phaclofen has been researched along with baclofen in 241 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 26 (10.79) | 18.7374 |
1990's | 135 (56.02) | 18.2507 |
2000's | 53 (21.99) | 29.6817 |
2010's | 26 (10.79) | 24.3611 |
2020's | 1 (0.41) | 2.80 |
Authors | Studies |
---|---|
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Del Bianco, E; Giuliani, S; Lecci, A; Maggi, CA; Santicioli, P | 1 |
Berger, TW; Nisenbaum, ES | 1 |
Blanchet, G; Gahery, Y; Luccarini, P; Pompeiano, O | 1 |
Douglas, WW; Kongsamut, S; Shibuya, I | 1 |
Libertun, C; Lux-Lantos, V; Rey, E | 1 |
Beani, L; Bianchi, C; Ferraro, L; Tanganelli, S | 1 |
Kawaguchi, Y | 1 |
Bonanno, G; Raiteri, M | 2 |
Donoso, AO; López, FJ; Negro-Vilar, A | 1 |
Bonanno, G; Gemignani, A; Lanza, M; Pende, M; Raiteri, M; Vellebuona, F | 1 |
Finch, DM; Mello, LE; Tan, AM | 1 |
Dunwiddie, TV; Lupica, CR; Proctor, WR | 1 |
Saito, H; Tamai, A; Ueno, H; Yoshida, K | 1 |
Bernardini, MC; Blandizzi, C; Del Tacca, M; Natale, G | 1 |
Allan, AM; Burnett, D; Harris, RA | 1 |
Bartolini, A; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P | 1 |
Kow, LM; Ogawa, S; Pfaff, DW | 1 |
Henry, JL; Hong, YG | 1 |
Henry, JL; Hong, Y | 1 |
Sanders, SK; Shekhar, A | 1 |
Sastry, BR; Xie, Z | 1 |
Aceves, J; Arias-Montaño, JA; Martínez-Fong, D | 1 |
Lacaille, JC | 1 |
Jones, AJ; Keen, P; Ray, NJ | 1 |
Couture, R; De Champlain, J; Hasséssian, H; Prat, A | 1 |
Lewis, DV; Morrisett, RA; Mott, DD; Swartzwelder, HS; Wilson, WA | 1 |
Henriksen, SJ; Steffensen, SC | 1 |
Aran, S; Hammond, DL | 1 |
Baldwin, BA; Ebenezer, IS | 1 |
Howson, W; Lacey, MG; Seabrook, GR | 1 |
Ebenezer, IS | 1 |
Alberch, J; Arenas, E; Marsal, J | 1 |
Alhaider, AA; Lei, SZ; Wilcox, GL | 1 |
Hankins, MW; Ikeda, H; Kay, CD | 1 |
Kamata, O; Nakagawa, T; Nakanishi, H; Ukai, K; Watanabe, S; Yamamoto, K | 1 |
Bonanno, G; Giralt, MT; Raiteri, M | 1 |
Bernardini, MC; Blandizzi, C; Del Tacca, M | 1 |
Dun, NJ; Wang, MY | 1 |
Allan, RD; Drew, CA; Ong, J; Tran, HW | 1 |
Huang, JH; Johnston, GA | 1 |
Drew, CA; Johnston, GA; Kerr, DI; Ong, J | 1 |
Barraclough, CA; Hartman, RD; He, JR | 1 |
Collingridge, GL; Davies, CH; Davies, SN | 1 |
Mehta, AK; Ticku, MK | 1 |
Karlsson, G; Olpe, HR | 3 |
De Luca, C; Massotti, M | 1 |
Michler, A | 1 |
Sved, AF; Sved, JC | 1 |
al-Dahan, MI; Tehrani, MH; Thalmann, RH | 1 |
Bittiger, H; Brugger, F; Fagg, G; Froestl, W; Hall, RG; Karlsson, G; Olpe, HR; Pozza, MF; Steinmann, M; Van Riezen, H | 1 |
Hicks, TP; Kaneko, T | 1 |
Bernardi, G; Calabresi, P; De Murtas, M; Mercuri, NB | 1 |
Slater, NT; Smith, RD; Turek, FW | 1 |
Furshpan, EJ; Segal, MM | 1 |
Fukuda, H; Hirayama, T; Ono, H | 1 |
Goto, Y; Hara, N; Hara, Y | 1 |
Bragdon, AC; Lewis, DV; Mott, DD | 1 |
Harrison, NL | 1 |
Malouf, AT; Robbins, CA; Schwartzkroin, PA | 1 |
Kulkarni, SK | 1 |
Johnston, GA; Kerr, DI; Ong, J; Prager, RH | 1 |
Asaro, D; Bonanno, G; Fontana, G; Pellegrini, G; Raiteri, M | 1 |
Böhmer, G; Gebauer, K; Schmid, K | 1 |
Dingsdale, RA; Dolle, RE; Hills, JM; Howson, W; Parsons, ME | 1 |
Erdö, SL; Michler, A | 1 |
Boar, BR; Cross, AJ; Green, AR; Robinson, TN; Toczek, JM | 1 |
Allan, AM; Harris, RA | 1 |
Bonanno, G; Cantoni, C; Pellegrini, G; Raiteri, M | 1 |
Gallagher, JP; Hasuo, H | 2 |
Chamberlin, NL; Dingledine, R | 1 |
Dutar, P; Lamour, Y; Rascol, O | 1 |
Neal, MJ; Shah, MA | 1 |
Klockgether, T; Sontag, KH; Wüllner, U | 1 |
Dutar, P; Nicoll, RA | 1 |
Crunelli, V; Haby, M; Leresche, N; Soltesz, I | 1 |
Karlsson, G; Olpe, HR; Pozza, M | 1 |
Brugger, F; Hall, RG; Olpe, HR; Pozza, MF; Steinmann, MW | 1 |
Albus, K; Baumfalk, U | 1 |
Enna, SJ; Ferkany, JW; Scherer, RW | 1 |
Bonanno, G; Fontana, G; Raiteri, M | 1 |
Curtis, DR; Gynther, BD; Kerr, DI; Ong, J; Prager, RH | 1 |
Borsini, F; Evangelista, S; Giuliani, S; Meli, A | 1 |
Alkon, DL; Axelrod, J; Collin, C; Dahl, D; Devane, WA; Lee, CJ | 1 |
Chad, JE; Stanford, IM; Wheal, HV | 1 |
Cano, J; Machado, A; Santiago, M | 1 |
Humeniuk, RE; Kerr, DI; Ong, J; White, JM | 1 |
Hyson, RL; Reyes, AD; Rubel, EW | 1 |
Boksa, P; Chaudieu, I; Quirion, R; St-Pierre, JA | 1 |
Caddick, SJ; Chad, JE; Stanford, IM | 1 |
Banerjee, PK; Snead, OC | 1 |
Slaughter, MM; Tian, N | 1 |
Bonanno, G; Cavazzani, P; Fassio, A; Raiteri, M | 1 |
Gean, PW; Huang, CC | 1 |
Humeniuk, RE; Ong, J; White, JM | 1 |
Araki, T; Endo, K; Kaneko, T; Kang, Y; Ohishi, H | 1 |
Carpenter, DO; Lin, Y | 1 |
Fisone, G; Greengard, P; Snyder, GL | 1 |
Bonanno, G; Gemignani, A; Paudice, P; Raiteri, M | 1 |
Finch, DM; Gigg, J; Tan, AM | 1 |
Domann, R; Westerhoff, CH; Witte, OW | 1 |
Drew, CA; Frydenvang, K; Hansen, JJ; Johnston, GA; Krogsgaard-Larsen, P; Mitrovic, A; Tran, H | 1 |
Beninger, RJ; Boegman, RJ; DeSousa, NJ; Jhamandas, K | 1 |
Bonanno, G; Lanza, M; Pende, M; Raiteri, M | 1 |
Lewis, DV; Mott, DD; Swartzwelder, HS; Wilson, WA; Xie, CW | 1 |
Hammond, DL; McGowan, MK | 1 |
Hasler, WL; Owyang, C; Roberts, DJ | 1 |
Cotman, CW; Kahle, JS | 1 |
Lacaille, JC; Samulack, DD | 1 |
Dutar, P; Lamour, Y; Potier, B | 1 |
Lennon, VA; Parkman, HP; Stapelfeldt, WH; Szurszewski, JH; Williams, CL | 1 |
Brikas, P | 1 |
DiScenna, PG; Nowicky, AV; Teyler, TJ | 1 |
Hoffman, DS; Kurata, K | 1 |
Haji, A; Takeda, R | 1 |
Clarke, IJ; Scott, CJ | 1 |
Guo, JZ; Ichinose, T; Murakoshi, T | 1 |
Eriksson, PS; Hansson, E; Nilsson, M; Rönnbäck, L | 1 |
Bradley, RM; Wang, L | 1 |
De Koning, HP; Jenks, BG; Roubos, EW | 1 |
el Manira, A; Grillner, S; Matsushima, T; Tegnér, J | 1 |
Kuramochi, T; Suga, T; Suzuki, M | 1 |
Billard, JM; Deisz, RA; Zieglgänsberger, W | 1 |
Albrecht, D; Henklein, P; Zippel, U | 1 |
Haugh-Scheidt, L; Malchow, RP; Ripps, H | 1 |
Chen, W; Hu, GY; Wu, CP; Zhang, JJ | 1 |
Ayata, G; Cutrer, FM; Limmroth, V; Moskowitz, MA | 1 |
Croucher, MJ; Patel, DR; Sundaralingam, J | 1 |
Hashemi, B; Toloui, V; Zarrindast, MR | 1 |
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G | 1 |
Antonelli, T; Ferraro, L; Fuxe, K; O'Connor, WT; Rambert, F; Tanganelli, S | 1 |
Brumberg, JC; Carvell, GE; Kyriazi, HT; Simons, DJ | 1 |
Kubota, K | 1 |
Chen, W; Cheng, JT; Terada, M | 1 |
Brailowsky, S; Di Scala, G; Meneses, S; Montiel, T | 1 |
Snead, OC | 2 |
Dar, MS | 1 |
Armony, JL; LeDoux, JE; Li, XF | 1 |
Itoh, T; Kamisaki, Y; Nakamoto, K; Wada, K | 1 |
Armstrong, DL; Cato, MJ; Gannon, RL; Kelley, KH; Rea, MA | 1 |
Chowdhury, SA; Kawashima, T; Konishi, T; Matsunami, K | 1 |
Chen, Y; Matsuki, N; Saito, H | 1 |
Pierau, FK; Sann, H; Schmid, HA; Yakimova, KS | 1 |
Kar, S; Quirion, R; Seto, D | 1 |
Hashemi, B; Semnanian, S; Shafizadeh, M; Zarrindast, MR | 1 |
El Manira, A; Grillner, S; Tegnér, J | 1 |
Chub, N; O'Donovan, MJ | 1 |
Celis, ME; Cremer, MC; De Barioglio, SR | 1 |
Gong, W; Justice, JB; Neill, DB | 1 |
Carlen, PL; Frantseva, MV; Perez Velazquez, JL | 1 |
Ciriello, J; Roder, S | 1 |
Chavkin, C; Jin, W | 1 |
Kerr, DI; Ong, J; Parnas, I; Rashkovan, G | 1 |
Cairns, BE; Hu, JW; Sessle, BJ | 1 |
Klejbor, I; Trojniar, W | 1 |
Dun, NJ; Hwang, BH; Mizoguchi, H; Nagase, H; Narita, M; Oji, DE; Tseng, LF | 1 |
Bonanno, G; Marcoli, M; Maura, G; Raiteri, M; Scarrone, S | 1 |
Ozdem, SS; Sadan, G; Taşatargil, A; Usta, C | 1 |
Hood, SC; Schwartz, NB | 1 |
Gotoh, S; Miwa, N; Nakayama, H; Suzuki, J; Terao, K | 1 |
Hartings, JA; Simons, DJ | 1 |
Elshourbagy, NA; Gager, TL; Hirst, WD; Jenkins, O; Minton, J; Murkitt, KL; Pangalos, M; Price, GW; Punia, PK; Rice, SQ; Shabon, U; Stammers, M; Taylor, SJ; Testa, T; Wood, MD | 1 |
Fendt, M; Koch, M; Kretschmer, BD | 1 |
Hayashi, Y; Miyakubo, H; Nomura, S; Okumura, T; Sakamaki, K; Tanaka, J | 1 |
Chase, MH; Morales, FR; Xi, MC | 1 |
Kerr, DI; Ong, J | 1 |
Shigenaga, Y; Shimada, T; Takemura, M | 1 |
Saleh, MC; Saleh, TM | 1 |
Hayashi, Y; Miyakubo, H; Nomura, M; Tanaka, J | 1 |
Bowles, W; Hargreaves, KM; Richardson, JD; Wurm, C | 1 |
Gietzen, DW; Magrum, LJ; Truong, BG | 1 |
Aguilar, E; González, LC; Pinilla, L; Tena-Sempere, M | 1 |
Chowdhury, SA; Matsunami, KI | 1 |
Hoffman, CS; Johnson, PL; Miner, HM; Renner, KJ; Summers, CH; Westin, TM | 1 |
Kawakami, A; Mashiko, N; Nomura, M; Tanaka, J; Ushigome, A | 1 |
Horie, S; Ishihara, S; Minowa, S; Murayama, T; Tsuchiya, S; Watanabe, K | 1 |
Nomura, M; Tanaka, J; Ushigome, A | 1 |
Cummings, RT; Grant, SK; Sklar, JG | 1 |
An, SJ; Hwang, IK; Kang, TC; Park, SK; Won, MH | 1 |
Gasior, M; Kaminski, R; Witkin, JM | 1 |
Enna, SJ | 1 |
Escher, T; Mittleman, G | 1 |
Nomura, M; Sakamaki, K; Tanaka, J; Yamato, K | 1 |
Fink, DJ; Glorioso, JC; Hao, S; Huang, S; Liu, J; Mata, M; Wolfe, D | 1 |
An, SJ; Choi, SY; Hwang, IK; Jeong, YG; Jung, JY; Kang, TC; Kim, DW; Kwon, OS; Park, SK; Won, MH | 1 |
Bradley, PM; Burns, BD; Gowland, CJ; Webb, AC | 1 |
He, S; Huang, J; Li, L; Wu, X | 1 |
Przekop, F; Tomaszewska-Zaremba, D | 1 |
Choi, SY; Jung, JY; Kang, TC; Kim, DS; Kim, JE; Kwak, SE; Kwon, OS; Won, MH | 1 |
Choi, KB; Jeong, JH; Moon, NJ; Park, ES; Sohn, UD | 1 |
Huang, J; Li, L; Wu, X; Yeomans, J | 1 |
Cremers, TI; Rea, K; Westerink, BH | 1 |
Bonte, JP; Foulon, C; Goossens, JF; Lipka, E; Vaccher, C; Vaccher, MP | 1 |
Iwa, M; Nakade, Y; Pappas, TN; Takahashi, T | 1 |
Chen, JS; Huang, CY; Lee, SD; Lo, MJ; Ting, H; Yang, AL | 1 |
Fuchs, PN; LaGraize, SC | 1 |
Balcar, VJ; Griffin, JL; Nasrallah, FA; Rae, C | 1 |
Chiappinelli, VA; Guo, JZ; Liu, YB | 1 |
Waraczynski, M | 1 |
Dubrovina, NI; Zinov'ev, DR | 1 |
Billings, HJ; Bogusz, AL; Connors, JM; Coolen, LM; Goodman, RL; Hardy, SL; Hileman, SM; Lehman, MN; McManus, CJ; Nestor, CC; Singh, SR; Sliwowska, JH; Valent, M | 1 |
Álvarez-Buylla, R; Cadenas, JL; de Álvarez-Buylla, ER; Lara, JJ; Lemus, M; Montero, S; Tejeda-Chávez, HR | 1 |
Yamada, T; Yamaguchi, K | 1 |
Franci, CR; Marques de Souza, L | 1 |
Adams, DJ; Berecki, G; Callaghan, B; Clark, RJ; Craik, DJ; Haythornthwaite, A | 1 |
Marazioti, A; Spyraki, C; Thermos, K | 1 |
Bowser, DN; Gibbs, ME | 1 |
Hasanein, P; Keshavarz, S; Moghaddam, AH; Rezvani, ME; Roohbakhsh, A | 1 |
Alves, N; Bosch, D; Daros, A; Schmid, S; Ure, RJ; Yeomans, JS | 1 |
Prado, WA; Silva, JR; Silva, ML | 1 |
Debold, JF; Kwa, C; Miczek, KA; Takahashi, A | 1 |
Jurkowlaniec, E; Kuśmierczak, M; Orzeł-Gryglewska, J | 1 |
Bianchini, P; Diaspro, A; Fato, M; Ferrando, S; Gallus, L; Ledda, FD; Manconi, R; Ramoino, P; Tagliafierro, G | 1 |
Chen, SH; Li, SF; Lin, CT; Lue, JH; Tsai, YJ; Wang, HY | 1 |
Al-Qahtani, MH; Ansari, SA; Bibi, F; Karim, S; Kim, MO; Naseer, MI; Ullah, I; Ullah, N | 1 |
Bolton, MM; Heaney, CF; Kinney, JW; Magcalas, CM; Murtishaw, AS; Sabbagh, JJ | 2 |
Artola, A; Dallel, R; Jacquot, F; Melin, C | 1 |
Cui, N; Jiang, C; Jin, X; Jin, XT; Zhong, W | 1 |
Choi, MG; Jung, JS; Kang, YJ; Kim, CH; Kim, SJ; Kim, SS; Park, SH; Ryu, OH; Sim, YB; Suh, HW | 1 |
Bailey, CP; Dewey, WL; Gabra, BH; Henderson, G; Hull, LC | 1 |
Acquas, E; Cotti, E; Kasture, SB; Muggironi, G; Peana, AT; Rosas, M; Spina, L | 1 |
Fais, RS; Prado, WA; Reis, GM | 1 |
Khanegheini, A; Nasehi, M; Zarrindast, MR | 1 |
Hatam, M; Nasimi, A; Rasoulpanah, M | 1 |
Akbarabadi, A; Bakhtazad, A; Farahmandfar, M; Zarrindast, MR | 1 |
Dias, QM; Prado, WA | 1 |
Nomura, M; Takahashi, M; Tanaka, J | 1 |
Ågmo, A; Dominguez, G; Gómora-Arrati, P | 1 |
Johnston, GAR | 1 |
Takahashi, M; Tanaka, J | 1 |
Alaghmandan-Motlagh, N; Ebrahimi-Ghiri, M; Nami, M; Nasehi, M; Zarrindast, MR | 1 |
Farrahizadeh, M; Nasehi, M; Zarrabian, S; Zarrindast, MR | 1 |
de Melo, JR; de Paula, BB; Leite-Panissi, CRA | 1 |
Khakpoor, M; Mohammadi-Mahdiabadi-Hasani, MH; Nasehi, M; Vaseghi, S | 1 |
4 review(s) available for phaclofen and baclofen
Article | Year |
---|---|
GABAB receptors and phaclofen.
Topics: Baclofen; Humans; Receptors, GABA-A | 1989 |
Recent advances in GABAB receptors: from pharmacology to molecular biology.
Topics: Animals; Baclofen; Cloning, Molecular; GABA Agonists; GABA Antagonists; Potassium Channels; Receptors, GABA-B | 2000 |
A GABA(B) mystery: the search for pharmacologically distinct GABA(B) receptors.
Topics: Acetates; Amines; Animals; Anticonvulsants; Baclofen; Benzylamines; Cyclohexanecarboxylic Acids; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Molecular Structure; Morpholines; Phosphinic Acids; Protein Isoforms; Receptors, GABA-B; RNA, Messenger | 2001 |
GABA Australis, some reflections on the history of GABA receptor research in Australia.
Topics: Animals; Australia; Baclofen; Bicuculline; Cyclic AMP; Humans; Isoxazoles; Muscimol; Receptors, GABA | 2017 |
237 other study(ies) available for phaclofen and baclofen
Article | Year |
---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Effect of the GABAB antagonist, phaclofen, on baclofen-induced inhibition of micturition reflex in urethane-anesthetized rats.
Topics: Animals; Baclofen; Capsaicin; Cerebral Ventricles; Fenclonine; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Reflex; Urethane; Urinary Bladder; Urination | 1992 |
Functionally distinct subpopulations of striatal neurons are differentially regulated by GABAergic and dopaminergic inputs--I. In vivo analysis.
Topics: Animals; Baclofen; Benzazepines; Bicuculline; Corpus Striatum; Dopamine; Electric Stimulation; Electrophysiology; gamma-Aminobutyric Acid; Male; Neural Pathways; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Sulpiride; Sympathectomy, Chemical | 1992 |
GABA receptors in Deiters nucleus modulate posturokinetic responses to cortical stimulation in the cat.
Topics: Animals; Baclofen; Bicuculline; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Extremities; Male; Microinjections; Motor Cortex; Muscimol; Posture; Receptors, GABA-A; Vestibular Nucleus, Lateral | 1992 |
Effectiveness of GABAB antagonists in inhibiting baclofen-induced reductions in cytosolic free Ca concentration in isolated melanotrophs of rat.
Topics: Animals; Baclofen; Calcium; Cytosol; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Organophosphorus Compounds; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains | 1992 |
Activation of GABA B receptors in the anterior pituitary inhibits prolactin and luteinizing hormone secretion.
Topics: Animals; Baclofen; Butylamines; Cells, Cultured; Female; GABA Antagonists; Gonadotropin-Releasing Hormone; Lactation; Luteinizing Hormone; Organophosphorus Compounds; Pituitary Gland, Anterior; Proestrus; Prolactin; Propylamines; Rats; Receptors, GABA-A; Thyrotropin-Releasing Hormone | 1992 |
Changes in gamma-aminobutyric acid release induced by topical administration of drugs affecting its metabolism and receptors: studies in freely moving guinea pigs with epidural cups.
Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Baclofen; beta-Alanine; Calcium; Cerebral Cortex; Epidural Space; Ethanolamines; Feedback; Female; gamma-Aminobutyric Acid; Guinea Pigs; Kinetics; Male; Nipecotic Acids; Norepinephrine; Receptors, GABA-A; Sodium; Tetrodotoxin | 1992 |
Receptor subtypes involved in callosally-induced postsynaptic potentials in rat frontal agranular cortex in vitro.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Corpus Callosum; Electric Stimulation; Evoked Potentials; Frontal Lobe; GABA Antagonists; In Vitro Techniques; Male; Picrotoxin; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Synapses | 1992 |
Functional evidence for multiple gamma-aminobutyric acidB receptor subtypes in the rat cerebral cortex.
Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Male; Organophosphorus Compounds; Peptides; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
Cross-talk between excitatory and inhibitory amino acids in the regulation of luteinizing hormone-releasing hormone secretion.
Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Bicuculline; Drug Interactions; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Gonadotropin-Releasing Hormone; In Vitro Techniques; Male; Median Eminence; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
Pharmacologically distinct GABAB receptor subtypes modulate neurotransmitter release in the rat brain cortex.
Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; GABA-A Receptor Antagonists; Glutamates; Glutamic Acid; Muscimol; Neurotransmitter Agents; Organophosphorus Compounds; Rats; Receptors, GABA-A; Somatostatin; Synaptosomes | 1992 |
GABAergic synaptic transmission in projections from the basal forebrain and hippocampal formation to the amygdala: an in vivo iontophoretic study.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Electric Stimulation; gamma-Aminobutyric Acid; Hippocampus; Iontophoresis; Male; Neural Pathways; Prosencephalon; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Neurotransmitter; Synapses; Synaptic Transmission | 1992 |
Dissociation of mu and delta opioid receptor-mediated reductions in evoked and spontaneous synaptic inhibition in the rat hippocampus in vitro.
Topics: 2-Amino-5-phosphonovalerate; Analgesics; Animals; Axons; Baclofen; Bicuculline; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Evoked Potentials; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Neurons; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Synapses | 1992 |
[Effect of GABA antagonists on the rat electroretinogram].
Topics: Animals; Baclofen; Bicuculline; Electroretinography; GABA Antagonists; Male; Rats; Rats, Inbred Strains; Retina | 1992 |
Phaclofen-sensitive GABA-B receptors do not mediate excitatory effects of baclofen on gastric secretion.
Topics: Animals; Baclofen; Gastric Fundus; Gastric Juice; Injections, Intravenous; Injections, Intraventricular; Male; Pylorus; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Ethanol-induced changes in chloride flux are mediated by both GABA(A) and GABA(B) receptors.
Topics: Alcohol Drinking; Animals; Baclofen; Bicuculline; Cerebral Cortex; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Drug Synergism; Ethanol; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Receptors, GABA-A | 1991 |
CGP 35348, a new GABAB antagonist, prevents antinociception and muscle-relaxant effect induced by baclofen.
Topics: Analgesics; Animals; Baclofen; GABA Antagonists; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Mice; Morphine; Muscle Relaxation; Muscles; Organophosphorus Compounds; Oxotremorine; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time | 1991 |
Effects of GABA and related agents on the electrical activity of hypothalamic ventromedial nucleus neurons in vitro.
Topics: Animals; Baclofen; Bicuculline; Electrophysiology; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Neurons; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ventromedial Hypothalamic Nucleus | 1991 |
Effects of phaclofen and the enantiomers of baclofen on cardiovascular responses to intrathecal administration of L- and D-baclofen in the rat.
Topics: Animals; Baclofen; Blood Pressure; Cardiovascular System; Drug Interactions; GABA-A Receptor Antagonists; Heart Rate; Injections, Spinal; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Time Factors | 1991 |
Phaclofen-reversible effects of GABA in the spinal cord of the rat.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heart Rate; Injections, Spinal; Lidocaine; Male; Rats; Rats, Inbred Strains; Spinal Cord; Stereoisomerism; Sympathetic Nervous System | 1991 |
Blockade of GABAA receptors in the region of the anterior basolateral amygdala of rats elicits increases in heart rate and blood pressure.
Topics: Amygdala; Analysis of Variance; Anesthesia, General; Animals; Baclofen; Bicuculline; Blood Pressure; Consciousness; Dose-Response Relationship, Drug; Electroencephalography; Heart Rate; Hippocampus; Male; Microinjections; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Strychnine; Temporal Lobe | 1991 |
Inhibition of protein kinase activity enhances long-term potentiation of hippocampal IPSPs.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Acetates; Acetic Acid; Animals; Baclofen; Carbazoles; Evoked Potentials; Guinea Pigs; Hippocampus; In Vitro Techniques; Indole Alkaloids; Neurons; Picrotoxin; Potentiometry; Protein Kinase C; Pyramidal Tracts; Quinoxalines; Sesterterpenes | 1991 |
Gamma-aminobutyric acid (GABAB) receptor-mediated inhibition of tyrosine hydroxylase activity in the striatum of rat.
Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Baclofen; Calcium; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; gamma-Aminobutyric Acid; Hydrazines; In Vitro Techniques; Male; Muscimol; Neural Pathways; Picrotoxin; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Tyrosine 3-Monooxygenase | 1991 |
Postsynaptic potentials mediated by excitatory and inhibitory amino acids in interneurons of stratum pyramidale of the CA1 region of rat hippocampal slices in vitro.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Amino Acids; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Interneurons; Male; Membrane Potentials; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Synapses | 1991 |
GABAB receptor modulation of the release of substance P from capsaicin-sensitive neurones in the rat trachea in vitro.
Topics: Animals; Baclofen; Bicuculline; Capsaicin; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Neurons; Potassium; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substance P; Taurine; Trachea | 1991 |
Regulation of cardiovascular sympathetic neurons by substance P and gamma-aminobutyric acid in the rat spinal cord.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Capsaicin; Cardiovascular Physiological Phenomena; Cardiovascular System; Catecholamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Heart Rate; Injections, Spinal; Male; Muscimol; Neurons; Neuropeptide Y; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Substance P; Sympathetic Nervous System | 1991 |
GABAB-receptor-mediated inhibition of the N-methyl-D-aspartate component of synaptic transmission in the rat hippocampus.
Topics: Animals; Baclofen; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Picrotoxin; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission | 1991 |
Effects of baclofen and bicuculline on inhibition in the fascia dentata and hippocampus regio superior.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; Hippocampus; Interneurons; Iontophoresis; Male; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synapses | 1991 |
Antagonism of baclofen-induced antinociception by intrathecal administration of phaclofen or 2-hydroxy-saclofen, but not delta-aminovaleric acid in the rat.
Topics: Amino Acids; Amino Acids, Neutral; Analgesia; Animals; Baclofen; Injections, Spinal; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Effect of intracerebroventricular administration of the GABAB-receptor agonist baclofen on operant feeding in satiated pigs.
Topics: Animals; Baclofen; Central Nervous System; Conditioning, Operant; Drinking Behavior; Feeding Behavior; Female; Injections, Intraventricular; Male; Receptors, GABA-A; Satiation; Swine | 1990 |
Electrophysiological characterization of potent agonists and antagonists at pre- and postsynaptic GABAB receptors on neurones in rat brain slices.
Topics: Animals; Baclofen; Bicuculline; Brain; Corpus Striatum; Electrophysiology; GABA-A Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Neurons; Organophosphorus Compounds; Rats; Receptors, GABA-A; Substantia Nigra; Synapses | 1990 |
The effect of intracerebroventricular administration of baclofen on food intake in rats.
Topics: Animals; Ataxia; Baclofen; Brain; Dose-Response Relationship, Drug; Eating; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
GABAA and GABAB antagonists prevent the opioid inhibition of endogenous acetylcholine release evoked by glutamate from rat neostriatal slices.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; GABA Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Morphine; Narcotics; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Spinal 5-HT3 receptor-mediated antinociception: possible release of GABA.
Topics: Analgesia; Animals; Baclofen; Behavior, Animal; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; N-Methylaspartate; Neurons; Nociceptors; Pain Measurement; Picrotoxin; Receptors, Serotonin; Serotonin; Spinal Cord | 1991 |
Actions of baclofen and phaclofen upon ON- and OFF-ganglion cells in the cat retina.
Topics: Animals; Baclofen; Bicuculline; Cats; Iontophoresis; Microelectrodes; Muscimol; Retinal Ganglion Cells | 1990 |
Enhancement of NMDA receptor-mediated synaptic potential evoked in rat medial-amygdala neuron following olfactory bulbectomy.
Topics: Action Potentials; Amygdala; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; In Vitro Techniques; Kynurenic Acid; Male; Membrane Potentials; Neurons; Olfactory Bulb; Organophosphorus Compounds; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Synapses | 1990 |
GABA terminal autoreceptors in the pars compacta and in the pars reticulata of the rat substantia nigra are GABAB.
Topics: Animals; Anticonvulsants; Baclofen; gamma-Aminobutyric Acid; Male; Muscimol; Nipecotic Acids; Potassium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Synaptosomes; Tritium | 1990 |
Central GABAA excitatory and GABAB inhibitory receptors regulate gastric acid secretion in rats.
Topics: Anesthesia; Animals; Baclofen; Bicuculline; Central Nervous System; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Gastric Acid; Injections, Intraventricular; Male; Muscimol; Pylorus; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Phaclofen-insensitive presynaptic inhibitory action of (+/-)-baclofen in neonatal rat motoneurones in vitro.
Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Evoked Potentials; Glutamates; In Vitro Techniques; Membrane Potentials; Motor Neurons; Nipecotic Acids; Potassium Channels; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereotyped Behavior; Synapses | 1990 |
Thioether analogues of baclofen, phaclofen and saclofen.
Topics: Animals; Baclofen; Binding, Competitive; Cerebellum; Guinea Pigs; Ileum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vas Deferens | 1990 |
(+)-Hydrastine, a potent competitive antagonist at mammalian GABAA receptors.
Topics: Acetylcholine; Alkaloids; Animals; Baclofen; Benzylisoquinolines; Bicuculline; Binding, Competitive; Brain Chemistry; Convulsants; Diazepam; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Membranes; Muscimol; Muscle, Smooth; Muscle, Smooth, Vascular; Rats; Receptors, GABA-A; Stereoisomerism | 1990 |
Inhibition of baclofen binding to rat cerebellar membranes by phaclofen, saclofen, 3-aminopropylphosphonic acid and related GABAB receptor antagonists.
Topics: Animals; Baclofen; Cerebellum; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Propylamines; Rats; Rats, Inbred Strains | 1990 |
Gamma-aminobutyric acid-A and -B receptor antagonists increase luteinizing hormone-releasing hormone neuronal responsiveness to intracerebroventricular norepinephrine in ovariectomized estrogen-treated rats.
Topics: Animals; Baclofen; Bicuculline; Estradiol; Female; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Hypothalamus; Kinetics; Luteinizing Hormone; Neurons; Norepinephrine; Ovariectomy; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Paired-pulse depression of monosynaptic GABA-mediated inhibitory postsynaptic responses in rat hippocampus.
Topics: Action Potentials; Animals; Baclofen; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Picrotoxin; Rats; Synapses; Synaptic Transmission; Tetrodotoxin | 1990 |
Are GABAB receptors involved in the pharmacological effects of ethanol?
Topics: Animals; Baclofen; Cells, Cultured; Chlorine; Diazepam; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; N-Methylaspartate; Picrotoxin; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Spinal Cord | 1990 |
The effects of baclofen and two GABAB-receptor antagonists on long-term potentiation.
Topics: Animals; Baclofen; Electric Stimulation; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Male; Neurons; Organophosphorus Compounds; Rats; Rats, Inbred Strains; Synapses | 1990 |
Phaclofen antagonizes the antinociceptive but not the sedative effects of (-)-baclofen.
Topics: Analgesics; Animals; Baclofen; Behavior, Animal; Electrocardiography; Hypnotics and Sedatives; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscle Relaxants, Central; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Stereoisomerism | 1990 |
Involvement of GABA receptors in the regulation of neurite growth in cultured embryonic chick tectum.
Topics: Animals; Axons; Baclofen; Cells, Cultured; Chick Embryo; Culture Media; gamma-Aminobutyric Acid; Isoxazoles; Ligands; Muscimol; Receptors, GABA-A; Superior Colliculi | 1990 |
Endogenous GABA acts on GABAB receptors in nucleus tractus solitarius to increase blood pressure.
Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Medulla Oblongata; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vigabatrin | 1990 |
Effect of 2-hydroxy-saclofen, an antagonist of GABAB action, upon the binding of baclofen and other receptor ligands in rat cerebrum.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Baclofen; Brain; GABA Antagonists; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
CGP 35348: a centrally active blocker of GABAB receptors.
Topics: Adenylyl Cyclase Inhibitors; Animals; Animals, Newborn; Anticonvulsants; Baclofen; Behavior, Animal; Brain Chemistry; Cyclic AMP; Electrophysiology; Hippocampus; In Vitro Techniques; Iontophoresis; Organophosphorus Compounds; Postural Balance; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord | 1990 |
GABA(B)-related activity involved in synaptic processing of somatosensory information in S1 cortex of the anaesthetized cat.
Topics: Anesthesia; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrodes; Female; gamma-Aminobutyric Acid; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Physical Stimulation; Somatosensory Cortex; Synapses | 1990 |
Endogenous GABA mediates presynaptic inhibition of spontaneous and evoked excitatory synaptic potentials in the rat neostriatum.
Topics: Animals; Baclofen; Corpus Striatum; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Synapses; Tetrodotoxin | 1990 |
Bicuculline and picrotoxin block phase advances induced by GABA agonists in the circadian rhythm of locomotor activity in the golden hamster by a phaclofen-insensitive mechanism.
Topics: Animals; Baclofen; Bicuculline; Circadian Rhythm; Cricetinae; gamma-Aminobutyric Acid; Male; Mesocricetus; Microinjections; Motor Activity; Muscimol; Picrotoxin; Stereotaxic Techniques; Triazolam | 1990 |
Epileptiform activity in microcultures containing small numbers of hippocampal neurons.
Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Cells, Cultured; Epilepsy; Evoked Potentials; Hippocampus; Kynurenic Acid; Neurons; Rats; Synapses | 1990 |
Effects of excitatory and inhibitory amino acid agonists and antagonists of ventral horn cells in slices of spinal cord isolated from adult rats.
Topics: Action Potentials; Amino Acids; Animals; Anterior Horn Cells; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Strychnine; Synapses | 1990 |
Effects of GABA antagonists and structural GABA analogues on baclofen stimulated gastric acid secretion in the rat.
Topics: Amino Acids; Anesthesia; Animals; Baclofen; Bethanechol Compounds; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Gastric Acid; Male; Rats; Rats, Inbred Strains | 1990 |
Phaclofen antagonizes post-tetanic disinhibition in the rat dentate gyrus.
Topics: Animals; Baclofen; Electric Stimulation; Hippocampus; In Vitro Techniques; Male; Neural Inhibition; Rats; Rats, Inbred Strains | 1990 |
On the presynaptic action of baclofen at inhibitory synapses between cultured rat hippocampal neurones.
Topics: Action Potentials; Animals; Baclofen; Calcium; Cells, Cultured; gamma-Aminobutyric Acid; Hippocampus; Neurons; Pertussis Toxin; Rats; Synapses; Virulence Factors, Bordetella | 1990 |
Phaclofen inhibition of the slow inhibitory postsynaptic potential in hippocampal slice cultures: a possible role for the GABAB-mediated inhibitory postsynaptic potential.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neural Inhibition; Organ Culture Techniques; Rats | 1990 |
GABAB-receptor-mediated actions of baclofen in rat isolated neocortical slice preparations: antagonism by phosphono-analogues of GABA.
Topics: Animals; Baclofen; Cerebral Cortex; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Propylamines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
GABAB autoreceptors in rat cortex synaptosomes: response under different depolarizing and ionic conditions.
Topics: Animals; Baclofen; Calcium; Cerebral Cortex; In Vitro Techniques; Male; Muscimol; Neuromuscular Depolarizing Agents; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes; Veratrine | 1989 |
Inhibitory processes in normal and epileptic-like rat hippocampal slices: the role of GABAB receptors.
Topics: Animals; Baclofen; Bicuculline; Epilepsy; Hippocampus; In Vitro Techniques; Male; Penicillins; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
GABAB receptor mediated effects on central respiratory system and their antagonism by phaclofen.
Topics: Animals; Baclofen; Phrenic Nerve; Rabbits; Receptors, GABA-A; Reference Values; Respiration; Vagotomy | 1989 |
3-Aminopropylphosphinic acid--a potent, selective GABAB receptor agonist in the guinea-pig ileum and rat anococcygeus muscle.
Topics: Animals; Baclofen; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscles; Organophosphorus Compounds; Parasympathetic Nervous System; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Stimulation by phaclofen of inositol 1,4,5-triphosphate production in cultured neurons from chick tectum.
Topics: Animals; Baclofen; Chick Embryo; gamma-Aminobutyric Acid; Inosine Nucleotides; Inosine Triphosphate; Isoxazoles; Neurons; Receptors, GABA-A; Superior Colliculi | 1989 |
Effects of the putative antagonists phaclofen and delta-aminovaleric acid on GABAB receptor biochemistry.
Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Cerebral Cortex; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Kinetics; Male; Proteins; Radioligand Assay; Rats; Receptors, GABA-A | 1989 |
A new alcohol antagonist: phaclofen.
Topics: Animals; Baclofen; Behavior, Animal; Body Temperature; Ethanol; GABA-A Receptor Antagonists; Male; Mice; Mice, Inbred ICR; Motor Activity; Receptors, GABA-A; Sleep | 1989 |
A novel type of GABA receptor in rat spinal cord?
Topics: Animals; Baclofen; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Synaptosomes | 1989 |
Late inhibitory postsynaptic potentials in rat prefrontal cortex may be mediated by GABAB receptors.
Topics: Animals; Baclofen; Electric Conductivity; Electric Stimulation; Evoked Potentials; Frontal Lobe; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Isoxazoles; Male; Membrane Potentials; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synapses | 1989 |
Bicuculline- and phaclofen-sensitive components of N-methyl-D-aspartate-induced hyperpolarizations in rat dorsolateral septal nucleus neurones.
Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Baclofen; Bicuculline; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Membrane Potentials; N-Methylaspartate; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Septal Nuclei; Tetrodotoxin | 1989 |
Control of epileptiform burst rate by CA3 hippocampal cell afterhyperpolarizations in vitro.
Topics: Action Potentials; Animals; Baclofen; Epilepsy; Hippocampus; In Vitro Techniques; Membrane Potentials; Phorbol Esters; Potassium; Rats | 1989 |
Rhythmical bursting activity and GABAergic mechanisms in the medial septum of normal and pertussis toxin-pretreated rats.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Hippocampus; Male; Neurons; Nipecotic Acids; Pertussis Toxin; Proline; Rats; Rats, Inbred Strains; Septum Pellucidum; Virulence Factors, Bordetella | 1989 |
Baclofen and phaclofen modulate GABA release from slices of rat cerebral cortex and spinal cord but not from retina.
Topics: Amino Acids; Aminocaproates; Aminolevulinic Acid; Animals; Baclofen; Calcium; Cerebral Cortex; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Potassium; Rats; Rats, Inbred Strains; Retina; Spinal Cord; Vigabatrin | 1989 |
Phaclofen antagonizes the depressant effect of baclofen on spinal reflex transmission in rats.
Topics: Animals; Baclofen; H-Reflex; Male; Neural Inhibition; Rats; Rats, Inbred Strains; Reflex, Monosynaptic; Spinal Cord | 1989 |
A physiological role for GABAB receptors in the central nervous system.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Potassium; Rats; Receptors, GABA-A; Serotonin; Synapses | 1988 |
The GABAB antagonist phaclofen inhibits the late K+-dependent IPSP in cat and rat thalamic and hippocampal neurones.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Geniculate Bodies; Hippocampus; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Phaclofen: a GABAB blocker reduces long-duration inhibition in the neocortex.
Topics: Animals; Baclofen; Cerebral Cortex; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
GABAA and GABAB receptors in locus coeruleus: effects of blockers.
Topics: Animals; Baclofen; In Vitro Techniques; Locus Coeruleus; Male; Muscimol; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Phaclofen antagonizes baclofen-induced suppression of visually evoked responses in the cat's striate cortex.
Topics: Animals; Baclofen; Cats; Evoked Potentials, Visual; gamma-Aminobutyric Acid; Receptors, GABA-A; Visual Cortex | 1988 |
Evidence for pharmacologically distinct subsets of GABAB receptors.
Topics: Animals; Baclofen; Binding, Competitive; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Propylamines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Phaclofen antagonizes GABA at autoreceptors regulating release in rat cerebral cortex.
Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; GABA Antagonists; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1988 |
Phaclofen: a peripheral and central baclofen antagonist.
Topics: Animals; Baclofen; Cats; Cholinergic Fibers; Colon; Guinea Pigs; Ileum; In Vitro Techniques; Interneurons; Intestines; Receptors, GABA-A; Spinal Cord; Synaptic Transmission | 1987 |
Intracerebroventricular phaclofen antagonizes baclofen antinociceptive activity in hot plate test with mice.
Topics: Analgesics; Animals; Baclofen; Injections, Intraventricular; Male; Mice; Reaction Time; Time Factors | 1988 |
Comparison of antagonism by phaclofen of baclofen induced hyperpolarizations and synaptically mediated late hyperpolarizing potentials recorded intracellularly from rat dorsolateral septal neurons.
Topics: Animals; Baclofen; In Vitro Techniques; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Septal Nuclei | 1988 |
Long-term synaptic transformation of hippocampal CA1 gamma-aminobutyric acid synapses and the effect of anandamide.
Topics: Animals; Arachidonic Acids; Baclofen; Calcium Channel Blockers; Chloride Channels; Endocannabinoids; Furosemide; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Models, Neurological; Polyunsaturated Alkamides; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Snails; Synapses; Synaptic Transmission | 1995 |
Bicuculline enhances the late GABAB receptor-mediated paired-pulse inhibition observed in rat hippocampal slices.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Electric Stimulation; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Neurons; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B | 1995 |
Regulation of the prefrontal cortical dopamine release by GABAA and GABAB receptor agonists and antagonists.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Microdialysis; Muscimol; Nomifensine; Picrotoxin; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B | 1993 |
Characterization of GABAB ligands in vivo.
Topics: Animals; Baclofen; beta-Alanine; Drug Interactions; Female; GABA Antagonists; GABA-B Receptor Antagonists; Ligands; Mice; Mice, Inbred BALB C; Muscle Relaxation; Organophosphorus Compounds | 1995 |
A depolarizing inhibitory response to GABA in brainstem auditory neurons of the chick.
Topics: Animals; Baclofen; Basal Ganglia; Bicuculline; Brain Stem; Chickens; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Neuromuscular Depolarizing Agents; Neurons, Afferent; Patch-Clamp Techniques | 1995 |
GABAA receptor-mediated inhibition of N-methyl-D-aspartate-evoked [3H]dopamine release from mesencephalic cell cultures.
Topics: Animals; Baclofen; Cells, Cultured; Dopamine; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Kainic Acid; Mesencephalon; Muscimol; N-Methylaspartate; Picrotoxin; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA; Ventral Tegmental Area | 1994 |
2-Hydroxy-saclofen causes a phaclofen-reversible reduction in population spike amplitude in the rat hippocampal slice.
Topics: Animals; Baclofen; Bicuculline; Evoked Potentials; GABA Antagonists; Hippocampus; Male; Microelectrodes; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B; Synaptic Transmission | 1995 |
Presynaptic gamma-hydroxybutyric acid (GHB) and gamma-aminobutyric acidB (GABAB) receptor-mediated release of GABA and glutamate (GLU) in rat thalamic ventrobasal nucleus (VB): a possible mechanism for the generation of absence-like seizures induced by GH
Topics: Action Potentials; Animals; Baclofen; Epilepsy, Absence; Extracellular Space; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Organophosphorus Compounds; Potassium; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, GABA-B; Sodium Oxybate; Thalamic Nuclei | 1995 |
Pharmacology of the GABAB receptor in amphibian retina.
Topics: Ambystoma; Animals; Baclofen; Butylamines; Evoked Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Necturus; Organophosphorus Compounds; Propylamines; Receptors, GABA-B; Retina; Retinal Ganglion Cells; Stereoisomerism; Structure-Activity Relationship | 1994 |
Characterization of the GABA autoreceptor in human neocortex as a pharmacological subtype of the GABAB receptor.
Topics: Adolescent; Adult; Aged; Animals; Baclofen; Benzylamines; Binding, Competitive; Brain Neoplasms; Cerebral Cortex; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Humans; Male; Middle Aged; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B | 1994 |
Paired-pulse depression of the N-methyl-D-aspartate receptor-mediated synaptic potentials in the amygdala.
Topics: Amygdala; Animals; Baclofen; In Vitro Techniques; Male; Potassium; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission | 1994 |
The effects of GABAB ligands on alcohol withdrawal in mice.
Topics: Animals; Baclofen; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; GABA-B Receptor Antagonists; Mice; Mice, Inbred C57BL; Organophosphorus Compounds; Phenylalanine; Receptors, GABA-B; Seizures; Substance Withdrawal Syndrome; Tremor | 1994 |
Spatiotemporally differential inhibition of pyramidal cells in the cat motor cortex.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Axons; Baclofen; Bicuculline; Cats; Electric Stimulation; Interneurons; Membrane Potentials; Microelectrodes; Motor Cortex; Pyramidal Cells; Quinoxalines; Synapses | 1994 |
Medial vestibular neurons are endogenous pacemakers whose discharge is modulated by neurotransmitters.
Topics: Amino Acids; Animals; Baclofen; Bicuculline; Calcium; In Vitro Techniques; Kynurenic Acid; Magnesium; Male; Membrane Potentials; Nerve Fibers; Neurons; Neurotransmitter Agents; Rats; Rats, Wistar; Receptors, GABA-A; Synapses; Vestibular Nuclei | 1993 |
Phosphorylation of DARPP-32 is regulated by GABA in rat striatum and substantia nigra.
Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine and cAMP-Regulated Phosphoprotein 32; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra | 1994 |
Pharmacological discrimination between gamma-aminobutyric acid type B receptors regulating cholecystokinin and somatostatin release from rat neocortex synaptosomes.
Topics: Animals; Baclofen; Benzylamines; Cerebral Cortex; Cholecystokinin; GABA Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ligands; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes | 1994 |
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus | 1994 |
Inhibitory mechanisms terminating paroxysmal depolarization shifts in hippocampal neurons of rats.
Topics: Animals; Baclofen; Bicuculline; Calcium; Egtazic Acid; GABA Antagonists; Hippocampus; In Vitro Techniques; Magnesium; Membrane Potentials; Neurons; Penicillins; Potassium Channel Blockers; Potassium Channels; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Tetraethylammonium; Tetraethylammonium Compounds | 1994 |
GABAB antagonists: resolution, absolute stereochemistry, and pharmacology of (R)- and (S)-phaclofen.
Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; Crystallography, X-Ray; GABA Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Models, Molecular; Molecular Conformation; Molecular Structure; Rats; Stereoisomerism; Structure-Activity Relationship | 1994 |
Stimulation of GABAB receptors in the basal forebrain selectively impairs working memory of rats in the double Y-maze.
Topics: Animals; Baclofen; Exploratory Behavior; Male; Memory; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Stereoisomerism; Substantia Innominata | 1994 |
Release of endogenous glutamic and aspartic acids from cerebrocortex synaptosomes and its modulation through activation of a gamma-aminobutyric acidB (GABAB) receptor subtype.
Topics: Animals; Aspartic Acid; Baclofen; Bicuculline; Cerebral Cortex; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Kinetics; Male; Organophosphorus Compounds; Picrotoxin; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptosomes | 1993 |
GABAB autoreceptors mediate activity-dependent disinhibition and enhance signal transmission in the dentate gyrus.
Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Culture Techniques; GABA-A Receptor Antagonists; Hippocampus; Male; Membrane Potentials; Nerve Fibers; Neural Inhibition; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Theta Rhythm | 1993 |
Intrathecal GABAB antagonists attenuate the antinociception produced by microinjection of L-glutamate into the ventromedial medulla of the rat.
Topics: Analgesics; Animals; Baclofen; Basal Ganglia; Behavior, Animal; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glutamates; Glutamic Acid; Injections, Spinal; Medulla Oblongata; Methysergide; Microinjections; Organophosphorus Compounds; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Skin Temperature | 1993 |
GABA mediation of the dual effects of somatostatin on guinea pig ileal myenteric cholinergic transmission.
Topics: Acetylcholine; Adenylate Cyclase Toxin; Animals; Baclofen; Bicuculline; Cholecystokinin; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Pertussis Toxin; Receptors, GABA-A; Somatostatin; Virulence Factors, Bordetella | 1993 |
L-2-amino-4-phosphonobutanoic acid and 1S,3R-1-aminocyclopentane-1,3-dicarboxylic acid reduce paired-pulse depression recorded from medial perforant path in the dentate gyrus of rat hippocampal slices.
Topics: Aminobutyrates; Animals; Atropine; Baclofen; Carbachol; Cycloleucine; Depression, Chemical; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Neural Pathways; Neurotransmitter Uptake Inhibitors; Picrotoxin; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Theophylline | 1993 |
Hyperpolarizing synaptic potentials evoked in CA1 pyramidal cells by glutamate stimulation of interneurons from the oriens/alveus border of rat hippocampal slices. II. Sensitivity to GABA antagonists.
Topics: Animals; Baclofen; Bicuculline; Electrophysiology; Evoked Potentials; GABA Antagonists; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Neurons; Rats; Synapses | 1993 |
Different effects of omega-conotoxin GVIA at excitatory and inhibitory synapses in rat CA1 hippocampal neurons.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Mollusk Venoms; Neurons; omega-Conotoxin GVIA; Peptides; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Synapses | 1993 |
Enteric GABA-containing nerves projecting to the guinea-pig inferior mesenteric ganglion modulate acetylcholine release.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Colon; Diazepam; Electric Stimulation; gamma-Aminobutyric Acid; Ganglia, Sympathetic; Guinea Pigs; In Vitro Techniques; Male; Mesentery; Muscimol; Neural Pathways; Receptors, GABA-A; Receptors, GABA-B; Splanchnic Nerves; Synaptic Transmission | 1993 |
The role of GABA receptors in the control of the omasal myoelectrical activity in sheep.
Topics: Animals; Baclofen; Bicuculline; Female; GABA Antagonists; Muscimol; Myoelectric Complex, Migrating; Omasum; Receptors, GABA; Sheep | 1994 |
The development of GABAB-mediated activity in the rat dentate gyrus.
Topics: Animals; Baclofen; Electric Stimulation; Evoked Potentials; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Organophosphorus Compounds; Rats; Receptors, GABA-A; Receptors, GABA-B | 1994 |
Differential effects of muscimol microinjection into dorsal and ventral aspects of the premotor cortex of monkeys.
Topics: Animals; Appetitive Behavior; Attention; Baclofen; Brain Mapping; Macaca; Male; Membrane Potentials; Microinjections; Motor Cortex; Motor Skills; Muscimol; Neurons; Orientation; Psychomotor Performance; Receptors, GABA-A | 1994 |
Microiontophoresis of baclofen on membrane potential and input resistance in bulbar respiratory neurons in the cat.
Topics: Action Potentials; Animals; Baclofen; Cats; Iontophoresis; Medulla Oblongata; Membrane Potentials; Neurons; Respiratory System; Tetrodotoxin | 1993 |
Evidence that changes in the function of the subtypes of the receptors for gamma-amino butyric acid may be involved in the seasonal changes in the negative-feedback effects of estrogen on gonadotropin-releasing hormone secretion and plasma luteinizing hor
Topics: Animals; Baclofen; Bicuculline; Estrogens; Feedback; Female; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Muscimol; Receptors, GABA; Seasons; Sheep | 1993 |
Electrophysiological identification of horizontal synaptic connections in rat visual cortex in vitro.
Topics: Animals; Baclofen; Calcium; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kynurenic Acid; Magnesium; Quinoxalines; Rats; Receptors, GABA-B; Synapses; Synaptic Transmission; Visual Cortex | 1993 |
GABA induces Ca2+ transients in astrocytes.
Topics: Animals; Astrocytes; Baclofen; Bicuculline; Calcium; Cells, Cultured; Cerebral Cortex; Cytosol; gamma-Aminobutyric Acid; Immunohistochemistry; Muscimol; Nicotinic Acids; Nifedipine; Rats | 1993 |
Influence of GABA on neurons of the gustatory zone of the rat nucleus of the solitary tract.
Topics: Animals; Baclofen; Bicuculline; Brain Mapping; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Male; Medulla Oblongata; Membrane Potentials; Muscimol; Neurons; Perfusion; Rats; Taste; Tetrodotoxin | 1993 |
Analysis of gamma-aminobutyric acidB receptor function in the in vitro and in vivo regulation of alpha-melanotropin-stimulating hormone secretion from melanotrope cells of Xenopus laevis.
Topics: alpha-MSH; Animals; Baclofen; Butylamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Homeostasis; In Vitro Techniques; Kinetics; Organophosphorus Compounds; Perfusion; Pituitary Gland, Posterior; Radioimmunoassay; Receptors, GABA-A; Xenopus laevis | 1993 |
The spinal GABA system modulates burst frequency and intersegmental coordination in the lamprey: differential effects of GABAA and GABAB receptors.
Topics: Animals; Baclofen; Bicuculline; Culture Techniques; Diazepam; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Lampreys; Locomotion; Motor Neurons; Muscimol; Muscles; N-Methylaspartate; Nerve Net; Neurons; Nipecotic Acids; Proline; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Spinal Nerve Roots; Synaptic Transmission | 1993 |
gamma-Aminobutyric acid (GABA) autoreceptors in rat cerebral cortex and spinal cord represent pharmacologically distinct subtypes of the GABAB receptor.
Topics: Animals; Baclofen; Cerebral Cortex; gamma-Aminobutyric Acid; Male; Organophosphorus Compounds; Potassium; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Synaptosomes | 1993 |
GABA receptor subtypes involved in the neuronal mechanisms of baroreceptor reflex in the nucleus tractus solitarii of rabbits.
Topics: Animals; Baclofen; Bicuculline; Brain Stem; Electrophysiology; gamma-Aminobutyric Acid; Male; Neurons; Phenylephrine; Pressoreceptors; Rabbits; Receptors, GABA-A | 1993 |
Pre- and postsynaptic GABAB receptors of rat neocortical neurons differ in their pharmacological properties.
Topics: Animals; Baclofen; Cerebral Cortex; Electric Stimulation; Feedback; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Membrane Potentials; Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses | 1993 |
Inhibitory effects of cholecystokinin on rat's geniculate activity can be blocked by GABA-antagonists.
Topics: Animals; Baclofen; Bicuculline; Cholecystokinin; Extracellular Space; GABA Antagonists; Geniculate Bodies; Interneurons; Iontophoresis; Male; Rats; Rats, Wistar; Trypan Blue | 1995 |
GABA transport and calcium dynamics in horizontal cells from the skate retina.
Topics: Animals; Baclofen; Bicuculline; Biological Transport; Calcium; Calcium Channel Blockers; Dantrolene; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Muscle Relaxants, Central; Nifedipine; Picrotoxin; Retina; Skates, Fish | 1995 |
GABAA receptor-mediated feedback inhibition in pyramidal neurons of cat motor cortex.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Cats; Dendrites; Feedback; Female; GABA Antagonists; Male; Motor Cortex; Neurotransmitter Agents; Patch-Clamp Techniques; Potassium Chloride; Pyramidal Cells; Receptors, GABA-A | 1995 |
Attenuation by valproate of c-fos immunoreactivity in trigeminal nucleus caudalis induced by intracisternal capsaicin.
Topics: Animals; Baclofen; Bicuculline; Brain Stem; Capsaicin; GABA Agents; GABA Antagonists; Guinea Pigs; Injections, Intraventricular; Male; Proto-Oncogene Proteins c-fos; Trigeminal Nuclei; Valproic Acid | 1995 |
Actions of the anticonvulsant agent 2-amino-4-phosphonobutyrate on the release of [3H]D-aspartate from rat forebrain slices.
Topics: Aminobutyrates; Animals; Anticonvulsants; Aspartic Acid; Baclofen; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isomerism; Kynurenic Acid; Prosencephalon; Rats | 1996 |
Effects of GABAergic drugs on physostigmine-induced yawning in rats.
Topics: Animals; Baclofen; Bicuculline; Cholinesterase Inhibitors; Drug Interactions; GABA Agonists; GABA Antagonists; Male; Muscimol; Physostigmine; Picrotoxin; Rats; Rats, Wistar; Yawning | 1995 |
Role of peripheral GABAB receptors in the regulation of pepsinogen secretion in anaesthetized rats.
Topics: Anesthesia; Animals; Baclofen; Capsaicin; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gastric Mucosa; Male; Organophosphorus Compounds; p-Methoxy-N-methylphenethylamine; Pepsinogens; Perfusion; Rats; Rats, Wistar; Receptors, GABA-B; Vagotomy | 1995 |
The vigilance promoting drug modafinil increases dopamine release in the rat nucleus accumbens via the involvement of a local GABAergic mechanism.
Topics: Analysis of Variance; Animals; Baclofen; Benzhydryl Compounds; Central Nervous System Stimulants; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Modafinil; Muscimol; Nipecotic Acids; Nucleus Accumbens; Rats; Rats, Sprague-Dawley | 1996 |
Effects of baclofen and phaclofen on receptive field properties of rat whisker barrel neurons.
Topics: Animals; Baclofen; Extracellular Space; Female; GABA Agonists; GABA Antagonists; Iontophoresis; Mechanoreceptors; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Somatosensory Cortex; Vibrissae | 1996 |
Delayed response deficits induced by local injection of GABA antagonists (bicuculline and phaclofen) into area 46 in infant rhesus monkeys.
Topics: Animals; Baclofen; Cerebral Cortex; Functional Laterality; GABA Antagonists; Hand; Injections; Macaca mulatta; Male; Neural Pathways; Psychomotor Performance | 1996 |
Characterization of subtypes of gamma-aminobutyric acid receptors in an Ascaris muscle preparation by binding assay and binding of PF1022A, a new anthelmintic, on the receptors.
Topics: Animals; Anthelmintics; Ascaris suum; Baclofen; Depsipeptides; Dose-Response Relationship, Drug; GABA Antagonists; Muscles; Peptides, Cyclic; Radioligand Assay; Receptors, GABA; Time Factors | 1996 |
Potentiation by baclofen of gastric acid secretion stimulated by secretagogues in vagotomized rats under anesthesia.
Topics: Anesthesia; Animals; Baclofen; Bethanechol Compounds; Body Temperature; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; GABA Agonists; GABA Antagonists; Gastric Acid; Male; Pentagastrin; Rats; Rats, Wistar; Urethane; Vagotomy; Vagus Nerve | 1996 |
Effects of GABAB receptor antagonists on two models of focal epileptogenesis.
Topics: Animals; Baclofen; Disease Models, Animal; Epilepsies, Partial; GABA Antagonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Rats; Rats, Wistar; Time Factors | 1995 |
Antiabsence seizure activity of specific GABAB and gamma-Hydroxybutyric acid receptor antagonists.
Topics: Animals; Anticonvulsants; Baclofen; Benzocycloheptenes; Electroencephalography; Epilepsy, Absence; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Injections, Intraventricular; Isomerism; Male; Pentylenetetrazole; Rats; Rats, Sprague-Dawley | 1996 |
Mouse cerebellar GABAB participation in the expression of acute ethanol-induced ataxia and in its modulation by the cerebellar adenosinergic A1 system.
Topics: Adenosine; Adenylate Cyclase Toxin; Animals; Ataxia; Baclofen; Behavior, Animal; Cerebellum; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; GTP-Binding Proteins; Male; Mice; Mice, Inbred Strains; Microinjections; Motor Activity; Muscimol; Pertussis Toxin; Receptors, GABA-B; Receptors, Purinergic P1; Virulence Factors, Bordetella | 1996 |
GABAA and GABAB receptors differentially regulate synaptic transmission in the auditory thalamo-amygdala pathway: an in vivo microiontophoretic study and a model.
Topics: Amygdala; Animals; Baclofen; GABA Antagonists; Male; Models, Neurological; Neural Pathways; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamus | 1996 |
Release of taurine and its effects on release of neurotransmitter amino acids in rat cerebral cortex.
Topics: Animals; Aspartic Acid; Baclofen; Bicuculline; Calcium; Cerebral Cortex; Chromatography, High Pressure Liquid; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Kinetics; Male; Membrane Potentials; Potassium Chloride; Rats; Rats, Wistar; Spectrometry, Fluorescence; Synaptosomes; Taurine; Time Factors | 1996 |
Relation of the [3H] gamma-hydroxybutyric acid (GHB) binding site to the gamma-aminobutyric acidB (GABAB) receptor in rat brain.
Topics: Animals; Autoradiography; Baclofen; Benzocycloheptenes; Binding Sites; Brain; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Guanosine Triphosphate; In Vitro Techniques; Male; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Seizures; Sodium Oxybate; Stereoisomerism | 1996 |
GABAergic modulation of optic nerve-evoked field potentials in the rat suprachiasmatic nucleus.
Topics: Animals; Baclofen; Bicuculline; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Optic Nerve; Rats; Rats, Sprague-Dawley; Suprachiasmatic Nucleus | 1995 |
GABAergic characteristics of transcallosal activity of cat motor cortical neurons.
Topics: Animals; Baclofen; Bicuculline; Cats; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Motor Cortex; Organophosphorus Compounds | 1996 |
Ethanol-induced emesis in the house musk shrew, Suncus murinus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaldehyde; Alcohol Deterrents; Animals; Antiemetics; Baclofen; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Disulfiram; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; Indoles; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Subcutaneous; Male; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Tiopronin; Tropisetron; Vagotomy; Vomiting | 1997 |
Specific action of GABAB ligands on the temperature sensitivity of hypothalamic neurons.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Body Temperature Regulation; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hot Temperature; Hypothalamus, Anterior; In Vitro Techniques; Male; Neurons; Preoptic Area; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Thermoreceptors | 1997 |
Evidence for direct and indirect mechanisms in the potent modulatory action of interleukin-2 on the release of acetylcholine in rat hippocampal slices.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; GABA Antagonists; Hippocampus; In Vitro Techniques; Interleukin-2; Male; Rats; Rats, Sprague-Dawley; Receptors, Interleukin-2; Sodium Channel Blockers; Sodium Channels; Tetrodotoxin | 1997 |
Involvement of GABAB receptors in the antinociception induced by baclofen in the formalin test.
Topics: Animals; Baclofen; Bicuculline; Formaldehyde; GABA Agonists; GABA Antagonists; Male; Pain Threshold; Picrotoxin; Rats; Receptors, GABA-B | 1997 |
Locomotor-related presynaptic modulation of primary afferents in the lamprey.
Topics: Afferent Pathways; Animals; Axons; Baclofen; Bicuculline; Functional Laterality; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Lampreys; Locomotion; Membrane Potentials; Motor Activity; N-Methylaspartate; Neurons, Afferent; Receptors, GABA-A; Receptors, GABA-B; Skin; Spinal Cord; Synapses | 1997 |
Blockade and recovery of spontaneous rhythmic activity after application of neurotransmitter antagonists to spinal networks of the chick embryo.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Chick Embryo; Cholinergic Antagonists; Dihydro-beta-Erythroidine; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glycine; Glycine Agents; Mecamylamine; Motor Neurons; Neuronal Plasticity; Neurotransmitter Agents; Nicotinic Antagonists; Periodicity; Spinal Cord; Strychnine | 1998 |
Interaction between alpha-MSH and gabaergic agents upon striatal cAMP levels: an in vitro model.
Topics: alpha-MSH; Animals; Baclofen; Benzazepines; Corpus Striatum; Cyclic AMP; Diazepam; Drug Interactions; Flumazenil; GABA Agents; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Models, Neurological; Rats; Rats, Wistar; Receptors, Dopamine D1 | 1998 |
GABAergic modulation of ventral pallidal dopamine release studied by in vivo microdialysis in the freely moving rat.
Topics: Animals; Baclofen; Cocaine; Dopamine; Dopamine Uptake Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Microdialysis; Picrotoxin; Piperazines; Rats; Rats, Wistar | 1998 |
Changes in membrane and synaptic properties of thalamocortical circuitry caused by hydrogen peroxide.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Free Radicals; GABA Antagonists; Hydrogen Peroxide; Membrane Potentials; Neural Inhibition; Neural Pathways; Oxidants; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, GABA-B; Somatosensory Cortex; Synaptic Transmission; Thalamus | 1998 |
GABAergic effects on the depressor responses elicited by stimulation of central nucleus of the amygdala.
Topics: Amygdala; Animals; Baclofen; Bicuculline; Blood Pressure; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heart Rate; Male; Microinjections; Neurons; Rats; Rats, Wistar | 1999 |
Mu opioids enhance mossy fiber synaptic transmission indirectly by reducing GABAB receptor activation.
Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Antagonists; Long-Term Potentiation; Male; Membrane Potentials; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Somatostatin; Synaptic Transmission | 1999 |
Tonic activation of presynaptic GABAB receptors in the opener neuromuscular junction of crayfish.
Topics: Animals; Astacoidea; Axons; Baclofen; GABA Agonists; GABA Antagonists; Logistic Models; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; Pronase; Quantum Theory; Receptors, GABA-B; Receptors, Presynaptic | 1999 |
Activation of peripheral GABAA receptors inhibits temporomandibular joint-evoked jaw muscle activity.
Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Electromyography; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Masseter Muscle; Motor Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Temporomandibular Joint | 1999 |
Facilitatory effect of unilateral lesion of the ventral tegmental area on locomotor response to stimulation of the contralateral ventral tegmental area: involvement of GABAergic transmission.
Topics: Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Functional Laterality; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Male; Models, Neurological; Motor Activity; Muscimol; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Ventral Tegmental Area | 1999 |
Identification of the G-protein-coupled ORL1 receptor in the mouse spinal cord by [35S]-GTPgammaS binding and immunohistochemistry.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Autoradiography; Baclofen; Binding, Competitive; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Haloperidol; Immunohistochemistry; In Vitro Techniques; Male; Membranes; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Propranolol; Receptors, Opioid; Somatostatin; Spinal Cord; Sulfur Radioisotopes; Yohimbine | 1999 |
A subtype of the gamma-aminobutyric acid(B) receptor regulates cholinergic twitch response in the guinea pig ileum.
Topics: Animals; Baclofen; Binding, Competitive; Electric Stimulation; GABA Agonists; GABA Antagonists; Guinea Pigs; Ileum; In Vitro Techniques; Ligands; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Parasympathetic Nervous System; Receptors, GABA-B; Spinal Cord | 2000 |
Effect of experimental diabetes on GABA-mediated inhibition of neurally induced contractions in rat isolated trachea.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscle Contraction; Rats; Rats, Wistar; Taurine; Tetrodotoxin; Trachea; Vasodilator Agents | 2000 |
Sex difference in serum luteinizing hormone postgonadectomy in the rat: role of gamma-aminobutyric acid-ergic inhibition.
Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Enzyme Inhibitors; Female; GABA Agents; GABA Antagonists; Kinetics; Luteinizing Hormone; Male; Orchiectomy; Ovariectomy; Rats; Sex Characteristics; Transaminases | 2000 |
Autoimmune hemolytic anemia (AIHA) in an infant rhesus macaque (Macaca mulatta).
Topics: Anemia, Hemolytic, Autoimmune; Animals; Baclofen; Benzazepines; Bicuculline; Bromocriptine; Drug Therapy, Combination; Lymphocyte Subsets; Macaca mulatta; Primate Diseases; Spleen | 2000 |
Inhibition suppresses transmission of tonic vibrissa-evoked activity in the rat ventrobasal thalamus.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Intralaminar Thalamic Nuclei; Iontophoresis; Neural Inhibition; Neurons; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamus; Vibrissae | 2000 |
The human GABA(B1b) and GABA(B2) heterodimeric recombinant receptor shows low sensitivity to phaclofen and saclofen.
Topics: Animals; Baclofen; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Receptors, GABA; Receptors, GABA-B | 2000 |
Role of the substantia nigra pars reticulata in sensorimotor gating, measured by prepulse inhibition of startle in rats.
Topics: 2-Amino-5-phosphonovalerate; Acoustic Stimulation; Animals; Baclofen; Central Nervous System Stimulants; Dextroamphetamine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Exploratory Behavior; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Male; Neostriatum; Picrotoxin; Proactive Inhibition; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Stereotyped Behavior; Substantia Nigra | 2000 |
GABAergic modulation of neurons in the nucleus of the solitary tract with ascending projections to the subfornical organ in the rat.
Topics: Animals; Baclofen; Bicuculline; Electric Stimulation; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Male; Neural Pathways; Neurons; Pressoreceptors; Rats; Rats, Wistar; Solitary Nucleus; Subfornical Organ | 2001 |
Induction of wakefulness and inhibition of active (REM) sleep by GABAergic processes in the nucleus pontis oralis.
Topics: Animals; Baclofen; Bicuculline; Cats; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Neural Inhibition; Pons; Receptors, GABA-A; Reticular Formation; Sleep, REM; Wakefulness | 2001 |
GABA B receptor-mediated effects on expression of c-Fos in rat trigeminal nucleus following high- and low-intensity afferent stimulation.
Topics: Animals; Baclofen; Electric Stimulation; GABA Agonists; GABA Antagonists; Male; Neurons, Afferent; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Trigeminal Nuclei | 2001 |
Inhibitory effect of 17beta-estradiol in the parabrachial nucleus is mediated by GABA.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Estradiol; Estrogen Antagonists; Female; Fulvestrant; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Neural Inhibition; Neural Pathways; Neurons; Ovariectomy; Pons; Rats; Receptors, Estrogen; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Vagus Nerve; Ventral Thalamic Nuclei; Visceral Afferents | 2001 |
Hemorrhage activates catecholaminergic neurons sensitive to GABA in the nucleus of the solitary tract with ascending projections to the subfornical organ in rats.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; Blood Pressure; Catecholamines; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Hemorrhage; Iontophoresis; Male; Neurons; Oxidopamine; Pressoreceptors; Rats; Rats, Wistar; Solitary Nucleus; Subfornical Organ; Sympatholytics | 2001 |
Evaluation of functional GABA(B) receptors in dental pulp.
Topics: Animals; Baclofen; Biotransformation; Cattle; Dental Pulp; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Radiopharmaceuticals; Receptors, GABA-B; Receptors, Opioid; Statistics, Nonparametric; Sulfur Radioisotopes | 2001 |
GABA(A) and GABA(B) receptors in the anterior piriform cortex modulate feeding in rats.
Topics: Amino Acids; Animals; Baclofen; Bicuculline; Feeding Behavior; Food Deprivation; Food, Formulated; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Neural Inhibition; Neurons; Olfactory Pathways; Oligonucleotide Array Sequence Analysis; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; RNA, Messenger; Threonine | 2002 |
Interactions between GABAergic and aminoacidergic pathways in the control of gonadotropin and GH secretion in pre-pubertal female rats.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Bicuculline; Excitatory Amino Acids; Female; Follicle Stimulating Hormone; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Human Growth Hormone; Kainic Acid; Luteinizing Hormone; Male; N-Methylaspartate; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sex Characteristics; Sexual Maturation | 2002 |
GABA-B-related activity in processing of transcallosal response in cat motor cortex.
Topics: Animals; Baclofen; Bicuculline; Cats; Corpus Callosum; Female; GABA Agonists; GABA Antagonists; Male; Motor Cortex; Organophosphorus Compounds; Receptors, GABA-A; Receptors, GABA-B; Receptors, Presynaptic; Synaptic Transmission | 2002 |
GABAergic drugs alter hypothalamic serotonin release and lordosis in estrogen-primed rats.
Topics: Animals; Baclofen; Estradiol; Female; GABA Agents; GABA Agonists; GABA Antagonists; Hypothalamus; Muscimol; Rats; Rats, Sprague-Dawley; Serotonin; Sexual Behavior, Animal | 2002 |
GABAergic systems in the nucleus tractus solitarius regulate noradrenaline release in the subfornical organ area in the rat.
Topics: Analysis of Variance; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Muscimol; Norepinephrine; Rats; Rats, Wistar; Solitary Nucleus; Subfornical Organ | 2002 |
Involvement of glutamate and gamma-amino-butyric acid receptor systems on gastric acid secretion induced by activation of kappa-opioid receptors in the central nervous system in rats.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Benzeneacetamides; Benzomorphans; Bicuculline; Brain; Dynorphins; gamma-Aminobutyric Acid; Gastric Acid; Injections, Intraventricular; Ketanserin; Male; Perfusion; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, Serotonin; Stomach | 2003 |
Modulation of noradrenaline release in the median preoptic area by GABAergic inputs from the organum vasculosum of the lamina terminalis in the rat.
Topics: Animals; Baclofen; Bicuculline; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Microdialysis; Norepinephrine; Preoptic Area; Rats; Rats, Wistar | 2004 |
Development of novel assays for proteolytic enzymes using rhodamine-based fluorogenic substrates.
Topics: Baclofen; Biological Assay; Combinatorial Chemistry Techniques; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Endopeptidases; Fluorescent Dyes; Inhibitory Concentration 50; Leucyl Aminopeptidase; Pentamidine; Peptides; Protease Inhibitors; Rhodamines; Substrate Specificity | 2002 |
GABA(B) receptor-mediated regulation of P2X7 receptor expression in the gerbil hippocampus.
Topics: Analysis of Variance; Animals; Baclofen; Bicuculline; Cell Count; GABA Agonists; GABA Antagonists; Gerbillinae; Hippocampus; Immunohistochemistry; Mossy Fibers, Hippocampal; Muscimol; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Seizures; Severity of Illness Index | 2004 |
Pharmacological modulation of GABA(B) receptors affects cocaine-induced seizures in mice.
Topics: Animals; Baclofen; Cocaine; Dopamine Uptake Inhibitors; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Kindling, Neurologic; Male; Mice; Piperazines; Receptors, GABA-A; Receptors, GABA-B; Seizures | 2004 |
Effects of ethanol and GABAB drugs on working memory in C57BL/6J and DBA/2J mice.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Drug Combinations; Ethanol; Female; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Memory; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Receptors, GABA-B; Species Specificity | 2004 |
GABA-mediated attenuation of noradrenaline release in the rat median preoptic area caused by intravenous injection of metaraminol.
Topics: Adrenergic alpha-Agonists; Animals; Baclofen; Baroreflex; Bicuculline; Blood Pressure; GABA Antagonists; gamma-Aminobutyric Acid; Injections, Intravenous; Male; Metaraminol; Microdialysis; Norepinephrine; Preoptic Area; Rats; Rats, Wistar; Receptors, GABA | 2004 |
Peripherally delivered glutamic acid decarboxylase gene therapy for spinal cord injury pain.
Topics: Animals; Baclofen; Bicuculline; Calcitonin Gene-Related Peptide; gamma-Aminobutyric Acid; Ganglia, Spinal; Genetic Therapy; Genetic Vectors; Glutamate Decarboxylase; Hyperalgesia; Injections, Subcutaneous; Isoenzymes; Neurons; Pain; Rats; Simplexvirus; Spinal Cord Injuries; Tissue Distribution; Transduction, Genetic | 2004 |
Altered GABAB receptor immunoreactivity in the gerbil hippocampus induced by baclofen and phaclofen, not seizure activity.
Topics: Animals; Baclofen; Blotting, Western; Cell Count; Dose-Response Relationship, Drug; Enzyme Inhibitors; GABA Antagonists; Gene Expression Regulation; Gerbillinae; Hippocampus; Immunohistochemistry; Proline; Receptors, GABA-B; Vigabatrin | 2004 |
Post-synaptic GABA(B) receptors--possible controllers of coincidence detection?
Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Baclofen; Chickens; Electric Impedance; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; In Vitro Techniques; Neurons; Prosencephalon; Receptors, GABA-B; Synapses; Synaptic Transmission; Valine | 2004 |
Glutamate and GABA(B) transmissions in lateral amygdala are involved in startle-like electromyographic (EMG) potentiation caused by activation of auditory thalamus.
Topics: Amygdala; Animals; Baclofen; Electric Stimulation; Electromyography; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; Kynurenic Acid; Male; Microinjections; Rats; Rats, Wistar; Receptors, GABA-A; Reflex, Startle; Synaptic Transmission; Time Factors; Trigeminal Nuclei | 2005 |
Effects of GABAB receptor modulation on gonadotropin-releasing hormone and beta-endorphin release, and on catecholaminergic activity in the ventromedial hypothalamus-infundibular nucleus region of anoestrous ewes.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; beta-Endorphin; Dopamine; Estrous Cycle; Extracellular Space; Female; GABA Agonists; GABA Antagonists; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Methoxyhydroxyphenylglycol; Norepinephrine; Pituitary Gland, Posterior; Receptors, GABA-B; Sheep; Ventromedial Hypothalamic Nucleus | 2005 |
Effects of GABAergic transmissions on the immunoreactivities of calcium binding proteins in the gerbil hippocampus.
Topics: Animals; Baclofen; Bicuculline; Calbindin 2; Calbindins; Calcium-Binding Proteins; Cell Count; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Gerbillinae; Hippocampus; Immunohistochemistry; Muscimol; Neurons; Parvalbumins; S100 Calcium Binding Protein G; Seizures; Synaptic Transmission | 2005 |
Benzodiazepine system is involved in hyperalgesia in rats induced by the exposure to extremely low frequency magnetic fields.
Topics: Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Diazepam; Electromagnetic Fields; Flumazenil; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hot Temperature; Hyperalgesia; Injections, Intraventricular; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A | 2005 |
Opposite effects of tetanic stimulation of the auditory thalamus or auditory cortex on the acoustic startle reflex in awake rats.
Topics: Acoustic Stimulation; Analysis of Variance; Animals; Auditory Cortex; Baclofen; Behavior, Animal; Electric Stimulation; Functional Laterality; GABA Antagonists; Geniculate Bodies; Male; Models, Biological; Rats; Rats, Wistar; Reflex, Startle; Time Factors; Wakefulness | 2005 |
HPLC conditions are critical for the detection of GABA by microdialysis.
Topics: Anesthetics, Local; Animals; Baclofen; Benzylamines; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Nipecotic Acids; Phosphinic Acids; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Time Factors | 2005 |
Enantiomeric analysis of baclofen analogs by capillary zone electrophoresis, using highly sulfated cyclodextrins: Inclusion ionization constant pKa determination.
Topics: Baclofen; Buffers; Cyclodextrins; Electrophoresis, Capillary; GABA Agonists; GABA-B Receptor Agonists; Hydrogen-Ion Concentration; Stereoisomerism; Sulfonic Acids | 2005 |
Electroacupuncture improves restraint stress-induced delay of gastric emptying via central glutaminergic pathways in conscious rats.
Topics: Animals; Baclofen; Bicuculline; Electroacupuncture; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Gastric Emptying; Kynurenic Acid; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Receptors, Glutamate; Restraint, Physical; Stomach; Stress, Psychological | 2006 |
GABA(A) and GABA(B) receptors differentially modulate volume and frequency in ventilatory compensation in obese Zucker rats.
Topics: Animals; Baclofen; Bicuculline; Dimethyl Sulfoxide; GABA Antagonists; Hypercapnia; Hypoxia; Male; Obesity; Oxygen Consumption; Physical Conditioning, Animal; Pulmonary Ventilation; Rats; Rats, Zucker; Receptors, GABA-A; Receptors, GABA-B; Respiratory Mechanics; Tidal Volume | 2007 |
GABAA but not GABAB receptors in the rostral anterior cingulate cortex selectively modulate pain-induced escape/avoidance behavior.
Topics: Animals; Avoidance Learning; Baclofen; Bicuculline; Escape Reaction; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gyrus Cinguli; Male; Microinjections; Muscimol; Pain; Pain Threshold; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B | 2007 |
Understanding your inhibitions: modulation of brain cortical metabolism by GABA(B) receptors.
Topics: Animals; Baclofen; Benzylamines; Carbon Isotopes; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Guinea Pigs; Molecular Structure; Morpholines; Nuclear Magnetic Resonance, Biomolecular; Organophosphorus Compounds; Phosphinic Acids; Principal Component Analysis; Receptors, GABA-B | 2007 |
Nicotinic receptor-mediated biphasic effect on neuronal excitability in chick lateral spiriform neurons.
Topics: Action Potentials; Animals; Baclofen; Brain; Calcium; Carbachol; Chick Embryo; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; GABA Antagonists; In Vitro Techniques; Neural Inhibition; Neurons; Nicotine; Nicotinic Antagonists; Receptors, Nicotinic; Time Factors | 2007 |
GABA receptor agonism in the sublenticular central extended amygdala impairs medial forebrain bundle self-stimulation but GABA blockade does not enhance it.
Topics: Amygdala; Animals; Baclofen; Bicuculline; Electric Stimulation; Functional Laterality; GABA Agonists; GABA Antagonists; Male; Medial Forebrain Bundle; Muscimol; Rats; Rats, Long-Evans; Receptors, GABA; Reinforcement, Psychology; Self Stimulation; Substantia Innominata | 2008 |
[Contribution of GABA receptors in extinction of memory trace in norm and depressive-like state].
Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Depression; Fear; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Memory; Mice; Muscimol; Receptors, GABA-A; Receptors, GABA-B | 2007 |
Evidence that gamma-aminobutyric acid is part of the neural circuit mediating estradiol negative feedback in anestrous ewes.
Topics: Anestrus; Animals; Baclofen; Bicuculline; Dopamine; Estradiol; Feedback; Female; gamma-Aminobutyric Acid; Muscimol; Neurons; Ovariectomy; Sheep | 2008 |
GabaB receptors activation in the NTS blocks the glycemic responses induced by carotid body receptor stimulation.
Topics: Analysis of Variance; Animals; Baclofen; Bicuculline; Blood Glucose; Carotid Body; GABA Agonists; GABA Antagonists; Glucose; Microinjections; Muscimol; Rats; Receptors, GABA-A; Receptors, GABA-B; Solitary Nucleus | 2008 |
Roles of forebrain GABA receptors in controlling vasopressin secretion and related phenomena under basal and hyperosmotic circumstances in conscious rats.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Consciousness; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Glucose; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Muscimol; Osmolar Concentration; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA; Saline Solution, Hypertonic; Sodium; Vasopressins | 2008 |
GABAergic mediation of stress-induced secretion of corticosterone and oxytocin, but not prolactin, by the hypothalamic paraventricular nucleus.
Topics: Animals; Baclofen; Bicuculline; Corticosterone; Dose-Response Relationship, Drug; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Microinjections; Oxytocin; Paraventricular Hypothalamic Nucleus; Prolactin; Rats; Rats, Wistar; Stress, Psychological | 2008 |
Analgesic alpha-conotoxins Vc1.1 and Rg1A inhibit N-type calcium channels in rat sensory neurons via GABAB receptor activation.
Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Barium; Calcium Channel Blockers; Calcium Channels, N-Type; Cells, Cultured; Conotoxins; Dose-Response Relationship, Radiation; Electric Stimulation; GABA Antagonists; Ganglia, Spinal; Membrane Potentials; omega-Conotoxins; Patch-Clamp Techniques; Pertussis Toxin; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA; Sensory Receptor Cells | 2008 |
GABA antagonists reverse the somatostatin dependent attenuation of rat locomotor activity.
Topics: Animals; Baclofen; Basal Ganglia; Bicuculline; GABA Antagonists; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Somatostatin | 2009 |
Astrocytes and interneurons in memory processing in the chick hippocampus: roles for G-coupled protein receptors, GABA(B) and mGluR1.
Topics: Animals; Animals, Newborn; Astrocytes; Baclofen; Chickens; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hippocampus; Housing, Animal; Interneurons; Male; Memory; Methoxyhydroxyphenylglycol; Receptors, G-Protein-Coupled; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Time Factors | 2009 |
Role of endocannabinoid system in the ventral hippocampus of rats in the modulation of anxiety-like behaviours.
Topics: Amidohydrolases; Animals; Anxiety; Baclofen; Behavior, Animal; Benzamides; Bicuculline; Cannabinoid Receptor Modulators; Carbamates; Dose-Response Relationship, Drug; Endocannabinoids; GABA Antagonists; Hippocampus; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1 | 2009 |
GABA receptors and prepulse inhibition of acoustic startle in mice and rats.
Topics: Acoustic Stimulation; Animals; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Muscimol; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, GABA; Reflex, Startle; Scopolamine; Time Factors | 2010 |
Analgesia induced by 2- or 100-Hz electroacupuncture in the rat tail-flick test depends on the activation of different descending pain inhibitory mechanisms.
Topics: Adjuvants, Anesthesia; Adrenergic alpha-Antagonists; Analgesia; Anesthetics, Intravenous; Animals; Atropine; Baclofen; Bicuculline; Biophysics; Dioxanes; Disease Models, Animal; Electroacupuncture; GABA Agents; Male; Methysergide; Models, Biological; Multivariate Analysis; Naloxone; Narcotic Antagonists; Pain; Pain Management; Pain Measurement; Rats; Rats, Wistar; Reaction Time; Serotonin Antagonists; Tail; Thiopental; Time Factors | 2011 |
GABA(A) receptors in the dorsal raphé nucleus of mice: escalation of aggression after alcohol consumption.
Topics: Aggression; Animals; Baclofen; Behavior, Animal; Bicuculline; Ethanol; GABA Agonists; GABA Antagonists; Male; Mice; Muscimol; Raphe Nuclei; Receptors, GABA-A; Receptors, GABA-B; Self Administration | 2010 |
Involvement of GABAergic transmission in the midbrain ventral tegmental area in the regulation of hippocampal theta rhythm.
Topics: Animals; Baclofen; Bicuculline; Electroencephalography; Fourier Analysis; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Muscimol; Rats; Rats, Wistar; Theta Rhythm; Ventral Tegmental Area | 2010 |
Metabotropic γ-aminobutyric acid (GABAB) receptors modulate feeding behavior in the calcisponge Leucandra aspera.
Topics: Animals; Baclofen; Drug Interactions; Endocytosis; Feeding Behavior; GABA Antagonists; GABA-B Receptor Agonists; Pertussis Toxin; Porifera; Receptors, GABA-B | 2011 |
Changes in GABA and GABA(B) receptor expressions are involved in neuropathy in the rat cuneate nucleus following median nerve transection.
Topics: Animals; Baclofen; Electric Stimulation; GABA Antagonists; Gait; gamma-Aminobutyric Acid; Ganglia, Spinal; Male; Median Nerve; Median Neuropathy; Medulla Oblongata; Neuropeptide Y; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-B | 2012 |
Decreased GABABR expression and increased neuronal cell death in developing rat brain after PTZ-induced seizure.
Topics: Animals; Animals, Newborn; Baclofen; Caspase 3; Cell Death; Disease Models, Animal; Electroencephalography; GABA Antagonists; GABA-B Receptor Agonists; Gene Expression Regulation, Developmental; Hippocampus; Microscopy, Confocal; Neurons; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Seizures | 2013 |
Baclofen administration alters fear extinction and GABAergic protein levels.
Topics: Amygdala; Animals; Baclofen; Conditioning, Psychological; Cues; Extinction, Psychological; Fear; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Male; Rats; Rats, Sprague-Dawley; Reflex, Startle | 2012 |
Segmental disinhibition suppresses C-fiber inputs to the rat superficial medullary dorsal horn via the activation of GABAB receptors.
Topics: Action Potentials; Animals; Baclofen; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Morphine; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Posterior Horn Cells; Rats; Rats, Inbred Strains; Receptors, GABA-B; Receptors, Glycine; Synaptic Transmission | 2013 |
GABAergic synaptic inputs of locus coeruleus neurons in wild-type and Mecp2-null mice.
Topics: Animals; Baclofen; Female; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; GABAergic Neurons; gamma-Aminobutyric Acid; Humans; Locus Coeruleus; Male; Membrane Potentials; Methyl-CpG-Binding Protein 2; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscimol; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Presynaptic Terminals; Receptors, GABA-A; Receptors, GABA-B; Rett Syndrome; Synaptic Membranes; Synaptic Transmission | 2013 |
Effect of GABA receptor agonists or antagonists injected spinally on the blood glucose level in mice.
Topics: Animals; Baclofen; Blood Glucose; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Receptors, GABA | 2013 |
Reversal of morphine analgesic tolerance by ethanol in the mouse.
Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethanol; GABA Antagonists; Hypnotics and Sedatives; Immersion; Injections, Intraventricular; Male; Mice; Morphine; Pain Measurement; Receptors, GABA-A; Receptors, GABA-B | 2013 |
Effects of Withania somnifera on oral ethanol self-administration in rats.
Topics: Administration, Oral; Alcohol Drinking; Animals; Baclofen; Conditioning, Operant; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Ethanol; Male; Plant Extracts; Rats; Rats, Wistar; Receptors, GABA-B; Reinforcement Schedule; Saccharin; Self Administration; Withania | 2014 |
Postnatal alterations in GABAB receptor tone produce sensorimotor gating deficits and protein level differences in adulthood.
Topics: Acoustic Stimulation; Age Factors; Animals; Animals, Newborn; Baclofen; Body Weight; Brain; Disease Models, Animal; Female; GABA Antagonists; GABA-B Receptor Agonists; Gait Disorders, Neurologic; Gene Expression Regulation, Developmental; Male; Pregnancy; Prepulse Inhibition; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Sensory Gating; Signal Transduction | 2015 |
The antinociceptive effect of stimulating the retrosplenial cortex in the rat tail-flick test but not in the formalin test involves the rostral anterior cingulate cortex.
Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; Cobalt; Electric Stimulation; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Gyrus Cinguli; Male; Pain Measurement; Pain Perception; Rats; Rats, Wistar; Tail | 2015 |
The modulatory effect of CA1 GABAb receptors on ketamine-induced spatial and non-spatial novelty detection deficits with respect to Ca(2+).
Topics: Analysis of Variance; Animals; Baclofen; CA1 Region, Hippocampal; Calcium; Calcium Channel Blockers; Disease Models, Animal; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Exploratory Behavior; GABA Antagonists; Imidazoles; Ketamine; Male; Memory Disorders; Mice; Receptors, GABA-A; Signal Detection, Psychological; Spatial Processing | 2015 |
GABA modulates baroreflex in the ventral tegmental area in rat.
Topics: Animals; Baclofen; Baroreflex; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Wistar; Ventral Tegmental Area | 2015 |
Recovery from ketamine-induced amnesia by blockade of GABA-A receptor in the medial prefrontal cortex of mice.
Topics: Amnesia; Animals; Baclofen; Bicuculline; Catheters, Indwelling; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; Ketamine; Male; Memory; Mice; Muscimol; Neuropsychological Tests; Prefrontal Cortex; Receptors, GABA-A; Time Factors | 2017 |
The lesion of dorsolateral funiculus changes the antiallodynic effect of the intrathecal muscimol and baclofen in distinct phases of neuropathic pain induced by spinal nerve ligation in rats.
Topics: Animals; Baclofen; Bicuculline; Functional Laterality; GABA Agents; Hyperalgesia; Injections, Spinal; Ligation; Male; Muscimol; Neuralgia; Pain Measurement; Pain Threshold; Physical Stimulation; Rats; Rats, Wistar; Spinal Cord Dorsal Horn; Spinal Nerves; Statistics, Nonparametric | 2016 |
GABAergic modulation of serotonin release in the rat subfornical organ area.
Topics: Animals; Baclofen; Bicuculline; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hydroxyindoleacetic Acid; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Serotonin; Subfornical Organ | 2016 |
GABA Receptors in the Medial Preoptic Area Modulate the Onset of Oestradiol-Induced Maternal Behaviour in Hysterectomised-Ovariectomised, Pregnant Rats.
Topics: Animals; Baclofen; Bicuculline; Estradiol; Female; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hysterectomy; Maternal Behavior; Nesting Behavior; Ovariectomy; Pregnancy; Preoptic Area; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B | 2016 |
GABAergic modulation of noradrenaline release caused by blood pressure changes in the rat median preoptic area.
Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Baclofen; Bicuculline; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Metaraminol; Microdialysis; Norepinephrine; Preoptic Area; Rats; Rats, Wistar | 2017 |
The interaction between hippocampal GABA-B and cannabinoid receptors upon spatial change and object novelty discrimination memory function.
Topics: Animals; Baclofen; Discrimination Learning; Dose-Response Relationship, Drug; Exploratory Behavior; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hippocampus; Male; Memory; Mice; Microinjections; Receptor, Cannabinoid, CB1; Receptors, Cannabinoid; Receptors, GABA-B; Spatial Behavior | 2017 |
The role of CA3 GABA
Topics: 2-Amino-5-phosphonovalerate; Animals; Anxiety; Avoidance Learning; Baclofen; CA3 Region, Hippocampal; Calcium; Calcium Channel Blockers; Cations, Divalent; Disease Models, Animal; GABA Antagonists; GABA-B Receptor Agonists; Imidazoles; Male; Memory Disorders; Motor Activity; Psychotropic Drugs; Random Allocation; Rats, Wistar; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate | 2017 |
Modulation of tonic immobility by GABAA and GABAB receptors of the medial amygdala.
Topics: Animals; Baclofen; Bicuculline; Corticomedial Nuclear Complex; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Guinea Pigs; Immobility Response, Tonic; Male; Microinjections; Motor Activity; Muscimol | 2019 |
The effect of GABA-B receptors in the basolateral amygdala on passive avoidance memory impairment induced by MK-801 in rats.
Topics: Animals; Avoidance Learning; Baclofen; Basolateral Nuclear Complex; Behavior, Animal; Disease Models, Animal; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Memory Disorders; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate | 2021 |