phenazocine has been researched along with morphine in 96 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 86 (89.58) | 18.7374 |
1990's | 8 (8.33) | 18.2507 |
2000's | 1 (1.04) | 29.6817 |
2010's | 1 (1.04) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Creveling, CR; Jacobson, AE; Klee, WA; Rice, KC; Shiotani, S | 1 |
Burke, TR; Konicki, PE; Pert, CB; Quirion, R; Rice, KC | 1 |
Metcalf, G; Rees, JM; Ward, SJ | 1 |
Creese, I; Feinberg, AP; Snyder, SH | 1 |
Eades, CG; Gilbert, PE; Huppler, RE; Martin, WR; Thompson, JA | 1 |
Bridges, RS; Kinsley, CH; Mann, PE | 1 |
Chiba, S; Nishida, N; Yasuhara, Y | 1 |
Dykstra, LA; Picker, MJ; Powell, K | 1 |
Bolen, JB; Burke, TR; Chapekar, M; Gang, Y; Glazer, RI; Li, ZH; Marquez, VE; Rice, KC | 1 |
Cone, EJ; Johnson, RE; Su, TP; Vaupel, DB | 1 |
Goldberg, SR; Schindler, CW; White, MF | 1 |
Bronson, ME; Moerschbaecher, JM | 1 |
Carino, MA; Horita, A; Yamawaki, S | 1 |
Holtzman, SG | 1 |
Cowan, A; Jacoby, HI; Vaught, JL | 1 |
Cooper, SJ; Jackson, A; Kirkham, TC | 1 |
Chung, JM; Kim, J; Shin, HK; Willcockson, WS; Willis, WD | 1 |
Cohen, S; Ouyang, A; Vos, P | 1 |
Adler, MW; Geller, EB; Rowan, CH | 1 |
George, R; Pechnick, R; Poland, RE | 2 |
Burks, TF; Hirning, LD; Porreca, F | 1 |
Calligaro, D; el-Fakahany, EE; Hong, O; Khazan, N; Young, GA | 1 |
Eisenberg, RM | 1 |
Baba, Y; Ban, M; Fujimura, H; Hori, M; Imai, E; Iwata, N; Morita, T; Niwa, M; Nozaki, M; Suzuki, Y | 1 |
Greenberg, BD; Segal, DS | 1 |
Hiramatsu, M; Kameyama, T; Nabeshima, T | 2 |
Dykstra, LA; Slifer, BL | 1 |
Harris, LS | 1 |
Dykstra, LA; Picker, M | 1 |
Gormezano, I; Harvey, JA; Lamb, MR; Schindler, CW | 1 |
Dykstra, LA; Heise, JW; Picker, M | 1 |
Risner, ME; Shannon, HE; Vaupel, DB | 1 |
Clark, RD; Katz, JL; Spealman, RD | 1 |
Pierson, AK | 1 |
Röthig, J | 1 |
Dole, VP | 1 |
Aceto, MD; McKean, DB; Pearl, J | 1 |
Bowman, WC; Buwembo, JB | 1 |
Pert, CB; Snyder, SH | 1 |
Pittman, KA; Williams, TA | 1 |
Armstrong Davison, MH | 1 |
Hopton, D | 1 |
Fennessy, MR; Heimans, RL; Rand, MJ | 1 |
Dundee, JW; Loan, WB; Morrison, JD | 1 |
McKean, DB; Pearl, J; Stander, H | 1 |
Rogers, KJ; Thornton, JA | 1 |
DeGraff, AC; Fisch, S; Hotz, MM; Kopeloff, A; Lustgarten, BP | 1 |
Chernov, HI; Grumbach, L | 1 |
Gyand, EA; Kosterlitz, HW | 1 |
Hopton, DS; Torrance, HB | 1 |
Clarke, RS; Dundee, JW; Hamilton, RC; Loan, WB; Morrison, JD | 1 |
Hein, GE; Powell, K | 1 |
Casy, AF; Kupchan, SM | 1 |
Contreras, E; Quijada, L; Tamayo, L | 1 |
Cowan, A; Gmerek, DE | 2 |
Calligaro, D; El-Fakany, EE; Hong, O; Khazan, N; Young, GA | 1 |
Khazan, N; Young, GA | 1 |
Miller, RJ | 1 |
Enger, M; Grynne, BH; Holmen, AT; Maurset, AR | 1 |
Holtzman, SG; Teal, JJ | 1 |
Harris, RA; Snell, D | 1 |
Shannon, HE; Su, TP | 1 |
Kandasamy, SB; Williams, BA | 1 |
Cicero, TJ; Meyer, ER; Owens, DP; Schmoeker, PF | 1 |
Aceto, MD; May, EL | 1 |
Vaupel, DB | 1 |
Gosnell, BA; Levine, AS; Morley, JE | 1 |
Greenfield, LJ; Guyenet, PG; Hackett, JT; Stringer, JL | 1 |
Michne, WF; Pierson, AK; Ward, SJ | 1 |
Bajorek, JG; Lee, RJ; Lomax, P | 1 |
Holtzman, SG; White, JM | 1 |
Cowan, A; Porreca, F; Raffa, RB; Tallarida, RJ | 1 |
Johnson, KM; Leventer, SM | 1 |
Mastropaolo, J; Moerschbaecher, JM; Thompson, DM; Winsauer, PJ | 1 |
Colpaert, FC; Janssen, PA | 1 |
Iwamoto, ET | 1 |
Herling, S; Woods, JH | 1 |
Adler, MW; Geller, EB; Hawk, C; Keinath, SH; Tallarida, RJ | 1 |
Carter, FE; Chau, TT; Harris, LS | 1 |
Moerschbaecher, JM; Thompson, DM | 1 |
Franklin, SR; Tang, AH | 1 |
Brent, PJ; Chahl, LA | 1 |
Brusa, L; D'Amore, A; Lorenzini, P; Massotti, M | 1 |
David Clark, J; Demirci, H; Gharagozlou, P; Lameh, J | 1 |
LATSHAW, WE; MACDONNELL, DR | 1 |
FELLOWS, EJ; TEDESCHI, DH; TEDESCHI, RE | 1 |
DAW, RH; MURRAY, A; SWERDLOW, M | 1 |
WANG, RI | 1 |
HARRIS, LS; PIERSON, AK | 1 |
LASAGNA, L | 1 |
SHEMANO, I; WENDEL, H | 1 |
DAW, RH; STARMER, G; SWERDLOW, M | 1 |
Hall, FS; Kitanaka, J; Kitanaka, N; Nishiyama, N; Takemura, M; Tanaka, K; Uhl, GR | 1 |
7 review(s) available for phenazocine and morphine
Article | Year |
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Drug discrimination studies.
Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response | 1985 |
Assays for narcotic antagonist activity in rodents.
Topics: Analgesics; Animals; Depression, Chemical; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Heroin; Hot Temperature; Lens, Crystalline; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Nalorphine; Naloxone; Narcotic Antagonists; Oxymorphone; Phenazocine; Pressure; Rabbits; Rats; Reaction Time; Reflex; Respiration; Tail | 1973 |
[Analgesics. 32].
Topics: Alphaprodine; Analgesics; Azepines; Benzimidazoles; Bridged-Ring Compounds; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Fentanyl; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Levallorphan; Levorphanol; Lysergic Acid Diethylamide; Methadone; Morphinans; Morphine; Nalorphine; Naphthoquinones; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine | 1969 |
Biochemistry of addiction.
Topics: Animals; Azepines; Brain; Drug Tolerance; Humans; Methadone; Morphinans; Morphine; Opium; Phenazocine; Piperidines; Receptors, Drug; Substance-Related Disorders; Synapses; Synaptic Transmission | 1970 |
Multiple opiate receptors for multiple opioid peptides.
Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission | 1982 |
THE CLINICAL EVALUATION OF MORPHINE AND ITS SUBSTITUTES AS ANALGESICS.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Biomedical Research; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Meperidine; Methadone; Methotrimeprazine; Morphine; Nalorphine; Narcotic Antagonists; Oxymorphone; Pentazocine; Phenazocine; Substance-Related Disorders; Toxicology | 1964 |
3 trial(s) available for phenazocine and morphine
Article | Year |
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Nathan B. Eddy Memorial Award lecture.
Topics: Analgesics; Animals; Clinical Trials as Topic; Humans; Meperidine; Morphine; Narcotic Antagonists; Phenazocine; Structure-Activity Relationship | 1986 |
Double-blind clinical trial of the analgesic effects of phenazocine hydrobromide (Narphen) compared with morphine sulphate in patients with acute abdominal pain.
Topics: Abdomen; Acute Disease; Adult; Aged; Ampulla of Vater; Biliary Tract Diseases; Clinical Trials as Topic; Female; Humans; Injections, Intramuscular; Male; Middle Aged; Morphine; Pain; Pancreatic Neoplasms; Pancreatitis; Phenazocine | 1971 |
Studies of drugs given before anaesthesia. 13. Pentazocine and other opiate antagonists.
Topics: Adult; Central Nervous System; Drug Antagonism; Female; Humans; Levallorphan; Meperidine; Morphine; Nalorphine; Pentazocine; Phenazocine; Preanesthetic Medication; Psychoses, Substance-Induced | 1967 |
86 other study(ies) available for phenazocine and morphine
Article | Year |
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N-(2,4,5-Trihydroxyphenehtyl)normetazocine, a potential irreversible inhibitor of the narcotic receptor.
Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Benzomorphans; Brain; Cyclazocine; Depression, Chemical; In Vitro Techniques; Male; Mice; Morphinans; Neoplasms, Experimental; Neuroblastoma; Norepinephrine; Protein Binding; Rats; Receptors, Opioid | 1977 |
Synthesis and pharmacological characterization of (+/-)-5,9 alpha-dimethyl-2-[2-(4-fluorophenyl)ethyl]-2'-hydroxy-6,7-benzomorphan (fluorophen), a ligand suitable for visualization of opiate receptors in vivo.
Topics: Animals; Benzomorphans; Biological Assay; Brain; Guinea Pigs; Ileum; Indicators and Reagents; Male; Morphinans; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
The comparative pharmacology of morphine, ketocyclazocine and 2'-hydroxy-5,9-dimethyl-2-allyl-6,7-benzomorphan in rodents [proceedings].
Topics: Animals; Behavior, Animal; Body Temperature; Cyclazocine; Mice; Morphine; Phenazocine; Rats; Respiration | 1977 |
The opiate receptor: a model explaining structure-activity relationships of opiate agonists and antagonists.
Topics: Allosteric Regulation; Dextropropoxyphene; Fentanyl; Methadone; Models, Biological; Models, Molecular; Molecular Conformation; Morphine; Nalorphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Protein Conformation; Receptors, Opioid; Structure-Activity Relationship | 1976 |
The effects of morphine- and nalorphine- like drugs in the nondependent and morphine-dependent chronic spinal dog.
Topics: Animals; Apomorphine; Cyclazocine; Cyclopropanes; Dextropropoxyphene; Dogs; Ethylketocyclazocine; Humans; Morphinans; Morphine; Morphine Dependence; Nalorphine; Naltrexone; Phenazocine; Spinal Cord | 1976 |
Opioid receptor subtype involvement in maternal behavior in lactating rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; beta-Endorphin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Lactation; Maternal Behavior; Morphine; Phenazocine; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu | 1991 |
[Evaluation of the discriminative stimulus effect of an enkephalin analog, EK-399, in the rat].
Topics: Animals; Discrimination, Psychological; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1991 |
Stereospecificity of mixed-action opioid agonist/antagonists in morphine-tolerant squirrel monkeys.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Morphine; Narcotic Antagonists; Narcotics; Pentazocine; Phenazocine; Saimiri; Stereoisomerism | 1990 |
Examination of the possible mediation of antineoplastic effects of opiates through the inhibition of tyrosine-specific protein kinases.
Topics: Antineoplastic Agents; Cell Line; ErbB Receptors; Humans; Hydroquinones; Morphine; Narcotics; Phenazocine; Phosphorylation; Protein-Tyrosine Kinases; Structure-Activity Relationship | 1991 |
Kappa opioid partial agonist activity of the enkephalin-like pentapeptide BW942C based on urination and in vitro studies in humans and animals.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adult; Amino Acid Sequence; Animals; Diuresis; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Methionine; Enkephalins; Humans; In Vitro Techniques; Male; Molecular Sequence Data; Morphine; Naltrexone; Oligopeptides; Phenazocine; Pyrrolidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Urination; Vas Deferens | 1990 |
Effects of morphine, ethylketocyclazocine, N-allylnormetazocine and naloxone on locomotor activity in the rabbit.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Female; Male; Morphine; Motor Activity; Naloxone; Nictitating Membrane; Phenazocine; Rabbits | 1990 |
Effects of mu, kappa and sigma opioids on fixed consecutive number responding in rats.
Topics: Animals; Buprenorphine; Conditioning, Operant; Cyclazocine; Dextroamphetamine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Phenazocine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1987 |
Analeptic effect of opiate receptor agonists in rabbits.
Topics: Animals; Arousal; Brain; Central Nervous System Stimulants; Codeine; Cyclazocine; Dose-Response Relationship, Drug; Enkephalin, Methionine; Ethylketocyclazocine; Etorphine; Male; Meperidine; Methadone; Morphine; Naltrexone; Narcotics; Phenazocine; Rabbits; Receptors, Opioid; Reflex | 1985 |
Mu and delta, but not kappa, opioid agonists induce contractions of the canine small intestine in vivo.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dogs; Duodenum; Dynorphins; Electric Stimulation; Enkephalin, Methionine; Female; Gastrointestinal Motility; Male; Morphine; Morphine Derivatives; Naloxone; Peptide Fragments; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Actions of opioids on primate spinothalamic tract neurons.
Topics: Animals; Dynorphins; Enkephalin, Methionine; Macaca fascicularis; Morphine; Naloxone; Narcotics; Neurons; Phenazocine; Phencyclidine; Spinal Cord; Thalamus | 1986 |
Sites of action of mu-, kappa- and sigma-opiate receptor agonists at the feline ileocecal sphincter.
Topics: Animals; Atropine; Cats; Dynorphins; Ganglionic Blockers; Ileocecal Valve; Morphine; Naloxone; Phenazocine; Receptors, Opioid; Tachyphylaxis; Tetrodotoxin; Vagotomy | 1988 |
Body temperature effects of opioids in rats: intracerebroventricular administration.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1986 |
Identification of multiple opiate receptors through neuroendocrine responses. I. Effects of agonists.
Topics: Animals; Corticosterone; Cyclazocine; Ethylketocyclazocine; Growth Hormone; Injections, Subcutaneous; Luteinizing Hormone; Male; Morphine; Phenazocine; Pituitary Hormones, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid | 1985 |
Identification of multiple opiate receptors through neuroendocrine responses. II. Antagonism of mu, kappa and sigma agonists by naloxone and WIN 44,441-3.
Topics: Animals; Azocines; Corticosterone; Cyclazocine; Drug Interactions; Ethylketocyclazocine; Growth Hormone; Luteinizing Hormone; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Pituitary Hormones, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid | 1985 |
Mu, but not kappa, opioid agonists induce contractions of the canine small intestine ex vivo.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Cyclazocine; Dimethylphenylpiperazinium Iodide; Dogs; Ethylketocyclazocine; Gastrointestinal Motility; In Vitro Techniques; Intestine, Small; Morphine; Nalorphine; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Sigma opioid receptors; SKF-10,047 update.
Topics: Animals; Electroencephalography; Female; Hallucinogens; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1985 |
Plasma corticosterone changes in response to central or peripheral administration of kappa and sigma opiate agonists.
Topics: Animals; Brain; Corticosterone; Cyclazocine; Ethylketocyclazocine; Humans; Hypothalamo-Hypophyseal System; Male; Morphine; Naloxone; Naltrexone; Opioid-Related Disorders; Phenazocine; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1985 |
Novel nonnarcotic analgesics with an improved therapeutic ratio. Structure-activity relationships of 8-(methylthio)- and 8-(acylthio)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines.
Topics: Acylation; Analgesia; Animals; Brain; Chemical Phenomena; Chemistry; Methylation; Mice; Morphinans; Morphine; Naloxone; Oxygen; Phenazocine; Rabbits; Rats; Receptors, Opioid; Structure-Activity Relationship; Sulfur | 1985 |
Evidence for multiple opiate receptor involvement in different phencyclidine-induced unconditioned behaviors in rats.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Eating; Habituation, Psychophysiologic; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereotyped Behavior | 1986 |
Phencyclidine-induced stereotyped behaviors after injection of morphine and N-allylnormetazocine (SKF 10,047) in rats.
Topics: Animals; Male; Morphine; Motor Activity; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereotyped Behavior | 1986 |
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid | 1986 |
The effects of N-allylnormetazocine on electric shock titration in squirrel monkeys.
Topics: Animals; Avoidance Learning; Electroshock; Male; Morphine; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma; Reinforcement Schedule; Saimiri; Stereoisomerism | 1987 |
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors | 1987 |
Effects of morphine, ethylketocyclazocine, and N-allylnormetazocine on classical conditioning of the rabbit nictitating membrane response.
Topics: Animals; Conditioning, Classical; Conditioning, Eyelid; Cyclazocine; Ethylketocyclazocine; Female; Light; Male; Morphine; Nictitating Membrane; Phenazocine; Rabbits; Sound | 1986 |
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule | 1987 |
Pharmacologic and reinforcing properties of phencyclidine and the enantiomers of N-allylnormetazocine in the dog.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Decerebrate State; Dogs; Female; Morphine; Naltrexone; Phenazocine; Phencyclidine; Reinforcement Schedule; Self Administration; Stereoisomerism | 1986 |
Stereoselective behavioral effects of N-allylnormetazocine in pigeons and squirrel monkeys.
Topics: Animals; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Morphine; Naloxone; Phenazocine; Phencyclidine; Reinforcement Schedule; Saimiri; Stereoisomerism | 1985 |
Effects of opiates and opiate antagonists on the Straub tail reaction in mice.
Topics: Analgesics; Animals; Atropine; Bridged-Ring Compounds; Codeine; Cyclazocine; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Narcotic Antagonists; Pentazocine; Phenazocine; Stereoisomerism; Tail | 1969 |
Effects of narcotic analgesics on contractions of the chick isolated, innervated oesophagus.
Topics: Acetylcholine; Analgesics; Animals; Chickens; Cyclazocine; Dextropropoxyphene; Electric Stimulation; Esophagus; Heroin; In Vitro Techniques; Meperidine; Methadone; Morphinans; Morphine; Muscle Contraction; Nalorphine; Pentazocine; Phenazocine; Serotonin; Tachyphylaxis; Time Factors | 1972 |
Opiate receptor: demonstration in nervous tissue.
Topics: Analgesics; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Codeine; Colchicine; Dextromethorphan; Dextropropoxyphene; Guinea Pigs; Histamine; Intestinal Mucosa; Levallorphan; Methadone; Mice; Morphine; Nalorphine; Naloxone; Phenazocine; Phenobarbital; Rats; Receptors, Drug; Serotonin; Tritium | 1973 |
Pentazocine radioimmunoassay.
Topics: Ammonium Sulfate; Animals; Antibody Specificity; Antigen-Antibody Reactions; Azo Compounds; Carboxylic Acids; Chromatography, Gas; Cross Reactions; Cyclazocine; Levallorphan; Levorphanol; Methods; Molecular Weight; Morphine; Nalorphine; Oxidation-Reduction; Pentazocine; Phenazocine; Rabbits; Radioimmunoassay; Tritium; Urine | 1974 |
Heavy sedation in ophthalmic surgery.
Topics: Cataract Extraction; Corneal Transplantation; Eye Diseases; Glaucoma; Humans; Hypnotics and Sedatives; Injections, Intramuscular; Injections, Intravenous; Morphine; Phenazocine; Promazine; Promethazine; Retinal Detachment; Transplantation, Homologous | 1967 |
Comparison of effect of morphine-like analgesics on transmurally stimulated guinea-pig ileum.
Topics: Analgesics; Animals; Codeine; Cyclic N-Oxides; Drug Tolerance; Electric Stimulation; Female; Fentanyl; Guinea Pigs; Heroin; Humans; Ileum; In Vitro Techniques; Male; Meperidine; Morphinans; Morphine; Muscle Contraction; Muscle, Smooth; Nalorphine; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine; Rats; Substance-Related Disorders; Urinary Bladder | 1969 |
Studies of drugs given before anaesthesia. XIX. The opiates.
Topics: Analgesics; Diazepam; Female; Fentanyl; Heroin; Humans; Levorphanol; Male; Meperidine; Methadone; Morphine; Papaverine; Phenazocine; Preanesthetic Medication; Vomiting | 1970 |
Effects of analgesics and other drugs on mice in phenylquinone and rotarod tests.
Topics: Analgesics; Animals; Chemical Phenomena; Chemistry; Chlorpromazine; Cyclazocine; Dextroamphetamine; Levallorphan; Male; Mice; Morphine; Motor Activity; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Pilocarpine; Quinones; Salivation | 1969 |
The interaction between monoamine oxidase inhibitors and narcotic analgesics in mice.
Topics: Analgesics; Animals; Drug Synergism; Iproniazid; Meperidine; Mice; Monoamine Oxidase Inhibitors; Morphine; Pentazocine; Phenazocine; Tranylcypromine | 1969 |
The effects of phenazocine hydrobromide on water and mercurial diuresis in man.
Topics: Diuresis; Heart Failure; Humans; Infusions, Parenteral; Kidney Function Tests; Morphine; Organomercury Compounds; Phenazocine; Water-Electrolyte Balance | 1965 |
The analgesic effect of opiate-opiate antagonist combinations in the rat.
Topics: Analgesics; Animals; Levallorphan; Meperidine; Methadone; Morphine; Nalorphine; Narcotic Antagonists; Phenazocine; Rats; Sensory Receptor Cells | 1965 |
Agonist and antagonist actions of morphine-like drugs on the guinea-pig isolated ileum.
Topics: Analgesics; Animals; Cyclazocine; Drug Synergism; Guinea Pigs; Ileum; Levallorphan; Levorphanol; Morphine; Muscle, Smooth; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Reflex | 1966 |
Action of various new analgesic drugs on the human common bile duct.
Topics: Analgesics; Common Bile Duct; Dextromoramide; Dextropropoxyphene; Humans; Injections, Intramuscular; Levorphanol; Meperidine; Morphine; Pain; Phenazocine; Phenoperidine | 1967 |
Evaluation of kinetic constants for mixed inhibitors of cholinesterase.
Topics: Animals; Bridged-Ring Compounds; Cattle; Cholinesterase Inhibitors; Cholinesterases; Edrophonium; Hallucinogens; Kinetics; Levallorphan; Lysergic Acid Diethylamide; Mathematics; Morphine; Nalorphine; Neostigmine; Phenazocine; Phenethylamines; Phenols; Physostigmine; Quaternary Ammonium Compounds | 1967 |
Drug latentiation. II. Labile ether derivatives of phenolic analgesics.
Topics: Analgesics; Animals; Chemistry, Pharmaceutical; Ethers; Mice; Morphine; Phenazocine; Phenols | 1967 |
Antagonistic action of tolazoline upon the analgesic effect of some morphine analogues.
Topics: Analgesia; Animals; Drug Antagonism; Meperidine; Methadone; Morphine; Phenazocine; Rats; Tolazoline | 1967 |
An in vivo pharmacological analysis of benzomorphan binding sites in rats.
Topics: Animals; Benzomorphans; Bombesin; Brain; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Grooming; Humans; Male; Morphinans; Morphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism; Stereotyped Behavior | 1984 |
Sigma receptors mediated the psychotomimetic effects of N-allylnormetazocine (SKF-10,047), but not its opioid agonistic-antagonistic properties.
Topics: Animals; Binding, Competitive; Brain; Dihydromorphine; Electroencephalography; Female; Hallucinogens; Humans; Morphine; Morphine Dependence; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1984 |
Differential neuropharmacological effects of mu, kappa and sigma opioid agonists on cortical EEG power spectra in the rat. Stereospecificity and naloxone antagonism.
Topics: Animals; Cerebral Cortex; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Methadone; Molecular Conformation; Morphine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1984 |
The effect of two different buffers on the high affinity 3H-ethylketocyclazocine and 3H-SKF10047 binding to guinea pig brain membranes.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Ethylketocyclazocine; Guinea Pigs; HEPES; In Vitro Techniques; Morphine; Naloxone; Phenazocine; Piperazines; Receptors, Opioid; Tritium; Tromethamine | 1984 |
In vivo evidence for benzomorphan-selective receptors in rats.
Topics: Analgesics, Opioid; Animals; Benzomorphans; Bombesin; Buprenorphine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Male; Morphinans; Morphine; Naloxone; Phenazocine; Pruritus; Rats; Rats, Inbred Strains; Receptors, Opioid | 1984 |
Discriminative stimulus effects of prototype opiate receptor agonists in monkeys.
Topics: Animals; Apomorphine; Cyclazocine; Ethylketocyclazocine; Female; Generalization, Stimulus; Haloperidol; Male; Models, Biological; Morphine; Naltrexone; Phenazocine; Prejudice; Receptors, Opioid; Saimiri | 1980 |
Interactions between narcotic agonists, partial agonists andd antagonists evaluated by punished an unpunished behavior in the rat.
Topics: Animals; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Phenazocine; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid | 1982 |
Effects of the combination of tripelennamine and pentazocine at the behavioral and molecular levels.
Topics: Animals; Brain; Diphenhydramine; Discrimination, Psychological; Drug Synergism; Guinea Pigs; Ileum; Learning; Male; Morphine; Pentazocine; Phenazocine; Rats; Receptors, Opioid; Synaptic Membranes; Tripelennamine | 1982 |
Peptide and non-peptide opioid-induced hyperthermia in rabbits.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptides; Phenazocine; Rats | 1983 |
Opiate-induced enhancement of the effects of naloxone on serum luteinizing hormone levels in the male rat: specificity for Mu agonists.
Topics: Animals; Binding, Competitive; Cyclazocine; Ethanol; Ethylketocyclazocine; Kinetics; Luteinizing Hormone; Male; Morphine; Naloxone; Pentobarbital; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
Antinociceptive studies of the optical isomers of N-allylnormetazocine (SKF 10,047).
Topics: Analgesics; Animals; Male; Mice; Mice, Inbred ICR; Morphine; Naloxone; Phenazocine; Receptors, Adrenergic, alpha; Receptors, Opioid; Stereoisomerism; Yohimbine | 1983 |
Naltrexone fails to antagonize the sigma effects of PCP and SKF 10,047 in the dog.
Topics: Animals; Body Temperature; Dogs; Female; Heart Rate; Morphine; Naloxone; Naltrexone; Paraplegia; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Reflex | 1983 |
N-allylnormetazocine (SKF-10,047): the induction of feeding by a putative sigma agonist.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Interactions; Eating; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
Blockade of long-term potentiation by phencyclidine and sigma opiates in the hippocampus in vivo and in vitro.
Topics: Animals; Cyclazocine; Drug Synergism; Hippocampus; Male; Membrane Potentials; Morphine; Naloxone; Narcotics; Phenazocine; Phencyclidine; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synapses; Synaptic Transmission | 1983 |
Multiple opioid receptor profile in vitro and activity in vivo of the potent opioid antagonist Win 44,441-3.
Topics: Animals; Azocines; Guinea Pigs; Ileum; Male; Mice; Morphine; Muscle Contraction; Naloxone; Narcotic Antagonists; Phenazocine; Receptors, Opioid; Vas Deferens | 1983 |
Similar anticonvulsant, but unique, behavioural effects of opioid agonists in the seizure-sensitive Mongolian gerbil.
Topics: Animals; Anticonvulsants; Behavior, Animal; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Gerbillinae; Male; Morphine; Narcotics; Phenazocine; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures | 1984 |
Further characterization of the three-choice morphine, cyclazocine and saline discrimination paradigm: opioids with agonist and antagonist properties.
Topics: Animals; Cyclazocine; Discrimination Learning; Discrimination, Psychological; Ethylketocyclazocine; Male; Morphine; Narcotic Antagonists; Narcotics; Phenazocine; Phencyclidine; Rats; Sodium Chloride; Stereoisomerism | 1983 |
Ketazocines and morphine: effects on gastrointestinal transit after central and peripheral administration.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Gastrointestinal Motility; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Phenazocine; Rats; Rats, Inbred Strains | 1983 |
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains | 1984 |
Effects of opioids on accuracy of a fixed-ratio discrimination in monkeys and rats.
Topics: Animals; Buprenorphine; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Isomerism; Macaca mulatta; Male; Methadone; Morphinans; Morphine; Phenazocine; Rats | 1984 |
Agonist and antagonist effects of prototype opiate drugs in rats discriminating fentanyl from saline: characteristics of partial generalization.
Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Male; Morphine; Nalorphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Sodium Chloride | 1984 |
Pharmacologic effects of N-allylnormetazocine (SKF-10047).
Topics: Analgesics; Animals; Behavior, Animal; Clonidine; Cyclazocine; Ethylketocyclazocine; Male; Morphine; Motor Activity; Phenazocine; Rats; Receptors, Dopamine; Spiperone | 1981 |
Discriminative stimulus effects of etorphine in Rhesus monkeys.
Topics: Animals; Codeine; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Etorphine; Macaca mulatta; Male; Meperidine; Morphinans; Morphine; Pentazocine; Phenazocine; Sodium Chloride | 1981 |
Subclasses of opioids based on body temperature change in rats: acute subcutaneous administration.
Topics: Animals; Body Temperature; Buprenorphine; Dose-Response Relationship, Drug; Endorphins; Injections, Subcutaneous; Male; Meperidine; Morphine; Nalbuphine; Naloxone; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1983 |
Antitussive effect of the optical isomers of mu, kappa and sigma opiate agonists/antagonists in the cat.
Topics: Animals; Antitussive Agents; Blood Pressure; Cats; Codeine; Cyclazocine; Dextromethorphan; Female; Heart Rate; Male; Methadone; Morphine; Narcotics; Phenazocine; Stereoisomerism | 1983 |
Differential effects of prototype opioid agonists on the acquisition of conditional discriminations in monkeys.
Topics: Animals; Behavior, Animal; Conditioning, Psychological; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Male; Morphine; Pentazocine; Phenazocine; Psychomotor Performance | 1983 |
Acquisition of brightness discrimination in the rat is impaired by opiates with psychotomimetic properties.
Topics: Animals; Avoidance Learning; Cyclazocine; Discrimination Learning; Male; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Phenazocine; Photic Stimulation; Psychotropic Drugs; Rats; Rats, Inbred F344 | 1983 |
Enhancement of the opiate withdrawal response by antipsychotic drugs in guinea-pigs is not mediated by sigma binding sites.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Atropine; Behavior, Animal; Clozapine; Dizocilpine Maleate; Female; Guinea Pigs; Ketamine; Kinetics; Male; Morphine; Motor Activity; Naloxone; Phenazocine; Raclopride; Radioligand Assay; Receptors, sigma; Remoxipride; Salicylamides; Substance Withdrawal Syndrome | 1993 |
Area tempestas modulates the behavioural responses to nociceptive stimuli in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anticonvulsants; Azocines; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Escape Reaction; Foot; Hot Temperature; Male; Morphine; Naltrexone; Narcotic Antagonists; Olfactory Pathways; Pain; Phenazocine; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Seizures; Tail | 1993 |
Activity of opioid ligands in cells expressing cloned mu opioid receptors.
Topics: Azocines; beta-Endorphin; Binding, Competitive; Butorphanol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Humans; Hydromorphone; Ligands; Morphine; Naltrexone; Phenazocine; Radioligand Assay; Receptors, Opioid, mu; Tritium | 2003 |
Phenazocine hydrobromide: pharmaceutical aspects of a new benzomorphan analgesic related to morphine.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Benzomorphans; Morphine; Pharmacy; Phenazocine | 1961 |
Analgesic and other neuropharmacologic effects of phenazocine (NIH 7519, prinadol) compared with morphine.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Morphine; Phenazocine | 1960 |
A study of postoperative pain.
Topics: Dextromoramide; Humans; Hydromorphone; Morphine; Pain; Pain, Postoperative; Phenazocine; Postoperative Care | 1963 |
ANALGESICS FOR THE RELIEF OF PAIN. I. NARCOTIC ANALGESICS.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Codeine; Humans; Hydromorphone; Meperidine; Methadone; Morphine; Narcotics; Oxymorphone; Pain; Phenazocine; Piperidines | 1964 |
SOME NARCOTIC ANTAGONISTS IN THE BENZOMORPHAN SERIES.
Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Antipyretics; Azocines; Benzomorphans; Cats; Cyclazocine; Haplorhini; Heterocyclic Compounds; Meperidine; Mice; Morphine; Nalorphine; Narcotic Antagonists; Pentazocine; Pharmacology; Phenazocine; Rats; Research; Toxicology | 1964 |
A RAPID SCREENING TEST FOR POTENTIAL ADDICTION LIABILITY OF NEW ANALGESIC AGENTS.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Behavior, Addictive; Codeine; Dextropropoxyphene; Heroin; Hydromorphone; Meperidine; Methadone; Mice; Morphine; Phenazocine; Research; Substance-Related Disorders; Toxicology | 1964 |
A COMPARISON OF MORPHINE AND PHENAZOCINE IN POSTOPERATIVE PAIN.
Topics: Drug Therapy; Humans; Laparotomy; Morphine; Pain; Pain, Postoperative; Phenazocine; Postoperative Complications | 1964 |
Straub tail reaction in mice treated with σ(1) receptor antagonist in combination with methamphetamine.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Antipsychotic Agents; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Male; Methamphetamine; Mice; Mice, Inbred Strains; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Pyrimidines; Receptors, Opioid, delta; Reflex; Tail; Time Factors | 2012 |