pentylenetetrazole and ethosuximide
pentylenetetrazole has been researched along with ethosuximide in 77 studies
Research
Studies (77)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 29 (37.66) | 18.7374 |
1990's | 18 (23.38) | 18.2507 |
2000's | 13 (16.88) | 29.6817 |
2010's | 12 (15.58) | 24.3611 |
2020's | 5 (6.49) | 2.80 |
Authors
Authors | Studies |
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Butler, DE; L'Italien, YJ; Marriott, JG; Nordin, IC; Poschel, PH; Zweisler, L | 1 |
Butler, DE; Marriott, JG; Poschel, BP | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Alkskas, IA; Azam, F; Khokra, SL; Prakash, O | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Consroe, PF; Wolkin, AL | 1 |
Ferrendelli, JA; Kinscherf, DA | 1 |
Banerjee, U; Yeoh, PN | 1 |
Frey, HH; Löscher, W | 1 |
Mares, P; Stanková, L | 1 |
Goehring, RR; Greenwood, TD; Pisipati, JS; Wolfe, JF | 1 |
Aguilar-Veiga, E; Galán-Valiente, J; Méndez-Alvarez, E; Sierra-Marcuño, G; Sierra-Paredes, G; Soto-Otero, R | 1 |
Coulter, DA; Huguenard, JR; Prince, DA | 2 |
Czuczwar, SJ; Kleinrok, Z; Małek, U | 1 |
Kulhánková, I; Mares, P; Mirvaldová, H; Roztocilová, L; Velísek, L; Velísková, J | 1 |
Rahwan, RG; Wong, WS | 1 |
Jakubow, JJ; Poling, A; Schlinger, H | 1 |
Aburada, M; Hosoya, E; Iizuka, S; Ishige, A; Matsuzaki, Y; Sakamoto, K; Sekiguchi, K; Sugaya, E | 1 |
Bender, AS; Hertz, L | 1 |
Mares, P; Velísek, L | 2 |
Chweh, AY; Lin-Michell, E; Swinyard, EA | 1 |
Centra, M; Keeting, PE; Lysz, TW; Markey, K | 1 |
Kaneda, H; Kaneto, H; Kawatani, S | 1 |
Piredda, SG; Swinyard, EA; Woodhead, JH | 1 |
Lasek, R; Müller, M | 1 |
Zetler, G | 1 |
Forrest, TP; Gilroy, ML; Vohra, MM; Yung, DK | 1 |
Millichap, JG | 1 |
Kästner, I; Müller, M; Schmiedel, R; Wenzel, J | 1 |
Frey, HH; Meyer, H | 1 |
Krüger, E; Müller, M; Wenzel, J | 1 |
Geschwind, N; Sherwin, I | 1 |
Karler, R; Turkanis, SA | 1 |
Mares, P; Maresová, D; Schickerová, R | 1 |
Mares, P; Zouhar, A | 1 |
Carey, MP; Fry, JP | 1 |
Kubová, H; Mares, P; Pohl, M; Zelízko, M | 1 |
Mares, P; Micianiková, D; Rokyta, R; Velísek, L; Velísková, J | 1 |
Pleuvry, BJ; Rodger, C | 1 |
Becker, A; Brosz, M; Grecksch, G | 1 |
Brudniak, T; Czuczwar, SJ; Gasior, M; Kamiński, R; Kleinrok, Z | 1 |
Stringer, JL | 1 |
Mares, P | 1 |
Czuczwar, SJ; Gasior, M; Kleinrok, Z; Kozicka, M; Pietrasiewicz, T; Turski, WA | 1 |
David, J; Joseph, S; Joseph, T | 1 |
Czuczwar, SJ; Kleinrok, Z; Klonowski, P; Tutka, P | 1 |
Fanaee, GH; Javadi, M; Kamalinejad, M; Majzoob, S; Pourgholami, MH; Sayyah, M | 1 |
Borowicz, KK; Czuczwar, SJ; Kleinrok, Z; Luszczki, J | 1 |
David, J; Joseph, T; Kumaresan, S | 1 |
Shaw, FZ | 1 |
FREY, HH | 1 |
Borowicz, KK; Czuczwar, SJ; Luszczki, JJ | 1 |
Czuczwar, SJ; Dekundy, A; Kaminski, RM; Tochman, AM; Turski, WA | 1 |
Czuczwar, SJ; Luszczki, JJ; Patsalos, PN; Ratnaraj, N | 2 |
Brevard, ME; Ferris, CF; King, JA; Kulkarni, P | 1 |
Calderon, A; Palencia, G; Sotelo, J | 1 |
Luszczki, JJ | 1 |
Andres-Mach, MM; Czuczwar, SJ; Dudra-Jastrzebska, M; Luszczki, JJ; Patsalos, PN; Ratnaraj, N | 1 |
Garg, S; Hinich, MJ; Mirski, MA; Sherman, D; Thakor, NV; White, MA; Zhang, N | 1 |
Chen, SD; Huang, YH; Shaw, FZ; Yeh, KH | 1 |
Andres-Mach, M; Barcicka-Klosowska, B; Czuczwar, SJ; Florek-Luszczki, M; Haratym-Maj, A; Luszczki, JJ | 1 |
Kamiński, K; Obniska, J; Rzepka, S | 1 |
Borowicz, KK; Czuczwar, SJ; Piskorska, B; Stępniak, B | 1 |
Abdar, M; Mandegary, A; Sharififar, F | 1 |
Filipek, B; Kamiński, K; Obniska, J; Rapacz, A; Rybka, S | 1 |
Asadi-Shekaari, M; Eslami, A; Joukar, S; Kalantaripour, T | 1 |
Godwin, DW; Masicampo, ML; Riegle, MA; Shan, HQ; Xu, V | 1 |
Borowicz, KK; Popławska, M; Wróblewska, D | 1 |
Barclay, JW; Burgoyne, RD; Cunliffe, VT; Dodd, S; Grimes, D; Jones, A; Marson, AG; Morgan, A; Sills, GJ; Wong, SQ | 1 |
Abram, M; Andres-Mach, M; Esguerra, CV; Gawel, K; Jakubiec, M; Kamiński, K; Latacz, G; Lubelska, A; Nieoczym, D; Pieróg, M; Rapacz, A; Socała, K; Szewczyk, A; Szulczyk, B; Wlaź, P; Zagaja, M; Łuszczki, JJ | 1 |
Abram, M; Andres-Mach, M; Kaminski, K; Luszczki, J; Maj, M; Rola, R; Szewczyk, A; Zagaja, M | 1 |
Czuczwar, SJ; Krzyżanowski, M; Świąder, K; Świąder, MJ; Wróbel, A; Zakrocka, I; Łuszczki, JJ | 1 |
Contreras-Murillo, G; González-Trujano, ME; Hidalgo-Flores, FJ; López-Najera, CA; Magdaleno-Madrigal, VM; Navarrete-Castro, A; Sánchez, CG | 1 |
Dziubina, A; Jarzyński, S; Pękala, E; Piska, K; Popiół, J; Rapacz, A; Rudolf, B; Wojtulewski, S | 1 |
Reviews
1 review(s) available for pentylenetetrazole and ethosuximide
Article | Year |
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Relation of laboratory evaluation to clinical effectiveness of antiepileptic drugs.
Topics: Acetazolamide; Adrenocorticotropic Hormone; Animals; Anticonvulsants; Benzazepines; Clinical Trials as Topic; Drug Tolerance; Electroencephalography; Electroshock; Epilepsy; Ethosuximide; Humans; Pentylenetetrazole; Phenobarbital; Phenytoin; Primidone; Seizures; Trimethadione; Urea | 1969 |
Trials
2 trial(s) available for pentylenetetrazole and ethosuximide
Article | Year |
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Relation of laboratory evaluation to clinical effectiveness of antiepileptic drugs.
Topics: Acetazolamide; Adrenocorticotropic Hormone; Animals; Anticonvulsants; Benzazepines; Clinical Trials as Topic; Drug Tolerance; Electroencephalography; Electroshock; Epilepsy; Ethosuximide; Humans; Pentylenetetrazole; Phenobarbital; Phenytoin; Primidone; Seizures; Trimethadione; Urea | 1969 |
Effects of fluoxetine on the anticonvulsant action of valproate and ethosuximide in mouse model of myoclonic convulsions.
Topics: Animals; Anticonvulsants; Antidepressive Agents, Second-Generation; Avoidance Learning; Convulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Epilepsies, Myoclonic; Ethosuximide; Fluorescent Antibody Technique; Fluoxetine; Male; Memory, Long-Term; Mice; Motor Activity; Pentylenetetrazole; Seizures; Selective Serotonin Reuptake Inhibitors; Valproic Acid | 2012 |
Other Studies
75 other study(ies) available for pentylenetetrazole and ethosuximide
Article | Year |
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Amnesia-reversal activity of a series of N-[(disubstituted-amino)alkyl] -2-oxo-1-pyrrolidineacetamides, including pramiracetam.
Topics: Amnesia; Animals; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Electroshock; Humans; Male; Mice; Mice, Inbred Strains; Pyrrolidines; Structure-Activity Relationship | 1984 |
Cognition-activating properties of 3-(Aryloxy)pyridines.
Topics: Animals; Cognition; Dose-Response Relationship, Drug; Male; Mice; Psychotropic Drugs; Pyridines; Structure-Activity Relationship | 1981 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Synthesis of some novel N4-(naphtha[1,2-d]thiazol-2-yl)semicarbazides as potential anticonvulsants.
Topics: Animals; Anticonvulsants; Brain Chemistry; Glutathione Peroxidase; Malondialdehyde; Mice; Motor Activity; Rats; Seizures; Semicarbazides; Structure-Activity Relationship; Superoxide Dismutase | 2009 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Anticonvulsant interaction of cannabidiol and ethosuximide in rats.
Topics: Animals; Anticonvulsants; Cannabidiol; Cannabinoids; Drug Interactions; Ethosuximide; Male; Pentylenetetrazole; Proadifen; Rats | 1977 |
Cyclic nucleotides in epileptic brain: effects of pentylenetetrazol on regional cyclic AMP and cyclic GMP levels in vivo.
Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Cyclic AMP; Cyclic GMP; Ethosuximide; Female; Hippocampus; Mice; Pentylenetetrazole; Phenobarbital; Phenytoin; Seizures; Thalamus | 1977 |
The temporal dimensions of anticonvulsant action of some newer benzodiazepines against metrazol induced seizures in mice and rats.
Topics: Animals; Benzodiazepines; Clonazepam; Diazepam; Drug Evaluation, Preclinical; Ethosuximide; Female; Flurazepam; Male; Mice; Nitrazepam; Pentylenetetrazole; Phenobarbital; Seizures; Trimethadione | 1977 |
Di-n-propylacetic acid--profile of anticonvulsant activity in mice.
Topics: Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Electroshock; Ethosuximide; Female; Male; Mice; Pentylenetetrazole; Phenobarbital; Picrotoxin; Seizures; Strychnine; Trimethadione; Valerates; Valproic Acid | 1976 |
Influence of phenobarbital on ECoG phenomena induced by metrazol in rats during ontogenesis.
Topics: Aging; Animals; Cerebral Cortex; Clonazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Electrodes; Electroencephalography; Epilepsy; Ethosuximide; Injections, Intraperitoneal; Male; Pentylenetetrazole; Phenobarbital; Prohibitins; Rats; Rats, Wistar; Valproic Acid | 1992 |
Synthesis and anticonvulsant evaluation of some new 2-benzylsuccinimides.
Topics: Animals; Anticonvulsants; Chemical Phenomena; Chemistry, Physical; Electroshock; Ethosuximide; Male; Mice; Pentylenetetrazole; Postural Balance; Succinimides | 1991 |
Correlation between ethosuximide brain levels measured by high performance liquid chromatography and its antiepileptic potential.
Topics: Animals; Anticonvulsants; Blood-Brain Barrier; Brain; Chromatography, High Pressure Liquid; Electrophysiology; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Tissue Distribution | 1991 |
Differential effects of petit mal anticonvulsants and convulsants on thalamic neurones: GABA current blockade.
Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Epilepsy, Absence; Ethosuximide; gamma-Aminobutyric Acid; In Vitro Techniques; Iontophoresis; Neurons; Pentylenetetrazole; Picrotoxin; Rats; Succinimides; Thalamus | 1990 |
Differential effects of petit mal anticonvulsants and convulsants on thalamic neurones: calcium current reduction.
Topics: Animals; Anticonvulsants; Calcium Channels; Convulsants; Epilepsy, Absence; Ethosuximide; gamma-Aminobutyric Acid; Neurons; Pentylenetetrazole; Rats; Structure-Activity Relationship; Succinimides; Thalamus | 1990 |
Influence of calcium channel inhibitors upon the anticonvulsant efficacy of common antiepileptics against pentylenetetrazol-induced convulsions in mice.
Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Diltiazem; Drug Therapy, Combination; Ethosuximide; Male; Mice; Nifedipine; Pentylenetetrazole; Phenobarbital; Reference Values; Seizures; Valproic Acid; Verapamil | 1990 |
Ethosuximide affects both pentylenetetrazole- and kainate-induced clonic seizures but differentiates between tonic-clonic seizures.
Topics: Animals; Anticonvulsants; Ethosuximide; Kainic Acid; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures | 1989 |
Examination of the potential antiepileptic activity of calcium antagonists with different sites of action.
Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Electroshock; Endoplasmic Reticulum; Ethosuximide; Female; In Vitro Techniques; Mice; Mice, Inbred ICR; Pentylenetetrazole; Seizures | 1989 |
Pentylenetetrazol-induced seizures in pigeons and the effects of ethosuximide thereon.
Topics: Animals; Anticonvulsants; Columbidae; Ethosuximide; Pentylenetetrazole; Seizures; Time Factors | 1989 |
Effect of anticonvulsants on pentylenetetrazol-induced power spectrum changes in electroencephalograms in rats.
Topics: Animals; Anticonvulsants; Cerebral Cortex; Cyclic AMP; Electroencephalography; Ethosuximide; Male; Pentylenetetrazole; Phenobarbital; Rats; Rats, Inbred Strains; Seizures; Valproic Acid | 1987 |
Evidence for involvement of the astrocytic benzodiazepine receptor in the mechanism of action of convulsant and anticonvulsant drugs.
Topics: Animals; Anticonvulsants; Astrocytes; Barbiturates; Benzodiazepinones; Brain; Carbamazepine; Cells, Cultured; Convulsants; Diazepam; Ethosuximide; Mice; Neurons; Pentylenetetrazole; Phenobarbital; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Trimethadione; Valproic Acid | 1988 |
Influence of ethosuximide and dipropylacetate on metrazol-induced electrocorticographic changes during ontogenesis in rats.
Topics: Animals; Brain; Electroencephalography; Ethosuximide; Pentylenetetrazole; Rats; Rats, Inbred Strains; Theta Rhythm; Valproic Acid | 1986 |
Effect of ethosuximide alone and in combination with gamma-aminobutyric acid receptor agonists on brain gamma-aminobutyric acid concentration, anticonvulsant activity and neurotoxicity in mice.
Topics: Animals; Brain Chemistry; Ethosuximide; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Mice, Inbred Strains; Nervous System; Pentylenetetrazole; Receptors, GABA-A; Seizures | 1986 |
Evidence for increased activity of mouse brain fatty acid cyclooxygenase following drug-induced convulsions.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Brain; Dinoprost; Dinoprostone; Ethosuximide; Female; Kinetics; Mice; Microsomes; Pentylenetetrazole; Picrotoxin; Prostaglandin-Endoperoxide Synthases; Prostaglandins E; Prostaglandins F; Seizures; Strychnine | 1987 |
Differentiation of alcohol and barbital physical dependence.
Topics: Animals; Barbital; Barbiturates; Diazepam; Ethanol; Ethosuximide; Male; Mice; Morphine; Naloxone; Pentylenetetrazole; Phenytoin; Substance Withdrawal Syndrome | 1986 |
Effect of stimulus intensity on the profile of anticonvulsant activity of phenytoin, ethosuximide and valproate.
Topics: Animals; Anticonvulsants; Bicuculline; Electroshock; Ethosuximide; Male; Mice; Pentylenetetrazole; Phenytoin; Picrotoxin; Seizures; Valproic Acid | 1985 |
[The anticonvulsant action of propranolol in pentylenetetrazole-induced convulsions].
Topics: Animals; Anticonvulsants; Dose-Response Relationship, Drug; Ethosuximide; Male; Mice; Pentylenetetrazole; Phenobarbital; Propranolol | 1985 |
Drug-induced catalepsy as influenced by convulsant and anticonvulsant drugs.
Topics: Animals; Anticonvulsants; Arecoline; Bemegride; Caffeine; Catalepsy; Central Nervous System Stimulants; Drug Synergism; Ethosuximide; Haloperidol; Humans; Lobeline; Male; Mice; Mice, Inbred Strains; Nicotine; Nikethamide; Paraoxon; Pentylenetetrazole; Pilocarpine; Tetrabenazine; Tremorine; Trifluoperazine | 1973 |
Alkylation reactions of hydantoins and succinimides.
Topics: Alkylation; Animals; Anticonvulsants; Benzyl Compounds; Chemical Phenomena; Chemistry; Ethosuximide; Hydantoins; Magnetic Resonance Spectroscopy; Male; Mice; Nitro Compounds; Pentylenetetrazole; Phenytoin; Spectrophotometry, Infrared; Succinimides | 1973 |
[Pharmacology of 2,4-dimethysulfolane].
Topics: Animals; Anticonvulsants; Blood Circulation; Cats; Central Nervous System; Central Nervous System Stimulants; Electroencephalography; Ethosuximide; Guinea Pigs; Heart; Male; Mice; Pentylenetetrazole; Rats | 1971 |
Dependence of anticonvulsant drug action on central monoamines.
Topics: Animals; Anticonvulsants; Dopamine; Drug Interactions; Electroshock; Ethosuximide; Lethal Dose 50; Male; Mice; Mice, Inbred Strains; Norepinephrine; Pentylenetetrazole; Phenobarbital; Phenytoin; Receptors, Drug; Seizures; Serotonin; Time Factors | 1973 |
[Inhibition of pentetrazole-induced hypersynchronous activity in thalamocortical system by ethosuximide].
Topics: Animals; Electrodes, Implanted; Electroencephalography; Ethosuximide; Male; Motor Cortex; Muscle Tonus; Olfactory Bulb; Pentylenetetrazole; Photic Stimulation; Rats; Rats, Inbred Strains; Reflex, Startle; Thalamus; Time Factors; Visual Cortex | 1971 |
Language-induced epilepsy.
Topics: Electroencephalography; Epilepsy; Ethosuximide; Humans; Male; Middle Aged; Movement Disorders; Pentylenetetrazole; Phenobarbital; Reading; Speech; Speech Disorders; Unconsciousness; Writing | 1967 |
Excitatory and depressant effects of delta 9-tetrahydrocannabinol and cannabidiol on cortical evoked responses in the conscious rat.
Topics: Animals; Anticonvulsants; Cannabidiol; Cannabinoids; Cerebral Cortex; Convulsants; Dronabinol; Ethosuximide; Evoked Potentials; Pentylenetetrazole; Phenytoin; Rats; Rats, Inbred Strains | 1981 |
Effect of antiepileptic drugs on metrazol convulsions during ontogenesis in the rat.
Topics: Age Factors; Animals; Anticonvulsants; Clonazepam; Ethosuximide; Male; Pentylenetetrazole; Rats; Seizures; Valproic Acid | 1981 |
Influence of ethosuximide on metrazol-induced seizures during ontogenesis in rats.
Topics: Aging; Animals; Dose-Response Relationship, Drug; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures | 1983 |
Influence of clonazepam and ethosuximide on ECoG pattern induced by metrazol during ontogenesis in rats.
Topics: Age Factors; Animals; Benzodiazepinones; Cerebral Cortex; Clonazepam; Dose-Response Relationship, Drug; Electroencephalography; Ethosuximide; Evoked Potentials; Male; Pentylenetetrazole; Rats; Seizures | 1982 |
A behavioural and pharmacological evaluation of the discriminative stimulus induced by pentylenetetrazole in the pig.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Cues; Diazepam; Discrimination, Psychological; Electroshock; Emotions; Ethosuximide; Male; Pentylenetetrazole; Reinforcement Schedule; Swine | 1993 |
Is the site of action of ethosuximide in the hindbrain?
Topics: Animals; Anticonvulsants; Brain Stem; Clonazepam; Decerebrate State; Electrocardiography; Electroencephalography; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Wistar; Rhombencephalon; Seizures; Valproic Acid | 1994 |
Ethosuximide suppresses seizures and lethality induced by picrotoxin in developing rats.
Topics: Animals; Anticonvulsants; Behavior, Animal; Epilepsies, Myoclonic; Epilepsy, Tonic-Clonic; Ethosuximide; Male; Pentylenetetrazole; Picrotoxin; Rats; Rats, Wistar; Seizures | 1993 |
Protective effect of flunarizine and nifedipine alone and in combination with anticonvulsant drugs against PTZ-induced seizures in mice.
Topics: Animals; Anticonvulsants; Carbamazepine; Dose-Response Relationship, Drug; Drug Interactions; Ethosuximide; Female; Flunarizine; Male; Mice; Nifedipine; Pentylenetetrazole; Phenytoin; Seizures | 1993 |
Antiepileptic drugs--their effects on kindled seizures and kindling-induced learning impairments.
Topics: Animals; Anticonvulsants; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Ethosuximide; Kindling, Neurologic; Learning Disabilities; Male; Pentylenetetrazole; Phenobarbital; Rats; Rats, Wistar; Seizures; Valproic Acid | 1995 |
Influence of nicardipine, nimodipine and flunarizine on the anticonvulsant efficacy of antiepileptics against pentylenetetrazol in mice.
Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Clonazepam; Drug Interactions; Ethosuximide; Flunarizine; Male; Mice; Mice, Inbred Strains; Motor Activity; Nicardipine; Nimodipine; Pentylenetetrazole; Random Allocation; Seizures; Valproic Acid | 1996 |
Ethosuximide specifically antagonizes the effect of pentylenetetrazol in the rat entorhinal cortex.
Topics: Animals; Dose-Response Relationship, Drug; Entorhinal Cortex; Ethosuximide; Evoked Potentials; Male; Pentylenetetrazole; Rats; Rats, Sprague-Dawley | 1996 |
Ontogeny of ethosuximide action against two seizure models in rats is different.
Topics: Action Potentials; Animals; Anticonvulsants; Disease Models, Animal; Electroencephalography; Ethosuximide; Pentylenetetrazole; Rats; Seizures | 1998 |
A potential anti-asthmatic drug, CR 2039, enhances the anticonvulsive activity of some antiepileptic drugs against pentetrazol in mice.
Topics: Animals; Anticonvulsants; Benzamides; Bronchodilator Agents; Clonazepam; Convulsants; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Ethosuximide; Male; Mice; Pentylenetetrazole; Seizures; Tetrazoles | 1998 |
Additive anticonvulsant effect of flunarizine and sodium valproate on electroshock and chemoshock induced seizures in mice.
Topics: Animals; Anticonvulsants; Carbamazepine; Disease Models, Animal; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Electroshock; Ethosuximide; Flunarizine; Male; Mice; Motor Activity; Pentylenetetrazole; Phenytoin; Seizures; Valproic Acid | 1998 |
N(G)-nitro-L-arginine impairs the anticonvulsive action of ethosuximide against pentylenetetrazol.
Topics: Animals; Anticonvulsants; Arginine; Convulsants; Diazepam; Drug Interactions; Enzyme Inhibitors; Ethosuximide; Male; Mice; Nitroarginine; Pentylenetetrazole; Phenobarbital; Psychomotor Performance; Seizures; Valproic Acid | 1999 |
The fruit essential oil of Pimpinella anisum exerts anticonvulsant effects in mice.
Topics: Animals; Anticonvulsants; Apiaceae; Convulsants; Electroshock; Ethosuximide; Fruit; India; Iran; Lethal Dose 50; Male; Mice; Oils, Volatile; Pentylenetetrazole; Postural Balance; Seizures; Turkey | 1999 |
7-Nitroindazole, a nitric oxide synthase inhibitor, enhances the anticonvulsive action of ethosuximide and clonazepam against pentylenetetrazol-induced convulsions.
Topics: Animals; Anticonvulsants; Avoidance Learning; Clonazepam; Disease Models, Animal; Drug Interactions; Epilepsies, Myoclonic; Ethosuximide; Indazoles; Male; Mice; Motor Skills; Neuroprotective Agents; Nitric Oxide; Nitric Oxide Synthase; Pentylenetetrazole; Seizures | 2000 |
Comparative profiles of sodium valproate and ethosuximide on electro-behavioural correlates in gamma-hydroxybutyrate and pentylenetetrazol induced absence seizures in rats.
Topics: Animals; Anticonvulsants; Convulsants; Disease Models, Animal; Electroencephalography; Epilepsy, Absence; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Wistar; Sodium Oxybate; Species Specificity; Valproic Acid | 2000 |
Is spontaneous high-voltage rhythmic spike discharge in Long Evans rats an absence-like seizure activity?
Topics: Animals; Anticonvulsants; Arousal; Behavior, Animal; Cerebral Cortex; Disease Models, Animal; Electric Stimulation; Electrodes, Implanted; Electroencephalography; Electromyography; Epilepsy, Absence; Ethosuximide; Female; Immobilization; Penicillins; Pentylenetetrazole; Rats; Rats, Inbred Strains; Rats, Long-Evans; Sleep; Time Factors; Wakefulness | 2004 |
NOTE ON THE INTERACTIONS OF AMPHETAMINE WITH ANTICONVULSANT DRUGS.
Topics: Amphetamine; Amphetamines; Animals; Anticonvulsants; Electricity; Electroshock; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Ethosuximide; Mice; Pentylenetetrazole; Pharmacology; Phenobarbital; Phenytoin; Research; Seizures | 1964 |
Isobolographic and subthreshold analysis of interactions among felbamate and four conventional antiepileptic drugs in pentylenetetrazole-induced seizures in mice.
Topics: Animals; Anticonvulsants; Behavior, Animal; Clonazepam; Disease Models, Animal; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Epilepsies, Myoclonic; Ethosuximide; Felbamate; Female; Humans; Lethal Dose 50; Mice; Motor Activity; Neurotoxicity Syndromes; Pentylenetetrazole; Phenobarbital; Phenylcarbamates; Propylene Glycols; Seizures; Valproic Acid | 2004 |
Ethosuximide and valproate display high efficacy against lindane-induced seizures in mice.
Topics: Animals; Anticonvulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethosuximide; GABA Agents; Hexachlorocyclohexane; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Mice; Pentylenetetrazole; Seizures; Valproic Acid | 2004 |
Pharmacodynamic and/or pharmacokinetic characteristics of interactions between loreclezole and four conventional antiepileptic drugs in pentylenetetrazole-induced seizures in mice: an isobolographic analysis.
Topics: Animals; Anticonvulsants; Clonazepam; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Ethosuximide; Kindling, Neurologic; Linear Models; Male; Mice; Pentylenetetrazole; Phenobarbital; Seizures; Triazoles; Valproic Acid | 2005 |
Imaging the neural substrates involved in the genesis of pentylenetetrazol-induced seizures.
Topics: Animals; Brain Mapping; Dentate Gyrus; Disease Models, Animal; Electroencephalography; Epilepsy, Absence; Ethosuximide; Hippocampus; Magnetic Resonance Imaging; Male; Neural Pathways; Oxygen; Pentylenetetrazole; Pilot Projects; Prosencephalon; Rats; Rats, Sprague-Dawley; Seizures; Thalamic Nuclei; Thalamus | 2006 |
Characterization of the anticonvulsant, behavioral and pharmacokinetic interaction profiles of stiripentol in combination with clonazepam, ethosuximide, phenobarbital, and valproate using isobolographic analysis.
Topics: Animals; Anticonvulsants; Brain Chemistry; Clonazepam; Dioxolanes; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Ethosuximide; Male; Mice; Neurotoxicity Syndromes; Pentylenetetrazole; Phenobarbital; Seizures; Valproic Acid | 2006 |
Thalidomide inhibits pentylenetetrazole-induced seizures.
Topics: Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Wistar; Seizures; Severity of Illness Index; Valproic Acid | 2007 |
Interactions of tiagabine with ethosuximide in the mouse pentylenetetrazole-induced seizure model: an isobolographic analysis for non-parallel dose-response relationship curves.
Topics: Animals; Anticonvulsants; Brain; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Ethosuximide; Fluorescence Polarization Immunoassay; Male; Mice; Nipecotic Acids; Pentylenetetrazole; Seizures; Tiagabine; Tissue Distribution | 2008 |
Isobolographic characterization of the anticonvulsant interaction profiles of levetiracetam in combination with clonazepam, ethosuximide, phenobarbital and valproate in the mouse pentylenetetrazole-induced seizure model.
Topics: Animals; Anticonvulsants; Clonazepam; Convulsants; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Ethosuximide; Levetiracetam; Male; Mice; Pentylenetetrazole; Phenobarbital; Piracetam; Seizures; Valproic Acid | 2009 |
Detection of nonlinear interactions of EEG alpha waves in the brain by a new coherence measure and its application to epilepsy and anti-epileptic drug therapy.
Topics: Animals; Anticonvulsants; Cerebral Cortex; Convulsants; Electroencephalography; Epilepsy; Ethosuximide; Humans; Mathematics; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Seizures; Thalamus | 2011 |
Effect of intracranial administration of ethosuximide in rats with spontaneous or pentylenetetrazol-induced spike-wave discharges.
Topics: Animals; Anticonvulsants; Brain; Disease Models, Animal; Epilepsy, Absence; Ethosuximide; Infusions, Intraventricular; Male; Pentylenetetrazole; Rats; Rats, Long-Evans; Rats, Wistar | 2011 |
Effects of WIN 55,212-2 mesylate (a synthetic cannabinoid) on the protective action of clonazepam, ethosuximide, phenobarbital and valproate against pentylenetetrazole-induced clonic seizures in mice.
Topics: Animals; Anticonvulsants; Avoidance Learning; Benzoxazines; Brain; Cannabinoid Receptor Agonists; Clonazepam; Disease Models, Animal; Drug Synergism; Ethosuximide; Hand Strength; Male; Mice; Morpholines; Naphthalenes; Pentylenetetrazole; Phenobarbital; Seizures; Valproic Acid | 2011 |
Synthesis and anticonvulsant activity of new 1-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-diones.
Topics: Administration, Oral; Animals; Anticonvulsants; Convulsants; Dose-Response Relationship, Drug; Drug Design; Drug Evaluation, Preclinical; Electroshock; Ethosuximide; Injections, Intraperitoneal; Mice; Molecular Structure; Motor Activity; Pentylenetetrazole; Phenytoin; Piperazines; Rats; Seizures; Structure-Activity Relationship; Succinimides; Time Factors | 2011 |
Anticonvulsant effect of the essential oil and methanolic extracts of Zataria multiflora Boiss.
Topics: Animals; Anticonvulsants; Distillation; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Electroshock; Ethosuximide; Injections, Intraperitoneal; Lamiaceae; Male; Methanol; Mice; Oils, Volatile; Pentylenetetrazole; Phenytoin; Phytotherapy; Plant Extracts; Plant Oils; Plants, Medicinal; Postural Balance; Rotarod Performance Test; Seizures; Sesame Oil; Solvents | 2013 |
Synthesis, physicochemical, and anticonvulsant properties of new N-Mannich bases derived from pyrrolidine-2,5-dione and its 3-methyl analog.
Topics: Animals; Anticonvulsants; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Design; Electroshock; Ethosuximide; Male; Mannich Bases; Mice; Molecular Structure; Motor Activity; Neurotoxicity Syndromes; Pentylenetetrazole; Pyrrolidines; Rotarod Performance Test; Seizures; Structure-Activity Relationship; Valproic Acid | 2014 |
Potential mechanisms involved in the anticonvulsant effect of walnut extract on pentylenetetrazole-induced seizure.
Topics: Animals; Anticonvulsants; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Ethosuximide; Flumazenil; Juglans; Male; Pentylenetetrazole; Plant Extracts; Rats; Rats, Wistar; Seizures | 2014 |
Ethosuximide Reduces Mortality and Seizure Severity in Response to Pentylenetetrazole Treatment During Ethanol Withdrawal.
Topics: Alcoholism; Animals; Anticonvulsants; Ethosuximide; Male; Mice; Mice, Inbred DBA; Mortality; Pentylenetetrazole; Seizures; Severity of Illness Index; Substance Withdrawal Syndrome | 2015 |
Interactions between an antidepressant reboxetine and four classic antiepileptic drugs in the mouse model of myoclonic seizures.
Topics: Animals; Anticonvulsants; Antidepressive Agents; Avoidance Learning; Clonazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Epilepsies, Myoclonic; Ethosuximide; Male; Mice; Morpholines; Motor Skills; Pentylenetetrazole; Phenobarbital; Reboxetine; Valproic Acid | 2015 |
A Caenorhabditis elegans assay of seizure-like activity optimised for identifying antiepileptic drugs and their mechanisms of action.
Topics: Animals; Anticonvulsants; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Convulsants; Disease Models, Animal; Drug Evaluation, Preclinical; Ethosuximide; Pentylenetetrazole; Receptors, GABA-A; Seizures | 2018 |
N-Benzyl-(2,5-dioxopyrrolidin-1-yl)propanamide (AS-1) with Hybrid Structure as a Candidate for a Broad-Spectrum Antiepileptic Drug.
Topics: Animals; Anticonvulsants; Behavior, Animal; Dose-Response Relationship, Drug; Epilepsy; Ethosuximide; Lacosamide; Levetiracetam; Male; Mice; Pentylenetetrazole; Pyrrolidines; Seizures; Valproic Acid; Zebrafish | 2020 |
Evaluation of the impact of compound C11 a new anticonvulsant candidate on cognitive functions and hippocampal neurogenesis in mouse brain.
Topics: Animals; Anticonvulsants; Brain; Cognition; Epilepsy; Ethosuximide; Hippocampus; Lacosamide; Levetiracetam; Male; Mice; Mice, Inbred C57BL; Neurogenesis; Pentylenetetrazole; Spatial Memory | 2020 |
Long-term vigabatrin treatment modifies pentylenetetrazole-induced seizures in mice: focused on GABA brain concentration.
Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Brain; Clonazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethosuximide; gamma-Aminobutyric Acid; Mice; Pentylenetetrazole; Seizures; Time Factors; Valproic Acid; Vigabatrin | 2020 |
Anticonvulsant activity of Valeriana edulis roots and valepotriates on the pentylenetetrazole-induced seizures in rats.
Topics: Animals; Anticonvulsants; Computer Simulation; Disease Models, Animal; Electroencephalography; Ethosuximide; Iridoids; Male; Pentylenetetrazole; Plant Extracts; Plant Roots; Rats; Rats, Wistar; Seizures; Time Factors; Valerian | 2021 |
Mechanochemical synthesis and anticonvulsant activity of 3-aminopyrrolidine-2,5-dione derivatives.
Topics: Animals; Anticonvulsants; Ethosuximide; Humans; Mice; Molecular Structure; Neuroblastoma; Pentylenetetrazole; Seizures; Spectroscopy, Fourier Transform Infrared; Structure-Activity Relationship | 2023 |