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pentylenetetrazole and ethosuximide

pentylenetetrazole has been researched along with ethosuximide in 77 studies

Research

Studies (77)

TimeframeStudies, this research(%)All Research%
pre-199029 (37.66)18.7374
1990's18 (23.38)18.2507
2000's13 (16.88)29.6817
2010's12 (15.58)24.3611
2020's5 (6.49)2.80

Authors

AuthorsStudies
Butler, DE; L'Italien, YJ; Marriott, JG; Nordin, IC; Poschel, PH; Zweisler, L1
Butler, DE; Marriott, JG; Poschel, BP1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Alkskas, IA; Azam, F; Khokra, SL; Prakash, O1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Consroe, PF; Wolkin, AL1
Ferrendelli, JA; Kinscherf, DA1
Banerjee, U; Yeoh, PN1
Frey, HH; Löscher, W1
Mares, P; Stanková, L1
Goehring, RR; Greenwood, TD; Pisipati, JS; Wolfe, JF1
Aguilar-Veiga, E; Galán-Valiente, J; Méndez-Alvarez, E; Sierra-Marcuño, G; Sierra-Paredes, G; Soto-Otero, R1
Coulter, DA; Huguenard, JR; Prince, DA2
Czuczwar, SJ; Kleinrok, Z; Małek, U1
Kulhánková, I; Mares, P; Mirvaldová, H; Roztocilová, L; Velísek, L; Velísková, J1
Rahwan, RG; Wong, WS1
Jakubow, JJ; Poling, A; Schlinger, H1
Aburada, M; Hosoya, E; Iizuka, S; Ishige, A; Matsuzaki, Y; Sakamoto, K; Sekiguchi, K; Sugaya, E1
Bender, AS; Hertz, L1
Mares, P; Velísek, L2
Chweh, AY; Lin-Michell, E; Swinyard, EA1
Centra, M; Keeting, PE; Lysz, TW; Markey, K1
Kaneda, H; Kaneto, H; Kawatani, S1
Piredda, SG; Swinyard, EA; Woodhead, JH1
Lasek, R; Müller, M1
Zetler, G1
Forrest, TP; Gilroy, ML; Vohra, MM; Yung, DK1
Millichap, JG1
Kästner, I; Müller, M; Schmiedel, R; Wenzel, J1
Frey, HH; Meyer, H1
Krüger, E; Müller, M; Wenzel, J1
Geschwind, N; Sherwin, I1
Karler, R; Turkanis, SA1
Mares, P; Maresová, D; Schickerová, R1
Mares, P; Zouhar, A1
Carey, MP; Fry, JP1
Kubová, H; Mares, P; Pohl, M; Zelízko, M1
Mares, P; Micianiková, D; Rokyta, R; Velísek, L; Velísková, J1
Pleuvry, BJ; Rodger, C1
Becker, A; Brosz, M; Grecksch, G1
Brudniak, T; Czuczwar, SJ; Gasior, M; Kamiński, R; Kleinrok, Z1
Stringer, JL1
Mares, P1
Czuczwar, SJ; Gasior, M; Kleinrok, Z; Kozicka, M; Pietrasiewicz, T; Turski, WA1
David, J; Joseph, S; Joseph, T1
Czuczwar, SJ; Kleinrok, Z; Klonowski, P; Tutka, P1
Fanaee, GH; Javadi, M; Kamalinejad, M; Majzoob, S; Pourgholami, MH; Sayyah, M1
Borowicz, KK; Czuczwar, SJ; Kleinrok, Z; Luszczki, J1
David, J; Joseph, T; Kumaresan, S1
Shaw, FZ1
FREY, HH1
Borowicz, KK; Czuczwar, SJ; Luszczki, JJ1
Czuczwar, SJ; Dekundy, A; Kaminski, RM; Tochman, AM; Turski, WA1
Czuczwar, SJ; Luszczki, JJ; Patsalos, PN; Ratnaraj, N2
Brevard, ME; Ferris, CF; King, JA; Kulkarni, P1
Calderon, A; Palencia, G; Sotelo, J1
Luszczki, JJ1
Andres-Mach, MM; Czuczwar, SJ; Dudra-Jastrzebska, M; Luszczki, JJ; Patsalos, PN; Ratnaraj, N1
Garg, S; Hinich, MJ; Mirski, MA; Sherman, D; Thakor, NV; White, MA; Zhang, N1
Chen, SD; Huang, YH; Shaw, FZ; Yeh, KH1
Andres-Mach, M; Barcicka-Klosowska, B; Czuczwar, SJ; Florek-Luszczki, M; Haratym-Maj, A; Luszczki, JJ1
Kamiński, K; Obniska, J; Rzepka, S1
Borowicz, KK; Czuczwar, SJ; Piskorska, B; Stępniak, B1
Abdar, M; Mandegary, A; Sharififar, F1
Filipek, B; Kamiński, K; Obniska, J; Rapacz, A; Rybka, S1
Asadi-Shekaari, M; Eslami, A; Joukar, S; Kalantaripour, T1
Godwin, DW; Masicampo, ML; Riegle, MA; Shan, HQ; Xu, V1
Borowicz, KK; Popławska, M; Wróblewska, D1
Barclay, JW; Burgoyne, RD; Cunliffe, VT; Dodd, S; Grimes, D; Jones, A; Marson, AG; Morgan, A; Sills, GJ; Wong, SQ1
Abram, M; Andres-Mach, M; Esguerra, CV; Gawel, K; Jakubiec, M; Kamiński, K; Latacz, G; Lubelska, A; Nieoczym, D; Pieróg, M; Rapacz, A; Socała, K; Szewczyk, A; Szulczyk, B; Wlaź, P; Zagaja, M; Łuszczki, JJ1
Abram, M; Andres-Mach, M; Kaminski, K; Luszczki, J; Maj, M; Rola, R; Szewczyk, A; Zagaja, M1
Czuczwar, SJ; Krzyżanowski, M; Świąder, K; Świąder, MJ; Wróbel, A; Zakrocka, I; Łuszczki, JJ1
Contreras-Murillo, G; González-Trujano, ME; Hidalgo-Flores, FJ; López-Najera, CA; Magdaleno-Madrigal, VM; Navarrete-Castro, A; Sánchez, CG1
Dziubina, A; Jarzyński, S; Pękala, E; Piska, K; Popiół, J; Rapacz, A; Rudolf, B; Wojtulewski, S1

Reviews

1 review(s) available for pentylenetetrazole and ethosuximide

ArticleYear
Relation of laboratory evaluation to clinical effectiveness of antiepileptic drugs.
    Epilepsia, 1969, Volume: 10, Issue:2

    Topics: Acetazolamide; Adrenocorticotropic Hormone; Animals; Anticonvulsants; Benzazepines; Clinical Trials as Topic; Drug Tolerance; Electroencephalography; Electroshock; Epilepsy; Ethosuximide; Humans; Pentylenetetrazole; Phenobarbital; Phenytoin; Primidone; Seizures; Trimethadione; Urea

1969

Trials

2 trial(s) available for pentylenetetrazole and ethosuximide

ArticleYear
Relation of laboratory evaluation to clinical effectiveness of antiepileptic drugs.
    Epilepsia, 1969, Volume: 10, Issue:2

    Topics: Acetazolamide; Adrenocorticotropic Hormone; Animals; Anticonvulsants; Benzazepines; Clinical Trials as Topic; Drug Tolerance; Electroencephalography; Electroshock; Epilepsy; Ethosuximide; Humans; Pentylenetetrazole; Phenobarbital; Phenytoin; Primidone; Seizures; Trimethadione; Urea

1969
Effects of fluoxetine on the anticonvulsant action of valproate and ethosuximide in mouse model of myoclonic convulsions.
    Annals of agricultural and environmental medicine : AAEM, 2012, Volume: 19, Issue:3

    Topics: Animals; Anticonvulsants; Antidepressive Agents, Second-Generation; Avoidance Learning; Convulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Epilepsies, Myoclonic; Ethosuximide; Fluorescent Antibody Technique; Fluoxetine; Male; Memory, Long-Term; Mice; Motor Activity; Pentylenetetrazole; Seizures; Selective Serotonin Reuptake Inhibitors; Valproic Acid

2012

Other Studies

75 other study(ies) available for pentylenetetrazole and ethosuximide

ArticleYear
Amnesia-reversal activity of a series of N-[(disubstituted-amino)alkyl] -2-oxo-1-pyrrolidineacetamides, including pramiracetam.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:5

    Topics: Amnesia; Animals; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Electroshock; Humans; Male; Mice; Mice, Inbred Strains; Pyrrolidines; Structure-Activity Relationship

1984
Cognition-activating properties of 3-(Aryloxy)pyridines.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Animals; Cognition; Dose-Response Relationship, Drug; Male; Mice; Psychotropic Drugs; Pyridines; Structure-Activity Relationship

1981
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Synthesis of some novel N4-(naphtha[1,2-d]thiazol-2-yl)semicarbazides as potential anticonvulsants.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:1

    Topics: Animals; Anticonvulsants; Brain Chemistry; Glutathione Peroxidase; Malondialdehyde; Mice; Motor Activity; Rats; Seizures; Semicarbazides; Structure-Activity Relationship; Superoxide Dismutase

2009
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Anticonvulsant interaction of cannabidiol and ethosuximide in rats.
    The Journal of pharmacy and pharmacology, 1977, Volume: 29, Issue:8

    Topics: Animals; Anticonvulsants; Cannabidiol; Cannabinoids; Drug Interactions; Ethosuximide; Male; Pentylenetetrazole; Proadifen; Rats

1977
Cyclic nucleotides in epileptic brain: effects of pentylenetetrazol on regional cyclic AMP and cyclic GMP levels in vivo.
    Epilepsia, 1977, Volume: 18, Issue:4

    Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Cyclic AMP; Cyclic GMP; Ethosuximide; Female; Hippocampus; Mice; Pentylenetetrazole; Phenobarbital; Phenytoin; Seizures; Thalamus

1977
The temporal dimensions of anticonvulsant action of some newer benzodiazepines against metrazol induced seizures in mice and rats.
    Medical biology, 1977, Volume: 55, Issue:6

    Topics: Animals; Benzodiazepines; Clonazepam; Diazepam; Drug Evaluation, Preclinical; Ethosuximide; Female; Flurazepam; Male; Mice; Nitrazepam; Pentylenetetrazole; Phenobarbital; Seizures; Trimethadione

1977
Di-n-propylacetic acid--profile of anticonvulsant activity in mice.
    Arzneimittel-Forschung, 1976, Volume: 26, Issue:2

    Topics: Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Electroshock; Ethosuximide; Female; Male; Mice; Pentylenetetrazole; Phenobarbital; Picrotoxin; Seizures; Strychnine; Trimethadione; Valerates; Valproic Acid

1976
Influence of phenobarbital on ECoG phenomena induced by metrazol in rats during ontogenesis.
    Physiological research, 1992, Volume: 41, Issue:2

    Topics: Aging; Animals; Cerebral Cortex; Clonazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Electrodes; Electroencephalography; Epilepsy; Ethosuximide; Injections, Intraperitoneal; Male; Pentylenetetrazole; Phenobarbital; Prohibitins; Rats; Rats, Wistar; Valproic Acid

1992
Synthesis and anticonvulsant evaluation of some new 2-benzylsuccinimides.
    Journal of pharmaceutical sciences, 1991, Volume: 80, Issue:8

    Topics: Animals; Anticonvulsants; Chemical Phenomena; Chemistry, Physical; Electroshock; Ethosuximide; Male; Mice; Pentylenetetrazole; Postural Balance; Succinimides

1991
Correlation between ethosuximide brain levels measured by high performance liquid chromatography and its antiepileptic potential.
    Research communications in chemical pathology and pharmacology, 1991, Volume: 71, Issue:3

    Topics: Animals; Anticonvulsants; Blood-Brain Barrier; Brain; Chromatography, High Pressure Liquid; Electrophysiology; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Tissue Distribution

1991
Differential effects of petit mal anticonvulsants and convulsants on thalamic neurones: GABA current blockade.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Epilepsy, Absence; Ethosuximide; gamma-Aminobutyric Acid; In Vitro Techniques; Iontophoresis; Neurons; Pentylenetetrazole; Picrotoxin; Rats; Succinimides; Thalamus

1990
Differential effects of petit mal anticonvulsants and convulsants on thalamic neurones: calcium current reduction.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Animals; Anticonvulsants; Calcium Channels; Convulsants; Epilepsy, Absence; Ethosuximide; gamma-Aminobutyric Acid; Neurons; Pentylenetetrazole; Rats; Structure-Activity Relationship; Succinimides; Thalamus

1990
Influence of calcium channel inhibitors upon the anticonvulsant efficacy of common antiepileptics against pentylenetetrazol-induced convulsions in mice.
    Neuropharmacology, 1990, Volume: 29, Issue:10

    Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Diltiazem; Drug Therapy, Combination; Ethosuximide; Male; Mice; Nifedipine; Pentylenetetrazole; Phenobarbital; Reference Values; Seizures; Valproic Acid; Verapamil

1990
Ethosuximide affects both pentylenetetrazole- and kainate-induced clonic seizures but differentiates between tonic-clonic seizures.
    Canadian journal of physiology and pharmacology, 1989, Volume: 67, Issue:10

    Topics: Animals; Anticonvulsants; Ethosuximide; Kainic Acid; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures

1989
Examination of the potential antiepileptic activity of calcium antagonists with different sites of action.
    General pharmacology, 1989, Volume: 20, Issue:3

    Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Electroshock; Endoplasmic Reticulum; Ethosuximide; Female; In Vitro Techniques; Mice; Mice, Inbred ICR; Pentylenetetrazole; Seizures

1989
Pentylenetetrazol-induced seizures in pigeons and the effects of ethosuximide thereon.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:1

    Topics: Animals; Anticonvulsants; Columbidae; Ethosuximide; Pentylenetetrazole; Seizures; Time Factors

1989
Effect of anticonvulsants on pentylenetetrazol-induced power spectrum changes in electroencephalograms in rats.
    Epilepsy research, 1987, Volume: 1, Issue:5

    Topics: Animals; Anticonvulsants; Cerebral Cortex; Cyclic AMP; Electroencephalography; Ethosuximide; Male; Pentylenetetrazole; Phenobarbital; Rats; Rats, Inbred Strains; Seizures; Valproic Acid

1987
Evidence for involvement of the astrocytic benzodiazepine receptor in the mechanism of action of convulsant and anticonvulsant drugs.
    Life sciences, 1988, Volume: 43, Issue:6

    Topics: Animals; Anticonvulsants; Astrocytes; Barbiturates; Benzodiazepinones; Brain; Carbamazepine; Cells, Cultured; Convulsants; Diazepam; Ethosuximide; Mice; Neurons; Pentylenetetrazole; Phenobarbital; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Trimethadione; Valproic Acid

1988
Influence of ethosuximide and dipropylacetate on metrazol-induced electrocorticographic changes during ontogenesis in rats.
    Physiologia Bohemoslovaca, 1986, Volume: 35, Issue:2

    Topics: Animals; Brain; Electroencephalography; Ethosuximide; Pentylenetetrazole; Rats; Rats, Inbred Strains; Theta Rhythm; Valproic Acid

1986
Effect of ethosuximide alone and in combination with gamma-aminobutyric acid receptor agonists on brain gamma-aminobutyric acid concentration, anticonvulsant activity and neurotoxicity in mice.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Brain Chemistry; Ethosuximide; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Mice, Inbred Strains; Nervous System; Pentylenetetrazole; Receptors, GABA-A; Seizures

1986
Evidence for increased activity of mouse brain fatty acid cyclooxygenase following drug-induced convulsions.
    Brain research, 1987, Apr-07, Volume: 408, Issue:1-2

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Brain; Dinoprost; Dinoprostone; Ethosuximide; Female; Kinetics; Mice; Microsomes; Pentylenetetrazole; Picrotoxin; Prostaglandin-Endoperoxide Synthases; Prostaglandins E; Prostaglandins F; Seizures; Strychnine

1987
Differentiation of alcohol and barbital physical dependence.
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1986, Volume: 6, Issue:2

    Topics: Animals; Barbital; Barbiturates; Diazepam; Ethanol; Ethosuximide; Male; Mice; Morphine; Naloxone; Pentylenetetrazole; Phenytoin; Substance Withdrawal Syndrome

1986
Effect of stimulus intensity on the profile of anticonvulsant activity of phenytoin, ethosuximide and valproate.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:3

    Topics: Animals; Anticonvulsants; Bicuculline; Electroshock; Ethosuximide; Male; Mice; Pentylenetetrazole; Phenytoin; Picrotoxin; Seizures; Valproic Acid

1985
[The anticonvulsant action of propranolol in pentylenetetrazole-induced convulsions].
    Die Pharmazie, 1985, Volume: 40, Issue:4

    Topics: Animals; Anticonvulsants; Dose-Response Relationship, Drug; Ethosuximide; Male; Mice; Pentylenetetrazole; Phenobarbital; Propranolol

1985
Drug-induced catalepsy as influenced by convulsant and anticonvulsant drugs.
    Neuropharmacology, 1973, Volume: 12, Issue:8

    Topics: Animals; Anticonvulsants; Arecoline; Bemegride; Caffeine; Catalepsy; Central Nervous System Stimulants; Drug Synergism; Ethosuximide; Haloperidol; Humans; Lobeline; Male; Mice; Mice, Inbred Strains; Nicotine; Nikethamide; Paraoxon; Pentylenetetrazole; Pilocarpine; Tetrabenazine; Tremorine; Trifluoperazine

1973
Alkylation reactions of hydantoins and succinimides.
    Journal of pharmaceutical sciences, 1973, Volume: 62, Issue:11

    Topics: Alkylation; Animals; Anticonvulsants; Benzyl Compounds; Chemical Phenomena; Chemistry; Ethosuximide; Hydantoins; Magnetic Resonance Spectroscopy; Male; Mice; Nitro Compounds; Pentylenetetrazole; Phenytoin; Spectrophotometry, Infrared; Succinimides

1973
[Pharmacology of 2,4-dimethysulfolane].
    Acta biologica et medica Germanica, 1971, Volume: 26, Issue:5

    Topics: Animals; Anticonvulsants; Blood Circulation; Cats; Central Nervous System; Central Nervous System Stimulants; Electroencephalography; Ethosuximide; Guinea Pigs; Heart; Male; Mice; Pentylenetetrazole; Rats

1971
Dependence of anticonvulsant drug action on central monoamines.
    Neuropharmacology, 1973, Volume: 12, Issue:10

    Topics: Animals; Anticonvulsants; Dopamine; Drug Interactions; Electroshock; Ethosuximide; Lethal Dose 50; Male; Mice; Mice, Inbred Strains; Norepinephrine; Pentylenetetrazole; Phenobarbital; Phenytoin; Receptors, Drug; Seizures; Serotonin; Time Factors

1973
[Inhibition of pentetrazole-induced hypersynchronous activity in thalamocortical system by ethosuximide].
    Acta biologica et medica Germanica, 1971, Volume: 26, Issue:3

    Topics: Animals; Electrodes, Implanted; Electroencephalography; Ethosuximide; Male; Motor Cortex; Muscle Tonus; Olfactory Bulb; Pentylenetetrazole; Photic Stimulation; Rats; Rats, Inbred Strains; Reflex, Startle; Thalamus; Time Factors; Visual Cortex

1971
Language-induced epilepsy.
    Archives of neurology, 1967, Volume: 16, Issue:1

    Topics: Electroencephalography; Epilepsy; Ethosuximide; Humans; Male; Middle Aged; Movement Disorders; Pentylenetetrazole; Phenobarbital; Reading; Speech; Speech Disorders; Unconsciousness; Writing

1967
Excitatory and depressant effects of delta 9-tetrahydrocannabinol and cannabidiol on cortical evoked responses in the conscious rat.
    Psychopharmacology, 1981, Volume: 75, Issue:3

    Topics: Animals; Anticonvulsants; Cannabidiol; Cannabinoids; Cerebral Cortex; Convulsants; Dronabinol; Ethosuximide; Evoked Potentials; Pentylenetetrazole; Phenytoin; Rats; Rats, Inbred Strains

1981
Effect of antiepileptic drugs on metrazol convulsions during ontogenesis in the rat.
    Physiologia Bohemoslovaca, 1981, Volume: 30, Issue:2

    Topics: Age Factors; Animals; Anticonvulsants; Clonazepam; Ethosuximide; Male; Pentylenetetrazole; Rats; Seizures; Valproic Acid

1981
Influence of ethosuximide on metrazol-induced seizures during ontogenesis in rats.
    Activitas nervosa superior, 1983, Volume: 25, Issue:4

    Topics: Aging; Animals; Dose-Response Relationship, Drug; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures

1983
Influence of clonazepam and ethosuximide on ECoG pattern induced by metrazol during ontogenesis in rats.
    Activitas nervosa superior, 1982, Volume: 24, Issue:1

    Topics: Age Factors; Animals; Benzodiazepinones; Cerebral Cortex; Clonazepam; Dose-Response Relationship, Drug; Electroencephalography; Ethosuximide; Evoked Potentials; Male; Pentylenetetrazole; Rats; Seizures

1982
A behavioural and pharmacological evaluation of the discriminative stimulus induced by pentylenetetrazole in the pig.
    Psychopharmacology, 1993, Volume: 111, Issue:2

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Cues; Diazepam; Discrimination, Psychological; Electroshock; Emotions; Ethosuximide; Male; Pentylenetetrazole; Reinforcement Schedule; Swine

1993
Is the site of action of ethosuximide in the hindbrain?
    Physiological research, 1994, Volume: 43, Issue:1

    Topics: Animals; Anticonvulsants; Brain Stem; Clonazepam; Decerebrate State; Electrocardiography; Electroencephalography; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Wistar; Rhombencephalon; Seizures; Valproic Acid

1994
Ethosuximide suppresses seizures and lethality induced by picrotoxin in developing rats.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Animals; Anticonvulsants; Behavior, Animal; Epilepsies, Myoclonic; Epilepsy, Tonic-Clonic; Ethosuximide; Male; Pentylenetetrazole; Picrotoxin; Rats; Rats, Wistar; Seizures

1993
Protective effect of flunarizine and nifedipine alone and in combination with anticonvulsant drugs against PTZ-induced seizures in mice.
    Neuropharmacology, 1993, Volume: 32, Issue:3

    Topics: Animals; Anticonvulsants; Carbamazepine; Dose-Response Relationship, Drug; Drug Interactions; Ethosuximide; Female; Flunarizine; Male; Mice; Nifedipine; Pentylenetetrazole; Phenytoin; Seizures

1993
Antiepileptic drugs--their effects on kindled seizures and kindling-induced learning impairments.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:3

    Topics: Animals; Anticonvulsants; Avoidance Learning; Cognition; Dose-Response Relationship, Drug; Ethosuximide; Kindling, Neurologic; Learning Disabilities; Male; Pentylenetetrazole; Phenobarbital; Rats; Rats, Wistar; Seizures; Valproic Acid

1995
Influence of nicardipine, nimodipine and flunarizine on the anticonvulsant efficacy of antiepileptics against pentylenetetrazol in mice.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:7

    Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Clonazepam; Drug Interactions; Ethosuximide; Flunarizine; Male; Mice; Mice, Inbred Strains; Motor Activity; Nicardipine; Nimodipine; Pentylenetetrazole; Random Allocation; Seizures; Valproic Acid

1996
Ethosuximide specifically antagonizes the effect of pentylenetetrazol in the rat entorhinal cortex.
    Epilepsy research, 1996, Volume: 25, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Entorhinal Cortex; Ethosuximide; Evoked Potentials; Male; Pentylenetetrazole; Rats; Rats, Sprague-Dawley

1996
Ontogeny of ethosuximide action against two seizure models in rats is different.
    Life sciences, 1998, Volume: 63, Issue:3

    Topics: Action Potentials; Animals; Anticonvulsants; Disease Models, Animal; Electroencephalography; Ethosuximide; Pentylenetetrazole; Rats; Seizures

1998
A potential anti-asthmatic drug, CR 2039, enhances the anticonvulsive activity of some antiepileptic drugs against pentetrazol in mice.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1998, Volume: 8, Issue:3

    Topics: Animals; Anticonvulsants; Benzamides; Bronchodilator Agents; Clonazepam; Convulsants; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Ethosuximide; Male; Mice; Pentylenetetrazole; Seizures; Tetrazoles

1998
Additive anticonvulsant effect of flunarizine and sodium valproate on electroshock and chemoshock induced seizures in mice.
    Indian journal of physiology and pharmacology, 1998, Volume: 42, Issue:3

    Topics: Animals; Anticonvulsants; Carbamazepine; Disease Models, Animal; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Electroshock; Ethosuximide; Flunarizine; Male; Mice; Motor Activity; Pentylenetetrazole; Phenytoin; Seizures; Valproic Acid

1998
N(G)-nitro-L-arginine impairs the anticonvulsive action of ethosuximide against pentylenetetrazol.
    European journal of pharmacology, 1999, Feb-05, Volume: 366, Issue:2-3

    Topics: Animals; Anticonvulsants; Arginine; Convulsants; Diazepam; Drug Interactions; Enzyme Inhibitors; Ethosuximide; Male; Mice; Nitroarginine; Pentylenetetrazole; Phenobarbital; Psychomotor Performance; Seizures; Valproic Acid

1999
The fruit essential oil of Pimpinella anisum exerts anticonvulsant effects in mice.
    Journal of ethnopharmacology, 1999, Volume: 66, Issue:2

    Topics: Animals; Anticonvulsants; Apiaceae; Convulsants; Electroshock; Ethosuximide; Fruit; India; Iran; Lethal Dose 50; Male; Mice; Oils, Volatile; Pentylenetetrazole; Postural Balance; Seizures; Turkey

1999
7-Nitroindazole, a nitric oxide synthase inhibitor, enhances the anticonvulsive action of ethosuximide and clonazepam against pentylenetetrazol-induced convulsions.
    Journal of neural transmission (Vienna, Austria : 1996), 2000, Volume: 107, Issue:10

    Topics: Animals; Anticonvulsants; Avoidance Learning; Clonazepam; Disease Models, Animal; Drug Interactions; Epilepsies, Myoclonic; Ethosuximide; Indazoles; Male; Mice; Motor Skills; Neuroprotective Agents; Nitric Oxide; Nitric Oxide Synthase; Pentylenetetrazole; Seizures

2000
Comparative profiles of sodium valproate and ethosuximide on electro-behavioural correlates in gamma-hydroxybutyrate and pentylenetetrazol induced absence seizures in rats.
    Indian journal of physiology and pharmacology, 2000, Volume: 44, Issue:4

    Topics: Animals; Anticonvulsants; Convulsants; Disease Models, Animal; Electroencephalography; Epilepsy, Absence; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Wistar; Sodium Oxybate; Species Specificity; Valproic Acid

2000
Is spontaneous high-voltage rhythmic spike discharge in Long Evans rats an absence-like seizure activity?
    Journal of neurophysiology, 2004, Volume: 91, Issue:1

    Topics: Animals; Anticonvulsants; Arousal; Behavior, Animal; Cerebral Cortex; Disease Models, Animal; Electric Stimulation; Electrodes, Implanted; Electroencephalography; Electromyography; Epilepsy, Absence; Ethosuximide; Female; Immobilization; Penicillins; Pentylenetetrazole; Rats; Rats, Inbred Strains; Rats, Long-Evans; Sleep; Time Factors; Wakefulness

2004
NOTE ON THE INTERACTIONS OF AMPHETAMINE WITH ANTICONVULSANT DRUGS.
    Acta pharmacologica et toxicologica, 1964, Volume: 21

    Topics: Amphetamine; Amphetamines; Animals; Anticonvulsants; Electricity; Electroshock; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Ethosuximide; Mice; Pentylenetetrazole; Pharmacology; Phenobarbital; Phenytoin; Research; Seizures

1964
Isobolographic and subthreshold analysis of interactions among felbamate and four conventional antiepileptic drugs in pentylenetetrazole-induced seizures in mice.
    Epilepsia, 2004, Volume: 45, Issue:10

    Topics: Animals; Anticonvulsants; Behavior, Animal; Clonazepam; Disease Models, Animal; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Epilepsies, Myoclonic; Ethosuximide; Felbamate; Female; Humans; Lethal Dose 50; Mice; Motor Activity; Neurotoxicity Syndromes; Pentylenetetrazole; Phenobarbital; Phenylcarbamates; Propylene Glycols; Seizures; Valproic Acid

2004
Ethosuximide and valproate display high efficacy against lindane-induced seizures in mice.
    Toxicology letters, 2004, Dec-01, Volume: 154, Issue:1-2

    Topics: Animals; Anticonvulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethosuximide; GABA Agents; Hexachlorocyclohexane; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Mice; Pentylenetetrazole; Seizures; Valproic Acid

2004
Pharmacodynamic and/or pharmacokinetic characteristics of interactions between loreclezole and four conventional antiepileptic drugs in pentylenetetrazole-induced seizures in mice: an isobolographic analysis.
    Epilepsy & behavior : E&B, 2005, Volume: 7, Issue:4

    Topics: Animals; Anticonvulsants; Clonazepam; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Ethosuximide; Kindling, Neurologic; Linear Models; Male; Mice; Pentylenetetrazole; Phenobarbital; Seizures; Triazoles; Valproic Acid

2005
Imaging the neural substrates involved in the genesis of pentylenetetrazol-induced seizures.
    Epilepsia, 2006, Volume: 47, Issue:4

    Topics: Animals; Brain Mapping; Dentate Gyrus; Disease Models, Animal; Electroencephalography; Epilepsy, Absence; Ethosuximide; Hippocampus; Magnetic Resonance Imaging; Male; Neural Pathways; Oxygen; Pentylenetetrazole; Pilot Projects; Prosencephalon; Rats; Rats, Sprague-Dawley; Seizures; Thalamic Nuclei; Thalamus

2006
Characterization of the anticonvulsant, behavioral and pharmacokinetic interaction profiles of stiripentol in combination with clonazepam, ethosuximide, phenobarbital, and valproate using isobolographic analysis.
    Epilepsia, 2006, Volume: 47, Issue:11

    Topics: Animals; Anticonvulsants; Brain Chemistry; Clonazepam; Dioxolanes; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Ethosuximide; Male; Mice; Neurotoxicity Syndromes; Pentylenetetrazole; Phenobarbital; Seizures; Valproic Acid

2006
Thalidomide inhibits pentylenetetrazole-induced seizures.
    Journal of the neurological sciences, 2007, Jul-15, Volume: 258, Issue:1-2

    Topics: Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Ethosuximide; Male; Pentylenetetrazole; Rats; Rats, Wistar; Seizures; Severity of Illness Index; Valproic Acid

2007
Interactions of tiagabine with ethosuximide in the mouse pentylenetetrazole-induced seizure model: an isobolographic analysis for non-parallel dose-response relationship curves.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 378, Issue:5

    Topics: Animals; Anticonvulsants; Brain; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Ethosuximide; Fluorescence Polarization Immunoassay; Male; Mice; Nipecotic Acids; Pentylenetetrazole; Seizures; Tiagabine; Tissue Distribution

2008
Isobolographic characterization of the anticonvulsant interaction profiles of levetiracetam in combination with clonazepam, ethosuximide, phenobarbital and valproate in the mouse pentylenetetrazole-induced seizure model.
    Seizure, 2009, Volume: 18, Issue:9

    Topics: Animals; Anticonvulsants; Clonazepam; Convulsants; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Ethosuximide; Levetiracetam; Male; Mice; Pentylenetetrazole; Phenobarbital; Piracetam; Seizures; Valproic Acid

2009
Detection of nonlinear interactions of EEG alpha waves in the brain by a new coherence measure and its application to epilepsy and anti-epileptic drug therapy.
    International journal of neural systems, 2011, Volume: 21, Issue:2

    Topics: Animals; Anticonvulsants; Cerebral Cortex; Convulsants; Electroencephalography; Epilepsy; Ethosuximide; Humans; Mathematics; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Seizures; Thalamus

2011
Effect of intracranial administration of ethosuximide in rats with spontaneous or pentylenetetrazol-induced spike-wave discharges.
    Epilepsia, 2011, Volume: 52, Issue:7

    Topics: Animals; Anticonvulsants; Brain; Disease Models, Animal; Epilepsy, Absence; Ethosuximide; Infusions, Intraventricular; Male; Pentylenetetrazole; Rats; Rats, Long-Evans; Rats, Wistar

2011
Effects of WIN 55,212-2 mesylate (a synthetic cannabinoid) on the protective action of clonazepam, ethosuximide, phenobarbital and valproate against pentylenetetrazole-induced clonic seizures in mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2011, Dec-01, Volume: 35, Issue:8

    Topics: Animals; Anticonvulsants; Avoidance Learning; Benzoxazines; Brain; Cannabinoid Receptor Agonists; Clonazepam; Disease Models, Animal; Drug Synergism; Ethosuximide; Hand Strength; Male; Mice; Morpholines; Naphthalenes; Pentylenetetrazole; Phenobarbital; Seizures; Valproic Acid

2011
Synthesis and anticonvulsant activity of new 1-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-diones.
    Bioorganic & medicinal chemistry letters, 2011, Oct-01, Volume: 21, Issue:19

    Topics: Administration, Oral; Animals; Anticonvulsants; Convulsants; Dose-Response Relationship, Drug; Drug Design; Drug Evaluation, Preclinical; Electroshock; Ethosuximide; Injections, Intraperitoneal; Mice; Molecular Structure; Motor Activity; Pentylenetetrazole; Phenytoin; Piperazines; Rats; Seizures; Structure-Activity Relationship; Succinimides; Time Factors

2011
Anticonvulsant effect of the essential oil and methanolic extracts of Zataria multiflora Boiss.
    Central nervous system agents in medicinal chemistry, 2013, Volume: 13, Issue:2

    Topics: Animals; Anticonvulsants; Distillation; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Electroshock; Ethosuximide; Injections, Intraperitoneal; Lamiaceae; Male; Methanol; Mice; Oils, Volatile; Pentylenetetrazole; Phenytoin; Phytotherapy; Plant Extracts; Plant Oils; Plants, Medicinal; Postural Balance; Rotarod Performance Test; Seizures; Sesame Oil; Solvents

2013
Synthesis, physicochemical, and anticonvulsant properties of new N-Mannich bases derived from pyrrolidine-2,5-dione and its 3-methyl analog.
    Archiv der Pharmazie, 2014, Volume: 347, Issue:10

    Topics: Animals; Anticonvulsants; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Design; Electroshock; Ethosuximide; Male; Mannich Bases; Mice; Molecular Structure; Motor Activity; Neurotoxicity Syndromes; Pentylenetetrazole; Pyrrolidines; Rotarod Performance Test; Seizures; Structure-Activity Relationship; Valproic Acid

2014
Potential mechanisms involved in the anticonvulsant effect of walnut extract on pentylenetetrazole-induced seizure.
    Medical principles and practice : international journal of the Kuwait University, Health Science Centre, 2014, Volume: 23, Issue:6

    Topics: Animals; Anticonvulsants; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Ethosuximide; Flumazenil; Juglans; Male; Pentylenetetrazole; Plant Extracts; Rats; Rats, Wistar; Seizures

2014
Ethosuximide Reduces Mortality and Seizure Severity in Response to Pentylenetetrazole Treatment During Ethanol Withdrawal.
    Alcohol and alcoholism (Oxford, Oxfordshire), 2015, Volume: 50, Issue:5

    Topics: Alcoholism; Animals; Anticonvulsants; Ethosuximide; Male; Mice; Mice, Inbred DBA; Mortality; Pentylenetetrazole; Seizures; Severity of Illness Index; Substance Withdrawal Syndrome

2015
Interactions between an antidepressant reboxetine and four classic antiepileptic drugs in the mouse model of myoclonic seizures.
    Pharmacological reports : PR, 2015, Volume: 67, Issue:6

    Topics: Animals; Anticonvulsants; Antidepressive Agents; Avoidance Learning; Clonazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Epilepsies, Myoclonic; Ethosuximide; Male; Mice; Morpholines; Motor Skills; Pentylenetetrazole; Phenobarbital; Reboxetine; Valproic Acid

2015
A Caenorhabditis elegans assay of seizure-like activity optimised for identifying antiepileptic drugs and their mechanisms of action.
    Journal of neuroscience methods, 2018, 11-01, Volume: 309

    Topics: Animals; Anticonvulsants; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Convulsants; Disease Models, Animal; Drug Evaluation, Preclinical; Ethosuximide; Pentylenetetrazole; Receptors, GABA-A; Seizures

2018
N-Benzyl-(2,5-dioxopyrrolidin-1-yl)propanamide (AS-1) with Hybrid Structure as a Candidate for a Broad-Spectrum Antiepileptic Drug.
    Neurotherapeutics : the journal of the American Society for Experimental NeuroTherapeutics, 2020, Volume: 17, Issue:1

    Topics: Animals; Anticonvulsants; Behavior, Animal; Dose-Response Relationship, Drug; Epilepsy; Ethosuximide; Lacosamide; Levetiracetam; Male; Mice; Pentylenetetrazole; Pyrrolidines; Seizures; Valproic Acid; Zebrafish

2020
Evaluation of the impact of compound C11 a new anticonvulsant candidate on cognitive functions and hippocampal neurogenesis in mouse brain.
    Neuropharmacology, 2020, Volume: 163

    Topics: Animals; Anticonvulsants; Brain; Cognition; Epilepsy; Ethosuximide; Hippocampus; Lacosamide; Levetiracetam; Male; Mice; Mice, Inbred C57BL; Neurogenesis; Pentylenetetrazole; Spatial Memory

2020
Long-term vigabatrin treatment modifies pentylenetetrazole-induced seizures in mice: focused on GABA brain concentration.
    Pharmacological reports : PR, 2020, Volume: 72, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Brain; Clonazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethosuximide; gamma-Aminobutyric Acid; Mice; Pentylenetetrazole; Seizures; Time Factors; Valproic Acid; Vigabatrin

2020
Anticonvulsant activity of Valeriana edulis roots and valepotriates on the pentylenetetrazole-induced seizures in rats.
    Journal of ethnopharmacology, 2021, Jan-30, Volume: 265

    Topics: Animals; Anticonvulsants; Computer Simulation; Disease Models, Animal; Electroencephalography; Ethosuximide; Iridoids; Male; Pentylenetetrazole; Plant Extracts; Plant Roots; Rats; Rats, Wistar; Seizures; Time Factors; Valerian

2021
Mechanochemical synthesis and anticonvulsant activity of 3-aminopyrrolidine-2,5-dione derivatives.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2023, Volume: 168

    Topics: Animals; Anticonvulsants; Ethosuximide; Humans; Mice; Molecular Structure; Neuroblastoma; Pentylenetetrazole; Seizures; Spectroscopy, Fourier Transform Infrared; Structure-Activity Relationship

2023
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