phenazocine has been researched along with cyclazocine in 96 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 89 (92.71) | 18.7374 |
1990's | 7 (7.29) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Metcalf, G; Rees, JM; Ward, SJ | 1 |
Coale, EH; Hein, DW; Herling, S; Valentino, RJ; Woods, JH | 1 |
Eades, CG; Gilbert, PE; Huppler, RE; Martin, WR; Thompson, JA | 1 |
Feuerstein, G; Gagnon, RC; Gu, JL; Lysko, PG; Yue, TL | 1 |
Baldessarini, RJ; Booth, RG | 1 |
Dykstra, LA; Picker, MJ; Powell, K | 1 |
Goldberg, SR; Schindler, CW; White, MF | 1 |
Barnette, MS; Barone, FC; Callahan, JF; Grous, M; Manning, CD | 1 |
Balster, RL | 1 |
Beart, PM; Manallack, DT; O'Shea, RD | 1 |
Martin, WR; Wu, KM | 2 |
Bronson, ME; Moerschbaecher, JM | 1 |
Junien, JL; Pascaud, X; Roman, F; Vauché, D | 1 |
Kamei, H; Kameyama, T; Nabeshima, T | 1 |
Carino, MA; Horita, A; Yamawaki, S | 1 |
Cooper, SJ; Jackson, A; Kirkham, TC | 1 |
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K | 1 |
Furukawa, H; Hiramatsu, M; Kameyama, T; Nabeshima, T | 1 |
Adler, MW; Geller, EB; Rowan, CH | 1 |
George, R; Pechnick, R; Poland, RE | 2 |
Adler, MW; Geller, EB; Kirby, A; Messner, S; Robin, M | 1 |
Burks, TF; Hirning, LD; Porreca, F | 1 |
Eisenberg, RM | 1 |
DeRossett, SE; Holtzman, SG | 1 |
Su, TP; Weissman, AD; Yeh, SY | 1 |
Contreras, PC; O'Donohue, TL; Quirion, R | 1 |
Hiramatsu, M; Kameyama, T; Nabeshima, T | 1 |
Dykstra, LA; Slifer, BL | 1 |
Cook, L; Steinfels, GF; Tam, SW | 1 |
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR | 1 |
Bartschat, DK; Blaustein, MP | 1 |
Dykstra, LA; Picker, M | 1 |
Gormezano, I; Harvey, JA; Lamb, MR; Schindler, CW | 1 |
Dykstra, LA; Heise, JW; Picker, M | 1 |
Costa, T; Dunn, LL; Hubbell, CL; Hunter, GA; Reid, LD | 1 |
Bergman, J; Hassoun, J; Schuster, CR | 1 |
Röthig, J | 1 |
Medzihradsky, F; Nandhasri, PS | 1 |
Aceto, MD; McKean, DB; Pearl, J | 1 |
Bowman, WC; Buwembo, JB | 1 |
Carr, EA; Marks, MJ; Medzihradsky, F | 1 |
Janssen, PA | 1 |
Pittman, KA; Williams, TA | 1 |
Ahmad, K; Medzihradsky, F | 1 |
McKean, DB; Pearl, J; Stander, H | 1 |
Gyand, EA; Kosterlitz, HW | 1 |
Cowan, A; Gmerek, DE | 2 |
Berry, SC; Dawkins, SL; Lodge, D | 1 |
Khazan, N; Young, GA | 2 |
Herz, A; Pfeiffer, A | 2 |
Dawson, G; McLawhon, RW; Miller, RJ; West, RE | 1 |
Zukin, RS; Zukin, SR | 1 |
Miller, RJ | 1 |
Tung, AS; Yaksh, TL | 1 |
Leander, JD | 1 |
Ben-Sreti, MM; Gonzalez, JP; Sewell, RD | 1 |
Enger, M; Grynne, BH; Holmen, AT; Maurset, AR | 1 |
Billington, CJ; Gerritsen, GC; Levine, AS; Morley, JE | 1 |
Balster, RL; Brady, KT; Slifer, BL; Zukin, SR | 1 |
Holtzman, SG; Teal, JJ | 1 |
Harris, RA; Snell, D | 1 |
Nishimura, S; Pasternak, GW; Wolozin, BL | 1 |
Nishimura, S; Pasternak, GW | 1 |
Guidotti, A; Saiani, L | 1 |
Bearden, LJ; Snead, OC | 1 |
Kandasamy, SB; Williams, BA | 1 |
Balster, RL; Slifer, BL | 1 |
Cicero, TJ; Meyer, ER; Owens, DP; Schmoeker, PF | 1 |
Johnson, N; Pasternak, GW | 1 |
Tam, SW | 1 |
Gosnell, BA; Levine, AS; Morley, JE | 1 |
Greenfield, LJ; Guyenet, PG; Hackett, JT; Stringer, JL | 1 |
Code, RA; Tang, AH | 1 |
Bajorek, JG; Lee, RJ; Lomax, P | 1 |
Holtzman, SG; White, JM | 2 |
Cowan, A; Porreca, F; Raffa, RB; Tallarida, RJ | 1 |
Johnson, KM; Leventer, SM | 1 |
Mastropaolo, J; Moerschbaecher, JM; Thompson, DM; Winsauer, PJ | 1 |
Commissaris, RL; Henck, JW; Mokler, DJ; Rech, RH | 1 |
Colpaert, FC; Janssen, PA | 1 |
Iwamoto, ET | 1 |
Herling, S; Woods, JH | 1 |
Holtzman, SG | 1 |
Carter, FE; Chau, TT; Harris, LS | 1 |
Moerschbaecher, JM; Thompson, DM | 1 |
Franklin, SR; Tang, AH | 1 |
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC | 1 |
Ichikawa, T; Ikeda, K; Kobayashi, T; Kumanishi, T; Togashi, S | 1 |
HARRIS, LS; PIERSON, AK | 1 |
LASAGNA, L | 1 |
4 review(s) available for phenazocine and cyclazocine
Article | Year |
---|---|
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response | 1985 |
[Analgesics. 32].
Topics: Alphaprodine; Analgesics; Azepines; Benzimidazoles; Bridged-Ring Compounds; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Fentanyl; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Levallorphan; Levorphanol; Lysergic Acid Diethylamide; Methadone; Morphinans; Morphine; Nalorphine; Naphthoquinones; Oxymorphone; Pentazocine; Phenazocine; Phenoperidine | 1969 |
Multiple opiate receptors for multiple opioid peptides.
Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission | 1982 |
THE CLINICAL EVALUATION OF MORPHINE AND ITS SUBSTITUTES AS ANALGESICS.
Topics: Analgesics; Analgesics, Non-Narcotic; Antipyretics; Biomedical Research; Codeine; Cyclazocine; Dextromoramide; Dextropropoxyphene; Heroin; Humans; Hydromorphone; Isonipecotic Acids; Meperidine; Methadone; Methotrimeprazine; Morphine; Nalorphine; Narcotic Antagonists; Oxymorphone; Pentazocine; Phenazocine; Substance-Related Disorders; Toxicology | 1964 |
92 other study(ies) available for phenazocine and cyclazocine
Article | Year |
---|---|
The comparative pharmacology of morphine, ketocyclazocine and 2'-hydroxy-5,9-dimethyl-2-allyl-6,7-benzomorphan in rodents [proceedings].
Topics: Animals; Behavior, Animal; Body Temperature; Cyclazocine; Mice; Morphine; Phenazocine; Rats; Respiration | 1977 |
Narcotic drug discriminations by rhesus monkeys and pigeons.
Topics: Animals; Columbidae; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Discrimination Learning; Dose-Response Relationship, Drug; Enkephalins; Ethylketocyclazocine; Etorphine; Hormones; Macaca; Macaca mulatta; Naltrexone; Narcotics; Phenazocine | 1979 |
The effects of morphine- and nalorphine- like drugs in the nondependent and morphine-dependent chronic spinal dog.
Topics: Animals; Apomorphine; Cyclazocine; Cyclopropanes; Dextropropoxyphene; Dogs; Ethylketocyclazocine; Humans; Morphinans; Morphine; Morphine Dependence; Nalorphine; Naltrexone; Phenazocine; Spinal Cord | 1976 |
Neuroprotective effects of SKF 10,047 in cultured rat cerebellar neurons and in gerbil global brain ischemia.
Topics: Animals; Body Temperature; Brain Ischemia; Cells, Cultured; Cerebellum; Cyclazocine; Dizocilpine Maleate; Gerbillinae; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Reference Values; Stereoisomerism | 1992 |
(+)-6,7-benzomorphan sigma ligands stimulate dopamine synthesis in rat corpus striatum tissue.
Topics: Animals; Benzomorphans; Catecholamines; Corpus Striatum; Cyclazocine; Dopamine; In Vitro Techniques; Ligands; Male; Nerve Endings; Neural Pathways; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Stimulation, Chemical; Tyrosine 3-Monooxygenase | 1991 |
Stereospecificity of mixed-action opioid agonist/antagonists in morphine-tolerant squirrel monkeys.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Morphine; Narcotic Antagonists; Narcotics; Pentazocine; Phenazocine; Saimiri; Stereoisomerism | 1990 |
Effects of morphine, ethylketocyclazocine, N-allylnormetazocine and naloxone on locomotor activity in the rabbit.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Female; Male; Morphine; Motor Activity; Naloxone; Nictitating Membrane; Phenazocine; Rabbits | 1990 |
Inhibition of neuronally induced relaxation of canine lower esophageal sphincter by opioid peptides.
Topics: Animals; Autonomic Nervous System; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Dogs; Electric Stimulation; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Esophagogastric Junction; Ethylketocyclazocine; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Neurons; Phenazocine | 1990 |
Substitution and antagonism in rats trained to discriminate (+)-N-allylnormetazocine from saline.
Topics: Animals; Binding Sites; Butaclamol; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Haloperidol; Male; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1989 |
Regulation of sigma-receptors: high- and low-affinity agonist states, GTP shifts, and up-regulation by rimcazole and 1,3-Di(2-tolyl)guanidine.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Binding, Competitive; Brain; Carbazoles; Cyclazocine; Dopamine; Dopamine Agents; GTP-Binding Proteins; Guanidines; Guanosine Triphosphate; Magnesium; Male; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma | 1989 |
Cardiovascular and respiratory effects of an opioid kappa agonist ethylketazocine and sigma agonist N-allylnormetazocine in acutely decerebrated dogs.
Topics: Animals; Blood Pressure; Cyclazocine; Decerebrate State; Dogs; Ethylketocyclazocine; Female; Heart Rate; Male; Phenazocine; Pulmonary Ventilation | 1989 |
Effects of mu, kappa and sigma opioids on fixed consecutive number responding in rats.
Topics: Animals; Buprenorphine; Conditioning, Operant; Cyclazocine; Dextroamphetamine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Phenazocine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1987 |
Evidence for a non-opioid sigma binding site in the guinea-pig myenteric plexus.
Topics: Animals; Binding, Competitive; Cell Membrane; Chlorpromazine; Cyclazocine; Ethylketocyclazocine; Guinea Pigs; Haloperidol; Imipramine; Male; Myenteric Plexus; Phenazocine; Propranolol; Receptors, Opioid; Receptors, sigma | 1988 |
A role played by sigma receptors in the conditioned suppression of motility in mice.
Topics: Animals; Conditioning, Psychological; Cyclazocine; Drug Tolerance; Male; Mice; Mice, Inbred Strains; Motor Activity; Naloxone; Phenazocine; Receptors, Opioid; Receptors, sigma; Synaptic Membranes | 1988 |
Analeptic effect of opiate receptor agonists in rabbits.
Topics: Animals; Arousal; Brain; Central Nervous System Stimulants; Codeine; Cyclazocine; Dose-Response Relationship, Drug; Enkephalin, Methionine; Ethylketocyclazocine; Etorphine; Male; Meperidine; Methadone; Morphine; Naltrexone; Narcotics; Phenazocine; Rabbits; Receptors, Opioid; Reflex | 1985 |
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid | 1987 |
Different effects of ethylketocyclazocine on phencyclidine- and N-allylnormetazocine-induced stereotyped behaviors in rats.
Topics: Analgesics, Opioid; Animals; Cyclazocine; Ethylketocyclazocine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Stereotyped Behavior | 1987 |
Body temperature effects of opioids in rats: intracerebroventricular administration.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1986 |
Identification of multiple opiate receptors through neuroendocrine responses. I. Effects of agonists.
Topics: Animals; Corticosterone; Cyclazocine; Ethylketocyclazocine; Growth Hormone; Injections, Subcutaneous; Luteinizing Hormone; Male; Morphine; Phenazocine; Pituitary Hormones, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid | 1985 |
Identification of multiple opiate receptors through neuroendocrine responses. II. Antagonism of mu, kappa and sigma agonists by naloxone and WIN 44,441-3.
Topics: Animals; Azocines; Corticosterone; Cyclazocine; Drug Interactions; Ethylketocyclazocine; Growth Hormone; Luteinizing Hormone; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Pituitary Hormones, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid | 1985 |
Differentiating opioids by their pupillary effects in the rat.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Methadone; Motor Activity; Naloxone; Narcotics; Nystagmus, Physiologic; Phenazocine; Pupil; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism | 1985 |
Mu, but not kappa, opioid agonists induce contractions of the canine small intestine ex vivo.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Cyclazocine; Dimethylphenylpiperazinium Iodide; Dogs; Ethylketocyclazocine; Gastrointestinal Motility; In Vitro Techniques; Intestine, Small; Morphine; Nalorphine; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Plasma corticosterone changes in response to central or peripheral administration of kappa and sigma opiate agonists.
Topics: Animals; Brain; Corticosterone; Cyclazocine; Ethylketocyclazocine; Humans; Hypothalamo-Hypophyseal System; Male; Morphine; Naloxone; Naltrexone; Opioid-Related Disorders; Phenazocine; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1985 |
Discriminative stimulus effects of the opioid antagonist diprenorphine in the squirrel monkey.
Topics: Animals; Cyclazocine; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Generalization, Stimulus; Morphinans; Naloxone; Narcotic Antagonists; Phenazocine; Psychotropic Drugs; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Saimiri | 1986 |
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays.
Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma | 1986 |
Agonistic and antagonistic effects of PCP-derivatives and sigma opioids in PCP behavioral and receptor assays.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclazocine; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereotyped Behavior; Structure-Activity Relationship; Tritium | 1986 |
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid | 1986 |
Discriminative stimulus effects of N-allylnormetazocine in rats trained to discriminate a kappa from a sigma agonist.
Topics: Animals; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, sigma; Stereoisomerism | 1987 |
Discriminative stimulus properties of (+)-N-allylnormetazocine in the rat: correlations with (+)-N-allylnormetazocine and phencyclidine receptor binding.
Topics: Animals; Brain; Cyclazocine; Discrimination Learning; Ketamine; Male; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism | 1987 |
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1987 |
Psychotomimetic sigma-ligands, dexoxadrol and phencyclidine block the same presynaptic potassium channel in rat brain.
Topics: Animals; Brain; Cyclazocine; Dioxolanes; Dioxoles; Dose-Response Relationship, Drug; Hallucinogens; In Vitro Techniques; Naloxone; Phenazocine; Phencyclidine; Piperidines; Potassium Channels; Rats; Synaptosomes | 1988 |
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors | 1987 |
Effects of morphine, ethylketocyclazocine, and N-allylnormetazocine on classical conditioning of the rabbit nictitating membrane response.
Topics: Animals; Conditioning, Classical; Conditioning, Eyelid; Cyclazocine; Ethylketocyclazocine; Female; Light; Male; Morphine; Nictitating Membrane; Phenazocine; Rabbits; Sound | 1986 |
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule | 1987 |
Selected opioids and responding for intracranial reinforcement.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Hypothalamic Area, Lateral; Naloxone; Phenazocine; Rats; Reinforcement, Psychology; Self Stimulation; Stereoisomerism | 1985 |
Behavioral effects of selected opiates and phencyclidine in the nondependent and cyclazocine-dependent rhesus monkey.
Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Food; Macaca mulatta; Male; Naloxone; Phenazocine; Phencyclidine; Stereoisomerism; Substance-Related Disorders | 1985 |
Effects of some analgesics and antidepressants on the (Na + + K + )-adenosine triphosphatase from cortices of brain and kidney.
Topics: Adenosine Triphosphatases; Amitriptyline; Analgesics; Animals; Antidepressive Agents; Cattle; Cerebral Cortex; Chlorpromazine; Cyclazocine; Desipramine; Dose-Response Relationship, Drug; Hydralazine; Imipramine; In Vitro Techniques; Kidney; Kidney Cortex; Pentazocine; Phenazocine; Phenelzine; Potassium; Sodium; Tranylcypromine | 1972 |
Effects of opiates and opiate antagonists on the Straub tail reaction in mice.
Topics: Analgesics; Animals; Atropine; Bridged-Ring Compounds; Codeine; Cyclazocine; Levallorphan; Meperidine; Mice; Morphinans; Morphine; Narcotic Antagonists; Pentazocine; Phenazocine; Stereoisomerism; Tail | 1969 |
Effects of narcotic analgesics on contractions of the chick isolated, innervated oesophagus.
Topics: Acetylcholine; Analgesics; Animals; Chickens; Cyclazocine; Dextropropoxyphene; Electric Stimulation; Esophagus; Heroin; In Vitro Techniques; Meperidine; Methadone; Morphinans; Morphine; Muscle Contraction; Nalorphine; Pentazocine; Phenazocine; Serotonin; Tachyphylaxis; Time Factors | 1972 |
Energy-dependent uptake of benzomorphans by leukocytes.
Topics: Animals; Cell Membrane; Chromatography, Gas; Cyclazocine; Fluorides; Glucose; Leukocytes; Male; Models, Biological; Oxygen Consumption; Pentazocine; Phenazocine; Potassium; Rats; Sodium; Structure-Activity Relationship; Time Factors | 1972 |
Potent long-acting antagonists of the 9,9-dialkylbenzomorphan series.
Topics: Alkylation; Analgesics; Animals; Butyrates; Cyclazocine; Cyclization; Isomerism; Methylation; Morphinans; Narcotic Antagonists; Pentazocine; Phenazocine; Phenols; Propionates; Rats; Structure-Activity Relationship; Time Factors | 1973 |
Pentazocine radioimmunoassay.
Topics: Ammonium Sulfate; Animals; Antibody Specificity; Antigen-Antibody Reactions; Azo Compounds; Carboxylic Acids; Chromatography, Gas; Cross Reactions; Cyclazocine; Levallorphan; Levorphanol; Methods; Molecular Weight; Morphine; Nalorphine; Oxidation-Reduction; Pentazocine; Phenazocine; Rabbits; Radioimmunoassay; Tritium; Urine | 1974 |
The determination of benzomorphan derivatives in plasma by gas chromatography.
Topics: Analgesics; Azocines; Cyclazocine; Humans; Methods; Narcotic Antagonists; Pentazocine; Phenazocine | 1971 |
Effects of analgesics and other drugs on mice in phenylquinone and rotarod tests.
Topics: Analgesics; Animals; Chemical Phenomena; Chemistry; Chlorpromazine; Cyclazocine; Dextroamphetamine; Levallorphan; Male; Mice; Morphine; Motor Activity; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Pilocarpine; Quinones; Salivation | 1969 |
Agonist and antagonist actions of morphine-like drugs on the guinea-pig isolated ileum.
Topics: Analgesics; Animals; Cyclazocine; Drug Synergism; Guinea Pigs; Ileum; Levallorphan; Levorphanol; Morphine; Muscle, Smooth; Nalorphine; Narcotic Antagonists; Pentazocine; Phenazocine; Reflex | 1966 |
An in vivo pharmacological analysis of benzomorphan binding sites in rats.
Topics: Animals; Benzomorphans; Bombesin; Brain; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Grooming; Humans; Male; Morphinans; Morphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism; Stereotyped Behavior | 1984 |
Comparison of sigma- and kappa-opiate receptor ligands as excitatory amino acid antagonists.
Topics: Acetylcholine; Amino Acids; Animals; Aspartic Acid; Cats; Cyclazocine; Ethylketocyclazocine; Kainic Acid; Ketamine; Ligands; Microelectrodes; N-Methylaspartate; Neurons; Oxadiazoles; Phenazocine; Quisqualic Acid; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, sigma; Stereoisomerism | 1984 |
Differential neuropharmacological effects of mu, kappa and sigma opioid agonists on cortical EEG power spectra in the rat. Stereospecificity and naloxone antagonism.
Topics: Animals; Cerebral Cortex; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Methadone; Molecular Conformation; Morphine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1984 |
Demonstration and distribution of an opiate binding site in rat brain with high affinity for ethylketocyclazocine and SKF 10,047.
Topics: Analgesics, Opioid; Animals; Brain; Cerebral Cortex; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Kinetics; Mesencephalon; Phenazocine; Rats; Receptors, Opioid; Thalamus; Tissue Distribution | 1981 |
Distinct high-affinity binding sites for benzomorphan drugs and enkephalin in a neuroblastoma--brain hybrid cell line.
Topics: Analgesics, Opioid; Animals; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Cell Line; Cyclazocine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hybrid Cells; Kinetics; Morphinans; Neuroblastoma; Phenazocine; Rats; Receptors, Opioid | 1981 |
Multiple opiate receptors: emerging concepts.
Topics: Analgesics, Opioid; Animals; Behavior; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Kinetics; Phenazocine; Rats; Receptors, Opioid; Structure-Activity Relationship | 1981 |
Discrimination of three opiate receptor binding sites with the use of a computerized curve-fitting technique.
Topics: Animals; Binding, Competitive; Brain; Computers; Cyclazocine; Dihydromorphine; Diprenorphine; Dynorphins; Endorphins; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Phenazocine; Rats; Receptors, Opioid | 1982 |
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord | 1982 |
Effects of ketazocine, ethylketazocine and phenazocine on schedule-controlled behavior: antagonism by naloxone.
Topics: Analgesics, Opioid; Animals; Columbidae; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Naloxone; Phenazocine | 1982 |
Effects of elevated calcium and calcium antagonists on 6,7-benzomorphan-induced analgesia.
Topics: Analgesia; Analgesics; Analgesics, Opioid; Animals; Benzomorphans; Calcium; Calcium Channel Blockers; Cyclazocine; Egtazic Acid; Ethylketocyclazocine; Gallopamil; Male; Mice; Morphinans; Pentazocine; Phenazocine | 1983 |
The effect of two different buffers on the high affinity 3H-ethylketocyclazocine and 3H-SKF10047 binding to guinea pig brain membranes.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Ethylketocyclazocine; Guinea Pigs; HEPES; In Vitro Techniques; Morphine; Naloxone; Phenazocine; Piperazines; Receptors, Opioid; Tritium; Tromethamine | 1984 |
In vivo evidence for benzomorphan-selective receptors in rats.
Topics: Analgesics, Opioid; Animals; Benzomorphans; Bombesin; Buprenorphine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Male; Morphinans; Morphine; Naloxone; Phenazocine; Pruritus; Rats; Rats, Inbred Strains; Receptors, Opioid | 1984 |
Feeding systems in Chinese hamsters.
Topics: Animals; Brain; Calcitonin; Circadian Rhythm; Cricetinae; Cyclazocine; Diabetes Mellitus; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Feeding Behavior; Haloperidol; Mesocricetus; Naloxone; Peptide Fragments; Phenazocine; Sincalide; Starvation | 1984 |
Behavioral and biochemical stereoselectivity of sigma opiate/PCP receptors.
Topics: Animals; Behavior, Animal; Brain; Cyclazocine; Hydromorphone; In Vitro Techniques; Ketamine; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism | 1984 |
Discriminative stimulus effects of prototype opiate receptor agonists in monkeys.
Topics: Animals; Apomorphine; Cyclazocine; Ethylketocyclazocine; Female; Generalization, Stimulus; Haloperidol; Male; Models, Biological; Morphine; Naltrexone; Phenazocine; Prejudice; Receptors, Opioid; Saimiri | 1980 |
Interactions between narcotic agonists, partial agonists andd antagonists evaluated by punished an unpunished behavior in the rat.
Topics: Animals; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Phenazocine; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid | 1982 |
The binding of kappa- and sigma-opiates in rat brain.
Topics: Animals; Binding Sites; Brain; Culture Techniques; Cyclazocine; Dihydromorphine; Enkephalins; Ethylketocyclazocine; Ligands; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Tritium | 1982 |
Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity.
Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Goldfish; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1982 |
Opiate receptor-mediated inhibition of catecholamine release in primary cultures of bovine adrenal chromaffin cells.
Topics: Acetylcholine; Adrenal Medulla; Animals; beta-Endorphin; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Phenazocine; Receptors, Opioid | 1982 |
The epileptogenic spectrum of opiate agonists.
Topics: Animals; Anticonvulsants; beta-Endorphin; Cyclazocine; Electroencephalography; Endorphins; Enkephalin, Leucine; Epilepsy; Ethylketocyclazocine; Injections, Intraventricular; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains | 1982 |
Peptide and non-peptide opioid-induced hyperthermia in rabbits.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptides; Phenazocine; Rats | 1983 |
Reinforcing properties of stereoisomers of the putative sigma agonists N-allylnormetazocine and cyclazocine in rhesus monkeys.
Topics: Animals; Cocaine; Cyclazocine; Dose-Response Relationship, Drug; Macaca mulatta; Male; Phenazocine; Receptors, Opioid; Receptors, sigma; Reinforcement, Psychology; Self Stimulation; Stereoisomerism; Structure-Activity Relationship | 1983 |
Differential stereospecific effects of mu, kappa, and sigma opioid agonists on cortical EEG power spectra in the rat.
Topics: Animals; Cerebral Cortex; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Methadone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma; Stereoisomerism | 1983 |
Opiate-induced enhancement of the effects of naloxone on serum luteinizing hormone levels in the male rat: specificity for Mu agonists.
Topics: Animals; Binding, Competitive; Cyclazocine; Ethanol; Ethylketocyclazocine; Kinetics; Luteinizing Hormone; Male; Morphine; Naloxone; Pentobarbital; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
The binding to rat brain homogenates of Mr2034, a universal opiate.
Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
An analysis of nicotinic and opioid processes in the medulla oblongata and nucleus ambiguus of the dog.
Topics: Animals; Blood Pressure; Cyclazocine; Decerebrate State; Dogs; Electric Stimulation; Endorphins; Ethylketocyclazocine; Female; Fentanyl; Heart Rate; Male; Mecamylamine; Medulla Oblongata; Naloxone; Nicotine; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma | 1983 |
Naloxone-inaccessible sigma receptor in rat central nervous system.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Enkephalins; Ethylketocyclazocine; Kinetics; Naloxone; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, sigma; Spinal Cord; Tissue Distribution | 1983 |
N-allylnormetazocine (SKF-10,047): the induction of feeding by a putative sigma agonist.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Interactions; Eating; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |
Blockade of long-term potentiation by phencyclidine and sigma opiates in the hippocampus in vivo and in vitro.
Topics: Animals; Cyclazocine; Drug Synergism; Hippocampus; Male; Membrane Potentials; Morphine; Naloxone; Narcotics; Phenazocine; Phencyclidine; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synapses; Synaptic Transmission | 1983 |
Discriminative stimulus properties of nalorphine in the rhesus monkeys.
Topics: Animals; Benzodiazepines; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Macaca mulatta; Male; Nalorphine; Naloxone; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa | 1983 |
Similar anticonvulsant, but unique, behavioural effects of opioid agonists in the seizure-sensitive Mongolian gerbil.
Topics: Animals; Anticonvulsants; Behavior, Animal; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Gerbillinae; Male; Morphine; Narcotics; Phenazocine; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures | 1984 |
Further characterization of the three-choice morphine, cyclazocine and saline discrimination paradigm: opioids with agonist and antagonist properties.
Topics: Animals; Cyclazocine; Discrimination Learning; Discrimination, Psychological; Ethylketocyclazocine; Male; Morphine; Narcotic Antagonists; Narcotics; Phenazocine; Phencyclidine; Rats; Sodium Chloride; Stereoisomerism | 1983 |
Ketazocines and morphine: effects on gastrointestinal transit after central and peripheral administration.
Topics: Animals; Cyclazocine; Ethylketocyclazocine; Gastrointestinal Motility; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Phenazocine; Rats; Rats, Inbred Strains | 1983 |
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains | 1984 |
Effects of opioids on accuracy of a fixed-ratio discrimination in monkeys and rats.
Topics: Animals; Buprenorphine; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Isomerism; Macaca mulatta; Male; Methadone; Morphinans; Morphine; Phenazocine; Rats | 1984 |
Three-choice drug discrimination: phencyclidine-like stimulus effects of opioids.
Topics: Animals; Choice Behavior; Cyclazocine; Dextroamphetamine; Discrimination, Psychological; Male; Naltrexone; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Secobarbital | 1983 |
Behavioral interactions of opioid agonists and antagonists with serotonergic systems.
Topics: Animals; Brain; Conditioning, Operant; Cyclazocine; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Lysergic Acid Diethylamide; Male; Metergoline; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement Schedule | 1984 |
Agonist and antagonist effects of prototype opiate drugs in rats discriminating fentanyl from saline: characteristics of partial generalization.
Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Male; Morphine; Nalorphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Sodium Chloride | 1984 |
Pharmacologic effects of N-allylnormetazocine (SKF-10047).
Topics: Analgesics; Animals; Behavior, Animal; Clonidine; Cyclazocine; Ethylketocyclazocine; Male; Morphine; Motor Activity; Phenazocine; Rats; Receptors, Dopamine; Spiperone | 1981 |
Discriminative stimulus effects of etorphine in Rhesus monkeys.
Topics: Animals; Codeine; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Etorphine; Macaca mulatta; Male; Meperidine; Morphinans; Morphine; Pentazocine; Phenazocine; Sodium Chloride | 1981 |
Phencyclidine-like discriminative stimulus properties of opioids in the squirrel monkey.
Topics: Animals; Cyclazocine; Discrimination Learning; Female; Male; Naltrexone; Narcotics; Phenazocine; Phencyclidine; Saimiri; Time Factors | 1982 |
Antitussive effect of the optical isomers of mu, kappa and sigma opiate agonists/antagonists in the cat.
Topics: Animals; Antitussive Agents; Blood Pressure; Cats; Codeine; Cyclazocine; Dextromethorphan; Female; Heart Rate; Male; Methadone; Morphine; Narcotics; Phenazocine; Stereoisomerism | 1983 |
Differential effects of prototype opioid agonists on the acquisition of conditional discriminations in monkeys.
Topics: Animals; Behavior, Animal; Conditioning, Psychological; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Male; Morphine; Pentazocine; Phenazocine; Psychomotor Performance | 1983 |
Acquisition of brightness discrimination in the rat is impaired by opiates with psychotomimetic properties.
Topics: Animals; Avoidance Learning; Cyclazocine; Discrimination Learning; Male; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Phenazocine; Photic Stimulation; Psychotropic Drugs; Rats; Rats, Inbred F344 | 1983 |
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma | 1995 |
Effects of sigma ligands on the cloned mu-, delta- and kappa-opioid receptors co-expressed with G-protein-activated K+ (GIRK) channel in Xenopus oocytes.
Topics: Animals; Brain Chemistry; Cyclazocine; Cyclopentanes; Dose-Response Relationship, Drug; GTP-Binding Proteins; Ligands; Oocytes; Phenazocine; Potassium Channels; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma; RNA, Messenger; Xenopus laevis | 1996 |
SOME NARCOTIC ANTAGONISTS IN THE BENZOMORPHAN SERIES.
Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Antipyretics; Azocines; Benzomorphans; Cats; Cyclazocine; Haplorhini; Heterocyclic Compounds; Meperidine; Mice; Morphine; Nalorphine; Narcotic Antagonists; Pentazocine; Pharmacology; Phenazocine; Rats; Research; Toxicology | 1964 |