pentobarbital and baclofen

pentobarbital has been researched along with baclofen in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199011 (28.95)18.7374
1990's19 (50.00)18.2507
2000's4 (10.53)29.6817
2010's4 (10.53)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Cankaya, A; Gepdiremen, A; Kutlu, N; Tan, U2
Bartolini, A; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P1
Gautam, SK; Kulkarni, SK1
Ho, IK; Kimura, T; Saunders, PA; Yamamoto, I1
Asprodini, EK; Rainnie, DG; Shinnick-Gallagher, P1
Miledi, R; Polenzani, L; Woodward, RM1
Araki, T; Kato, H; Kogure, K1
Hori, S; Ito, T; Kadokawa, T; Miura, Y; Miyahara, T; Shimada, J1
Ferrendelli, JA; Miller, JW1
Friedman, DL; Redburn, DA1
Kim, KH; Takeuchi, H1
Shimizu, M; Yamamoto, M1
Holden-Dye, L; Krogsgaard-Larsen, P; Nielsen, L; Walker, RJ1
Kontani, H; Nakagawa, M; Sakai, T1
Goodwin, GM; Gray, JA; Green, AR; Heal, DJ1
Georgiev, V; Getova, D1
Mehta, AK; Ticku, MK1
Iwai, S; Shirakawa, J; Tanaka, C; Taniyama, K1
Chweh, AY; Swinyard, EA; Wolf, HH1
Herling, S; Valentino, RJ; Winger, GD1
Lake, N; Potashner, SJ1
George, B; Kulkarni, SK1
Belachew, S; Coucke, P; Goffin, F; Lefebvre, PP; Malgrange, B; Moonen, G; Rigo, JM; Van de Water, TR; Xhauflaire, G1
Curtis, DR; Lacey, G1
Isshiki, A; Ito, H; Uchino, H; Watanabe, Y1
Davidoff, RA; Hackman, JC; Holohean, AM; Katz, JL; Valeyev, AY; Wood, PM1
Chen, CL; Chiu, TH; Yang, YR1
Huang, XL; Osawa, M; Saito, T; Takeichi, S; Yamamoto, I; Yukawa, N1
Advokat, C; Duke, M1
Menzikov, S; Menzikova, O1
Ariwodola, OJ; Weiner, JL1
Archer, DP; Nguyen, KQ; Roth, SH; Samanani, N1
Brogi, S; Carai, MA; Castelli, MP; Casti, P; Casu, A; Colombo, G; Corelli, F; Gessa, GL; Giunta, D; Lobina, C; Mugnaini, C; Pasquini, S; Solinas, M; Tafi, A1
Castelli, MP; Casti, A; Casu, A; Colombo, G; Corelli, F; Dragoni, S; Gessa, GL; Giunta, D; Lamponi, S; Lobina, C; Maccioni, P; Mugnaini, C; Pedani, V; Porcu, A; Solinas, M; Valoti, M1

Reviews

1 review(s) available for pentobarbital and baclofen

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

37 other study(ies) available for pentobarbital and baclofen

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Parkinsonian-like tremor induced by a combined application of chlorpromazine and pentobarbitone in cats with left-paw preference.
    The International journal of neuroscience, 1992, Volume: 63, Issue:3-4

    Topics: Animals; Atropine; Baclofen; Biperiden; Cats; Chlorpromazine; Feedback; Female; Functional Laterality; Male; Parkinson Disease, Secondary; Pentobarbital; Tremor

1992
Desensitization of GABAB receptors and antagonism by CGP 35348, prevent bicuculline- and picrotoxin-induced antinociception.
    Neuropharmacology, 1992, Volume: 31, Issue:8

    Topics: Analgesics; Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Drug Tolerance; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Mice; Motor Activity; Organophosphorus Compounds; Pain Measurement; Pentobarbital; Picrotoxin; Postural Balance; Rats; Rats, Inbred Strains; Receptors, GABA-A

1992
GABA/BZ-and NMDA-receptor interaction in digoxin-induced convulsions in rats.
    Indian journal of experimental biology, 1991, Volume: 29, Issue:7

    Topics: Animals; Baclofen; Diazepam; Digoxin; Dizocilpine Maleate; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Salts; Seizures

1991
Effects of pentobarbital tolerance to and dependence on GABAB receptor-binding.
    Neurochemical research, 1991, Volume: 16, Issue:10

    Topics: Animals; Baclofen; Cerebellum; Cerebral Cortex; Drug Tolerance; Kinetics; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values

1991
Inhibitory transmission in the basolateral amygdala.
    Journal of neurophysiology, 1991, Volume: 66, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Neural Inhibition; Pentobarbital; Potassium; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

1991
Expression of mammalian gamma-aminobutyric acid receptors with distinct pharmacology in Xenopus oocytes.
    Proceedings of the National Academy of Sciences of the United States of America, 1991, May-15, Volume: 88, Issue:10

    Topics: Animals; Baclofen; Bicuculline; Cattle; Cerebral Cortex; Electric Conductivity; gamma-Aminobutyric Acid; Gene Expression; Membrane Potentials; Oocytes; Pentobarbital; Picrotoxin; Poly A; Rats; Receptors, GABA-A; Retina; RNA; RNA, Messenger; Transfection; Xenopus

1991
Comparative protective effects of vinconate, baclofen, and pentobarbital against neuronal damage following repeated brief cerebral ischemia in the gerbil brain.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:6

    Topics: Animals; Baclofen; Behavior, Animal; Body Temperature; Brain Ischemia; Gerbillinae; Male; Neurons; Pentobarbital; Vinca Alkaloids

1991
A simple tremor model induced by pentobarbitone in guinea pig.
    The International journal of neuroscience, 1991, Volume: 61, Issue:1-2

    Topics: Animals; Baclofen; Biperiden; Electromyography; Guinea Pigs; Pentobarbital; Transducers; Tremor

1991
Effects of enoxacin and its combination with 4-biphenylacetate, an active metabolite of fenbufen, on population spikes in rat hippocampal slices.
    Pharmacology & toxicology, 1991, Volume: 68, Issue:3

    Topics: Action Potentials; Animals; Anti-Inflammatory Agents, Non-Steroidal; Baclofen; Bicuculline; Clorazepate Dipotassium; Drug Interactions; Electric Stimulation; Enoxacin; Hippocampus; In Vitro Techniques; Male; Muscimol; Pentobarbital; Phenylacetates; Phenylbutyrates; Rats; Rats, Inbred Strains

1991
Characterization of GABAergic seizure regulation in the midline thalamus.
    Neuropharmacology, 1990, Volume: 29, Issue:7

    Topics: Animals; Baclofen; Bicuculline; Electroencephalography; Epilepsy; Female; Flurazepam; gamma-Aminobutyric Acid; Pentobarbital; Pentylenetetrazole; Piperidines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thalamic Nuclei

1990
Evidence for functionally distinct subclasses of gamma-aminobutyric acid receptors in rabbit retina.
    Journal of neurochemistry, 1990, Volume: 55, Issue:4

    Topics: Acetylcholine; Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Binding, Competitive; Cell Fractionation; Flurazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Light; Models, Theoretical; Pentobarbital; Picrotoxin; Rabbits; Receptors, GABA-A; Retina

1990
Pharmacological characteristics of two different types of inhibitory GABA receptors on Achatina fulica neurones.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Crotonates; Diazepam; Dibenzazepines; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Neurons; Pentobarbital; Picrotoxin; Receptors, GABA-A; Snails

1990
Effects of a new analogue of thyrotropin-releasing hormone on pentobarbital-induced sleeping time in rodents.
    Neuropharmacology, 1989, Volume: 28, Issue:8

    Topics: Animals; Atropine; Azetidines; Azetines; Baclofen; Dipeptides; Haloperidol; Injections, Intramuscular; Injections, Intravenous; Male; Mice; Mice, Inbred ICR; Pentobarbital; Phentolamine; Rats; Sleep; Thyrotropin-Releasing Hormone; Time Factors

1989
GABA receptors on the somatic muscle cells of the parasitic nematode, Ascaris suum: stereoselectivity indicates similarity to a GABAA-type agonist recognition site.
    British journal of pharmacology, 1989, Volume: 98, Issue:3

    Topics: Animals; Ascaris; Baclofen; Binding, Competitive; Dieldrin; Electric Stimulation; Flurazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Muscles; Pentobarbital; Receptors, GABA-A; Stereoisomerism

1989
Effects of central nervous system-acting drugs on urinary bladder contraction in unanesthetized rats.
    Japanese journal of pharmacology, 1989, Volume: 50, Issue:3

    Topics: Anesthesia; Animals; Baclofen; Behavior, Animal; Central Nervous System Agents; Diazepam; Male; Morphine; Muscle Contraction; Muscle, Smooth; Pentobarbital; Rats; Rats, Inbred Strains; Urinary Bladder; Urination

1989
Hypothermia induced by baclofen, a possible index of GABAB receptor function in mice, is enhanced by antidepressant drugs and ECS.
    British journal of pharmacology, 1987, Volume: 92, Issue:4

    Topics: 5,7-Dihydroxytryptamine; Amitriptyline; Animals; Antidepressive Agents; Baclofen; Body Temperature; Electroshock; Flurazepam; Hypnotics and Sedatives; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Neural Pathways; Pentobarbital; Receptors, GABA-A

1987
GABA-ergic mechanisms in the anticonvulsive activity of newly synthesized barbiturates. II. Correlation of HB-7 with GABA-ergic agents.
    Acta physiologica et pharmacologica Bulgarica, 1988, Volume: 14, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Mice; Muscimol; Pentobarbital; Receptors, GABA-A

1988
Interactions of pentobarbital and phenobarbital with GABAergic drugs against chemoconvulsants in rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Convulsants; Diazepam; Drug Interactions; Isoxazoles; Male; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Strychnine

1988
Regulation of [3H]GABA release from strips of guinea pig urinary bladder.
    The American journal of physiology, 1988, Volume: 255, Issue:6 Pt 2

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Bicuculline; Clonazepam; Clonidine; Female; gamma-Aminobutyric Acid; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Male; Muscimol; Pentobarbital; Phenylephrine; Pirenzepine; Potassium; Prazosin; Tritium; Urinary Bladder; Yohimbine

1988
Hypnotic action of pentobarbital in mice: a possible mechanism.
    Experimental neurology, 1987, Volume: 97, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Isoxazoles; Male; Mice; Oxazoles; Pentobarbital; Receptors, GABA-A; Reflex; Sleep

1987
Discriminative stimulus effects of pentobarbital in pigeons.
    Psychopharmacology, 1980, Volume: 71, Issue:1

    Topics: Animals; Baclofen; Bemegride; Columbidae; Ethanol; gamma-Aminobutyric Acid; Muscimol; Pentobarbital; Prejudice

1980
Action of baclofen and pentobarbital on amino acid release.
    Advances in biochemical psychopharmacology, 1981, Volume: 27

    Topics: Amino Acids; Animals; Baclofen; Cerebral Cortex; Electric Stimulation; Humans; Pentobarbital

1981
Protective effects of GABAergic drugs and other anticonvulsants in lithium-pilocarpine-induced status epilepticus.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:5

    Topics: Animals; Anticonvulsants; Baclofen; Clonazepam; Diazepam; Dizocilpine Maleate; Ethanol; GABA Agents; gamma-Aminobutyric Acid; Lithium Chloride; Male; Neuroprotective Agents; Pentobarbital; Phenobarbital; Phenytoin; Pilocarpine; Rats; Rats, Wistar; Status Epilepticus; Valproic Acid

1996
Diazepam-insensitive GABAA receptors on postnatal spiral ganglion neurones in culture.
    Neuroreport, 1997, Feb-10, Volume: 8, Issue:3

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Carbolines; Cells, Cultured; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Spiral Ganglion; Zinc

1997
Prolonged GABA(B) receptor-mediated synaptic inhibition in the cat spinal cord: an in vivo study.
    Experimental brain research, 1998, Volume: 121, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrophysiology; Female; GABA Agonists; GABA Antagonists; GABA Modulators; Male; Membrane Potentials; Motor Neurons; Neural Inhibition; Pentobarbital; Phosphinic Acids; Propanolamines; Receptors, GABA-A; Receptors, GABA-B; Reflex; Spinal Cord; Synapses

1998
Neuroprotective properties of propofol and midazolam, but not pentobarbital, on neuronal damage induced by forebrain ischemia, based on the GABAA receptors.
    Acta anaesthesiologica Scandinavica, 1999, Volume: 43, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Baclofen; Brain Ischemia; Dose-Response Relationship, Drug; GABA Agonists; GABA Modulators; Gerbillinae; Histocytochemistry; Male; Midazolam; Muscimol; Neurons; Neuroprotective Agents; Pentobarbital; Propofol; Prosencephalon; Receptors, GABA-A; Reperfusion Injury

1999
GABA-Induced Cl- current in cultured embryonic human dorsal root ganglion neurons.
    Journal of neurophysiology, 1999, Volume: 82, Issue:1

    Topics: Adult; Baclofen; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chloride Channels; Convulsants; Crotonates; Embryo, Mammalian; gamma-Aminobutyric Acid; Ganglia, Spinal; Glycine; Humans; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pentobarbital; Potassium Channels; Pregnanediones; Receptors, GABA-A; Taurine

1999
Activation of rat locus coeruleus neuron GABA(A) receptors by propofol and its potentiation by pentobarbital or alphaxalone.
    European journal of pharmacology, 1999, Dec-15, Volume: 386, Issue:2-3

    Topics: Anesthetics; Anesthetics, Intravenous; Animals; Baclofen; Barium Compounds; Bicuculline; Chlorides; Diazepam; Drug Synergism; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ionophores; Locus Coeruleus; Male; Neurons; Pentobarbital; Picrotoxin; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zinc Compounds

1999
Effects of muscle relaxants on EEG, ABR and EMG in rabbits.
    Human & experimental toxicology, 1999, Volume: 18, Issue:12

    Topics: Acoustic Stimulation; Anesthesia; Animals; Baclofen; Dose-Response Relationship, Drug; Electric Stimulation; Electroencephalography; Electromyography; Evoked Potentials; Evoked Potentials, Auditory, Brain Stem; Male; Muscle Relaxants, Central; Neuromuscular Nondepolarizing Agents; Pancuronium; Pentobarbital; Rabbits; Reaction Time

1999
Pentobarbital-induced modulation of flexor and H-reflexes in spinal rats.
    Brain research, 2000, Oct-27, Volume: 881, Issue:2

    Topics: Adjuvants, Anesthesia; Animals; Baclofen; Electric Stimulation; H-Reflex; Male; Muscle Relaxants, Central; Pentobarbital; Rats; Rats, Sprague-Dawley; Reflex; Spinal Cord Injuries

2000
Interaction of pentobarbital with gabaergic drugs acting on the Cl(-)-ATPase activity of the plasma membranes from bream brain (Abramis brama L.).
    Neuroscience letters, 2002, Dec-16, Volume: 334, Issue:3

    Topics: Adenosine Triphosphatases; Animals; Anion Transport Proteins; Baclofen; Bicuculline; Brain; Cell Membrane; Chlorides; Dose-Response Relationship, Drug; Drug Interactions; GABA Agents; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Pentobarbital; Picrotoxin; Receptors, GABA-A; Sea Bream

2002
Ethanol potentiation of GABAergic synaptic transmission may be self-limiting: role of presynaptic GABA(B) receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Nov-24, Volume: 24, Issue:47

    Topics: Animals; Autoreceptors; Baclofen; Bicuculline; Central Nervous System Depressants; Electric Stimulation; Electrophysiology; Ethanol; Flunitrazepam; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Male; Morpholines; Neural Inhibition; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission

2004
Pentobarbital enhances gamma-aminobutyric acid-mediated excitation without altering synaptic plasticity in rat hippocampus.
    Anesthesia and analgesia, 2007, Volume: 104, Issue:4

    Topics: Adjuvants, Anesthesia; Animals; Baclofen; Bicarbonates; Bicuculline; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Neuronal Plasticity; Neurons; Pentobarbital; Rats; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Time Factors

2007
Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA(B) receptor.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:3

    Topics: Adamantane; Allosteric Regulation; Animals; Baclofen; Binding Sites; GABA Modulators; Guanosine 5'-O-(3-Thiotriphosphate); Male; Mice; Mice, Inbred DBA; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Thiophenes

2012
Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor.
    Journal of medicinal chemistry, 2013, May-09, Volume: 56, Issue:9

    Topics: Administration, Oral; Allosteric Regulation; Animals; Baclofen; Chemistry Techniques, Synthetic; Drug Design; Drug Stability; Guanosine 5'-O-(3-Thiotriphosphate); Immobility Response, Tonic; Mice; Microsomes, Liver; NIH 3T3 Cells; Pentobarbital; Rats; Receptors, GABA-B; Thiophenes

2013