Page last updated: 2024-08-21

phenazocine and naloxone

phenazocine has been researched along with naloxone in 72 studies

Research

Studies (72)

TimeframeStudies, this research(%)All Research%
pre-199063 (87.50)18.7374
1990's7 (9.72)18.2507
2000's1 (1.39)29.6817
2010's1 (1.39)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creese, I; Feinberg, AP; Snyder, SH1
Chiba, S; Nishida, N; Yasuhara, Y1
Defaux, JP; Junien, JL; Pascaud, X; Rozé, C1
Goldberg, SR; Schindler, CW; White, MF1
Kobylyansky, AG1
Kamei, H; Kameyama, T; Nabeshima, T1
Holtzman, SG1
Cowan, A; Jacoby, HI; Vaught, JL1
Chung, JM; Kim, J; Shin, HK; Willcockson, WS; Willis, WD1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Cohen, S; Ouyang, A; Vos, P1
Adler, MW; Geller, EB; Rowan, CH1
George, R; Pechnick, R; Poland, RE1
Adler, MW; Geller, EB; Kirby, A; Messner, S; Robin, M1
Calligaro, D; el-Fakahany, EE; Hong, O; Khazan, N; Young, GA1
Eisenberg, RM1
Baba, Y; Ban, M; Fujimura, H; Hori, M; Imai, E; Iwata, N; Morita, T; Niwa, M; Nozaki, M; Suzuki, Y1
Starr, MS1
Greenberg, BD; Segal, DS1
DeRossett, SE; Holtzman, SG1
Ieni, JR; Nichtenhauser, R; Sircar, R; Zukin, SR1
Su, TP; Weissman, AD; Yeh, SY1
Contreras, PC; O'Donohue, TL; Quirion, R1
Hiramatsu, M; Kameyama, T; Nabeshima, T1
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR1
Giles, TD; Given, MB; Lowe, RF; Sander, GE1
Bartschat, DK; Blaustein, MP1
Dzhumbaev, SU; Egamov, IuS; Polonskiĭ, VM; Vinogradov, VA1
Dykstra, LA; Picker, M1
Dykstra, LA; Heise, JW; Picker, M1
Harris, LS; May, EL1
Costa, T; Dunn, LL; Hubbell, CL; Hunter, GA; Reid, LD1
Clark, RD; Katz, JL; Spealman, RD1
Bergman, J; Hassoun, J; Schuster, CR1
Pierson, AK1
Pert, CB; Snyder, SH1
Cowan, A; Gmerek, DE2
Miller, RJ1
Tung, AS; Yaksh, TL1
Leander, JD1
Enger, M; Grynne, BH; Holmen, AT; Maurset, AR1
Billington, CJ; Gerritsen, GC; Levine, AS; Morley, JE1
Rackham, A; Wood, PL1
Balster, RL; Brady, KT; May, EL1
Harris, RA; Snell, D1
Nishimura, S; Pasternak, GW; Wolozin, BL1
Nishimura, S; Pasternak, GW1
Bearden, LJ; Snead, OC1
Kandasamy, SB; Williams, BA1
Cicero, TJ; Meyer, ER; Owens, DP; Schmoeker, PF1
Johnson, N; Pasternak, GW1
Aceto, MD; May, EL1
Vaupel, DB1
Martin, WR; Wu, KM1
Tam, SW1
Gosnell, BA; Levine, AS; Morley, JE1
Greenfield, LJ; Guyenet, PG; Hackett, JT; Stringer, JL1
Code, RA; Tang, AH1
Michne, WF; Pierson, AK; Ward, SJ1
Johnson, KM; Leventer, SM1
Commissaris, RL; Henck, JW; Mokler, DJ; Rech, RH1
Colpaert, FC; Janssen, PA1
Shannon, HE2
Adler, MW; Geller, EB; Hawk, C; Keinath, SH; Tallarida, RJ1
Gonzalez-Alvear, GM; Werling, LL1
Brent, PJ; Chahl, LA1
Su, TP; Tsao, LI1
Lashkari, SB; Shafiee, A; Tabatabai, SA; Zarrindast, MR1
Botros, M; Carlsson, A; Fransson, R; Gordh, T; Hallberg, M; Nyberg, F; Sandström, A; Zhou, Q1
Hall, FS; Kitanaka, J; Kitanaka, N; Nishiyama, N; Takemura, M; Tanaka, K; Uhl, GR1

Reviews

3 review(s) available for phenazocine and naloxone

ArticleYear
Drug discrimination studies.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Assays for narcotic antagonist activity in rodents.
    Advances in biochemical psychopharmacology, 1973, Volume: 8, Issue:0

    Topics: Analgesics; Animals; Depression, Chemical; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Heroin; Hot Temperature; Lens, Crystalline; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Nalorphine; Naloxone; Narcotic Antagonists; Oxymorphone; Phenazocine; Pressure; Rabbits; Rats; Reaction Time; Reflex; Respiration; Tail

1973
Multiple opiate receptors for multiple opioid peptides.
    Medical biology, 1982, Volume: 60, Issue:1

    Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission

1982

Other Studies

69 other study(ies) available for phenazocine and naloxone

ArticleYear
The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists.
    Proceedings of the National Academy of Sciences of the United States of America, 1976, Volume: 73, Issue:11

    Topics: Allosteric Regulation; Dextropropoxyphene; Fentanyl; Methadone; Models, Biological; Models, Molecular; Molecular Conformation; Morphine; Nalorphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Protein Conformation; Receptors, Opioid; Structure-Activity Relationship

1976
[Evaluation of the discriminative stimulus effect of an enkephalin analog, EK-399, in the rat].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 97, Issue:6

    Topics: Animals; Discrimination, Psychological; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1991
Effect of selective sigma ligands on duodenal alkaline secretion in the rat.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: Animals; Atropine; Bicarbonates; Dose-Response Relationship, Drug; Duodenum; Guanidines; Haloperidol; Injections, Intravenous; Intestinal Mucosa; Intestinal Secretions; Male; Naloxone; Phenazocine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Yohimbine

1990
Effects of morphine, ethylketocyclazocine, N-allylnormetazocine and naloxone on locomotor activity in the rabbit.
    Psychopharmacology, 1990, Volume: 101, Issue:2

    Topics: Animals; Cyclazocine; Ethylketocyclazocine; Female; Male; Morphine; Motor Activity; Naloxone; Nictitating Membrane; Phenazocine; Rabbits

1990
Opioids induce postural asymmetry in spinal rat: the side of the flexed limb depends upon the type of opioid agonist.
    Brain research, 1989, Feb-20, Volume: 480, Issue:1-2

    Topics: Animals; Benzomorphans; Decerebrate State; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Functional Laterality; Male; Muscles; Naloxone; Narcotics; Phenazocine; Posture; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord; Time Factors

1989
A role played by sigma receptors in the conditioned suppression of motility in mice.
    Psychopharmacology, 1988, Volume: 94, Issue:4

    Topics: Animals; Conditioning, Psychological; Cyclazocine; Drug Tolerance; Male; Mice; Mice, Inbred Strains; Motor Activity; Naloxone; Phenazocine; Receptors, Opioid; Receptors, sigma; Synaptic Membranes

1988
Mu and delta, but not kappa, opioid agonists induce contractions of the canine small intestine in vivo.
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dogs; Duodenum; Dynorphins; Electric Stimulation; Enkephalin, Methionine; Female; Gastrointestinal Motility; Male; Morphine; Morphine Derivatives; Naloxone; Peptide Fragments; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Actions of opioids on primate spinothalamic tract neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:9

    Topics: Animals; Dynorphins; Enkephalin, Methionine; Macaca fascicularis; Morphine; Naloxone; Narcotics; Neurons; Phenazocine; Phencyclidine; Spinal Cord; Thalamus

1986
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:3

    Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid

1987
Sites of action of mu-, kappa- and sigma-opiate receptor agonists at the feline ileocecal sphincter.
    The American journal of physiology, 1988, Volume: 254, Issue:2 Pt 1

    Topics: Animals; Atropine; Cats; Dynorphins; Ganglionic Blockers; Ileocecal Valve; Morphine; Naloxone; Phenazocine; Receptors, Opioid; Tachyphylaxis; Tetrodotoxin; Vagotomy

1988
Body temperature effects of opioids in rats: intracerebroventricular administration.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:6

    Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains

1986
Identification of multiple opiate receptors through neuroendocrine responses. II. Antagonism of mu, kappa and sigma agonists by naloxone and WIN 44,441-3.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1

    Topics: Animals; Azocines; Corticosterone; Cyclazocine; Drug Interactions; Ethylketocyclazocine; Growth Hormone; Luteinizing Hormone; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Pituitary Hormones, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid

1985
Differentiating opioids by their pupillary effects in the rat.
    Life sciences, 1985, Apr-29, Volume: 36, Issue:17

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Methadone; Motor Activity; Naloxone; Narcotics; Nystagmus, Physiologic; Phenazocine; Pupil; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism

1985
Sigma opioid receptors; SKF-10,047 update.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: Animals; Electroencephalography; Female; Hallucinogens; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism

1985
Plasma corticosterone changes in response to central or peripheral administration of kappa and sigma opiate agonists.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:3

    Topics: Animals; Brain; Corticosterone; Cyclazocine; Ethylketocyclazocine; Humans; Hypothalamo-Hypophyseal System; Male; Morphine; Naloxone; Naltrexone; Opioid-Related Disorders; Phenazocine; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma

1985
Novel nonnarcotic analgesics with an improved therapeutic ratio. Structure-activity relationships of 8-(methylthio)- and 8-(acylthio)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:11

    Topics: Acylation; Analgesia; Animals; Brain; Chemical Phenomena; Chemistry; Methylation; Mice; Morphinans; Morphine; Naloxone; Oxygen; Phenazocine; Rabbits; Rats; Receptors, Opioid; Structure-Activity Relationship; Sulfur

1985
Multiple opiate receptors may be involved in suppressing gamma-aminobutyrate release in substantia nigra.
    Life sciences, 1985, Dec-16, Volume: 37, Issue:24

    Topics: Aminooxyacetic Acid; Animals; Benzomorphans; Dopamine; Enkephalin, Methionine; Female; gamma-Aminobutyric Acid; Male; Naloxone; Nialamide; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Secretory Rate; Substantia Nigra

1985
Evidence for multiple opiate receptor involvement in different phencyclidine-induced unconditioned behaviors in rats.
    Psychopharmacology, 1986, Volume: 88, Issue:1

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Eating; Habituation, Psychophysiologic; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereotyped Behavior

1986
Discriminative stimulus effects of the opioid antagonist diprenorphine in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Cyclazocine; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Generalization, Stimulus; Morphinans; Naloxone; Narcotic Antagonists; Phenazocine; Psychotropic Drugs; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Saimiri

1986
Characterization and autoradiographic visualization of (+)-[3H]SKF10,047 binding in rat and mouse brain: further evidence for phencyclidine/"sigma opiate" receptor commonality.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Autoradiography; Brain Chemistry; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Species Specificity; Tritium

1986
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays.
    Life sciences, 1986, Jun-16, Volume: 38, Issue:24

    Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma

1986
Agonistic and antagonistic effects of PCP-derivatives and sigma opioids in PCP behavioral and receptor assays.
    NIDA research monograph, 1986, Volume: 64

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclazocine; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereotyped Behavior; Structure-Activity Relationship; Tritium

1986
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
    Journal of pharmacobio-dynamics, 1986, Volume: 9, Issue:5

    Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid

1986
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
    Life sciences, 1987, Jun-01, Volume: 40, Issue:22

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism

1987
N-allylnormetazocine: hemodynamic actions and inhibition of leucine-enkephalin hemodynamic activity in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Blood Pressure; Dogs; Enkephalin, Leucine; Female; Heart Rate; Hemodynamics; Male; Naloxone; Phenazocine; Stereoisomerism

1988
Psychotomimetic sigma-ligands, dexoxadrol and phencyclidine block the same presynaptic potassium channel in rat brain.
    The Journal of physiology, 1988, Volume: 403

    Topics: Animals; Brain; Cyclazocine; Dioxolanes; Dioxoles; Dose-Response Relationship, Drug; Hallucinogens; In Vitro Techniques; Naloxone; Phenazocine; Phencyclidine; Piperidines; Potassium Channels; Rats; Synaptosomes

1988
[Effect of opioid peptides on the lymphatic drainage of the pancreas in the rat and dog].
    Biulleten' eksperimental'noi biologii i meditsiny, 1988, Volume: 105, Issue:3

    Topics: Animals; Dogs; Dose-Response Relationship, Drug; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Evans Blue; Female; Lymph; Male; Naloxone; Pancreas; Phenazocine; Rats; Rats, Inbred Strains

1988
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors

1987
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule

1987
Historical introduction and review of chemistry.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Analgesics; Chemistry; History, 20th Century; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Phenazocine

1985
Selected opioids and responding for intracranial reinforcement.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: Animals; Cyclazocine; Ethylketocyclazocine; Hypothalamic Area, Lateral; Naloxone; Phenazocine; Rats; Reinforcement, Psychology; Self Stimulation; Stereoisomerism

1985
Stereoselective behavioral effects of N-allylnormetazocine in pigeons and squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:2

    Topics: Animals; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Morphine; Naloxone; Phenazocine; Phencyclidine; Reinforcement Schedule; Saimiri; Stereoisomerism

1985
Behavioral effects of selected opiates and phencyclidine in the nondependent and cyclazocine-dependent rhesus monkey.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Food; Macaca mulatta; Male; Naloxone; Phenazocine; Phencyclidine; Stereoisomerism; Substance-Related Disorders

1985
Opiate receptor: demonstration in nervous tissue.
    Science (New York, N.Y.), 1973, Mar-09, Volume: 179, Issue:4077

    Topics: Analgesics; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Codeine; Colchicine; Dextromethorphan; Dextropropoxyphene; Guinea Pigs; Histamine; Intestinal Mucosa; Levallorphan; Methadone; Mice; Morphine; Nalorphine; Naloxone; Phenazocine; Phenobarbital; Rats; Receptors, Drug; Serotonin; Tritium

1973
An in vivo pharmacological analysis of benzomorphan binding sites in rats.
    NIDA research monograph, 1984, Volume: 49

    Topics: Animals; Benzomorphans; Bombesin; Brain; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Grooming; Humans; Male; Morphinans; Morphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism; Stereotyped Behavior

1984
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord.
    Brain research, 1982, Sep-09, Volume: 247, Issue:1

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord

1982
Effects of ketazocine, ethylketazocine and phenazocine on schedule-controlled behavior: antagonism by naloxone.
    Neuropharmacology, 1982, Volume: 21, Issue:9

    Topics: Analgesics, Opioid; Animals; Columbidae; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Naloxone; Phenazocine

1982
The effect of two different buffers on the high affinity 3H-ethylketocyclazocine and 3H-SKF10047 binding to guinea pig brain membranes.
    Acta pharmacologica et toxicologica, 1984, Volume: 54, Issue:3

    Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Ethylketocyclazocine; Guinea Pigs; HEPES; In Vitro Techniques; Morphine; Naloxone; Phenazocine; Piperazines; Receptors, Opioid; Tritium; Tromethamine

1984
In vivo evidence for benzomorphan-selective receptors in rats.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Analgesics, Opioid; Animals; Benzomorphans; Bombesin; Buprenorphine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Male; Morphinans; Morphine; Naloxone; Phenazocine; Pruritus; Rats; Rats, Inbred Strains; Receptors, Opioid

1984
Feeding systems in Chinese hamsters.
    The American journal of physiology, 1984, Volume: 247, Issue:3 Pt 2

    Topics: Animals; Brain; Calcitonin; Circadian Rhythm; Cricetinae; Cyclazocine; Diabetes Mellitus; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Feeding Behavior; Haloperidol; Mesocricetus; Naloxone; Peptide Fragments; Phenazocine; Sincalide; Starvation

1984
Actions of kappa, sigma and partial mu narcotic receptor agonists on rat brain acetylcholine turnover.
    Neuroscience letters, 1981, Apr-09, Volume: 23, Issue:1

    Topics: Acetylcholine; Animals; Brain; Buprenorphine; Male; Morphinans; Naloxone; Organ Specificity; Phenazocine; Rats; Receptors, Opioid

1981
Stereoisomers of N-allylnormetazocine: phencyclidine-like behavioral effects in squirrel monkeys and rats.
    Science (New York, N.Y.), 1982, Jan-08, Volume: 215, Issue:4529

    Topics: Animals; Behavior, Animal; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Saimiri; Stereoisomerism; Structure-Activity Relationship

1982
Interactions between narcotic agonists, partial agonists andd antagonists evaluated by punished an unpunished behavior in the rat.
    Psychopharmacology, 1982, Volume: 76, Issue:2

    Topics: Animals; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Phenazocine; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid

1982
The binding of kappa- and sigma-opiates in rat brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1982, Volume: 2, Issue:6

    Topics: Animals; Binding Sites; Brain; Culture Techniques; Cyclazocine; Dihydromorphine; Enkephalins; Ethylketocyclazocine; Ligands; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Tritium

1982
Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity.
    Brain research, 1982, Sep-23, Volume: 248, Issue:1

    Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Goldfish; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma

1982
The epileptogenic spectrum of opiate agonists.
    Neuropharmacology, 1982, Volume: 21, Issue:11

    Topics: Animals; Anticonvulsants; beta-Endorphin; Cyclazocine; Electroencephalography; Endorphins; Enkephalin, Leucine; Epilepsy; Ethylketocyclazocine; Injections, Intraventricular; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains

1982
Peptide and non-peptide opioid-induced hyperthermia in rabbits.
    Brain research, 1983, Apr-11, Volume: 265, Issue:1

    Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptides; Phenazocine; Rats

1983
Opiate-induced enhancement of the effects of naloxone on serum luteinizing hormone levels in the male rat: specificity for Mu agonists.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Animals; Binding, Competitive; Cyclazocine; Ethanol; Ethylketocyclazocine; Kinetics; Luteinizing Hormone; Male; Morphine; Naloxone; Pentobarbital; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
The binding to rat brain homogenates of Mr2034, a universal opiate.
    Life sciences, 1983, Sep-05, Volume: 33, Issue:10

    Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
Antinociceptive studies of the optical isomers of N-allylnormetazocine (SKF 10,047).
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Analgesics; Animals; Male; Mice; Mice, Inbred ICR; Morphine; Naloxone; Phenazocine; Receptors, Adrenergic, alpha; Receptors, Opioid; Stereoisomerism; Yohimbine

1983
Naltrexone fails to antagonize the sigma effects of PCP and SKF 10,047 in the dog.
    European journal of pharmacology, 1983, Sep-02, Volume: 92, Issue:3-4

    Topics: Animals; Body Temperature; Dogs; Female; Heart Rate; Morphine; Naloxone; Naltrexone; Paraplegia; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Reflex

1983
An analysis of nicotinic and opioid processes in the medulla oblongata and nucleus ambiguus of the dog.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:2

    Topics: Animals; Blood Pressure; Cyclazocine; Decerebrate State; Dogs; Electric Stimulation; Endorphins; Ethylketocyclazocine; Female; Fentanyl; Heart Rate; Male; Mecamylamine; Medulla Oblongata; Naloxone; Nicotine; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma

1983
Naloxone-inaccessible sigma receptor in rat central nervous system.
    Proceedings of the National Academy of Sciences of the United States of America, 1983, Volume: 80, Issue:21

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalins; Ethylketocyclazocine; Kinetics; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Spinal Cord; Tissue Distribution

1983
N-allylnormetazocine (SKF-10,047): the induction of feeding by a putative sigma agonist.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:5

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Interactions; Eating; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
Blockade of long-term potentiation by phencyclidine and sigma opiates in the hippocampus in vivo and in vitro.
    Brain research, 1983, Nov-28, Volume: 280, Issue:1

    Topics: Animals; Cyclazocine; Drug Synergism; Hippocampus; Male; Membrane Potentials; Morphine; Naloxone; Narcotics; Phenazocine; Phencyclidine; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synapses; Synaptic Transmission

1983
Discriminative stimulus properties of nalorphine in the rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:3

    Topics: Animals; Benzodiazepines; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Macaca mulatta; Male; Nalorphine; Naloxone; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa

1983
Multiple opioid receptor profile in vitro and activity in vivo of the potent opioid antagonist Win 44,441-3.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Animals; Azocines; Guinea Pigs; Ileum; Male; Mice; Morphine; Muscle Contraction; Naloxone; Narcotic Antagonists; Phenazocine; Receptors, Opioid; Vas Deferens

1983
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
    Life sciences, 1984, Feb-20, Volume: 34, Issue:8

    Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains

1984
Behavioral interactions of opioid agonists and antagonists with serotonergic systems.
    NIDA research monograph, 1984, Volume: 49

    Topics: Animals; Brain; Conditioning, Operant; Cyclazocine; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Lysergic Acid Diethylamide; Male; Metergoline; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement Schedule

1984
Agonist and antagonist effects of prototype opiate drugs in rats discriminating fentanyl from saline: characteristics of partial generalization.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Male; Morphine; Nalorphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Sodium Chloride

1984
Pharmacological evaluation of N-allynormetazocine (SKF 10,047) on the basis of its discriminative stimulus properties in the rat.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:1

    Topics: Animals; Benzomorphans; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Male; Naloxone; Phenazocine; Phencyclidine; Propranolol; Rats; Rats, Inbred F344; Stereoisomerism

1983
Subclasses of opioids based on body temperature change in rats: acute subcutaneous administration.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:2

    Topics: Animals; Body Temperature; Buprenorphine; Dose-Response Relationship, Drug; Endorphins; Injections, Subcutaneous; Male; Meperidine; Morphine; Nalbuphine; Naloxone; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains

1983
Phencyclidine-like discriminative stimuli of (+)- and (-)-N-allylnormetazocine in rats.
    European journal of pharmacology, 1982, Oct-22, Volume: 84, Issue:3-4

    Topics: Animals; Discrimination Learning; Discrimination, Psychological; Male; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Reinforcement Schedule; Stereoisomerism

1982
Regulation of [3H]dopamine release from rat striatal slices by sigma receptor ligands.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:1

    Topics: Animals; Atropine; Corpus Striatum; Dopamine; Flavonoids; In Vitro Techniques; N-Methylaspartate; Naloxone; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma

1994
Enhancement of the opiate withdrawal response by antipsychotic drugs in guinea-pigs is not mediated by sigma binding sites.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1993, Volume: 3, Issue:1

    Topics: Analysis of Variance; Animals; Antipsychotic Agents; Atropine; Behavior, Animal; Clozapine; Dizocilpine Maleate; Female; Guinea Pigs; Ketamine; Kinetics; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Raclopride; Radioligand Assay; Receptors, sigma; Remoxipride; Salicylamides; Substance Withdrawal Syndrome

1993
Naloxone-sensitive, haloperidol-sensitive, [3H](+)SKF-10047-binding protein partially purified from rat liver and rat brain membranes: an opioid/sigma receptor?
    Synapse (New York, N.Y.), 1997, Volume: 25, Issue:2

    Topics: Animals; Antipsychotic Agents; Brain; Haloperidol; Liver; Naloxone; Phenazocine; Radioligand Assay; Rats; Receptors, Opioid

1997
Synthesis, conformational analysis and antinociceptive activity of 1-[N-methyl-(2-phenylethyl)amino]methyl-1,2,3,4-tetrahydroisoquinoline derivatives.
    Arzneimittel-Forschung, 1999, Volume: 49, Issue:12

    Topics: Analgesics; Analgesics, Opioid; Animals; Isoquinolines; Male; Mice; Molecular Conformation; Naloxone; Narcotic Antagonists; Phenazocine; Reaction Time; Stereoisomerism

1999
The C-terminal amidated analogue of the substance P (SP) fragment SP(1-7) attenuates the expression of naloxone-precipitated withdrawal in morphine dependent rats.
    Peptides, 2009, Volume: 30, Issue:12

    Topics: Animals; Antipsychotic Agents; Brain; Male; Morphine Dependence; Naloxone; Peptide Fragments; Phenazocine; Rats; Rats, Wistar; Substance P; Substance Withdrawal Syndrome

2009
Straub tail reaction in mice treated with σ(1) receptor antagonist in combination with methamphetamine.
    Brain research, 2012, Oct-30, Volume: 1482

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Antipsychotic Agents; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Male; Methamphetamine; Mice; Mice, Inbred Strains; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Pyrimidines; Receptors, Opioid, delta; Reflex; Tail; Time Factors

2012