalline; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Nalorphine; Naloxone; Narcotic Antagonists; Oxymorphone; Phenazocine; Pressure; Rabbits; Rats; Reaction Time; Reflex; Respiration; Tail | 1973 |
Multiple opiate receptors for multiple opioid peptides.
Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission | 1982 |
69 other study(ies) available for phenazocine and naloxone
Article | Year |
---|---|
The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists.
Topics: Allosteric Regulation; Dextropropoxyphene; Fentanyl; Methadone; Models, Biological; Models, Molecular; Molecular Conformation; Morphine; Nalorphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Protein Conformation; Receptors, Opioid; Structure-Activity Relationship | 1976 |
[Evaluation of the discriminative stimulus effect of an enkephalin analog, EK-399, in the rat].
Topics: Animals; Discrimination, Psychological; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1991 |
Effect of selective sigma ligands on duodenal alkaline secretion in the rat.
Topics: Animals; Atropine; Bicarbonates; Dose-Response Relationship, Drug; Duodenum; Guanidines; Haloperidol; Injections, Intravenous; Intestinal Mucosa; Intestinal Secretions; Male; Naloxone; Phenazocine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Yohimbine | 1990 |
Effects of morphine, ethylketocyclazocine, N-allylnormetazocine and naloxone on locomotor activity in the rabbit.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Female; Male; Morphine; Motor Activity; Naloxone; Nictitating Membrane; Phenazocine; Rabbits | 1990 |
Opioids induce postural asymmetry in spinal rat: the side of the flexed limb depends upon the type of opioid agonist.
Topics: Animals; Benzomorphans; Decerebrate State; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Functional Laterality; Male; Muscles; Naloxone; Narcotics; Phenazocine; Posture; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord; Time Factors | 1989 |
A role played by sigma receptors in the conditioned suppression of motility in mice.
Topics: Animals; Conditioning, Psychological; Cyclazocine; Drug Tolerance; Male; Mice; Mice, Inbred Strains; Motor Activity; Naloxone; Phenazocine; Receptors, Opioid; Receptors, sigma; Synaptic Membranes | 1988 |
Mu and delta, but not kappa, opioid agonists induce contractions of the canine small intestine in vivo.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dogs; Duodenum; Dynorphins; Electric Stimulation; Enkephalin, Methionine; Female; Gastrointestinal Motility; Male; Morphine; Morphine Derivatives; Naloxone; Peptide Fragments; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Actions of opioids on primate spinothalamic tract neurons.
Topics: Animals; Dynorphins; Enkephalin, Methionine; Macaca fascicularis; Morphine; Naloxone; Narcotics; Neurons; Phenazocine; Phencyclidine; Spinal Cord; Thalamus | 1986 |
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid | 1987 |
Sites of action of mu-, kappa- and sigma-opiate receptor agonists at the feline ileocecal sphincter.
Topics: Animals; Atropine; Cats; Dynorphins; Ganglionic Blockers; Ileocecal Valve; Morphine; Naloxone; Phenazocine; Receptors, Opioid; Tachyphylaxis; Tetrodotoxin; Vagotomy | 1988 |
Body temperature effects of opioids in rats: intracerebroventricular administration.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1986 |
Identification of multiple opiate receptors through neuroendocrine responses. II. Antagonism of mu, kappa and sigma agonists by naloxone and WIN 44,441-3.
Topics: Animals; Azocines; Corticosterone; Cyclazocine; Drug Interactions; Ethylketocyclazocine; Growth Hormone; Luteinizing Hormone; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Pituitary Hormones, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid | 1985 |
Differentiating opioids by their pupillary effects in the rat.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Methadone; Motor Activity; Naloxone; Narcotics; Nystagmus, Physiologic; Phenazocine; Pupil; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism | 1985 |
Sigma opioid receptors; SKF-10,047 update.
Topics: Animals; Electroencephalography; Female; Hallucinogens; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1985 |
Plasma corticosterone changes in response to central or peripheral administration of kappa and sigma opiate agonists.
Topics: Animals; Brain; Corticosterone; Cyclazocine; Ethylketocyclazocine; Humans; Hypothalamo-Hypophyseal System; Male; Morphine; Naloxone; Naltrexone; Opioid-Related Disorders; Phenazocine; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1985 |
Novel nonnarcotic analgesics with an improved therapeutic ratio. Structure-activity relationships of 8-(methylthio)- and 8-(acylthio)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines.
Topics: Acylation; Analgesia; Animals; Brain; Chemical Phenomena; Chemistry; Methylation; Mice; Morphinans; Morphine; Naloxone; Oxygen; Phenazocine; Rabbits; Rats; Receptors, Opioid; Structure-Activity Relationship; Sulfur | 1985 |
Multiple opiate receptors may be involved in suppressing gamma-aminobutyrate release in substantia nigra.
Topics: Aminooxyacetic Acid; Animals; Benzomorphans; Dopamine; Enkephalin, Methionine; Female; gamma-Aminobutyric Acid; Male; Naloxone; Nialamide; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Secretory Rate; Substantia Nigra | 1985 |
Evidence for multiple opiate receptor involvement in different phencyclidine-induced unconditioned behaviors in rats.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Eating; Habituation, Psychophysiologic; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereotyped Behavior | 1986 |
Discriminative stimulus effects of the opioid antagonist diprenorphine in the squirrel monkey.
Topics: Animals; Cyclazocine; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Generalization, Stimulus; Morphinans; Naloxone; Narcotic Antagonists; Phenazocine; Psychotropic Drugs; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Saimiri | 1986 |
Characterization and autoradiographic visualization of (+)-[3H]SKF10,047 binding in rat and mouse brain: further evidence for phencyclidine/"sigma opiate" receptor commonality.
Topics: Animals; Autoradiography; Brain Chemistry; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Species Specificity; Tritium | 1986 |
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays.
Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma | 1986 |
Agonistic and antagonistic effects of PCP-derivatives and sigma opioids in PCP behavioral and receptor assays.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclazocine; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereotyped Behavior; Structure-Activity Relationship; Tritium | 1986 |
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid | 1986 |
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1987 |
N-allylnormetazocine: hemodynamic actions and inhibition of leucine-enkephalin hemodynamic activity in conscious dogs.
Topics: Animals; Blood Pressure; Dogs; Enkephalin, Leucine; Female; Heart Rate; Hemodynamics; Male; Naloxone; Phenazocine; Stereoisomerism | 1988 |
Psychotomimetic sigma-ligands, dexoxadrol and phencyclidine block the same presynaptic potassium channel in rat brain.
Topics: Animals; Brain; Cyclazocine; Dioxolanes; Dioxoles; Dose-Response Relationship, Drug; Hallucinogens; In Vitro Techniques; Naloxone; Phenazocine; Phencyclidine; Piperidines; Potassium Channels; Rats; Synaptosomes | 1988 |
[Effect of opioid peptides on the lymphatic drainage of the pancreas in the rat and dog].
Topics: Animals; Dogs; Dose-Response Relationship, Drug; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Evans Blue; Female; Lymph; Male; Naloxone; Pancreas; Phenazocine; Rats; Rats, Inbred Strains | 1988 |
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors | 1987 |
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule | 1987 |
Historical introduction and review of chemistry.
Topics: Analgesics; Chemistry; History, 20th Century; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Phenazocine | 1985 |
Selected opioids and responding for intracranial reinforcement.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Hypothalamic Area, Lateral; Naloxone; Phenazocine; Rats; Reinforcement, Psychology; Self Stimulation; Stereoisomerism | 1985 |
Stereoselective behavioral effects of N-allylnormetazocine in pigeons and squirrel monkeys.
Topics: Animals; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Morphine; Naloxone; Phenazocine; Phencyclidine; Reinforcement Schedule; Saimiri; Stereoisomerism | 1985 |
Behavioral effects of selected opiates and phencyclidine in the nondependent and cyclazocine-dependent rhesus monkey.
Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Food; Macaca mulatta; Male; Naloxone; Phenazocine; Phencyclidine; Stereoisomerism; Substance-Related Disorders | 1985 |
Opiate receptor: demonstration in nervous tissue.
Topics: Analgesics; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Codeine; Colchicine; Dextromethorphan; Dextropropoxyphene; Guinea Pigs; Histamine; Intestinal Mucosa; Levallorphan; Methadone; Mice; Morphine; Nalorphine; Naloxone; Phenazocine; Phenobarbital; Rats; Receptors, Drug; Serotonin; Tritium | 1973 |
An in vivo pharmacological analysis of benzomorphan binding sites in rats.
Topics: Animals; Benzomorphans; Bombesin; Brain; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Grooming; Humans; Male; Morphinans; Morphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism; Stereotyped Behavior | 1984 |
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord | 1982 |
Effects of ketazocine, ethylketazocine and phenazocine on schedule-controlled behavior: antagonism by naloxone.
Topics: Analgesics, Opioid; Animals; Columbidae; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Naloxone; Phenazocine | 1982 |
The effect of two different buffers on the high affinity 3H-ethylketocyclazocine and 3H-SKF10047 binding to guinea pig brain membranes.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Ethylketocyclazocine; Guinea Pigs; HEPES; In Vitro Techniques; Morphine; Naloxone; Phenazocine; Piperazines; Receptors, Opioid; Tritium; Tromethamine | 1984 |
In vivo evidence for benzomorphan-selective receptors in rats.
Topics: Analgesics, Opioid; Animals; Benzomorphans; Bombesin; Buprenorphine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Male; Morphinans; Morphine; Naloxone; Phenazocine; Pruritus; Rats; Rats, Inbred Strains; Receptors, Opioid | 1984 |
Feeding systems in Chinese hamsters.
Topics: Animals; Brain; Calcitonin; Circadian Rhythm; Cricetinae; Cyclazocine; Diabetes Mellitus; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Feeding Behavior; Haloperidol; Mesocricetus; Naloxone; Peptide Fragments; Phenazocine; Sincalide; Starvation | 1984 |
Actions of kappa, sigma and partial mu narcotic receptor agonists on rat brain acetylcholine turnover.
Topics: Acetylcholine; Animals; Brain; Buprenorphine; Male; Morphinans; Naloxone; Organ Specificity; Phenazocine; Rats; Receptors, Opioid | 1981 |
Stereoisomers of N-allylnormetazocine: phencyclidine-like behavioral effects in squirrel monkeys and rats.
Topics: Animals; Behavior, Animal; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Saimiri; Stereoisomerism; Structure-Activity Relationship | 1982 |
Interactions between narcotic agonists, partial agonists andd antagonists evaluated by punished an unpunished behavior in the rat.
Topics: Animals; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Phenazocine; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid | 1982 |
The binding of kappa- and sigma-opiates in rat brain.
Topics: Animals; Binding Sites; Brain; Culture Techniques; Cyclazocine; Dihydromorphine; Enkephalins; Ethylketocyclazocine; Ligands; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Tritium | 1982 |
Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity.
Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Goldfish; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1982 |
The epileptogenic spectrum of opiate agonists.
Topics: Animals; Anticonvulsants; beta-Endorphin; Cyclazocine; Electroencephalography; Endorphins; Enkephalin, Leucine; Epilepsy; Ethylketocyclazocine; Injections, Intraventricular; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains | 1982 |
Peptide and non-peptide opioid-induced hyperthermia in rabbits.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptides; Phenazocine; Rats | 1983 |
Opiate-induced enhancement of the effects of naloxone on serum luteinizing hormone levels in the male rat: specificity for Mu agonists.
Topics: Animals; Binding, Competitive; Cyclazocine; Ethanol; Ethylketocyclazocine; Kinetics; Luteinizing Hormone; Male; Morphine; Naloxone; Pentobarbital; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
The binding to rat brain homogenates of Mr2034, a universal opiate.
Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
Antinociceptive studies of the optical isomers of N-allylnormetazocine (SKF 10,047).
Topics: Analgesics; Animals; Male; Mice; Mice, Inbred ICR; Morphine; Naloxone; Phenazocine; Receptors, Adrenergic, alpha; Receptors, Opioid; Stereoisomerism; Yohimbine | 1983 |
Naltrexone fails to antagonize the sigma effects of PCP and SKF 10,047 in the dog.
Topics: Animals; Body Temperature; Dogs; Female; Heart Rate; Morphine; Naloxone; Naltrexone; Paraplegia; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Reflex | 1983 |
An analysis of nicotinic and opioid processes in the medulla oblongata and nucleus ambiguus of the dog.
Topics: Animals; Blood Pressure; Cyclazocine; Decerebrate State; Dogs; Electric Stimulation; Endorphins; Ethylketocyclazocine; Female; Fentanyl; Heart Rate; Male; Mecamylamine; Medulla Oblongata; Naloxone; Nicotine; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1983 |
Naloxone-inaccessible sigma receptor in rat central nervous system.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalins; Ethylketocyclazocine; Kinetics; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Spinal Cord; Tissue Distribution | 1983 |
N-allylnormetazocine (SKF-10,047): the induction of feeding by a putative sigma agonist.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Interactions; Eating; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
Blockade of long-term potentiation by phencyclidine and sigma opiates in the hippocampus in vivo and in vitro.
Topics: Animals; Cyclazocine; Drug Synergism; Hippocampus; Male; Membrane Potentials; Morphine; Naloxone; Narcotics; Phenazocine; Phencyclidine; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synapses; Synaptic Transmission | 1983 |
Discriminative stimulus properties of nalorphine in the rhesus monkeys.
Topics: Animals; Benzodiazepines; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Macaca mulatta; Male; Nalorphine; Naloxone; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa | 1983 |
Multiple opioid receptor profile in vitro and activity in vivo of the potent opioid antagonist Win 44,441-3.
Topics: Animals; Azocines; Guinea Pigs; Ileum; Male; Mice; Morphine; Muscle Contraction; Naloxone; Narcotic Antagonists; Phenazocine; Receptors, Opioid; Vas Deferens | 1983 |
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains | 1984 |
Behavioral interactions of opioid agonists and antagonists with serotonergic systems.
Topics: Animals; Brain; Conditioning, Operant; Cyclazocine; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Lysergic Acid Diethylamide; Male; Metergoline; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement Schedule | 1984 |
Agonist and antagonist effects of prototype opiate drugs in rats discriminating fentanyl from saline: characteristics of partial generalization.
Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Male; Morphine; Nalorphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Sodium Chloride | 1984 |
Pharmacological evaluation of N-allynormetazocine (SKF 10,047) on the basis of its discriminative stimulus properties in the rat.
Topics: Animals; Benzomorphans; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Male; Naloxone; Phenazocine; Phencyclidine; Propranolol; Rats; Rats, Inbred F344; Stereoisomerism | 1983 |
Subclasses of opioids based on body temperature change in rats: acute subcutaneous administration.
Topics: Animals; Body Temperature; Buprenorphine; Dose-Response Relationship, Drug; Endorphins; Injections, Subcutaneous; Male; Meperidine; Morphine; Nalbuphine; Naloxone; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1983 |
Phencyclidine-like discriminative stimuli of (+)- and (-)-N-allylnormetazocine in rats.
Topics: Animals; Discrimination Learning; Discrimination, Psychological; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Reinforcement Schedule; Stereoisomerism | 1982 |
Regulation of [3H]dopamine release from rat striatal slices by sigma receptor ligands.
Topics: Animals; Atropine; Corpus Striatum; Dopamine; Flavonoids; In Vitro Techniques; N-Methylaspartate; Naloxone; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma | 1994 |
Enhancement of the opiate withdrawal response by antipsychotic drugs in guinea-pigs is not mediated by sigma binding sites.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Atropine; Behavior, Animal; Clozapine; Dizocilpine Maleate; Female; Guinea Pigs; Ketamine; Kinetics; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Raclopride; Radioligand Assay; Receptors, sigma; Remoxipride; Salicylamides; Substance Withdrawal Syndrome | 1993 |
Naloxone-sensitive, haloperidol-sensitive, [3H](+)SKF-10047-binding protein partially purified from rat liver and rat brain membranes: an opioid/sigma receptor?
Topics: Animals; Antipsychotic Agents; Brain; Haloperidol; Liver; Naloxone; Phenazocine; Radioligand Assay; Rats; Receptors, Opioid | 1997 |
Synthesis, conformational analysis and antinociceptive activity of 1-[N-methyl-(2-phenylethyl)amino]methyl-1,2,3,4-tetrahydroisoquinoline derivatives.
Topics: Analgesics; Analgesics, Opioid; Animals; Isoquinolines; Male; Mice; Molecular Conformation; Naloxone; Narcotic Antagonists; Phenazocine; Reaction Time; Stereoisomerism | 1999 |
The C-terminal amidated analogue of the substance P (SP) fragment SP(1-7) attenuates the expression of naloxone-precipitated withdrawal in morphine dependent rats.
Topics: Animals; Antipsychotic Agents; Brain; Male; Morphine Dependence; Naloxone; Peptide Fragments; Phenazocine; Rats; Rats, Wistar; Substance P; Substance Withdrawal Syndrome | 2009 |
Straub tail reaction in mice treated with σ(1) receptor antagonist in combination with methamphetamine.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Antipsychotic Agents; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Male; Methamphetamine; Mice; Mice, Inbred Strains; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Pyrimidines; Receptors, Opioid, delta; Reflex; Tail; Time Factors | 2012 |