phaclofen and baclofen

phaclofen has been researched along with baclofen in 241 studies

Research

Studies (241)

TimeframeStudies, this research(%)All Research%
pre-199026 (10.79)18.7374
1990's135 (56.02)18.2507
2000's53 (21.99)29.6817
2010's26 (10.79)24.3611
2020's1 (0.41)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Del Bianco, E; Giuliani, S; Lecci, A; Maggi, CA; Santicioli, P1
Berger, TW; Nisenbaum, ES1
Blanchet, G; Gahery, Y; Luccarini, P; Pompeiano, O1
Douglas, WW; Kongsamut, S; Shibuya, I1
Libertun, C; Lux-Lantos, V; Rey, E1
Beani, L; Bianchi, C; Ferraro, L; Tanganelli, S1
Kawaguchi, Y1
Bonanno, G; Raiteri, M2
Donoso, AO; López, FJ; Negro-Vilar, A1
Bonanno, G; Gemignani, A; Lanza, M; Pende, M; Raiteri, M; Vellebuona, F1
Finch, DM; Mello, LE; Tan, AM1
Dunwiddie, TV; Lupica, CR; Proctor, WR1
Saito, H; Tamai, A; Ueno, H; Yoshida, K1
Bernardini, MC; Blandizzi, C; Del Tacca, M; Natale, G1
Allan, AM; Burnett, D; Harris, RA1
Bartolini, A; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P1
Kow, LM; Ogawa, S; Pfaff, DW1
Henry, JL; Hong, YG1
Henry, JL; Hong, Y1
Sanders, SK; Shekhar, A1
Sastry, BR; Xie, Z1
Aceves, J; Arias-Montaño, JA; Martínez-Fong, D1
Lacaille, JC1
Jones, AJ; Keen, P; Ray, NJ1
Couture, R; De Champlain, J; Hasséssian, H; Prat, A1
Lewis, DV; Morrisett, RA; Mott, DD; Swartzwelder, HS; Wilson, WA1
Henriksen, SJ; Steffensen, SC1
Aran, S; Hammond, DL1
Baldwin, BA; Ebenezer, IS1
Howson, W; Lacey, MG; Seabrook, GR1
Ebenezer, IS1
Alberch, J; Arenas, E; Marsal, J1
Alhaider, AA; Lei, SZ; Wilcox, GL1
Hankins, MW; Ikeda, H; Kay, CD1
Kamata, O; Nakagawa, T; Nakanishi, H; Ukai, K; Watanabe, S; Yamamoto, K1
Bonanno, G; Giralt, MT; Raiteri, M1
Bernardini, MC; Blandizzi, C; Del Tacca, M1
Dun, NJ; Wang, MY1
Allan, RD; Drew, CA; Ong, J; Tran, HW1
Huang, JH; Johnston, GA1
Drew, CA; Johnston, GA; Kerr, DI; Ong, J1
Barraclough, CA; Hartman, RD; He, JR1
Collingridge, GL; Davies, CH; Davies, SN1
Mehta, AK; Ticku, MK1
Karlsson, G; Olpe, HR3
De Luca, C; Massotti, M1
Michler, A1
Sved, AF; Sved, JC1
al-Dahan, MI; Tehrani, MH; Thalmann, RH1
Bittiger, H; Brugger, F; Fagg, G; Froestl, W; Hall, RG; Karlsson, G; Olpe, HR; Pozza, MF; Steinmann, M; Van Riezen, H1
Hicks, TP; Kaneko, T1
Bernardi, G; Calabresi, P; De Murtas, M; Mercuri, NB1
Slater, NT; Smith, RD; Turek, FW1
Furshpan, EJ; Segal, MM1
Fukuda, H; Hirayama, T; Ono, H1
Goto, Y; Hara, N; Hara, Y1
Bragdon, AC; Lewis, DV; Mott, DD1
Harrison, NL1
Malouf, AT; Robbins, CA; Schwartzkroin, PA1
Kulkarni, SK1
Johnston, GA; Kerr, DI; Ong, J; Prager, RH1
Asaro, D; Bonanno, G; Fontana, G; Pellegrini, G; Raiteri, M1
Böhmer, G; Gebauer, K; Schmid, K1
Dingsdale, RA; Dolle, RE; Hills, JM; Howson, W; Parsons, ME1
Erdö, SL; Michler, A1
Boar, BR; Cross, AJ; Green, AR; Robinson, TN; Toczek, JM1
Allan, AM; Harris, RA1
Bonanno, G; Cantoni, C; Pellegrini, G; Raiteri, M1
Gallagher, JP; Hasuo, H2
Chamberlin, NL; Dingledine, R1
Dutar, P; Lamour, Y; Rascol, O1
Neal, MJ; Shah, MA1
Klockgether, T; Sontag, KH; Wüllner, U1
Dutar, P; Nicoll, RA1
Crunelli, V; Haby, M; Leresche, N; Soltesz, I1
Karlsson, G; Olpe, HR; Pozza, M1
Brugger, F; Hall, RG; Olpe, HR; Pozza, MF; Steinmann, MW1
Albus, K; Baumfalk, U1
Enna, SJ; Ferkany, JW; Scherer, RW1
Bonanno, G; Fontana, G; Raiteri, M1
Curtis, DR; Gynther, BD; Kerr, DI; Ong, J; Prager, RH1
Borsini, F; Evangelista, S; Giuliani, S; Meli, A1
Alkon, DL; Axelrod, J; Collin, C; Dahl, D; Devane, WA; Lee, CJ1
Chad, JE; Stanford, IM; Wheal, HV1
Cano, J; Machado, A; Santiago, M1
Humeniuk, RE; Kerr, DI; Ong, J; White, JM1
Hyson, RL; Reyes, AD; Rubel, EW1
Boksa, P; Chaudieu, I; Quirion, R; St-Pierre, JA1
Caddick, SJ; Chad, JE; Stanford, IM1
Banerjee, PK; Snead, OC1
Slaughter, MM; Tian, N1
Bonanno, G; Cavazzani, P; Fassio, A; Raiteri, M1
Gean, PW; Huang, CC1
Humeniuk, RE; Ong, J; White, JM1
Araki, T; Endo, K; Kaneko, T; Kang, Y; Ohishi, H1
Carpenter, DO; Lin, Y1
Fisone, G; Greengard, P; Snyder, GL1
Bonanno, G; Gemignani, A; Paudice, P; Raiteri, M1
Finch, DM; Gigg, J; Tan, AM1
Domann, R; Westerhoff, CH; Witte, OW1
Drew, CA; Frydenvang, K; Hansen, JJ; Johnston, GA; Krogsgaard-Larsen, P; Mitrovic, A; Tran, H1
Beninger, RJ; Boegman, RJ; DeSousa, NJ; Jhamandas, K1
Bonanno, G; Lanza, M; Pende, M; Raiteri, M1
Lewis, DV; Mott, DD; Swartzwelder, HS; Wilson, WA; Xie, CW1
Hammond, DL; McGowan, MK1
Hasler, WL; Owyang, C; Roberts, DJ1
Cotman, CW; Kahle, JS1
Lacaille, JC; Samulack, DD1
Dutar, P; Lamour, Y; Potier, B1
Lennon, VA; Parkman, HP; Stapelfeldt, WH; Szurszewski, JH; Williams, CL1
Brikas, P1
DiScenna, PG; Nowicky, AV; Teyler, TJ1
Hoffman, DS; Kurata, K1
Haji, A; Takeda, R1
Clarke, IJ; Scott, CJ1
Guo, JZ; Ichinose, T; Murakoshi, T1
Eriksson, PS; Hansson, E; Nilsson, M; Rönnbäck, L1
Bradley, RM; Wang, L1
De Koning, HP; Jenks, BG; Roubos, EW1
el Manira, A; Grillner, S; Matsushima, T; Tegnér, J1
Kuramochi, T; Suga, T; Suzuki, M1
Billard, JM; Deisz, RA; Zieglgänsberger, W1
Albrecht, D; Henklein, P; Zippel, U1
Haugh-Scheidt, L; Malchow, RP; Ripps, H1
Chen, W; Hu, GY; Wu, CP; Zhang, JJ1
Ayata, G; Cutrer, FM; Limmroth, V; Moskowitz, MA1
Croucher, MJ; Patel, DR; Sundaralingam, J1
Hashemi, B; Toloui, V; Zarrindast, MR1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Antonelli, T; Ferraro, L; Fuxe, K; O'Connor, WT; Rambert, F; Tanganelli, S1
Brumberg, JC; Carvell, GE; Kyriazi, HT; Simons, DJ1
Kubota, K1
Chen, W; Cheng, JT; Terada, M1
Brailowsky, S; Di Scala, G; Meneses, S; Montiel, T1
Snead, OC2
Dar, MS1
Armony, JL; LeDoux, JE; Li, XF1
Itoh, T; Kamisaki, Y; Nakamoto, K; Wada, K1
Armstrong, DL; Cato, MJ; Gannon, RL; Kelley, KH; Rea, MA1
Chowdhury, SA; Kawashima, T; Konishi, T; Matsunami, K1
Chen, Y; Matsuki, N; Saito, H1
Pierau, FK; Sann, H; Schmid, HA; Yakimova, KS1
Kar, S; Quirion, R; Seto, D1
Hashemi, B; Semnanian, S; Shafizadeh, M; Zarrindast, MR1
El Manira, A; Grillner, S; Tegnér, J1
Chub, N; O'Donovan, MJ1
Celis, ME; Cremer, MC; De Barioglio, SR1
Gong, W; Justice, JB; Neill, DB1
Carlen, PL; Frantseva, MV; Perez Velazquez, JL1
Ciriello, J; Roder, S1
Chavkin, C; Jin, W1
Kerr, DI; Ong, J; Parnas, I; Rashkovan, G1
Cairns, BE; Hu, JW; Sessle, BJ1
Klejbor, I; Trojniar, W1
Dun, NJ; Hwang, BH; Mizoguchi, H; Nagase, H; Narita, M; Oji, DE; Tseng, LF1
Bonanno, G; Marcoli, M; Maura, G; Raiteri, M; Scarrone, S1
Ozdem, SS; Sadan, G; Taşatargil, A; Usta, C1
Hood, SC; Schwartz, NB1
Gotoh, S; Miwa, N; Nakayama, H; Suzuki, J; Terao, K1
Hartings, JA; Simons, DJ1
Elshourbagy, NA; Gager, TL; Hirst, WD; Jenkins, O; Minton, J; Murkitt, KL; Pangalos, M; Price, GW; Punia, PK; Rice, SQ; Shabon, U; Stammers, M; Taylor, SJ; Testa, T; Wood, MD1
Fendt, M; Koch, M; Kretschmer, BD1
Hayashi, Y; Miyakubo, H; Nomura, S; Okumura, T; Sakamaki, K; Tanaka, J1
Chase, MH; Morales, FR; Xi, MC1
Kerr, DI; Ong, J1
Shigenaga, Y; Shimada, T; Takemura, M1
Saleh, MC; Saleh, TM1
Hayashi, Y; Miyakubo, H; Nomura, M; Tanaka, J1
Bowles, W; Hargreaves, KM; Richardson, JD; Wurm, C1
Gietzen, DW; Magrum, LJ; Truong, BG1
Aguilar, E; González, LC; Pinilla, L; Tena-Sempere, M1
Chowdhury, SA; Matsunami, KI1
Hoffman, CS; Johnson, PL; Miner, HM; Renner, KJ; Summers, CH; Westin, TM1
Kawakami, A; Mashiko, N; Nomura, M; Tanaka, J; Ushigome, A1
Horie, S; Ishihara, S; Minowa, S; Murayama, T; Tsuchiya, S; Watanabe, K1
Nomura, M; Tanaka, J; Ushigome, A1
Cummings, RT; Grant, SK; Sklar, JG1
An, SJ; Hwang, IK; Kang, TC; Park, SK; Won, MH1
Gasior, M; Kaminski, R; Witkin, JM1
Enna, SJ1
Escher, T; Mittleman, G1
Nomura, M; Sakamaki, K; Tanaka, J; Yamato, K1
Fink, DJ; Glorioso, JC; Hao, S; Huang, S; Liu, J; Mata, M; Wolfe, D1
An, SJ; Choi, SY; Hwang, IK; Jeong, YG; Jung, JY; Kang, TC; Kim, DW; Kwon, OS; Park, SK; Won, MH1
Bradley, PM; Burns, BD; Gowland, CJ; Webb, AC1
He, S; Huang, J; Li, L; Wu, X1
Przekop, F; Tomaszewska-Zaremba, D1
Choi, SY; Jung, JY; Kang, TC; Kim, DS; Kim, JE; Kwak, SE; Kwon, OS; Won, MH1
Choi, KB; Jeong, JH; Moon, NJ; Park, ES; Sohn, UD1
Huang, J; Li, L; Wu, X; Yeomans, J1
Cremers, TI; Rea, K; Westerink, BH1
Bonte, JP; Foulon, C; Goossens, JF; Lipka, E; Vaccher, C; Vaccher, MP1
Iwa, M; Nakade, Y; Pappas, TN; Takahashi, T1
Chen, JS; Huang, CY; Lee, SD; Lo, MJ; Ting, H; Yang, AL1
Fuchs, PN; LaGraize, SC1
Balcar, VJ; Griffin, JL; Nasrallah, FA; Rae, C1
Chiappinelli, VA; Guo, JZ; Liu, YB1
Waraczynski, M1
Dubrovina, NI; Zinov'ev, DR1
Billings, HJ; Bogusz, AL; Connors, JM; Coolen, LM; Goodman, RL; Hardy, SL; Hileman, SM; Lehman, MN; McManus, CJ; Nestor, CC; Singh, SR; Sliwowska, JH; Valent, M1
Álvarez-Buylla, R; Cadenas, JL; de Álvarez-Buylla, ER; Lara, JJ; Lemus, M; Montero, S; Tejeda-Chávez, HR1
Yamada, T; Yamaguchi, K1
Franci, CR; Marques de Souza, L1
Adams, DJ; Berecki, G; Callaghan, B; Clark, RJ; Craik, DJ; Haythornthwaite, A1
Marazioti, A; Spyraki, C; Thermos, K1
Bowser, DN; Gibbs, ME1
Hasanein, P; Keshavarz, S; Moghaddam, AH; Rezvani, ME; Roohbakhsh, A1
Alves, N; Bosch, D; Daros, A; Schmid, S; Ure, RJ; Yeomans, JS1
Prado, WA; Silva, JR; Silva, ML1
Debold, JF; Kwa, C; Miczek, KA; Takahashi, A1
Jurkowlaniec, E; Kuśmierczak, M; Orzeł-Gryglewska, J1
Bianchini, P; Diaspro, A; Fato, M; Ferrando, S; Gallus, L; Ledda, FD; Manconi, R; Ramoino, P; Tagliafierro, G1
Chen, SH; Li, SF; Lin, CT; Lue, JH; Tsai, YJ; Wang, HY1
Al-Qahtani, MH; Ansari, SA; Bibi, F; Karim, S; Kim, MO; Naseer, MI; Ullah, I; Ullah, N1
Bolton, MM; Heaney, CF; Kinney, JW; Magcalas, CM; Murtishaw, AS; Sabbagh, JJ2
Artola, A; Dallel, R; Jacquot, F; Melin, C1
Cui, N; Jiang, C; Jin, X; Jin, XT; Zhong, W1
Choi, MG; Jung, JS; Kang, YJ; Kim, CH; Kim, SJ; Kim, SS; Park, SH; Ryu, OH; Sim, YB; Suh, HW1
Bailey, CP; Dewey, WL; Gabra, BH; Henderson, G; Hull, LC1
Acquas, E; Cotti, E; Kasture, SB; Muggironi, G; Peana, AT; Rosas, M; Spina, L1
Fais, RS; Prado, WA; Reis, GM1
Khanegheini, A; Nasehi, M; Zarrindast, MR1
Hatam, M; Nasimi, A; Rasoulpanah, M1
Akbarabadi, A; Bakhtazad, A; Farahmandfar, M; Zarrindast, MR1
Dias, QM; Prado, WA1
Nomura, M; Takahashi, M; Tanaka, J1
Ågmo, A; Dominguez, G; Gómora-Arrati, P1
Johnston, GAR1
Takahashi, M; Tanaka, J1
Alaghmandan-Motlagh, N; Ebrahimi-Ghiri, M; Nami, M; Nasehi, M; Zarrindast, MR1
Farrahizadeh, M; Nasehi, M; Zarrabian, S; Zarrindast, MR1
de Melo, JR; de Paula, BB; Leite-Panissi, CRA1
Khakpoor, M; Mohammadi-Mahdiabadi-Hasani, MH; Nasehi, M; Vaseghi, S1

Reviews

4 review(s) available for phaclofen and baclofen

ArticleYear
GABAB receptors and phaclofen.
    Methods and findings in experimental and clinical pharmacology, 1989, Volume: 11, Issue:2

    Topics: Baclofen; Humans; Receptors, GABA-A

1989
Recent advances in GABAB receptors: from pharmacology to molecular biology.
    Acta pharmacologica Sinica, 2000, Volume: 21, Issue:2

    Topics: Animals; Baclofen; Cloning, Molecular; GABA Agonists; GABA Antagonists; Potassium Channels; Receptors, GABA-B

2000
A GABA(B) mystery: the search for pharmacologically distinct GABA(B) receptors.
    Molecular interventions, 2001, Volume: 1, Issue:4

    Topics: Acetates; Amines; Animals; Anticonvulsants; Baclofen; Benzylamines; Cyclohexanecarboxylic Acids; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Molecular Structure; Morpholines; Phosphinic Acids; Protein Isoforms; Receptors, GABA-B; RNA, Messenger

2001
GABA Australis, some reflections on the history of GABA receptor research in Australia.
    Pharmacological research, 2017, Volume: 116

    Topics: Animals; Australia; Baclofen; Bicuculline; Cyclic AMP; Humans; Isoxazoles; Muscimol; Receptors, GABA

2017

Other Studies

237 other study(ies) available for phaclofen and baclofen

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Effect of the GABAB antagonist, phaclofen, on baclofen-induced inhibition of micturition reflex in urethane-anesthetized rats.
    Neuroscience, 1992, Volume: 48, Issue:1

    Topics: Animals; Baclofen; Capsaicin; Cerebral Ventricles; Fenclonine; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Reflex; Urethane; Urinary Bladder; Urination

1992
Functionally distinct subpopulations of striatal neurons are differentially regulated by GABAergic and dopaminergic inputs--I. In vivo analysis.
    Neuroscience, 1992, Volume: 48, Issue:3

    Topics: Animals; Baclofen; Benzazepines; Bicuculline; Corpus Striatum; Dopamine; Electric Stimulation; Electrophysiology; gamma-Aminobutyric Acid; Male; Neural Pathways; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, GABA-A; Sulpiride; Sympathectomy, Chemical

1992
GABA receptors in Deiters nucleus modulate posturokinetic responses to cortical stimulation in the cat.
    Archives italiennes de biologie, 1992, Volume: 130, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Extremities; Male; Microinjections; Motor Cortex; Muscimol; Posture; Receptors, GABA-A; Vestibular Nucleus, Lateral

1992
Effectiveness of GABAB antagonists in inhibiting baclofen-induced reductions in cytosolic free Ca concentration in isolated melanotrophs of rat.
    British journal of pharmacology, 1992, Volume: 105, Issue:4

    Topics: Animals; Baclofen; Calcium; Cytosol; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Organophosphorus Compounds; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains

1992
Activation of GABA B receptors in the anterior pituitary inhibits prolactin and luteinizing hormone secretion.
    Neuroendocrinology, 1992, Volume: 56, Issue:5

    Topics: Animals; Baclofen; Butylamines; Cells, Cultured; Female; GABA Antagonists; Gonadotropin-Releasing Hormone; Lactation; Luteinizing Hormone; Organophosphorus Compounds; Pituitary Gland, Anterior; Proestrus; Prolactin; Propylamines; Rats; Receptors, GABA-A; Thyrotropin-Releasing Hormone

1992
Changes in gamma-aminobutyric acid release induced by topical administration of drugs affecting its metabolism and receptors: studies in freely moving guinea pigs with epidural cups.
    Neurochemistry international, 1992, Volume: 21, Issue:1

    Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Baclofen; beta-Alanine; Calcium; Cerebral Cortex; Epidural Space; Ethanolamines; Feedback; Female; gamma-Aminobutyric Acid; Guinea Pigs; Kinetics; Male; Nipecotic Acids; Norepinephrine; Receptors, GABA-A; Sodium; Tetrodotoxin

1992
Receptor subtypes involved in callosally-induced postsynaptic potentials in rat frontal agranular cortex in vitro.
    Experimental brain research, 1992, Volume: 88, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Corpus Callosum; Electric Stimulation; Evoked Potentials; Frontal Lobe; GABA Antagonists; In Vitro Techniques; Male; Picrotoxin; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Synapses

1992
Functional evidence for multiple gamma-aminobutyric acidB receptor subtypes in the rat cerebral cortex.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Male; Organophosphorus Compounds; Peptides; Rats; Rats, Inbred Strains; Receptors, GABA-A

1992
Cross-talk between excitatory and inhibitory amino acids in the regulation of luteinizing hormone-releasing hormone secretion.
    Endocrinology, 1992, Volume: 131, Issue:3

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Bicuculline; Drug Interactions; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Gonadotropin-Releasing Hormone; In Vitro Techniques; Male; Median Eminence; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A

1992
Pharmacologically distinct GABAB receptor subtypes modulate neurotransmitter release in the rat brain cortex.
    Advances in biochemical psychopharmacology, 1992, Volume: 47

    Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; GABA-A Receptor Antagonists; Glutamates; Glutamic Acid; Muscimol; Neurotransmitter Agents; Organophosphorus Compounds; Rats; Receptors, GABA-A; Somatostatin; Synaptosomes

1992
GABAergic synaptic transmission in projections from the basal forebrain and hippocampal formation to the amygdala: an in vivo iontophoretic study.
    Brain research, 1992, Jul-31, Volume: 587, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Electric Stimulation; gamma-Aminobutyric Acid; Hippocampus; Iontophoresis; Male; Neural Pathways; Prosencephalon; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Neurotransmitter; Synapses; Synaptic Transmission

1992
Dissociation of mu and delta opioid receptor-mediated reductions in evoked and spontaneous synaptic inhibition in the rat hippocampus in vitro.
    Brain research, 1992, Oct-16, Volume: 593, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Analgesics; Animals; Axons; Baclofen; Bicuculline; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Evoked Potentials; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Neurons; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Synapses

1992
[Effect of GABA antagonists on the rat electroretinogram].
    Nippon Ganka Gakkai zasshi, 1992, Volume: 96, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Electroretinography; GABA Antagonists; Male; Rats; Rats, Inbred Strains; Retina

1992
Phaclofen-sensitive GABA-B receptors do not mediate excitatory effects of baclofen on gastric secretion.
    Pharmacology, 1991, Volume: 42, Issue:3

    Topics: Animals; Baclofen; Gastric Fundus; Gastric Juice; Injections, Intravenous; Injections, Intraventricular; Male; Pylorus; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Ethanol-induced changes in chloride flux are mediated by both GABA(A) and GABA(B) receptors.
    Alcoholism, clinical and experimental research, 1991, Volume: 15, Issue:2

    Topics: Alcohol Drinking; Animals; Baclofen; Bicuculline; Cerebral Cortex; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Drug Synergism; Ethanol; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Receptors, GABA-A

1991
CGP 35348, a new GABAB antagonist, prevents antinociception and muscle-relaxant effect induced by baclofen.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Analgesics; Animals; Baclofen; GABA Antagonists; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Mice; Morphine; Muscle Relaxation; Muscles; Organophosphorus Compounds; Oxotremorine; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time

1991
Effects of GABA and related agents on the electrical activity of hypothalamic ventromedial nucleus neurons in vitro.
    Experimental brain research, 1991, Volume: 85, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Electrophysiology; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Neurons; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ventromedial Hypothalamic Nucleus

1991
Effects of phaclofen and the enantiomers of baclofen on cardiovascular responses to intrathecal administration of L- and D-baclofen in the rat.
    European journal of pharmacology, 1991, Apr-24, Volume: 196, Issue:3

    Topics: Animals; Baclofen; Blood Pressure; Cardiovascular System; Drug Interactions; GABA-A Receptor Antagonists; Heart Rate; Injections, Spinal; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Time Factors

1991
Phaclofen-reversible effects of GABA in the spinal cord of the rat.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heart Rate; Injections, Spinal; Lidocaine; Male; Rats; Rats, Inbred Strains; Spinal Cord; Stereoisomerism; Sympathetic Nervous System

1991
Blockade of GABAA receptors in the region of the anterior basolateral amygdala of rats elicits increases in heart rate and blood pressure.
    Brain research, 1991, Dec-13, Volume: 567, Issue:1

    Topics: Amygdala; Analysis of Variance; Anesthesia, General; Animals; Baclofen; Bicuculline; Blood Pressure; Consciousness; Dose-Response Relationship, Drug; Electroencephalography; Heart Rate; Hippocampus; Male; Microinjections; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Strychnine; Temporal Lobe

1991
Inhibition of protein kinase activity enhances long-term potentiation of hippocampal IPSPs.
    Neuroreport, 1991, Volume: 2, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Acetates; Acetic Acid; Animals; Baclofen; Carbazoles; Evoked Potentials; Guinea Pigs; Hippocampus; In Vitro Techniques; Indole Alkaloids; Neurons; Picrotoxin; Potentiometry; Protein Kinase C; Pyramidal Tracts; Quinoxalines; Sesterterpenes

1991
Gamma-aminobutyric acid (GABAB) receptor-mediated inhibition of tyrosine hydroxylase activity in the striatum of rat.
    Neuropharmacology, 1991, Volume: 30, Issue:10

    Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Baclofen; Calcium; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; gamma-Aminobutyric Acid; Hydrazines; In Vitro Techniques; Male; Muscimol; Neural Pathways; Picrotoxin; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Tyrosine 3-Monooxygenase

1991
Postsynaptic potentials mediated by excitatory and inhibitory amino acids in interneurons of stratum pyramidale of the CA1 region of rat hippocampal slices in vitro.
    Journal of neurophysiology, 1991, Volume: 66, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Amino Acids; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Interneurons; Male; Membrane Potentials; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Synapses

1991
GABAB receptor modulation of the release of substance P from capsaicin-sensitive neurones in the rat trachea in vitro.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Capsaicin; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Neurons; Potassium; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substance P; Taurine; Trachea

1991
Regulation of cardiovascular sympathetic neurons by substance P and gamma-aminobutyric acid in the rat spinal cord.
    European journal of pharmacology, 1991, Sep-04, Volume: 202, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Capsaicin; Cardiovascular Physiological Phenomena; Cardiovascular System; Catecholamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Heart Rate; Injections, Spinal; Male; Muscimol; Neurons; Neuropeptide Y; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Substance P; Sympathetic Nervous System

1991
GABAB-receptor-mediated inhibition of the N-methyl-D-aspartate component of synaptic transmission in the rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1991, Volume: 11, Issue:1

    Topics: Animals; Baclofen; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Picrotoxin; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

1991
Effects of baclofen and bicuculline on inhibition in the fascia dentata and hippocampus regio superior.
    Brain research, 1991, Jan-04, Volume: 538, Issue:1

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; Hippocampus; Interneurons; Iontophoresis; Male; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synapses

1991
Antagonism of baclofen-induced antinociception by intrathecal administration of phaclofen or 2-hydroxy-saclofen, but not delta-aminovaleric acid in the rat.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Amino Acids; Amino Acids, Neutral; Analgesia; Animals; Baclofen; Injections, Spinal; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Effect of intracerebroventricular administration of the GABAB-receptor agonist baclofen on operant feeding in satiated pigs.
    British journal of pharmacology, 1990, Volume: 101, Issue:3

    Topics: Animals; Baclofen; Central Nervous System; Conditioning, Operant; Drinking Behavior; Feeding Behavior; Female; Injections, Intraventricular; Male; Receptors, GABA-A; Satiation; Swine

1990
Electrophysiological characterization of potent agonists and antagonists at pre- and postsynaptic GABAB receptors on neurones in rat brain slices.
    British journal of pharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Brain; Corpus Striatum; Electrophysiology; GABA-A Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Neurons; Organophosphorus Compounds; Rats; Receptors, GABA-A; Substantia Nigra; Synapses

1990
The effect of intracerebroventricular administration of baclofen on food intake in rats.
    Neuroreport, 1990, Volume: 1, Issue:1

    Topics: Animals; Ataxia; Baclofen; Brain; Dose-Response Relationship, Drug; Eating; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
GABAA and GABAB antagonists prevent the opioid inhibition of endogenous acetylcholine release evoked by glutamate from rat neostriatal slices.
    Neuroscience letters, 1990, Dec-11, Volume: 120, Issue:2

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; GABA Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Morphine; Narcotics; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Spinal 5-HT3 receptor-mediated antinociception: possible release of GABA.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1991, Volume: 11, Issue:7

    Topics: Analgesia; Animals; Baclofen; Behavior, Animal; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; N-Methylaspartate; Neurons; Nociceptors; Pain Measurement; Picrotoxin; Receptors, Serotonin; Serotonin; Spinal Cord

1991
Actions of baclofen and phaclofen upon ON- and OFF-ganglion cells in the cat retina.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Cats; Iontophoresis; Microelectrodes; Muscimol; Retinal Ganglion Cells

1990
Enhancement of NMDA receptor-mediated synaptic potential evoked in rat medial-amygdala neuron following olfactory bulbectomy.
    Brain research, 1990, Nov-05, Volume: 532, Issue:1-2

    Topics: Action Potentials; Amygdala; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; In Vitro Techniques; Kynurenic Acid; Male; Membrane Potentials; Neurons; Olfactory Bulb; Organophosphorus Compounds; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Synapses

1990
GABA terminal autoreceptors in the pars compacta and in the pars reticulata of the rat substantia nigra are GABAB.
    European journal of pharmacology, 1990, Jan-10, Volume: 175, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; gamma-Aminobutyric Acid; Male; Muscimol; Nipecotic Acids; Potassium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Synaptosomes; Tritium

1990
Central GABAA excitatory and GABAB inhibitory receptors regulate gastric acid secretion in rats.
    European journal of pharmacology, 1990, Feb-27, Volume: 177, Issue:3

    Topics: Anesthesia; Animals; Baclofen; Bicuculline; Central Nervous System; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Gastric Acid; Injections, Intraventricular; Male; Muscimol; Pylorus; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Phaclofen-insensitive presynaptic inhibitory action of (+/-)-baclofen in neonatal rat motoneurones in vitro.
    British journal of pharmacology, 1990, Volume: 99, Issue:2

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Evoked Potentials; Glutamates; In Vitro Techniques; Membrane Potentials; Motor Neurons; Nipecotic Acids; Potassium Channels; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereotyped Behavior; Synapses

1990
Thioether analogues of baclofen, phaclofen and saclofen.
    Neuroscience letters, 1990, May-04, Volume: 112, Issue:2-3

    Topics: Animals; Baclofen; Binding, Competitive; Cerebellum; Guinea Pigs; Ileum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vas Deferens

1990
(+)-Hydrastine, a potent competitive antagonist at mammalian GABAA receptors.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Baclofen; Benzylisoquinolines; Bicuculline; Binding, Competitive; Brain Chemistry; Convulsants; Diazepam; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Membranes; Muscimol; Muscle, Smooth; Muscle, Smooth, Vascular; Rats; Receptors, GABA-A; Stereoisomerism

1990
Inhibition of baclofen binding to rat cerebellar membranes by phaclofen, saclofen, 3-aminopropylphosphonic acid and related GABAB receptor antagonists.
    Neuroscience letters, 1990, May-18, Volume: 113, Issue:1

    Topics: Animals; Baclofen; Cerebellum; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Propylamines; Rats; Rats, Inbred Strains

1990
Gamma-aminobutyric acid-A and -B receptor antagonists increase luteinizing hormone-releasing hormone neuronal responsiveness to intracerebroventricular norepinephrine in ovariectomized estrogen-treated rats.
    Endocrinology, 1990, Volume: 127, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Estradiol; Female; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Hypothalamus; Kinetics; Luteinizing Hormone; Neurons; Norepinephrine; Ovariectomy; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Paired-pulse depression of monosynaptic GABA-mediated inhibitory postsynaptic responses in rat hippocampus.
    The Journal of physiology, 1990, Volume: 424

    Topics: Action Potentials; Animals; Baclofen; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Picrotoxin; Rats; Synapses; Synaptic Transmission; Tetrodotoxin

1990
Are GABAB receptors involved in the pharmacological effects of ethanol?
    European journal of pharmacology, 1990, Jul-17, Volume: 182, Issue:3

    Topics: Animals; Baclofen; Cells, Cultured; Chlorine; Diazepam; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; N-Methylaspartate; Picrotoxin; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Spinal Cord

1990
The effects of baclofen and two GABAB-receptor antagonists on long-term potentiation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:2

    Topics: Animals; Baclofen; Electric Stimulation; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Male; Neurons; Organophosphorus Compounds; Rats; Rats, Inbred Strains; Synapses

1990
Phaclofen antagonizes the antinociceptive but not the sedative effects of (-)-baclofen.
    Progress in neuro-psychopharmacology & biological psychiatry, 1990, Volume: 14, Issue:4

    Topics: Analgesics; Animals; Baclofen; Behavior, Animal; Electrocardiography; Hypnotics and Sedatives; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscle Relaxants, Central; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Stereoisomerism

1990
Involvement of GABA receptors in the regulation of neurite growth in cultured embryonic chick tectum.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1990, Volume: 8, Issue:4

    Topics: Animals; Axons; Baclofen; Cells, Cultured; Chick Embryo; Culture Media; gamma-Aminobutyric Acid; Isoxazoles; Ligands; Muscimol; Receptors, GABA-A; Superior Colliculi

1990
Endogenous GABA acts on GABAB receptors in nucleus tractus solitarius to increase blood pressure.
    Brain research, 1990, Sep-03, Volume: 526, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Medulla Oblongata; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vigabatrin

1990
Effect of 2-hydroxy-saclofen, an antagonist of GABAB action, upon the binding of baclofen and other receptor ligands in rat cerebrum.
    Brain research, 1990, Sep-03, Volume: 526, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Baclofen; Brain; GABA Antagonists; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1990
CGP 35348: a centrally active blocker of GABAB receptors.
    European journal of pharmacology, 1990, Oct-02, Volume: 187, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Animals, Newborn; Anticonvulsants; Baclofen; Behavior, Animal; Brain Chemistry; Cyclic AMP; Electrophysiology; Hippocampus; In Vitro Techniques; Iontophoresis; Organophosphorus Compounds; Postural Balance; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord

1990
GABA(B)-related activity involved in synaptic processing of somatosensory information in S1 cortex of the anaesthetized cat.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Anesthesia; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrodes; Female; gamma-Aminobutyric Acid; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Physical Stimulation; Somatosensory Cortex; Synapses

1990
Endogenous GABA mediates presynaptic inhibition of spontaneous and evoked excitatory synaptic potentials in the rat neostriatum.
    Neuroscience letters, 1990, Oct-02, Volume: 118, Issue:1

    Topics: Animals; Baclofen; Corpus Striatum; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Synapses; Tetrodotoxin

1990
Bicuculline and picrotoxin block phase advances induced by GABA agonists in the circadian rhythm of locomotor activity in the golden hamster by a phaclofen-insensitive mechanism.
    Brain research, 1990, Oct-22, Volume: 530, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Circadian Rhythm; Cricetinae; gamma-Aminobutyric Acid; Male; Mesocricetus; Microinjections; Motor Activity; Muscimol; Picrotoxin; Stereotaxic Techniques; Triazolam

1990
Epileptiform activity in microcultures containing small numbers of hippocampal neurons.
    Journal of neurophysiology, 1990, Volume: 64, Issue:5

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Cells, Cultured; Epilepsy; Evoked Potentials; Hippocampus; Kynurenic Acid; Neurons; Rats; Synapses

1990
Effects of excitatory and inhibitory amino acid agonists and antagonists of ventral horn cells in slices of spinal cord isolated from adult rats.
    Neuropharmacology, 1990, Volume: 29, Issue:12

    Topics: Action Potentials; Amino Acids; Animals; Anterior Horn Cells; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Strychnine; Synapses

1990
Effects of GABA antagonists and structural GABA analogues on baclofen stimulated gastric acid secretion in the rat.
    Japanese journal of pharmacology, 1990, Volume: 52, Issue:2

    Topics: Amino Acids; Anesthesia; Animals; Baclofen; Bethanechol Compounds; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Gastric Acid; Male; Rats; Rats, Inbred Strains

1990
Phaclofen antagonizes post-tetanic disinhibition in the rat dentate gyrus.
    Neuroscience letters, 1990, Mar-02, Volume: 110, Issue:1-2

    Topics: Animals; Baclofen; Electric Stimulation; Hippocampus; In Vitro Techniques; Male; Neural Inhibition; Rats; Rats, Inbred Strains

1990
On the presynaptic action of baclofen at inhibitory synapses between cultured rat hippocampal neurones.
    The Journal of physiology, 1990, Volume: 422

    Topics: Action Potentials; Animals; Baclofen; Calcium; Cells, Cultured; gamma-Aminobutyric Acid; Hippocampus; Neurons; Pertussis Toxin; Rats; Synapses; Virulence Factors, Bordetella

1990
Phaclofen inhibition of the slow inhibitory postsynaptic potential in hippocampal slice cultures: a possible role for the GABAB-mediated inhibitory postsynaptic potential.
    Neuroscience, 1990, Volume: 35, Issue:1

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neural Inhibition; Organ Culture Techniques; Rats

1990
GABAB-receptor-mediated actions of baclofen in rat isolated neocortical slice preparations: antagonism by phosphono-analogues of GABA.
    Brain research, 1989, Feb-20, Volume: 480, Issue:1-2

    Topics: Animals; Baclofen; Cerebral Cortex; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Propylamines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
GABAB autoreceptors in rat cortex synaptosomes: response under different depolarizing and ionic conditions.
    European journal of pharmacology, 1989, Mar-07, Volume: 172, Issue:1

    Topics: Animals; Baclofen; Calcium; Cerebral Cortex; In Vitro Techniques; Male; Muscimol; Neuromuscular Depolarizing Agents; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes; Veratrine

1989
Inhibitory processes in normal and epileptic-like rat hippocampal slices: the role of GABAB receptors.
    European journal of pharmacology, 1989, Apr-25, Volume: 163, Issue:2-3

    Topics: Animals; Baclofen; Bicuculline; Epilepsy; Hippocampus; In Vitro Techniques; Male; Penicillins; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
GABAB receptor mediated effects on central respiratory system and their antagonism by phaclofen.
    Neuroscience letters, 1989, May-08, Volume: 99, Issue:3

    Topics: Animals; Baclofen; Phrenic Nerve; Rabbits; Receptors, GABA-A; Reference Values; Respiration; Vagotomy

1989
3-Aminopropylphosphinic acid--a potent, selective GABAB receptor agonist in the guinea-pig ileum and rat anococcygeus muscle.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Animals; Baclofen; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscles; Organophosphorus Compounds; Parasympathetic Nervous System; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Stimulation by phaclofen of inositol 1,4,5-triphosphate production in cultured neurons from chick tectum.
    European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3

    Topics: Animals; Baclofen; Chick Embryo; gamma-Aminobutyric Acid; Inosine Nucleotides; Inosine Triphosphate; Isoxazoles; Neurons; Receptors, GABA-A; Superior Colliculi

1989
Effects of the putative antagonists phaclofen and delta-aminovaleric acid on GABAB receptor biochemistry.
    British journal of pharmacology, 1989, Volume: 98, Issue:3

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Cerebral Cortex; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Kinetics; Male; Proteins; Radioligand Assay; Rats; Receptors, GABA-A

1989
A new alcohol antagonist: phaclofen.
    Life sciences, 1989, Volume: 45, Issue:19

    Topics: Animals; Baclofen; Behavior, Animal; Body Temperature; Ethanol; GABA-A Receptor Antagonists; Male; Mice; Mice, Inbred ICR; Motor Activity; Receptors, GABA-A; Sleep

1989
A novel type of GABA receptor in rat spinal cord?
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:6

    Topics: Animals; Baclofen; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Synaptosomes

1989
Late inhibitory postsynaptic potentials in rat prefrontal cortex may be mediated by GABAB receptors.
    Experientia, 1989, Feb-15, Volume: 45, Issue:2

    Topics: Animals; Baclofen; Electric Conductivity; Electric Stimulation; Evoked Potentials; Frontal Lobe; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Isoxazoles; Male; Membrane Potentials; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synapses

1989
Bicuculline- and phaclofen-sensitive components of N-methyl-D-aspartate-induced hyperpolarizations in rat dorsolateral septal nucleus neurones.
    The Journal of physiology, 1989, Volume: 418

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Baclofen; Bicuculline; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Membrane Potentials; N-Methylaspartate; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Septal Nuclei; Tetrodotoxin

1989
Control of epileptiform burst rate by CA3 hippocampal cell afterhyperpolarizations in vitro.
    Brain research, 1989, Jul-17, Volume: 492, Issue:1-2

    Topics: Action Potentials; Animals; Baclofen; Epilepsy; Hippocampus; In Vitro Techniques; Membrane Potentials; Phorbol Esters; Potassium; Rats

1989
Rhythmical bursting activity and GABAergic mechanisms in the medial septum of normal and pertussis toxin-pretreated rats.
    Experimental brain research, 1989, Volume: 77, Issue:2

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Hippocampus; Male; Neurons; Nipecotic Acids; Pertussis Toxin; Proline; Rats; Rats, Inbred Strains; Septum Pellucidum; Virulence Factors, Bordetella

1989
Baclofen and phaclofen modulate GABA release from slices of rat cerebral cortex and spinal cord but not from retina.
    British journal of pharmacology, 1989, Volume: 98, Issue:1

    Topics: Amino Acids; Aminocaproates; Aminolevulinic Acid; Animals; Baclofen; Calcium; Cerebral Cortex; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Potassium; Rats; Rats, Inbred Strains; Retina; Spinal Cord; Vigabatrin

1989
Phaclofen antagonizes the depressant effect of baclofen on spinal reflex transmission in rats.
    Brain research, 1989, Sep-04, Volume: 496, Issue:1-2

    Topics: Animals; Baclofen; H-Reflex; Male; Neural Inhibition; Rats; Rats, Inbred Strains; Reflex, Monosynaptic; Spinal Cord

1989
A physiological role for GABAB receptors in the central nervous system.
    Nature, 1988, Mar-10, Volume: 332, Issue:6160

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Potassium; Rats; Receptors, GABA-A; Serotonin; Synapses

1988
The GABAB antagonist phaclofen inhibits the late K+-dependent IPSP in cat and rat thalamic and hippocampal neurones.
    Brain research, 1988, May-17, Volume: 448, Issue:2

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Geniculate Bodies; Hippocampus; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Phaclofen: a GABAB blocker reduces long-duration inhibition in the neocortex.
    European journal of pharmacology, 1988, Apr-13, Volume: 148, Issue:3

    Topics: Animals; Baclofen; Cerebral Cortex; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
GABAA and GABAB receptors in locus coeruleus: effects of blockers.
    European journal of pharmacology, 1988, Apr-27, Volume: 149, Issue:1-2

    Topics: Animals; Baclofen; In Vitro Techniques; Locus Coeruleus; Male; Muscimol; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Phaclofen antagonizes baclofen-induced suppression of visually evoked responses in the cat's striate cortex.
    Brain research, 1988, Nov-01, Volume: 463, Issue:2

    Topics: Animals; Baclofen; Cats; Evoked Potentials, Visual; gamma-Aminobutyric Acid; Receptors, GABA-A; Visual Cortex

1988
Evidence for pharmacologically distinct subsets of GABAB receptors.
    Brain research bulletin, 1988, Volume: 21, Issue:3

    Topics: Animals; Baclofen; Binding, Competitive; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Propylamines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Phaclofen antagonizes GABA at autoreceptors regulating release in rat cerebral cortex.
    European journal of pharmacology, 1988, Sep-13, Volume: 154, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; GABA Antagonists; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1988
Phaclofen: a peripheral and central baclofen antagonist.
    Brain research, 1987, Mar-03, Volume: 405, Issue:1

    Topics: Animals; Baclofen; Cats; Cholinergic Fibers; Colon; Guinea Pigs; Ileum; In Vitro Techniques; Interneurons; Intestines; Receptors, GABA-A; Spinal Cord; Synaptic Transmission

1987
Intracerebroventricular phaclofen antagonizes baclofen antinociceptive activity in hot plate test with mice.
    European journal of pharmacology, 1988, Sep-13, Volume: 154, Issue:2

    Topics: Analgesics; Animals; Baclofen; Injections, Intraventricular; Male; Mice; Reaction Time; Time Factors

1988
Comparison of antagonism by phaclofen of baclofen induced hyperpolarizations and synaptically mediated late hyperpolarizing potentials recorded intracellularly from rat dorsolateral septal neurons.
    Neuroscience letters, 1988, Mar-21, Volume: 86, Issue:1

    Topics: Animals; Baclofen; In Vitro Techniques; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Septal Nuclei

1988
Long-term synaptic transformation of hippocampal CA1 gamma-aminobutyric acid synapses and the effect of anandamide.
    Proceedings of the National Academy of Sciences of the United States of America, 1995, Oct-24, Volume: 92, Issue:22

    Topics: Animals; Arachidonic Acids; Baclofen; Calcium Channel Blockers; Chloride Channels; Endocannabinoids; Furosemide; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Models, Neurological; Polyunsaturated Alkamides; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Snails; Synapses; Synaptic Transmission

1995
Bicuculline enhances the late GABAB receptor-mediated paired-pulse inhibition observed in rat hippocampal slices.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Electric Stimulation; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Neurons; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B

1995
Regulation of the prefrontal cortical dopamine release by GABAA and GABAB receptor agonists and antagonists.
    Brain research, 1993, Dec-10, Volume: 630, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Microdialysis; Muscimol; Nomifensine; Picrotoxin; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B

1993
Characterization of GABAB ligands in vivo.
    General pharmacology, 1995, Volume: 26, Issue:2

    Topics: Animals; Baclofen; beta-Alanine; Drug Interactions; Female; GABA Antagonists; GABA-B Receptor Antagonists; Ligands; Mice; Mice, Inbred BALB C; Muscle Relaxation; Organophosphorus Compounds

1995
A depolarizing inhibitory response to GABA in brainstem auditory neurons of the chick.
    Brain research, 1995, Apr-17, Volume: 677, Issue:1

    Topics: Animals; Baclofen; Basal Ganglia; Bicuculline; Brain Stem; Chickens; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Neuromuscular Depolarizing Agents; Neurons, Afferent; Patch-Clamp Techniques

1995
GABAA receptor-mediated inhibition of N-methyl-D-aspartate-evoked [3H]dopamine release from mesencephalic cell cultures.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Baclofen; Cells, Cultured; Dopamine; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Kainic Acid; Mesencephalon; Muscimol; N-Methylaspartate; Picrotoxin; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA; Ventral Tegmental Area

1994
2-Hydroxy-saclofen causes a phaclofen-reversible reduction in population spike amplitude in the rat hippocampal slice.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Animals; Baclofen; Bicuculline; Evoked Potentials; GABA Antagonists; Hippocampus; Male; Microelectrodes; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B; Synaptic Transmission

1995
Presynaptic gamma-hydroxybutyric acid (GHB) and gamma-aminobutyric acidB (GABAB) receptor-mediated release of GABA and glutamate (GLU) in rat thalamic ventrobasal nucleus (VB): a possible mechanism for the generation of absence-like seizures induced by GH
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 273, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Epilepsy, Absence; Extracellular Space; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Organophosphorus Compounds; Potassium; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, GABA-B; Sodium Oxybate; Thalamic Nuclei

1995
Pharmacology of the GABAB receptor in amphibian retina.
    Brain research, 1994, Oct-17, Volume: 660, Issue:2

    Topics: Ambystoma; Animals; Baclofen; Butylamines; Evoked Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Necturus; Organophosphorus Compounds; Propylamines; Receptors, GABA-B; Retina; Retinal Ganglion Cells; Stereoisomerism; Structure-Activity Relationship

1994
Characterization of the GABA autoreceptor in human neocortex as a pharmacological subtype of the GABAB receptor.
    European journal of pharmacology, 1994, Oct-03, Volume: 263, Issue:3

    Topics: Adolescent; Adult; Aged; Animals; Baclofen; Benzylamines; Binding, Competitive; Brain Neoplasms; Cerebral Cortex; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Humans; Male; Middle Aged; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B

1994
Paired-pulse depression of the N-methyl-D-aspartate receptor-mediated synaptic potentials in the amygdala.
    British journal of pharmacology, 1994, Volume: 113, Issue:3

    Topics: Amygdala; Animals; Baclofen; In Vitro Techniques; Male; Potassium; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

1994
The effects of GABAB ligands on alcohol withdrawal in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:3

    Topics: Animals; Baclofen; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; GABA-B Receptor Antagonists; Mice; Mice, Inbred C57BL; Organophosphorus Compounds; Phenylalanine; Receptors, GABA-B; Seizures; Substance Withdrawal Syndrome; Tremor

1994
Spatiotemporally differential inhibition of pyramidal cells in the cat motor cortex.
    Journal of neurophysiology, 1994, Volume: 71, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Axons; Baclofen; Bicuculline; Cats; Electric Stimulation; Interneurons; Membrane Potentials; Microelectrodes; Motor Cortex; Pyramidal Cells; Quinoxalines; Synapses

1994
Medial vestibular neurons are endogenous pacemakers whose discharge is modulated by neurotransmitters.
    Cellular and molecular neurobiology, 1993, Volume: 13, Issue:6

    Topics: Amino Acids; Animals; Baclofen; Bicuculline; Calcium; In Vitro Techniques; Kynurenic Acid; Magnesium; Male; Membrane Potentials; Nerve Fibers; Neurons; Neurotransmitter Agents; Rats; Rats, Wistar; Receptors, GABA-A; Synapses; Vestibular Nuclei

1993
Phosphorylation of DARPP-32 is regulated by GABA in rat striatum and substantia nigra.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine and cAMP-Regulated Phosphoprotein 32; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra

1994
Pharmacological discrimination between gamma-aminobutyric acid type B receptors regulating cholecystokinin and somatostatin release from rat neocortex synaptosomes.
    Molecular pharmacology, 1994, Volume: 46, Issue:3

    Topics: Animals; Baclofen; Benzylamines; Cerebral Cortex; Cholecystokinin; GABA Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ligands; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes

1994
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
    Hippocampus, 1994, Volume: 4, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus

1994
Inhibitory mechanisms terminating paroxysmal depolarization shifts in hippocampal neurons of rats.
    Neuroscience letters, 1994, Jul-18, Volume: 176, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Calcium; Egtazic Acid; GABA Antagonists; Hippocampus; In Vitro Techniques; Magnesium; Membrane Potentials; Neurons; Penicillins; Potassium Channel Blockers; Potassium Channels; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Tetraethylammonium; Tetraethylammonium Compounds

1994
GABAB antagonists: resolution, absolute stereochemistry, and pharmacology of (R)- and (S)-phaclofen.
    Chirality, 1994, Volume: 6, Issue:7

    Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; Crystallography, X-Ray; GABA Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Models, Molecular; Molecular Conformation; Molecular Structure; Rats; Stereoisomerism; Structure-Activity Relationship

1994
Stimulation of GABAB receptors in the basal forebrain selectively impairs working memory of rats in the double Y-maze.
    Brain research, 1994, Mar-28, Volume: 641, Issue:1

    Topics: Animals; Baclofen; Exploratory Behavior; Male; Memory; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Stereoisomerism; Substantia Innominata

1994
Release of endogenous glutamic and aspartic acids from cerebrocortex synaptosomes and its modulation through activation of a gamma-aminobutyric acidB (GABAB) receptor subtype.
    Brain research, 1993, Feb-26, Volume: 604, Issue:1-2

    Topics: Animals; Aspartic Acid; Baclofen; Bicuculline; Cerebral Cortex; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Kinetics; Male; Organophosphorus Compounds; Picrotoxin; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptosomes

1993
GABAB autoreceptors mediate activity-dependent disinhibition and enhance signal transmission in the dentate gyrus.
    Journal of neurophysiology, 1993, Volume: 69, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Culture Techniques; GABA-A Receptor Antagonists; Hippocampus; Male; Membrane Potentials; Nerve Fibers; Neural Inhibition; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Theta Rhythm

1993
Intrathecal GABAB antagonists attenuate the antinociception produced by microinjection of L-glutamate into the ventromedial medulla of the rat.
    Brain research, 1993, Apr-02, Volume: 607, Issue:1-2

    Topics: Analgesics; Animals; Baclofen; Basal Ganglia; Behavior, Animal; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glutamates; Glutamic Acid; Injections, Spinal; Medulla Oblongata; Methysergide; Microinjections; Organophosphorus Compounds; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Skin Temperature

1993
GABA mediation of the dual effects of somatostatin on guinea pig ileal myenteric cholinergic transmission.
    The American journal of physiology, 1993, Volume: 264, Issue:5 Pt 1

    Topics: Acetylcholine; Adenylate Cyclase Toxin; Animals; Baclofen; Bicuculline; Cholecystokinin; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Pertussis Toxin; Receptors, GABA-A; Somatostatin; Virulence Factors, Bordetella

1993
L-2-amino-4-phosphonobutanoic acid and 1S,3R-1-aminocyclopentane-1,3-dicarboxylic acid reduce paired-pulse depression recorded from medial perforant path in the dentate gyrus of rat hippocampal slices.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Aminobutyrates; Animals; Atropine; Baclofen; Carbachol; Cycloleucine; Depression, Chemical; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Neural Pathways; Neurotransmitter Uptake Inhibitors; Picrotoxin; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Theophylline

1993
Hyperpolarizing synaptic potentials evoked in CA1 pyramidal cells by glutamate stimulation of interneurons from the oriens/alveus border of rat hippocampal slices. II. Sensitivity to GABA antagonists.
    Hippocampus, 1993, Volume: 3, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Electrophysiology; Evoked Potentials; GABA Antagonists; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Neurons; Rats; Synapses

1993
Different effects of omega-conotoxin GVIA at excitatory and inhibitory synapses in rat CA1 hippocampal neurons.
    Brain research, 1993, Jul-09, Volume: 616, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Mollusk Venoms; Neurons; omega-Conotoxin GVIA; Peptides; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Synapses

1993
Enteric GABA-containing nerves projecting to the guinea-pig inferior mesenteric ganglion modulate acetylcholine release.
    The Journal of physiology, 1993, Volume: 471

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Colon; Diazepam; Electric Stimulation; gamma-Aminobutyric Acid; Ganglia, Sympathetic; Guinea Pigs; In Vitro Techniques; Male; Mesentery; Muscimol; Neural Pathways; Receptors, GABA-A; Receptors, GABA-B; Splanchnic Nerves; Synaptic Transmission

1993
The role of GABA receptors in the control of the omasal myoelectrical activity in sheep.
    Research in veterinary science, 1994, Volume: 56, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Female; GABA Antagonists; Muscimol; Myoelectric Complex, Migrating; Omasum; Receptors, GABA; Sheep

1994
The development of GABAB-mediated activity in the rat dentate gyrus.
    Brain research. Developmental brain research, 1994, Feb-18, Volume: 77, Issue:2

    Topics: Animals; Baclofen; Electric Stimulation; Evoked Potentials; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Organophosphorus Compounds; Rats; Receptors, GABA-A; Receptors, GABA-B

1994
Differential effects of muscimol microinjection into dorsal and ventral aspects of the premotor cortex of monkeys.
    Journal of neurophysiology, 1994, Volume: 71, Issue:3

    Topics: Animals; Appetitive Behavior; Attention; Baclofen; Brain Mapping; Macaca; Male; Membrane Potentials; Microinjections; Motor Cortex; Motor Skills; Muscimol; Neurons; Orientation; Psychomotor Performance; Receptors, GABA-A

1994
Microiontophoresis of baclofen on membrane potential and input resistance in bulbar respiratory neurons in the cat.
    Brain research, 1993, Sep-17, Volume: 622, Issue:1-2

    Topics: Action Potentials; Animals; Baclofen; Cats; Iontophoresis; Medulla Oblongata; Membrane Potentials; Neurons; Respiratory System; Tetrodotoxin

1993
Evidence that changes in the function of the subtypes of the receptors for gamma-amino butyric acid may be involved in the seasonal changes in the negative-feedback effects of estrogen on gonadotropin-releasing hormone secretion and plasma luteinizing hor
    Endocrinology, 1993, Volume: 133, Issue:6

    Topics: Animals; Baclofen; Bicuculline; Estrogens; Feedback; Female; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Muscimol; Receptors, GABA; Seasons; Sheep

1993
Electrophysiological identification of horizontal synaptic connections in rat visual cortex in vitro.
    Neuroscience letters, 1993, Dec-12, Volume: 163, Issue:2

    Topics: Animals; Baclofen; Calcium; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kynurenic Acid; Magnesium; Quinoxalines; Rats; Receptors, GABA-B; Synapses; Synaptic Transmission; Visual Cortex

1993
GABA induces Ca2+ transients in astrocytes.
    Neuroscience, 1993, Volume: 54, Issue:3

    Topics: Animals; Astrocytes; Baclofen; Bicuculline; Calcium; Cells, Cultured; Cerebral Cortex; Cytosol; gamma-Aminobutyric Acid; Immunohistochemistry; Muscimol; Nicotinic Acids; Nifedipine; Rats

1993
Influence of GABA on neurons of the gustatory zone of the rat nucleus of the solitary tract.
    Brain research, 1993, Jul-09, Volume: 616, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Brain Mapping; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Male; Medulla Oblongata; Membrane Potentials; Muscimol; Neurons; Perfusion; Rats; Taste; Tetrodotoxin

1993
Analysis of gamma-aminobutyric acidB receptor function in the in vitro and in vivo regulation of alpha-melanotropin-stimulating hormone secretion from melanotrope cells of Xenopus laevis.
    Endocrinology, 1993, Volume: 132, Issue:2

    Topics: alpha-MSH; Animals; Baclofen; Butylamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Homeostasis; In Vitro Techniques; Kinetics; Organophosphorus Compounds; Perfusion; Pituitary Gland, Posterior; Radioimmunoassay; Receptors, GABA-A; Xenopus laevis

1993
The spinal GABA system modulates burst frequency and intersegmental coordination in the lamprey: differential effects of GABAA and GABAB receptors.
    Journal of neurophysiology, 1993, Volume: 69, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Culture Techniques; Diazepam; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Lampreys; Locomotion; Motor Neurons; Muscimol; Muscles; N-Methylaspartate; Nerve Net; Neurons; Nipecotic Acids; Proline; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Spinal Nerve Roots; Synaptic Transmission

1993
gamma-Aminobutyric acid (GABA) autoreceptors in rat cerebral cortex and spinal cord represent pharmacologically distinct subtypes of the GABAB receptor.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: Animals; Baclofen; Cerebral Cortex; gamma-Aminobutyric Acid; Male; Organophosphorus Compounds; Potassium; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Synaptosomes

1993
GABA receptor subtypes involved in the neuronal mechanisms of baroreceptor reflex in the nucleus tractus solitarii of rabbits.
    Journal of the autonomic nervous system, 1993, Volume: 43, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Brain Stem; Electrophysiology; gamma-Aminobutyric Acid; Male; Neurons; Phenylephrine; Pressoreceptors; Rabbits; Receptors, GABA-A

1993
Pre- and postsynaptic GABAB receptors of rat neocortical neurons differ in their pharmacological properties.
    Neuroscience letters, 1993, May-14, Volume: 154, Issue:1-2

    Topics: Animals; Baclofen; Cerebral Cortex; Electric Stimulation; Feedback; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Membrane Potentials; Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

1993
Inhibitory effects of cholecystokinin on rat's geniculate activity can be blocked by GABA-antagonists.
    Neuroscience letters, 1995, Sep-01, Volume: 197, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Cholecystokinin; Extracellular Space; GABA Antagonists; Geniculate Bodies; Interneurons; Iontophoresis; Male; Rats; Rats, Wistar; Trypan Blue

1995
GABA transport and calcium dynamics in horizontal cells from the skate retina.
    The Journal of physiology, 1995, Nov-01, Volume: 488 ( Pt 3)

    Topics: Animals; Baclofen; Bicuculline; Biological Transport; Calcium; Calcium Channel Blockers; Dantrolene; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Muscle Relaxants, Central; Nifedipine; Picrotoxin; Retina; Skates, Fish

1995
GABAA receptor-mediated feedback inhibition in pyramidal neurons of cat motor cortex.
    Neuroscience letters, 1995, Sep-29, Volume: 198, Issue:2

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Cats; Dendrites; Feedback; Female; GABA Antagonists; Male; Motor Cortex; Neurotransmitter Agents; Patch-Clamp Techniques; Potassium Chloride; Pyramidal Cells; Receptors, GABA-A

1995
Attenuation by valproate of c-fos immunoreactivity in trigeminal nucleus caudalis induced by intracisternal capsaicin.
    British journal of pharmacology, 1995, Volume: 116, Issue:8

    Topics: Animals; Baclofen; Bicuculline; Brain Stem; Capsaicin; GABA Agents; GABA Antagonists; Guinea Pigs; Injections, Intraventricular; Male; Proto-Oncogene Proteins c-fos; Trigeminal Nuclei; Valproic Acid

1995
Actions of the anticonvulsant agent 2-amino-4-phosphonobutyrate on the release of [3H]D-aspartate from rat forebrain slices.
    Biochemical Society transactions, 1996, Volume: 24, Issue:2

    Topics: Aminobutyrates; Animals; Anticonvulsants; Aspartic Acid; Baclofen; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isomerism; Kynurenic Acid; Prosencephalon; Rats

1996
Effects of GABAergic drugs on physostigmine-induced yawning in rats.
    Psychopharmacology, 1995, Volume: 122, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Cholinesterase Inhibitors; Drug Interactions; GABA Agonists; GABA Antagonists; Male; Muscimol; Physostigmine; Picrotoxin; Rats; Rats, Wistar; Yawning

1995
Role of peripheral GABAB receptors in the regulation of pepsinogen secretion in anaesthetized rats.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Anesthesia; Animals; Baclofen; Capsaicin; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gastric Mucosa; Male; Organophosphorus Compounds; p-Methoxy-N-methylphenethylamine; Pepsinogens; Perfusion; Rats; Rats, Wistar; Receptors, GABA-B; Vagotomy

1995
The vigilance promoting drug modafinil increases dopamine release in the rat nucleus accumbens via the involvement of a local GABAergic mechanism.
    European journal of pharmacology, 1996, Jun-13, Volume: 306, Issue:1-3

    Topics: Analysis of Variance; Animals; Baclofen; Benzhydryl Compounds; Central Nervous System Stimulants; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Modafinil; Muscimol; Nipecotic Acids; Nucleus Accumbens; Rats; Rats, Sprague-Dawley

1996
Effects of baclofen and phaclofen on receptive field properties of rat whisker barrel neurons.
    Brain research, 1996, Mar-18, Volume: 712, Issue:2

    Topics: Animals; Baclofen; Extracellular Space; Female; GABA Agonists; GABA Antagonists; Iontophoresis; Mechanoreceptors; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Somatosensory Cortex; Vibrissae

1996
Delayed response deficits induced by local injection of GABA antagonists (bicuculline and phaclofen) into area 46 in infant rhesus monkeys.
    Neuroscience research, 1996, Volume: 24, Issue:3

    Topics: Animals; Baclofen; Cerebral Cortex; Functional Laterality; GABA Antagonists; Hand; Injections; Macaca mulatta; Male; Neural Pathways; Psychomotor Performance

1996
Characterization of subtypes of gamma-aminobutyric acid receptors in an Ascaris muscle preparation by binding assay and binding of PF1022A, a new anthelmintic, on the receptors.
    Parasitology research, 1996, Volume: 82, Issue:2

    Topics: Animals; Anthelmintics; Ascaris suum; Baclofen; Depsipeptides; Dose-Response Relationship, Drug; GABA Antagonists; Muscles; Peptides, Cyclic; Radioligand Assay; Receptors, GABA; Time Factors

1996
Potentiation by baclofen of gastric acid secretion stimulated by secretagogues in vagotomized rats under anesthesia.
    Research communications in molecular pathology and pharmacology, 1996, Volume: 91, Issue:2

    Topics: Anesthesia; Animals; Baclofen; Bethanechol Compounds; Body Temperature; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; GABA Agonists; GABA Antagonists; Gastric Acid; Male; Pentagastrin; Rats; Rats, Wistar; Urethane; Vagotomy; Vagus Nerve

1996
Effects of GABAB receptor antagonists on two models of focal epileptogenesis.
    Brain research, 1995, Dec-08, Volume: 702, Issue:1-2

    Topics: Animals; Baclofen; Disease Models, Animal; Epilepsies, Partial; GABA Antagonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Rats; Rats, Wistar; Time Factors

1995
Antiabsence seizure activity of specific GABAB and gamma-Hydroxybutyric acid receptor antagonists.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:1

    Topics: Animals; Anticonvulsants; Baclofen; Benzocycloheptenes; Electroencephalography; Epilepsy, Absence; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Injections, Intraventricular; Isomerism; Male; Pentylenetetrazole; Rats; Rats, Sprague-Dawley

1996
Mouse cerebellar GABAB participation in the expression of acute ethanol-induced ataxia and in its modulation by the cerebellar adenosinergic A1 system.
    Brain research bulletin, 1996, Volume: 41, Issue:1

    Topics: Adenosine; Adenylate Cyclase Toxin; Animals; Ataxia; Baclofen; Behavior, Animal; Cerebellum; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; GTP-Binding Proteins; Male; Mice; Mice, Inbred Strains; Microinjections; Motor Activity; Muscimol; Pertussis Toxin; Receptors, GABA-B; Receptors, Purinergic P1; Virulence Factors, Bordetella

1996
GABAA and GABAB receptors differentially regulate synaptic transmission in the auditory thalamo-amygdala pathway: an in vivo microiontophoretic study and a model.
    Synapse (New York, N.Y.), 1996, Volume: 24, Issue:2

    Topics: Amygdala; Animals; Baclofen; GABA Antagonists; Male; Models, Neurological; Neural Pathways; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamus

1996
Release of taurine and its effects on release of neurotransmitter amino acids in rat cerebral cortex.
    Advances in experimental medicine and biology, 1996, Volume: 403

    Topics: Animals; Aspartic Acid; Baclofen; Bicuculline; Calcium; Cerebral Cortex; Chromatography, High Pressure Liquid; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Kinetics; Male; Membrane Potentials; Potassium Chloride; Rats; Rats, Wistar; Spectrometry, Fluorescence; Synaptosomes; Taurine; Time Factors

1996
Relation of the [3H] gamma-hydroxybutyric acid (GHB) binding site to the gamma-aminobutyric acidB (GABAB) receptor in rat brain.
    Biochemical pharmacology, 1996, Oct-25, Volume: 52, Issue:8

    Topics: Animals; Autoradiography; Baclofen; Benzocycloheptenes; Binding Sites; Brain; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Guanosine Triphosphate; In Vitro Techniques; Male; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Seizures; Sodium Oxybate; Stereoisomerism

1996
GABAergic modulation of optic nerve-evoked field potentials in the rat suprachiasmatic nucleus.
    Brain research, 1995, Oct-02, Volume: 694, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Optic Nerve; Rats; Rats, Sprague-Dawley; Suprachiasmatic Nucleus

1995
GABAergic characteristics of transcallosal activity of cat motor cortical neurons.
    Neuroscience research, 1996, Volume: 26, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Motor Cortex; Organophosphorus Compounds

1996
Ethanol-induced emesis in the house musk shrew, Suncus murinus.
    Life sciences, 1997, Volume: 60, Issue:4-5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaldehyde; Alcohol Deterrents; Animals; Antiemetics; Baclofen; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Disulfiram; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; Indoles; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Subcutaneous; Male; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Tiopronin; Tropisetron; Vagotomy; Vomiting

1997
Specific action of GABAB ligands on the temperature sensitivity of hypothalamic neurons.
    Annals of the New York Academy of Sciences, 1997, Mar-15, Volume: 813

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Body Temperature Regulation; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hot Temperature; Hypothalamus, Anterior; In Vitro Techniques; Male; Neurons; Preoptic Area; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Thermoreceptors

1997
Evidence for direct and indirect mechanisms in the potent modulatory action of interleukin-2 on the release of acetylcholine in rat hippocampal slices.
    British journal of pharmacology, 1997, Volume: 120, Issue:6

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; GABA Antagonists; Hippocampus; In Vitro Techniques; Interleukin-2; Male; Rats; Rats, Sprague-Dawley; Receptors, Interleukin-2; Sodium Channel Blockers; Sodium Channels; Tetrodotoxin

1997
Involvement of GABAB receptors in the antinociception induced by baclofen in the formalin test.
    General pharmacology, 1997, Volume: 28, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Formaldehyde; GABA Agonists; GABA Antagonists; Male; Pain Threshold; Picrotoxin; Rats; Receptors, GABA-B

1997
Locomotor-related presynaptic modulation of primary afferents in the lamprey.
    The European journal of neuroscience, 1997, Volume: 9, Issue:4

    Topics: Afferent Pathways; Animals; Axons; Baclofen; Bicuculline; Functional Laterality; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Lampreys; Locomotion; Membrane Potentials; Motor Activity; N-Methylaspartate; Neurons, Afferent; Receptors, GABA-A; Receptors, GABA-B; Skin; Spinal Cord; Synapses

1997
Blockade and recovery of spontaneous rhythmic activity after application of neurotransmitter antagonists to spinal networks of the chick embryo.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jan-01, Volume: 18, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Chick Embryo; Cholinergic Antagonists; Dihydro-beta-Erythroidine; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glycine; Glycine Agents; Mecamylamine; Motor Neurons; Neuronal Plasticity; Neurotransmitter Agents; Nicotinic Antagonists; Periodicity; Spinal Cord; Strychnine

1998
Interaction between alpha-MSH and gabaergic agents upon striatal cAMP levels: an in vitro model.
    Peptides, 1998, Volume: 19, Issue:2

    Topics: alpha-MSH; Animals; Baclofen; Benzazepines; Corpus Striatum; Cyclic AMP; Diazepam; Drug Interactions; Flumazenil; GABA Agents; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Models, Neurological; Rats; Rats, Wistar; Receptors, Dopamine D1

1998
GABAergic modulation of ventral pallidal dopamine release studied by in vivo microdialysis in the freely moving rat.
    Synapse (New York, N.Y.), 1998, Volume: 29, Issue:4

    Topics: Animals; Baclofen; Cocaine; Dopamine; Dopamine Uptake Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Microdialysis; Picrotoxin; Piperazines; Rats; Rats, Wistar

1998
Changes in membrane and synaptic properties of thalamocortical circuitry caused by hydrogen peroxide.
    Journal of neurophysiology, 1998, Volume: 80, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Free Radicals; GABA Antagonists; Hydrogen Peroxide; Membrane Potentials; Neural Inhibition; Neural Pathways; Oxidants; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, GABA-B; Somatosensory Cortex; Synaptic Transmission; Thalamus

1998
GABAergic effects on the depressor responses elicited by stimulation of central nucleus of the amygdala.
    The American journal of physiology, 1999, Volume: 276, Issue:1

    Topics: Amygdala; Animals; Baclofen; Bicuculline; Blood Pressure; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heart Rate; Male; Microinjections; Neurons; Rats; Rats, Wistar

1999
Mu opioids enhance mossy fiber synaptic transmission indirectly by reducing GABAB receptor activation.
    Brain research, 1999, Mar-13, Volume: 821, Issue:2

    Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Antagonists; Long-Term Potentiation; Male; Membrane Potentials; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Somatostatin; Synaptic Transmission

1999
Tonic activation of presynaptic GABAB receptors in the opener neuromuscular junction of crayfish.
    Journal of neurophysiology, 1999, Volume: 81, Issue:3

    Topics: Animals; Astacoidea; Axons; Baclofen; GABA Agonists; GABA Antagonists; Logistic Models; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; Pronase; Quantum Theory; Receptors, GABA-B; Receptors, Presynaptic

1999
Activation of peripheral GABAA receptors inhibits temporomandibular joint-evoked jaw muscle activity.
    Journal of neurophysiology, 1999, Volume: 81, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Electromyography; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Masseter Muscle; Motor Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Temporomandibular Joint

1999
Facilitatory effect of unilateral lesion of the ventral tegmental area on locomotor response to stimulation of the contralateral ventral tegmental area: involvement of GABAergic transmission.
    Brain research, 1999, Sep-25, Volume: 842, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Functional Laterality; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Male; Models, Neurological; Motor Activity; Muscimol; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Ventral Tegmental Area

1999
Identification of the G-protein-coupled ORL1 receptor in the mouse spinal cord by [35S]-GTPgammaS binding and immunohistochemistry.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Autoradiography; Baclofen; Binding, Competitive; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Haloperidol; Immunohistochemistry; In Vitro Techniques; Male; Membranes; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Propranolol; Receptors, Opioid; Somatostatin; Spinal Cord; Sulfur Radioisotopes; Yohimbine

1999
A subtype of the gamma-aminobutyric acid(B) receptor regulates cholinergic twitch response in the guinea pig ileum.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:1

    Topics: Animals; Baclofen; Binding, Competitive; Electric Stimulation; GABA Agonists; GABA Antagonists; Guinea Pigs; Ileum; In Vitro Techniques; Ligands; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Parasympathetic Nervous System; Receptors, GABA-B; Spinal Cord

2000
Effect of experimental diabetes on GABA-mediated inhibition of neurally induced contractions in rat isolated trachea.
    Clinical and experimental pharmacology & physiology, 2000, Volume: 27, Issue:4

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscle Contraction; Rats; Rats, Wistar; Taurine; Tetrodotoxin; Trachea; Vasodilator Agents

2000
Sex difference in serum luteinizing hormone postgonadectomy in the rat: role of gamma-aminobutyric acid-ergic inhibition.
    Endocrine, 2000, Volume: 12, Issue:1

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Enzyme Inhibitors; Female; GABA Agents; GABA Antagonists; Kinetics; Luteinizing Hormone; Male; Orchiectomy; Ovariectomy; Rats; Sex Characteristics; Transaminases

2000
Autoimmune hemolytic anemia (AIHA) in an infant rhesus macaque (Macaca mulatta).
    Journal of medical primatology, 2000, Volume: 29, Issue:2

    Topics: Anemia, Hemolytic, Autoimmune; Animals; Baclofen; Benzazepines; Bicuculline; Bromocriptine; Drug Therapy, Combination; Lymphocyte Subsets; Macaca mulatta; Primate Diseases; Spleen

2000
Inhibition suppresses transmission of tonic vibrissa-evoked activity in the rat ventrobasal thalamus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Oct-01, Volume: 20, Issue:19

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Intralaminar Thalamic Nuclei; Iontophoresis; Neural Inhibition; Neurons; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamus; Vibrissae

2000
The human GABA(B1b) and GABA(B2) heterodimeric recombinant receptor shows low sensitivity to phaclofen and saclofen.
    British journal of pharmacology, 2000, Volume: 131, Issue:6

    Topics: Animals; Baclofen; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Receptors, GABA; Receptors, GABA-B

2000
Role of the substantia nigra pars reticulata in sensorimotor gating, measured by prepulse inhibition of startle in rats.
    Behavioural brain research, 2000, Dec-20, Volume: 117, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Acoustic Stimulation; Animals; Baclofen; Central Nervous System Stimulants; Dextroamphetamine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Exploratory Behavior; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Male; Neostriatum; Picrotoxin; Proactive Inhibition; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Stereotyped Behavior; Substantia Nigra

2000
GABAergic modulation of neurons in the nucleus of the solitary tract with ascending projections to the subfornical organ in the rat.
    Brain research, 2001, Jan-05, Volume: 888, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Electric Stimulation; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Male; Neural Pathways; Neurons; Pressoreceptors; Rats; Rats, Wistar; Solitary Nucleus; Subfornical Organ

2001
Induction of wakefulness and inhibition of active (REM) sleep by GABAergic processes in the nucleus pontis oralis.
    Archives italiennes de biologie, 2001, Volume: 139, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Cats; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Neural Inhibition; Pons; Receptors, GABA-A; Reticular Formation; Sleep, REM; Wakefulness

2001
GABA B receptor-mediated effects on expression of c-Fos in rat trigeminal nucleus following high- and low-intensity afferent stimulation.
    Neuroscience, 2001, Volume: 103, Issue:4

    Topics: Animals; Baclofen; Electric Stimulation; GABA Agonists; GABA Antagonists; Male; Neurons, Afferent; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Trigeminal Nuclei

2001
Inhibitory effect of 17beta-estradiol in the parabrachial nucleus is mediated by GABA.
    Brain research, 2001, Aug-24, Volume: 911, Issue:2

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Estradiol; Estrogen Antagonists; Female; Fulvestrant; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Neural Inhibition; Neural Pathways; Neurons; Ovariectomy; Pons; Rats; Receptors, Estrogen; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Vagus Nerve; Ventral Thalamic Nuclei; Visceral Afferents

2001
Hemorrhage activates catecholaminergic neurons sensitive to GABA in the nucleus of the solitary tract with ascending projections to the subfornical organ in rats.
    Autonomic neuroscience : basic & clinical, 2001, Aug-13, Volume: 91, Issue:1-2

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Blood Pressure; Catecholamines; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Hemorrhage; Iontophoresis; Male; Neurons; Oxidopamine; Pressoreceptors; Rats; Rats, Wistar; Solitary Nucleus; Subfornical Organ; Sympatholytics

2001
Evaluation of functional GABA(B) receptors in dental pulp.
    Journal of endodontics, 2001, Volume: 27, Issue:10

    Topics: Animals; Baclofen; Biotransformation; Cattle; Dental Pulp; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Radiopharmaceuticals; Receptors, GABA-B; Receptors, Opioid; Statistics, Nonparametric; Sulfur Radioisotopes

2001
GABA(A) and GABA(B) receptors in the anterior piriform cortex modulate feeding in rats.
    Brain research, 2002, Jan-04, Volume: 924, Issue:1

    Topics: Amino Acids; Animals; Baclofen; Bicuculline; Feeding Behavior; Food Deprivation; Food, Formulated; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Neural Inhibition; Neurons; Olfactory Pathways; Oligonucleotide Array Sequence Analysis; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; RNA, Messenger; Threonine

2002
Interactions between GABAergic and aminoacidergic pathways in the control of gonadotropin and GH secretion in pre-pubertal female rats.
    Journal of endocrinological investigation, 2002, Volume: 25, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Bicuculline; Excitatory Amino Acids; Female; Follicle Stimulating Hormone; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Human Growth Hormone; Kainic Acid; Luteinizing Hormone; Male; N-Methylaspartate; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sex Characteristics; Sexual Maturation

2002
GABA-B-related activity in processing of transcallosal response in cat motor cortex.
    Journal of neuroscience research, 2002, May-15, Volume: 68, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; Corpus Callosum; Female; GABA Agonists; GABA Antagonists; Male; Motor Cortex; Organophosphorus Compounds; Receptors, GABA-A; Receptors, GABA-B; Receptors, Presynaptic; Synaptic Transmission

2002
GABAergic drugs alter hypothalamic serotonin release and lordosis in estrogen-primed rats.
    Brain research, 2002, Aug-09, Volume: 946, Issue:1

    Topics: Animals; Baclofen; Estradiol; Female; GABA Agents; GABA Agonists; GABA Antagonists; Hypothalamus; Muscimol; Rats; Rats, Sprague-Dawley; Serotonin; Sexual Behavior, Animal

2002
GABAergic systems in the nucleus tractus solitarius regulate noradrenaline release in the subfornical organ area in the rat.
    Autonomic neuroscience : basic & clinical, 2002, Sep-30, Volume: 100, Issue:1-2

    Topics: Analysis of Variance; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Muscimol; Norepinephrine; Rats; Rats, Wistar; Solitary Nucleus; Subfornical Organ

2002
Involvement of glutamate and gamma-amino-butyric acid receptor systems on gastric acid secretion induced by activation of kappa-opioid receptors in the central nervous system in rats.
    British journal of pharmacology, 2003, Volume: 138, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Benzeneacetamides; Benzomorphans; Bicuculline; Brain; Dynorphins; gamma-Aminobutyric Acid; Gastric Acid; Injections, Intraventricular; Ketanserin; Male; Perfusion; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, Serotonin; Stomach

2003
Modulation of noradrenaline release in the median preoptic area by GABAergic inputs from the organum vasculosum of the lamina terminalis in the rat.
    Neurochemistry international, 2004, Volume: 44, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Microdialysis; Norepinephrine; Preoptic Area; Rats; Rats, Wistar

2004
Development of novel assays for proteolytic enzymes using rhodamine-based fluorogenic substrates.
    Journal of biomolecular screening, 2002, Volume: 7, Issue:6

    Topics: Baclofen; Biological Assay; Combinatorial Chemistry Techniques; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Endopeptidases; Fluorescent Dyes; Inhibitory Concentration 50; Leucyl Aminopeptidase; Pentamidine; Peptides; Protease Inhibitors; Rhodamines; Substrate Specificity

2002
GABA(B) receptor-mediated regulation of P2X7 receptor expression in the gerbil hippocampus.
    Brain research. Molecular brain research, 2004, Feb-05, Volume: 121, Issue:1-2

    Topics: Analysis of Variance; Animals; Baclofen; Bicuculline; Cell Count; GABA Agonists; GABA Antagonists; Gerbillinae; Hippocampus; Immunohistochemistry; Mossy Fibers, Hippocampal; Muscimol; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Seizures; Severity of Illness Index

2004
Pharmacological modulation of GABA(B) receptors affects cocaine-induced seizures in mice.
    Psychopharmacology, 2004, Volume: 174, Issue:2

    Topics: Animals; Baclofen; Cocaine; Dopamine Uptake Inhibitors; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Kindling, Neurologic; Male; Mice; Piperazines; Receptors, GABA-A; Receptors, GABA-B; Seizures

2004
Effects of ethanol and GABAB drugs on working memory in C57BL/6J and DBA/2J mice.
    Psychopharmacology, 2004, Volume: 176, Issue:2

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Drug Combinations; Ethanol; Female; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Memory; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Receptors, GABA-B; Species Specificity

2004
GABA-mediated attenuation of noradrenaline release in the rat median preoptic area caused by intravenous injection of metaraminol.
    Autonomic neuroscience : basic & clinical, 2004, Mar-31, Volume: 111, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Baclofen; Baroreflex; Bicuculline; Blood Pressure; GABA Antagonists; gamma-Aminobutyric Acid; Injections, Intravenous; Male; Metaraminol; Microdialysis; Norepinephrine; Preoptic Area; Rats; Rats, Wistar; Receptors, GABA

2004
Peripherally delivered glutamic acid decarboxylase gene therapy for spinal cord injury pain.
    Molecular therapy : the journal of the American Society of Gene Therapy, 2004, Volume: 10, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Calcitonin Gene-Related Peptide; gamma-Aminobutyric Acid; Ganglia, Spinal; Genetic Therapy; Genetic Vectors; Glutamate Decarboxylase; Hyperalgesia; Injections, Subcutaneous; Isoenzymes; Neurons; Pain; Rats; Simplexvirus; Spinal Cord Injuries; Tissue Distribution; Transduction, Genetic

2004
Altered GABAB receptor immunoreactivity in the gerbil hippocampus induced by baclofen and phaclofen, not seizure activity.
    Neuroscience research, 2004, Volume: 49, Issue:4

    Topics: Animals; Baclofen; Blotting, Western; Cell Count; Dose-Response Relationship, Drug; Enzyme Inhibitors; GABA Antagonists; Gene Expression Regulation; Gerbillinae; Hippocampus; Immunohistochemistry; Proline; Receptors, GABA-B; Vigabatrin

2004
Post-synaptic GABA(B) receptors--possible controllers of coincidence detection?
    Behavioural brain research, 2004, Nov-05, Volume: 155, Issue:1

    Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Baclofen; Chickens; Electric Impedance; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; In Vitro Techniques; Neurons; Prosencephalon; Receptors, GABA-B; Synapses; Synaptic Transmission; Valine

2004
Glutamate and GABA(B) transmissions in lateral amygdala are involved in startle-like electromyographic (EMG) potentiation caused by activation of auditory thalamus.
    Neuroscience letters, 2005, Feb-10, Volume: 374, Issue:2

    Topics: Amygdala; Animals; Baclofen; Electric Stimulation; Electromyography; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; Kynurenic Acid; Male; Microinjections; Rats; Rats, Wistar; Receptors, GABA-A; Reflex, Startle; Synaptic Transmission; Time Factors; Trigeminal Nuclei

2005
Effects of GABAB receptor modulation on gonadotropin-releasing hormone and beta-endorphin release, and on catecholaminergic activity in the ventromedial hypothalamus-infundibular nucleus region of anoestrous ewes.
    Journal of neuroendocrinology, 2005, Volume: 17, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; beta-Endorphin; Dopamine; Estrous Cycle; Extracellular Space; Female; GABA Agonists; GABA Antagonists; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Methoxyhydroxyphenylglycol; Norepinephrine; Pituitary Gland, Posterior; Receptors, GABA-B; Sheep; Ventromedial Hypothalamic Nucleus

2005
Effects of GABAergic transmissions on the immunoreactivities of calcium binding proteins in the gerbil hippocampus.
    The Journal of comparative neurology, 2005, May-02, Volume: 485, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Calbindin 2; Calbindins; Calcium-Binding Proteins; Cell Count; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Gerbillinae; Hippocampus; Immunohistochemistry; Muscimol; Neurons; Parvalbumins; S100 Calcium Binding Protein G; Seizures; Synaptic Transmission

2005
Benzodiazepine system is involved in hyperalgesia in rats induced by the exposure to extremely low frequency magnetic fields.
    Archives of pharmacal research, 2005, Volume: 28, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Diazepam; Electromagnetic Fields; Flumazenil; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hot Temperature; Hyperalgesia; Injections, Intraventricular; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A

2005
Opposite effects of tetanic stimulation of the auditory thalamus or auditory cortex on the acoustic startle reflex in awake rats.
    The European journal of neuroscience, 2005, Volume: 21, Issue:7

    Topics: Acoustic Stimulation; Analysis of Variance; Animals; Auditory Cortex; Baclofen; Behavior, Animal; Electric Stimulation; Functional Laterality; GABA Antagonists; Geniculate Bodies; Male; Models, Biological; Rats; Rats, Wistar; Reflex, Startle; Time Factors; Wakefulness

2005
HPLC conditions are critical for the detection of GABA by microdialysis.
    Journal of neurochemistry, 2005, Volume: 94, Issue:3

    Topics: Anesthetics, Local; Animals; Baclofen; Benzylamines; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Nipecotic Acids; Phosphinic Acids; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Time Factors

2005
Enantiomeric analysis of baclofen analogs by capillary zone electrophoresis, using highly sulfated cyclodextrins: Inclusion ionization constant pKa determination.
    Electrophoresis, 2005, Volume: 26, Issue:15

    Topics: Baclofen; Buffers; Cyclodextrins; Electrophoresis, Capillary; GABA Agonists; GABA-B Receptor Agonists; Hydrogen-Ion Concentration; Stereoisomerism; Sulfonic Acids

2005
Electroacupuncture improves restraint stress-induced delay of gastric emptying via central glutaminergic pathways in conscious rats.
    Neuroscience letters, 2006, May-15, Volume: 399, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Electroacupuncture; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Gastric Emptying; Kynurenic Acid; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Receptors, Glutamate; Restraint, Physical; Stomach; Stress, Psychological

2006
GABA(A) and GABA(B) receptors differentially modulate volume and frequency in ventilatory compensation in obese Zucker rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2007, Volume: 102, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Dimethyl Sulfoxide; GABA Antagonists; Hypercapnia; Hypoxia; Male; Obesity; Oxygen Consumption; Physical Conditioning, Animal; Pulmonary Ventilation; Rats; Rats, Zucker; Receptors, GABA-A; Receptors, GABA-B; Respiratory Mechanics; Tidal Volume

2007
GABAA but not GABAB receptors in the rostral anterior cingulate cortex selectively modulate pain-induced escape/avoidance behavior.
    Experimental neurology, 2007, Volume: 204, Issue:1

    Topics: Animals; Avoidance Learning; Baclofen; Bicuculline; Escape Reaction; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gyrus Cinguli; Male; Microinjections; Muscimol; Pain; Pain Threshold; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B

2007
Understanding your inhibitions: modulation of brain cortical metabolism by GABA(B) receptors.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2007, Volume: 27, Issue:8

    Topics: Animals; Baclofen; Benzylamines; Carbon Isotopes; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Guinea Pigs; Molecular Structure; Morpholines; Nuclear Magnetic Resonance, Biomolecular; Organophosphorus Compounds; Phosphinic Acids; Principal Component Analysis; Receptors, GABA-B

2007
Nicotinic receptor-mediated biphasic effect on neuronal excitability in chick lateral spiriform neurons.
    Neuroscience, 2007, Sep-21, Volume: 148, Issue:4

    Topics: Action Potentials; Animals; Baclofen; Brain; Calcium; Carbachol; Chick Embryo; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; GABA Antagonists; In Vitro Techniques; Neural Inhibition; Neurons; Nicotine; Nicotinic Antagonists; Receptors, Nicotinic; Time Factors

2007
GABA receptor agonism in the sublenticular central extended amygdala impairs medial forebrain bundle self-stimulation but GABA blockade does not enhance it.
    Behavioural brain research, 2008, Mar-05, Volume: 187, Issue:2

    Topics: Amygdala; Animals; Baclofen; Bicuculline; Electric Stimulation; Functional Laterality; GABA Agonists; GABA Antagonists; Male; Medial Forebrain Bundle; Muscimol; Rats; Rats, Long-Evans; Receptors, GABA; Reinforcement, Psychology; Self Stimulation; Substantia Innominata

2008
[Contribution of GABA receptors in extinction of memory trace in norm and depressive-like state].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2007, Volume: 93, Issue:11

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Depression; Fear; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Memory; Mice; Muscimol; Receptors, GABA-A; Receptors, GABA-B

2007
Evidence that gamma-aminobutyric acid is part of the neural circuit mediating estradiol negative feedback in anestrous ewes.
    Endocrinology, 2008, Volume: 149, Issue:6

    Topics: Anestrus; Animals; Baclofen; Bicuculline; Dopamine; Estradiol; Feedback; Female; gamma-Aminobutyric Acid; Muscimol; Neurons; Ovariectomy; Sheep

2008
GabaB receptors activation in the NTS blocks the glycemic responses induced by carotid body receptor stimulation.
    Autonomic neuroscience : basic & clinical, 2008, Aug-18, Volume: 141, Issue:1-2

    Topics: Analysis of Variance; Animals; Baclofen; Bicuculline; Blood Glucose; Carotid Body; GABA Agonists; GABA Antagonists; Glucose; Microinjections; Muscimol; Rats; Receptors, GABA-A; Receptors, GABA-B; Solitary Nucleus

2008
Roles of forebrain GABA receptors in controlling vasopressin secretion and related phenomena under basal and hyperosmotic circumstances in conscious rats.
    Brain research bulletin, 2008, Sep-05, Volume: 77, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Consciousness; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Glucose; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Muscimol; Osmolar Concentration; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA; Saline Solution, Hypertonic; Sodium; Vasopressins

2008
GABAergic mediation of stress-induced secretion of corticosterone and oxytocin, but not prolactin, by the hypothalamic paraventricular nucleus.
    Life sciences, 2008, Nov-07, Volume: 83, Issue:19-20

    Topics: Animals; Baclofen; Bicuculline; Corticosterone; Dose-Response Relationship, Drug; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Microinjections; Oxytocin; Paraventricular Hypothalamic Nucleus; Prolactin; Rats; Rats, Wistar; Stress, Psychological

2008
Analgesic alpha-conotoxins Vc1.1 and Rg1A inhibit N-type calcium channels in rat sensory neurons via GABAB receptor activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Oct-22, Volume: 28, Issue:43

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Barium; Calcium Channel Blockers; Calcium Channels, N-Type; Cells, Cultured; Conotoxins; Dose-Response Relationship, Radiation; Electric Stimulation; GABA Antagonists; Ganglia, Spinal; Membrane Potentials; omega-Conotoxins; Patch-Clamp Techniques; Pertussis Toxin; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA; Sensory Receptor Cells

2008
GABA antagonists reverse the somatostatin dependent attenuation of rat locomotor activity.
    Neuropeptides, 2009, Volume: 43, Issue:3

    Topics: Animals; Baclofen; Basal Ganglia; Bicuculline; GABA Antagonists; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Somatostatin

2009
Astrocytes and interneurons in memory processing in the chick hippocampus: roles for G-coupled protein receptors, GABA(B) and mGluR1.
    Neurochemical research, 2009, Volume: 34, Issue:10

    Topics: Animals; Animals, Newborn; Astrocytes; Baclofen; Chickens; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hippocampus; Housing, Animal; Interneurons; Male; Memory; Methoxyhydroxyphenylglycol; Receptors, G-Protein-Coupled; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Time Factors

2009
Role of endocannabinoid system in the ventral hippocampus of rats in the modulation of anxiety-like behaviours.
    Basic & clinical pharmacology & toxicology, 2009, Volume: 105, Issue:5

    Topics: Amidohydrolases; Animals; Anxiety; Baclofen; Behavior, Animal; Benzamides; Bicuculline; Cannabinoid Receptor Modulators; Carbamates; Dose-Response Relationship, Drug; Endocannabinoids; GABA Antagonists; Hippocampus; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2009
GABA receptors and prepulse inhibition of acoustic startle in mice and rats.
    The European journal of neuroscience, 2010, Volume: 31, Issue:11

    Topics: Acoustic Stimulation; Animals; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Muscimol; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, GABA; Reflex, Startle; Scopolamine; Time Factors

2010
Analgesia induced by 2- or 100-Hz electroacupuncture in the rat tail-flick test depends on the activation of different descending pain inhibitory mechanisms.
    The journal of pain, 2011, Volume: 12, Issue:1

    Topics: Adjuvants, Anesthesia; Adrenergic alpha-Antagonists; Analgesia; Anesthetics, Intravenous; Animals; Atropine; Baclofen; Bicuculline; Biophysics; Dioxanes; Disease Models, Animal; Electroacupuncture; GABA Agents; Male; Methysergide; Models, Biological; Multivariate Analysis; Naloxone; Narcotic Antagonists; Pain; Pain Management; Pain Measurement; Rats; Rats, Wistar; Reaction Time; Serotonin Antagonists; Tail; Thiopental; Time Factors

2011
GABA(A) receptors in the dorsal raphé nucleus of mice: escalation of aggression after alcohol consumption.
    Psychopharmacology, 2010, Volume: 211, Issue:4

    Topics: Aggression; Animals; Baclofen; Behavior, Animal; Bicuculline; Ethanol; GABA Agonists; GABA Antagonists; Male; Mice; Muscimol; Raphe Nuclei; Receptors, GABA-A; Receptors, GABA-B; Self Administration

2010
Involvement of GABAergic transmission in the midbrain ventral tegmental area in the regulation of hippocampal theta rhythm.
    Brain research bulletin, 2010, Nov-20, Volume: 83, Issue:6

    Topics: Animals; Baclofen; Bicuculline; Electroencephalography; Fourier Analysis; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Muscimol; Rats; Rats, Wistar; Theta Rhythm; Ventral Tegmental Area

2010
Metabotropic γ-aminobutyric acid (GABAB) receptors modulate feeding behavior in the calcisponge Leucandra aspera.
    Journal of experimental zoology. Part A, Ecological genetics and physiology, 2011, Mar-01, Volume: 315, Issue:3

    Topics: Animals; Baclofen; Drug Interactions; Endocytosis; Feeding Behavior; GABA Antagonists; GABA-B Receptor Agonists; Pertussis Toxin; Porifera; Receptors, GABA-B

2011
Changes in GABA and GABA(B) receptor expressions are involved in neuropathy in the rat cuneate nucleus following median nerve transection.
    Synapse (New York, N.Y.), 2012, Volume: 66, Issue:6

    Topics: Animals; Baclofen; Electric Stimulation; GABA Antagonists; Gait; gamma-Aminobutyric Acid; Ganglia, Spinal; Male; Median Nerve; Median Neuropathy; Medulla Oblongata; Neuropeptide Y; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-B

2012
Decreased GABABR expression and increased neuronal cell death in developing rat brain after PTZ-induced seizure.
    Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology, 2013, Volume: 34, Issue:4

    Topics: Animals; Animals, Newborn; Baclofen; Caspase 3; Cell Death; Disease Models, Animal; Electroencephalography; GABA Antagonists; GABA-B Receptor Agonists; Gene Expression Regulation, Developmental; Hippocampus; Microscopy, Confocal; Neurons; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Seizures

2013
Baclofen administration alters fear extinction and GABAergic protein levels.
    Neurobiology of learning and memory, 2012, Volume: 98, Issue:3

    Topics: Amygdala; Animals; Baclofen; Conditioning, Psychological; Cues; Extinction, Psychological; Fear; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Male; Rats; Rats, Sprague-Dawley; Reflex, Startle

2012
Segmental disinhibition suppresses C-fiber inputs to the rat superficial medullary dorsal horn via the activation of GABAB receptors.
    The European journal of neuroscience, 2013, Volume: 37, Issue:3

    Topics: Action Potentials; Animals; Baclofen; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Morphine; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Posterior Horn Cells; Rats; Rats, Inbred Strains; Receptors, GABA-B; Receptors, Glycine; Synaptic Transmission

2013
GABAergic synaptic inputs of locus coeruleus neurons in wild-type and Mecp2-null mice.
    American journal of physiology. Cell physiology, 2013, May-01, Volume: 304, Issue:9

    Topics: Animals; Baclofen; Female; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; GABAergic Neurons; gamma-Aminobutyric Acid; Humans; Locus Coeruleus; Male; Membrane Potentials; Methyl-CpG-Binding Protein 2; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscimol; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Presynaptic Terminals; Receptors, GABA-A; Receptors, GABA-B; Rett Syndrome; Synaptic Membranes; Synaptic Transmission

2013
Effect of GABA receptor agonists or antagonists injected spinally on the blood glucose level in mice.
    Neurochemical research, 2013, Volume: 38, Issue:5

    Topics: Animals; Baclofen; Blood Glucose; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Receptors, GABA

2013
Reversal of morphine analgesic tolerance by ethanol in the mouse.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 345, Issue:3

    Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethanol; GABA Antagonists; Hypnotics and Sedatives; Immersion; Injections, Intraventricular; Male; Mice; Morphine; Pain Measurement; Receptors, GABA-A; Receptors, GABA-B

2013
Effects of Withania somnifera on oral ethanol self-administration in rats.
    Behavioural pharmacology, 2014, Volume: 25, Issue:7

    Topics: Administration, Oral; Alcohol Drinking; Animals; Baclofen; Conditioning, Operant; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Ethanol; Male; Plant Extracts; Rats; Rats, Wistar; Receptors, GABA-B; Reinforcement Schedule; Saccharin; Self Administration; Withania

2014
Postnatal alterations in GABAB receptor tone produce sensorimotor gating deficits and protein level differences in adulthood.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 2015, Volume: 41

    Topics: Acoustic Stimulation; Age Factors; Animals; Animals, Newborn; Baclofen; Body Weight; Brain; Disease Models, Animal; Female; GABA Antagonists; GABA-B Receptor Agonists; Gait Disorders, Neurologic; Gene Expression Regulation, Developmental; Male; Pregnancy; Prepulse Inhibition; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Sensory Gating; Signal Transduction

2015
The antinociceptive effect of stimulating the retrosplenial cortex in the rat tail-flick test but not in the formalin test involves the rostral anterior cingulate cortex.
    Pharmacology, biochemistry, and behavior, 2015, Volume: 131

    Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; Cobalt; Electric Stimulation; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Gyrus Cinguli; Male; Pain Measurement; Pain Perception; Rats; Rats, Wistar; Tail

2015
The modulatory effect of CA1 GABAb receptors on ketamine-induced spatial and non-spatial novelty detection deficits with respect to Ca(2+).
    Neuroscience, 2015, Oct-01, Volume: 305

    Topics: Analysis of Variance; Animals; Baclofen; CA1 Region, Hippocampal; Calcium; Calcium Channel Blockers; Disease Models, Animal; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Exploratory Behavior; GABA Antagonists; Imidazoles; Ketamine; Male; Memory Disorders; Mice; Receptors, GABA-A; Signal Detection, Psychological; Spatial Processing

2015
GABA modulates baroreflex in the ventral tegmental area in rat.
    Synapse (New York, N.Y.), 2015, Volume: 69, Issue:12

    Topics: Animals; Baclofen; Baroreflex; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Wistar; Ventral Tegmental Area

2015
Recovery from ketamine-induced amnesia by blockade of GABA-A receptor in the medial prefrontal cortex of mice.
    Neuroscience, 2017, 03-06, Volume: 344

    Topics: Amnesia; Animals; Baclofen; Bicuculline; Catheters, Indwelling; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; Ketamine; Male; Memory; Mice; Muscimol; Neuropsychological Tests; Prefrontal Cortex; Receptors, GABA-A; Time Factors

2017
The lesion of dorsolateral funiculus changes the antiallodynic effect of the intrathecal muscimol and baclofen in distinct phases of neuropathic pain induced by spinal nerve ligation in rats.
    Brain research bulletin, 2016, Volume: 124

    Topics: Animals; Baclofen; Bicuculline; Functional Laterality; GABA Agents; Hyperalgesia; Injections, Spinal; Ligation; Male; Muscimol; Neuralgia; Pain Measurement; Pain Threshold; Physical Stimulation; Rats; Rats, Wistar; Spinal Cord Dorsal Horn; Spinal Nerves; Statistics, Nonparametric

2016
GABAergic modulation of serotonin release in the rat subfornical organ area.
    Neuroscience letters, 2016, Sep-06, Volume: 630

    Topics: Animals; Baclofen; Bicuculline; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hydroxyindoleacetic Acid; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Serotonin; Subfornical Organ

2016
GABA Receptors in the Medial Preoptic Area Modulate the Onset of Oestradiol-Induced Maternal Behaviour in Hysterectomised-Ovariectomised, Pregnant Rats.
    Journal of neuroendocrinology, 2016, Volume: 28, Issue:11

    Topics: Animals; Baclofen; Bicuculline; Estradiol; Female; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hysterectomy; Maternal Behavior; Nesting Behavior; Ovariectomy; Pregnancy; Preoptic Area; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B

2016
GABAergic modulation of noradrenaline release caused by blood pressure changes in the rat median preoptic area.
    Neuroreport, 2017, Jun-14, Volume: 28, Issue:9

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Baclofen; Bicuculline; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Metaraminol; Microdialysis; Norepinephrine; Preoptic Area; Rats; Rats, Wistar

2017
The interaction between hippocampal GABA-B and cannabinoid receptors upon spatial change and object novelty discrimination memory function.
    Psychopharmacology, 2017, Volume: 234, Issue:20

    Topics: Animals; Baclofen; Discrimination Learning; Dose-Response Relationship, Drug; Exploratory Behavior; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hippocampus; Male; Memory; Mice; Microinjections; Receptor, Cannabinoid, CB1; Receptors, Cannabinoid; Receptors, GABA-B; Spatial Behavior

2017
The role of CA3 GABA
    Progress in neuro-psychopharmacology & biological psychiatry, 2017, 10-03, Volume: 79, Issue:Pt B

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anxiety; Avoidance Learning; Baclofen; CA3 Region, Hippocampal; Calcium; Calcium Channel Blockers; Cations, Divalent; Disease Models, Animal; GABA Antagonists; GABA-B Receptor Agonists; Imidazoles; Male; Memory Disorders; Motor Activity; Psychotropic Drugs; Random Allocation; Rats, Wistar; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate

2017
Modulation of tonic immobility by GABAA and GABAB receptors of the medial amygdala.
    Neuroscience letters, 2019, 04-23, Volume: 699

    Topics: Animals; Baclofen; Bicuculline; Corticomedial Nuclear Complex; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Guinea Pigs; Immobility Response, Tonic; Male; Microinjections; Motor Activity; Muscimol

2019
The effect of GABA-B receptors in the basolateral amygdala on passive avoidance memory impairment induced by MK-801 in rats.
    Behavioural brain research, 2021, 07-09, Volume: 409

    Topics: Animals; Avoidance Learning; Baclofen; Basolateral Nuclear Complex; Behavior, Animal; Disease Models, Animal; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Memory Disorders; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate

2021