Page last updated: 2024-09-03

perospirone and ketanserin

perospirone has been researched along with ketanserin in 2 studies

Compound Research Comparison

Studies
(perospirone)
Trials
(perospirone)
Recent Studies (post-2010)
(perospirone)
Studies
(ketanserin)
Trials
(ketanserin)
Recent Studies (post-2010) (ketanserin)
11124263,094335283

Protein Interaction Comparison

ProteinTaxonomyperospirone (IC50)ketanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0021
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.015
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.015
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.265
5-hydroxytryptamine receptor 1BHomo sapiens (human)6.5
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0184
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0027
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.29
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.015
D(2) dopamine receptorRattus norvegicus (Norway rat)1.8
Synaptic vesicular amine transporterHomo sapiens (human)0.18
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.001

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hirose, A; Kato, T; Katsube, J; Nakamura, M; Ohno, Y; Shimizu, H; Tanaka, H1
Nakamura, M; Ohno, Y; Tanaka, H1

Other Studies

2 other study(ies) available for perospirone and ketanserin

ArticleYear
Pharmacological actions of SM-9018, a new neuroleptic drug with both potent 5-hydroxytryptamine2 and dopamine2 antagonistic actions.
    Japanese journal of pharmacology, 1990, Volume: 53, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Brain Chemistry; Catalepsy; Dopamine Antagonists; Indoles; Isoindoles; Ketanserin; Male; Methamphetamine; Mice; Mice, Inbred Strains; Motor Activity; Norepinephrine; Parasympatholytics; Psychomotor Performance; Rats; Rats, Inbred Strains; Serotonin Antagonists; Spiperone; Stereotyped Behavior; Thiazoles

1990
Localization and pharmacological characterization of [3H]perospirone-binding sites in rat brain.
    General pharmacology, 1998, Volume: 31, Issue:1

    Topics: Animals; Antipsychotic Agents; Benzazepines; Binding Sites; Brain; Domperidone; Dopamine Antagonists; Indoles; Isoindoles; Ketanserin; Male; Membranes; Radioligand Assay; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Thiazoles; Tritium

1998